Karl Barry Sharpless
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American chemist and Nobel Laureate
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Karl Barry Sharplesschemistry Degrees
Chemistry
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#90
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#16
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Organic Chemistry
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#18
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Chemistry
Karl Barry Sharpless's Degrees
- Bachelors Chemistry Dartmouth College
- PhD Chemistry Stanford University
Why Is Karl Barry Sharpless Influential?
(Suggest an Edit or Addition)According to Wikipedia, Karl Barry Sharpless is an American stereochemist. He is a two-time Nobel laureate in Chemistry known for his work on stereoselective reactions and click chemistry. Sharpless was awarded half of the 2001 Nobel Prize in Chemistry "for his work on chirally catalysed oxidation reactions", and one third of the 2022 prize, jointly with Carolyn R. Bertozzi and Morten P. Meldal, "for the development of click chemistry and bioorthogonal chemistry". Sharpless is the fifth person , to have twice been awarded a Nobel prize, along with Marie Curie, John Bardeen, Linus Pauling and Frederick Sanger, and the third to have been awarded two prizes in the same discipline .
Karl Barry Sharpless's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Click Chemistry: Diverse Chemical Function from a Few Good Reactions. (2001) (9531)
- A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. (2002) (8851)
- Catalytic Asymmetric Dihydroxylation (1994) (2645)
- The growing impact of click chemistry on drug discovery. (2003) (2514)
- Catalytic asymmetric epoxidation and kinetic resolution: modified procedures including in situ derivatization (1987) (1526)
- Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. (2003) (1359)
- Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates. (2004) (1345)
- "On water": unique reactivity of organic compounds in aqueous suspension. (2005) (1288)
- A greatly improved procedure for ruthenium tetroxide catalyzed oxidations of organic compounds (1981) (1266)
- Polytriazoles as copper(I)-stabilizing ligands in catalysis. (2004) (1174)
- The Osmium-Catalyzed Asymmetric Dihydroxylation: A New Ligand Class and a Process Improvement (1992) (1100)
- Efficiency and fidelity in a click-chemistry route to triazole dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. (2004) (980)
- Preparation of 5-substituted 1H-tetrazoles from nitriles in water. (2001) (783)
- The first practical method for asymmetric epoxidation (1980) (605)
- Kinetic resolution of racemic allylic alcohols by enantioselective epoxidation. A route to substances of absolute enantiomeric purity (1981) (588)
- High stereo- and regioselectivities in the transition metal catalyzed epoxidations of olefinic alcohols by tert-butyl hydroperoxide (1973) (585)
- Click chemistry in situ: acetylcholinesterase as a reaction vessel for the selective assembly of a femtomolar inhibitor from an array of building blocks. (2002) (584)
- Asymmetric dihydroxylation via ligand-accelerated catalysis (1988) (530)
- Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry. (2014) (507)
- Catalytic Asymmetric Aminohydroxylation (AA) of Olefins (1996) (483)
- Inhibitors of HIV-1 protease by using in situ click chemistry. (2006) (447)
- Ligand‐Accelerated Catalysis (1995) (420)
- Vicinal diol cyclic sulfates. Like epoxides only more reactive (1988) (417)
- Searching for new reactivity (Nobel lecture). (2002) (404)
- Allylic oxidation of olefins by catalytic and stoichiometric selenium dioxide with tert-butyl hydroperoxide (1977) (398)
- Mild procedure for the conversion of epoxides to allylic alcohols. First organoselenium reagent (1973) (397)
- Multivalent, bifunctional dendrimers prepared by click chemistry. (2005) (371)
- A Potent and Highly Selective Inhibitor of Human α-1,3-Fucosyltransferase via Click Chemistry (2003) (369)
- A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-sulfonyl tetrazoles from azides and sulfonyl cyanides. (2002) (351)
- Electrophilic and nucleophilic organoselenium reagents. New routes to .alpha.,.beta.-unsaturated carbonyl compounds (1973) (350)
- Click chemistry in materials synthesis. 1. Adhesive polymers from copper‐catalyzed azide‐alkyne cycloaddition (2004) (346)
- Procedure for the catalytic asymmetric epoxidation of allylic alcohols in the presence of molecular sieves (1986) (343)
- In situ click chemistry: enzyme inhibitors made to their own specifications. (2004) (342)
- Highly Efficient Epoxidation of Olefins Using Aqueous H2O2 and Catalytic Methyltrioxorhenium/Pyridine: Pyridine-Mediated Ligand Acceleration (1997) (319)
- Why is tetrazole formation by addition of azide to organic nitriles catalyzed by zinc(II) salts? (2003) (286)
- In situ selection of lead compounds by click chemistry: target-guided optimization of acetylcholinesterase inhibitors. (2005) (273)
- Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation. (2004) (270)
- Ruthenium-catalyzed cycloaddition of alkynes and organic azides. (2006) (263)
- Asymmetric epoxidation provides shortest routes to four chiral epoxy alcohols which are key intermediates in syntheses of methymycin, erythromycin, leukotriene C-1, and disparlure (1981) (263)
- Titanium isopropoxide-mediated nucleophilic openings of 2,3-epoxy alcohols. A mild procedure for regioselective ring-opening (1985) (261)
- Mechanisms of tetrazole formation by addition of azide to nitriles. (2002) (260)
- Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling selectivity. (2007) (251)
- Chromyl chloride oxidations of olefins. Possible role of organometallic intermediates in the oxidations of olefins by oxo transition metal species (1977) (250)
- Ti(O-i-Pr)4-mediated nucleophilic openings of 2,3-epoxy alcohols. A mild procedure for regioselective ring-opening (1985) (247)
- Mechanism of asymmetric epoxidation. 2. Catalyst structure (1991) (232)
- Olefin synthesis. Rate enhancement of the elimination of alkyl aryl selenoxides by electron-withdrawing substituents (1975) (226)
- A simplified procedure for the stereospecific transformation of 1,2-diols into epoxides (1992) (221)
- Total Synthesis of the L-Hexoses (1983) (219)
- Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. (2004) (219)
- An intramolecular [2 + 3] cycloaddition route to fused 5-heterosubstituted tetrazoles. (2001) (216)
- Bromine-Catalyzed Aziridination of Olefins. A Rare Example of Atom-Transfer Redox Catalysis by a Main Group Element (1998) (209)
- A New Ligand Class for the Asymmetric Dihydroxylation of Olefins (1996) (209)
- Synthetic applications of arylselenenic and arylseleninic acids. Conversion of olefins to allylic alcohols and epoxides (1978) (200)
- Asymmetric induction in the reaction of osmium tetroxide with olefins (1980) (197)
- In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II. (2004) (195)
- Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalization. (2006) (186)
- Selenium dioxide oxidation of olefins. Evidence for the intermediacy of allylseleninic acids (1972) (186)
- A Sulfilimine Bond Identified in Collagen IV (2009) (185)
- Mechanism of epoxidation of olefins by covalent peroxides of molybdenum(VI) (1972) (181)
- Nucleophilic opening of 2,3-epoxy acids and amides mediated by titanium isopropoxide. Highly enhanced C-3 selectivity (1985) (177)
- Stereo and regioselective openings of chiral 2,3-epoxy alcohols. Versatile routes to optically pure natural products and drugs. Unusual kinetic resolutions (1983) (174)
- Synthesis of saccharides and related polyhydroxylated natural products. 2. Simple deoxyalditols (1982) (173)
- Mechanistic studies on the Cu-catalyzed three-component reactions of sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. (2008) (168)
- Selective asymmetric dihydroxylation (AD) of dienes (1992) (163)
- Mechanism of the molybdenum and vanadium catalyzed epoxidation of olefins by alkyl hydroperoxides (1977) (163)
- New ligands double the scope of the catalytic asymmetric dihydroxylation of olefins (1991) (159)
- An Expedient Route to the Tetrazole Analogues of α-Amino Acids (2002) (156)
- Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation (AD). 1. Kinetics (1994) (155)
- SuFEx-based synthesis of polysulfates. (2014) (152)
- Arenesulfonate derivatives of homochiral glycidol: versatile chiral building blocks for organic synthesis (1989) (151)
- From Styrenes to Enantiopure α-Arylglycines in Two Steps (1998) (150)
- Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr Residue. (2016) (148)
- Lower valent tungsten halides. New class of reagents for deoxygenation of organic molecules (1972) (147)
- Experimental and Theoretical Kinetic Isotope Effects for Asymmetric Dihydroxylation. Evidence Supporting a Rate-Limiting “(3 + 2)” Cycloaddition (1997) (147)
- Cyclic sulfates containing acid-sensitive groups and chemoselective hydrolysis of sulfate esters (1989) (147)
- Improved enantioselectivity in asymmetric dihydroxylations of terminal olefins using pyrimidine ligands (1993) (145)
- Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the synthesis of polysulfates and polysulfonates. (2017) (145)
- "Inverse Drug Discovery" Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates. (2018) (142)
- Chiral hydroxamic acids as ligands in the vanadium catalyzed asymmetric epoxidation of allylic alcohols by tert-butyl hydroperoxide (1977) (141)
- In situ click chemistry: a powerful means for lead discovery (2006) (141)
- Efficient synthesis of 2-substituted-1,2,3-triazoles. (2008) (140)
- Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks (2002) (140)
- Regioselective azide opening of 2,3-epoxy alcohols by [Ti(O-i-Pr)2(N3)2]: synthesis of .alpha.-amino acids (1988) (139)
- Mechanism of asymmetric epoxidation. 1. Kinetics (1991) (137)
- Asymmetric epoxidation of allyl alcohol: efficient routes to homochiral .beta.-adrenergic blocking agents (1986) (135)
- A SIMPLE AND EFFICIENT METHOD FOR EPOXIDATION OF TERMINAL ALKENES (1997) (135)
- Synthesis of dioxobis(tert-alkylimido)osmium(VIII) and oxotris(tert-alkylimido)osmium(VIII) complexes. Stereospecific vicinal diamination of olefins (1977) (133)
- Bringing Efficiency to Materials Synthesis: The Philosophy of Click Chemistry (2007) (133)
- Selective transformations of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-3 or carbon-2 (1985) (132)
- Anhydrous tert-butyl hydroperoxide in toluene: the preferred reagent for applications requiring dry TBHP (1983) (131)
- Selective transformation of 2,3-epoxy alcohols and related derivatives. Strategies for nucleophilic attack at carbon-1 (1985) (131)
- Stereoselective epoxidations of acyclic allylic alcohols by transition metal--hydroperoxide reagents. Synthesis of dl-C18 Cecropia juvenile hormone from farnesol. (1974) (129)
- Osmium‐Catalyzed Vicinal Oxyamination of Olefins by Chloramine‐T: cis‐2‐(p‐Toluenesulfonamido)Cyclohexanol and 2‐Methyl‐3‐(p‐Toluenesulfonamido)‐2‐Pentanol (2003) (128)
- On the mechanism of titanium-tartrate catalyzed asymmetric epoxidation (1983) (124)
- Modular click chemistry libraries for functional screens using a diazotizing reagent (2019) (123)
- Aromatic sulfonyl fluorides covalently kinetically stabilize transthyretin to prevent amyloidogenesis while affording a fluorescent conjugate. (2013) (121)
- Asymmetric epoxidation of homoallylic alcohols. Synthesis of (-)-γ-amino-β(R)-hydroxybutyric acid (GABOB) (1984) (120)
- Copper(I)-catalyzed cycloaddition of organic azides and 1-iodoalkynes. (2010) (120)
- .alpha.-Hydroxy ketones in high enantiomeric purity from asymmetric dihydroxylation of enol ethers (1992) (119)
- SuFEx Click Chemistry Enabled Late-Stage Drug Functionalization. (2018) (119)
- N‐Halocarbamate Salts Lead to More Efficient Catalytic Asymmetric Aminohydroxylation (1996) (118)
- Iterative in situ click chemistry creates antibody-like protein-capture agents. (2009) (118)
- Asymmetric synthesis of both enantiomers of tomoxetine and fluoxetine. Selective reduction of 2,3-epoxycinnamyl alcohol with Red-Al (1988) (116)
- A SIMPLE AND EFFICIENT METHOD FOR THE PREPARATION OF PYRIDINE N-OXIDES (1998) (111)
- Osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide under alkaline conditions (1976) (110)
- GENERAL METHOD FOR DETERMINING ABSOLUTE CONFIGURATION OF ACYCLIC ALLYLIC ALCOHOLS (1982) (106)
- Polytriazoles as Copper(I)‐Stabilizing Ligands in Catalysis. (2004) (105)
- Stereoselective epoxidation of acyclic allylic alcohols. A correction of our previous work. (1979) (104)
- New Structural Scaffolds for Centrally Acting Oxime Reactivators of Phosphylated Cholinesterases* (2011) (104)
- Palladium-catalyzed, ligand-free Suzuki reaction in water using aryl fluorosulfates. (2015) (104)
- Allylic amination of olefins and acetylenes by imido selenium compounds (1976) (103)
- Preclusion of the “second cycle” in the osmium-catalyzed asymmetric dihydroxylation of olefins leads to a superior process (1990) (102)
- Reactions of selenoxides: Thermal -elimination and H218O exchange. (1973) (101)
- A general approach to γ-lactones via osmium-catalyzed asymmetric dihydroxylation. Synthesis of (−)- and (+)-muricatacin. (1992) (101)
- Syntheses and crystal structures of the cinchona alkaloid derivatives used as ligands in the osmium-catalyzed asymmetric dihydroxylation of olefins (1993) (100)
- Selective asymmetric dihydroxylation of polyenes (1995) (98)
- N‐Bromoacetamide—A New Nitrogen Source for the Catalytic Asymmetric Aminohydroxylation of Olefins (1997) (98)
- Catalytic asymmetric dihydroxylation of tetrasubstituted olefins (1992) (98)
- Large-scale and highly enantioselective synthesis of the taxol C-13 side chain through asymmetric dihydroxylation (1994) (98)
- One pot synthesis of homochiral aziridines and aminoalcohols from homochiral 1,2-cyclic sulfates (1989) (96)
- Electrophilic organoselenium reagents. New route to allylic acetates and ethers (1974) (95)
- Role of Architecture and Molecular Weight in the Formation of Tailor-Made Ultrathin Multilayers Using Dendritic Macromolecules and Click Chemistry (2007) (94)
- A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry. (2016) (92)
- Refinement of Structural Leads for Centrally Acting Oxime Reactivators of Phosphylated Cholinesterases* (2012) (90)
- The copper-mediated cross-coupling of phenylboronic acids and N-hydroxyphthalimide at room temperature: synthesis of aryloxyamines. (2001) (89)
- A Solid-to-Solid Asymmetric Dihydroxylation Procedure for Kilogram-Scale Preparation of Enantiopure Hydrobenzoin (1994) (89)
- Selective transformations of threo-2,3-dihydroxy esters (1991) (89)
- Bisaryloxime ethers as potent inhibitors of transthyretin amyloid fibril formation. (2005) (89)
- Selenium in natural products synthesis (1984) (88)
- Heterogeneous catalytic asymmetric dihydroxylation: Use of a polymer-bound alkaloid (1990) (88)
- Temperature Effects in Asymmetric Dihydroxylation: Evidence for a Stepwise Mechanism (1993) (87)
- A click chemistry approach to tetrazoles by Huisgen 1,3-dipolar cycloaddition: synthesis of 5-acyltetrazoles from azides and acyl cyanides. (2002) (87)
- The allylic azide rearrangement: achieving selectivity. (2005) (87)
- Ruthenium catalyzed oxidation of alcohols to aldehydes and ketones by amine-n-oxides (1976) (87)
- The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates. (1999) (86)
- Comparison of amine additives most effective in the new methyltrioxorhenium-catalyzed epoxidation process (1999) (86)
- SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts. (2017) (86)
- Kinetic resolution of racemic .beta.-hydroxy amines by enantioselective N-oxide formation (1983) (85)
- Crystal structures of two titanium tartrate asymmetric epoxidation catalysts (1984) (84)
- Smaller Substituents on Nitrogen Facilitate the Osmium‐Catalyzed Asymmetric Aminohydroxylation (1996) (83)
- Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub. (2017) (83)
- A major improvement in the osmium catalyzed vicinal hydroxylation of olefins by tert-butyl hydroperoxide (1978) (82)
- Click chemistry in materials synthesis. III. Metal‐adhesive polymers from Cu(I)‐catalyzed azide–alkyne cycloaddition (2007) (81)
- SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase (2019) (80)
- Asymmetric dihydroxylation of aryl allyl ethers (1993) (80)
- A New Portal to SuFEx Click Chemistry: A Stable Fluorosulfuryl Imidazolium Salt Emerging as an "F-SO2 +" Donor of Unprecedented Reactivity, Selectivity, and Scope. (2018) (79)
- 8 – On the Mechanism of Asymmetric Epoxidation with Titanium—Tartrate Catalysts (1985) (78)
- Selenium dioxide oxidations of olefins. Trapping of the allylic seleninic acid intermediate as a seleninolactone (1973) (75)
- Reversal of regioselection in the asymmetric aminohydroxylation of cinnamates (1998) (75)
- Documenting the scope of the catalytic asymmetric dihydroxylation (1989) (75)
- Additions and Corrections - Synthesis of Saccharides and Related Polyhydroxylated Natural Products. 3. Efficient Conversion of 2,3-erythro-Aldoses to 2,3-threo-Aldoses (1982) (74)
- Convenient synthesis of sulfinate esters from sulfonyl chlorides (1987) (73)
- Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation. 4. Electronic effects in amine-accelerated osmylations (1997) (73)
- Improvements in the osmium-catalyzed oxyamination of olefins by chloramine-T (1978) (72)
- Imidazole Aldoximes Effective in Assisting Butyrylcholinesterase Catalysis of Organophosphate Detoxification (2014) (72)
- Catalytic Asymmetric Dihydroxylation. (2010) (72)
- New reaction. Stereospecific vicinal oxyamination of olefins by alkyl imido osmium compounds (1975) (72)
- NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies. (2010) (71)
- A Highly Efficient Aminohydroxylation Process (1997) (69)
- New Ligands and Improved Enantioselectivities for the Asymmetric Dihydroxylation of Olefins (1995) (68)
- Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 2. A Qualitative Molecular Mechanics Approach (1994) (68)
- SuFEx Chemistry of Thionyl Tetrafluoride (SOF4 ) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates. (2018) (67)
- Squalene-2,3oxide, an intermediate in the enzymatic conversion of squalene to lanosterol and cholesterol. (1967) (67)
- Conversion of allylic phenylselenides to the rearranged allylic chlorides by N-chlorosuccinimide. Mechanism of selenium-catalyzed allylic chlorination of .beta.-pinene (1979) (67)
- Palladium-Catalyzed Fluorosulfonylvinylation of Organic Iodides. (2017) (67)
- Tert-butylsulfonamide. A new nitrogen source for catalytic aminohydroxylation and aziridination of olefins. (1999) (67)
- Unexpected diversity in the coordination chemistry of tartrate esters with titanium(IV) (1987) (66)
- Generation of candidate ligands for nicotinic acetylcholine receptors via in situ click chemistry with a soluble acetylcholine binding protein template. (2012) (66)
- Centrally acting oximes in reactivation of tabun-phosphoramidated AChE. (2013) (65)
- Kinetic role of the alkaloid ligands in asymmetric catalytic dihydroxylation (1989) (65)
- A practical route to enantiopure 1,2-aminoalcohols (1996) (62)
- The first d0 metallooxaziridines. Amination of olefins [1] (1978) (61)
- A New Approach to Osmium‐Catalyzed Asymmetric Dihydroxylation and Aminohydroxylation of Olefins (2002) (60)
- Epoxy alcohol rearrangements: hydroxyl-mediated delivery of Lewis acid promoters (1981) (60)
- A fluorogenic aryl fluorosulfate for intraorganellar transthyretin imaging in living cells and in Caenorhabditis elegans. (2015) (60)
- Two new asymmetric epoxidation catalysts. Unusual stoichiometry and inverse enantiofacial selection (1984) (60)
- Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. (2009) (59)
- Improved procedure for the tungstate-catalyzed epoxidation of .alpha.,.beta.-unsaturated acids (1985) (58)
- Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry (2014) (58)
- Stereospecific conversion of chiral 1,2-cyclic sulfates to chiral imidazolines (1991) (57)
- Short and practical syntheses of(R)-(−)-carnitine and (R)-(−)-γ-amino-β-hydroxybutyric acid (GABOB) (1993) (57)
- Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl Fluorosulfates. (2016) (56)
- Enantioselective synthesis of swainsonine, a trihydroxylated indolizidine alkaloid (1985) (56)
- Catalytic asymmetric synthesis (2002) (55)
- Allylic amination of olefins and acetylenes by imido sulfur compounds (1976) (55)
- Synthesis of saccharides and related polyhydroxylated natural products. 4. .alpha.-D- and .beta.-D-C-Glycopyranosides (2,6-dialkyl-substituted tetrahydropyrans) (1982) (55)
- Oxime-assisted Acetylcholinesterase Catalytic Scavengers of Organophosphates That Resist Aging* (2011) (55)
- Selective perhydroxylation of squalene: taming the arithmetic demon. (2010) (54)
- Stereospecific vicinal oxyamination of olefins by alkylimidoosmium compounds (1978) (54)
- Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF4 )-Derived Connective Hubs for Bioconjugation to DNA and Proteins. (2019) (54)
- Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity (2013) (52)
- Asymmetric dihydroxylation of primary allylic halides and a concise synthesis of (−)-diepoxybutane (1994) (51)
- Asymmetric dihydroxylation (AD) of N,N-dialkyl and N-methoxy-N-methyl α,β- and β,γ-unsaturated amides (1993) (51)
- Ethenesulfonyl Fluoride (ESF): An On-Water Procedure for the Kilogram-Scale Preparation. (2016) (51)
- Selenium-catalyzed nonradical chlorination of olefins with N-chlorosuccinimide (1979) (51)
- Asymmetric Dihydroxylation Enables Rapid Construction of Chiral Dendrimers Based on 1,2‐Diols (1996) (50)
- Synthesis of carbohydrates via tandem use of the osmium-catalyzed asymmetric dihydroxylation and enzyme-catalyzed aldol addition reactions (1994) (49)
- Allylic Amination and 1,2‐Diamination with a Modified Diimidoselenium Reagent (1996) (48)
- Asymmetric dihydroxylation of enynes (1992) (48)
- Oxidation of alcohols to aldehydes by reagents derived from chromyl chloride (1975) (48)
- Synthesis of All Four Isomers of Disparlure Using Osmium-Catalyzed Asymmetric Dihydroxylation. (1992) (48)
- Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry (2009) (47)
- Oxotransition metal oxidants as mimics for the action of mixed-function oxygenases. "NIH shift" with chromyl reagents. (1971) (47)
- Osmium-Catalyzed Asymmetric Dihydroxylation of Cyclic Cis-Disubstituted Olefins (1994) (45)
- Kinetic resolution of racemic olefins via asymmetric dihydroxylation (1993) (45)
- Selenium dioxide oxidation of ketones and aldehydes. Evidence for the intermediacy of .beta.-ketoseleninic (1976) (45)
- Catalytic asymmetric aminohydroxylation provides a short taxol side-chain synthesis. (1996) (44)
- Osmium‐catalyzed vicinal oxyamination of olefins by N‐chloro‐N‐argentocarbamates: ethyl threo‐[1‐(2‐hydroxy‐1,2‐diphenylethyl)]carbamate (1978) (44)
- Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 3. New Insights into Isomeric Forms of the Putative Osmaoxetane Intermediate (1996) (44)
- The chemistry of zerumbone. Part 5: Structural transformation of the dimethylamine derivatives (2003) (43)
- Using Sulfuramidimidoyl Fluorides that Undergo Sulfur(VI) Fluoride Exchange for Inverse Drug Discovery (2020) (43)
- Primary amides. A general nitrogen source for catalytic asymmetric aminohydroxylation of olefins. (2000) (43)
- Calculations on the reaction of ruthenium tetroxide with olefins using density functional theory (DFT). Implications for the possibility of intermediates in osmium-catalyzed asymmetric dihydroxylation (1994) (42)
- Iterative in situ click chemistry assembles a branched capture agent and allosteric inhibitor for Akt1. (2011) (42)
- SuFEx-enabled high-throughput medicinal chemistry. (2019) (42)
- Identification of a new endogenous metabolite and the characterization of its protein interactions through an immobilization approach. (2009) (42)
- Addition Reactions with Formation of Carbon–Oxygen Bonds: (ii) Asymmetric Methods of Epoxidation (1991) (42)
- Synthesis of a C3-symmetric phospha[2.2.2]cyclophane (1988) (41)
- A Practical and Highly Efficient Aminohydroxylation of Unsaturated Carboxylic Acids (2001) (41)
- Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries. (2009) (41)
- Permanganate in acetic anhydride. .alpha.-Diketones directly from olefins (1971) (40)
- Diversity Oriented Clicking (DOC): Divergent Synthesis of SuFExable Pharmacophores From 2-Substituted-Alkynyl-1-Sulfonyl Fluoride (SASF) Hubs. (2020) (39)
- CATALYTIC OSMYLATION OF CONJUGATED DIENES : A ONE-POT STEREOSELECTIVE SYNTHESIS OF POLYOLS (1991) (38)
- Selenium dioxide oxidation of endocyclic olefins. Evidence for a dissociation-recombination pathway (1982) (37)
- Double diastereoselection in asymmetric dihydroxylation (1993) (37)
- 1,2-Diamination of 1,3-dienes by imido selenium compounds (1976) (37)
- Automated Docking with Protein Flexibility in the Design of Femtomolar "Click Chemistry" Inhibitors of Acetylcholinesterase (2013) (36)
- On "The origin of high enantioselectivity in the dihydroxylation of olefins using osmium tetraoxide and cinchona alkaloid catalysts" (1993) (36)
- p-Nitrobenzoate esters of epoxy alcohols: convenient synthons for water-soluble epoxy alcohols (1987) (36)
- Osmium-catalyzed vicinal oxyamination of olefins by N-chloro-N-metallocarbamates (1980) (36)
- Reengineering Antibiotics to Combat Bacterial Resistance: Click Chemistry [1,2,3]-Triazole Vancomycin Dimers with Potent Activity against MRSA and VRE. (2017) (36)
- Ligand-Dependent Reversal of Facial Selectivity in the Asymmetric Dihydroxylation. (1996) (35)
- Asymmetric epoxidation models: An alkyl hydroperoxide dependent change in mehanism (1987) (35)
- Regioselective openings of 2,3-epoxy acids with organocuprates (1985) (35)
- On the timing of hydrolysis / reoxidation in the osmium-catalyzed asymmetric dihydroxylation of olefins using potassium ferricyanide as the reoxidant (1991) (35)
- Facile thermal rearrangements of allyl selenides and diselenides. [1,3] and [2,3] Shifts (1972) (35)
- Catalytic asymmetric aminohydroxylation with amino-substituted heterocycles as nitrogen sources. (1999) (35)
- In situ opening of epoxy alcohols: a convenient alternative to the isolation of unstable epoxy alcohols (1986) (35)
- Asymmetric dihydroxylation of squalene (1992) (35)
- Sulfur [18F]Fluoride Exchange Click Chemistry Enabled Ultrafast Late-Stage Radiosynthesis. (2021) (34)
- A Dramatic Ligand Effect on the Relative Reactive Reactivites of Substituted Alkenes with Osmium Tetroxide (1993) (34)
- Catalytic asymmetric synthesis of new halogenated chiral synthons (1997) (34)
- Ligand-based improvement of enantioselectivity in the catalytic asymmetric dihydroxylation of dialkyl substituted olefins (1990) (34)
- Study of the regio- and enantioselectivity of the reactions of osmium tetroxide with allylic alcohols and allylic sulfonamides (1994) (34)
- An efficient synthesis of enantiomerically pure trans-2-phenylcyclohexanol (1994) (34)
- A simple method for the preparation of N-sulfonylsulfilimines from sulfides. (2001) (34)
- Structural insights into conformational flexibility at the peripheral site and within the active center gorge of AChE. (2005) (33)
- Synthesis of dl-gabaculine utilizing direct allylic amination as the key step (1978) (33)
- Bis(trimethylsilyl) Peroxide Extends the Range of Oxorhenium Catalysts for Olefin Epoxidation (1997) (33)
- N-chloro-N-sodio-2-trimethylsilyl ethyl carbamate: A new nitrogen source for the catalytic asymmetric aminohydroxylation (1998) (33)
- A ligand structure-enantioselectivity relationship for the osmium-catalyzed asymmetric dihydroxylation of olefins (1991) (32)
- Bifluoride Ion Mediated SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides. (2018) (32)
- Synthesis of vicinal diamines from cyclic sulfates (1995) (31)
- Pharmacology, Pharmacokinetics, and Tissue Disposition of Zwitterionic Hydroxyiminoacetamido Alkylamines as Reactivating Antidotes for Organophosphate Exposure (2018) (31)
- Asymmetric dihydroxylation (AD) of α,β-unsaturated ketones (1993) (31)
- Coelacanths and catalysis (1994) (30)
- 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: a privileged, bivalent scaffold for the display of nucleophilic components. (2001) (30)
- Steric and Dynamic Parameters Influencing In Situ Cycloadditions to Form Triazole Inhibitors with Crystalline Acetylcholinesterase. (2016) (30)
- Synthesis and stereochemical assignments for goniobutenolides A and B (1994) (30)
- d,1-Malabaricanediol. First cyclic natural product derived from squalene in a nonenzymic process (1970) (29)
- Synthesis of Sulfotyrosine-Containing Peptides by Incorporating Fluorosulfated Tyrosine Using an Fmoc-Based Solid-Phase Strategy. (2016) (29)
- Asymmetric Synthesis of γ-Hydroxy α,β-Unsaturated Amides via an AD-elimination Process; Synthesis of (+)-Coriolic Acid (1993) (29)
- A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistry. (2003) (29)
- Tartrate-like ligands in the asymmetric epoxidation (1989) (28)
- Asymmetric dihydroxylation of acrolein acetals: synthesis of stable equivalents of Enantiopure glyceraldehyde and glycidaldehyde (1992) (28)
- Positional selectivity during controlled oxidation of polyolefins (1967) (28)
- Allylic deuteration and tritiation of olefins with N-sulfinylsulfonamides (1978) (28)
- A short route to β-lactams: Use of cyclic sulfites from syn-2,3-dihydroxy esters (1990) (28)
- Chromyl chloride in acetone. .alpha.-Chloro ketones and ketones directly from olefins (1973) (27)
- Molar Scale Synthesis of Enantiopure Stilbene Oxide. (1996) (27)
- THE OSMIUM-CATALYZED AMINOHYDROXYLATION OF BAYLIS-HILLMAN OLEFINS (1999) (27)
- Mechanism of interaction of novel uncharged, centrally active reactivators with OP-hAChE conjugates. (2013) (27)
- Design and synthesis via click chemistry of 8,9-anhydroerythromycin A 6,9-hemiketal analogues with anti-MRSA and -VRE activity. (2007) (27)
- The asymmetric dihydroxylation of cis-allylic and homoallylic alcohols (1994) (27)
- A simple and efficient method for the preparation of pyridine-N-oxides II (1998) (27)
- Bacterial glycosyltransferase-mediated cell-surface chemoenzymatic glycan modification (2019) (27)
- Titanium isopropoxide mediated formation of 2,3-epithio alcohols from 2,3-epoxy alcohols (1988) (26)
- CHLOROHYDROXYLATION OF OLEFINS WITH PEROXIDES AND TITANIUM TETRACHLORIDE (1985) (26)
- Removal of the 4,4-dimethyl carbons in the enzymic conversion of lanosterol to cholesterol. Initial loss of the 4-alpha-methyl group. (1970) (26)
- Applications of Aziridinium Ions: Selective Syntheses of Pyrazolidin-3-ones and Pyrazolo[1,2-a]pyrazoles (2000) (26)
- Modified cinchona alkaloid ligands: Improved selectivities in the osmium tetroxide catalyzed asymmetric dihydroxylation (AD) of terminal olefins (1993) (25)
- Some reactions of N-(2-hydroxyalkyl)-p-toluenesulfonamides and N-allyl-p-toluenesulfonamides (1979) (25)
- Subtle effects in the asymmetric epoxidation : dependence of kinetic resolution efficiency on the monodentate alkoxide ligands of the bystander titanium center (1991) (25)
- Highly Efficient Epoxidation of Olefins Using Aqueous H2O2 and Catalytic Methyltrioxorhenium/Pyridine: Pyridine‐Mediated Ligand Acceleration. (1997) (25)
- Mechanism of the titanium-promoted deoxygenative coupling of allyl and benzyl alcohols to hydrocarbons (1969) (25)
- OXIDATION OF ACETYLENES WITH TERT-BUTYL HYDROPEROXIDE CATALYZED BY SELENIUM DIOXIDE. α,α′-DIOXYGENATION OF INTERNAL ALKYNES (1980) (25)
- Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia (2020) (24)
- Catalytic Asymmetric Epoxidation of Allylic Alcohols (2010) (24)
- Biological demethylation of 4,4-dimethyl sterols. Initial removal of the 4.alpha.-methyl group (1968) (24)
- Enzymic cyclization of trans,trans,trans-18,19-dihydrosqualene 2,3-oxide. (1967) (24)
- Applications of Aziridinium Ions. Selective Syntheses of β-Aryl-α,β-diamino Esters (1999) (24)
- Asymmetric dihydroxylation of tertiary allylic alcohols (1993) (23)
- Comparing two models for the selectivity in the asymmetric dihydroxylation reaction (AD) (1994) (23)
- SELENIUM DIOXIDE OXIDATION OF D-LIMONENE, A REINVESTIGATION (1975) (23)
- Asymmetric dihydroxylation of olefins containing sulfur: Chemoselective oxidation of CC double bonds in the presence of sulfides, 1,3-dithianes, and disulfides (1994) (23)
- Dihydroxylation of Polyenes Using Narasaka's Modification of the Upjohn Procedure. (1998) (23)
- SuFExable polymers with helical structures derived from thionyl tetrafluoride (2019) (22)
- One-step synthesis of 1,5-dienes involving reductive coupling of allyl alcohols (1968) (22)
- Structural Characterization of the Pseudoenantiomeric cis-Dioxo Osmium(VI) Esters of Chiral Diols with Cinchona Alkaloid Ligands† (1990) (22)
- Quantitative and Orthogonal Formation and Reactivity of SuFEx Platforms (2018) (22)
- Effect of isomers of swainsonine on glycosidase activity and glycoprotein processing. (1987) (22)
- Interaction kinetics of oximes with native, phosphylated and aged human acetylcholinesterase. (2010) (22)
- Synthesis of Selective Agonists for the α7 Nicotinic Acetylcholine Receptor with In Situ Click-Chemistry on Acetylcholine-Binding Protein Templates (2012) (21)
- Carbonyl participation in the addition of p-chlorophenylselenenyl bromide to ()-4-hexenal: A new route to 2,6-dideoxylgycosides (1978) (21)
- Asymmetric Dihydroxylation Via Ligand-Accelerated Catalysis. (1988) (20)
- Cover Picture: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. Int. Ed. 21/2005) (2005) (20)
- Studies on the mechanism of the asymmetric epoxidation: a ligand variation approach (1989) (20)
- Observation of the controlled assembly of preclick components in the in situ click chemistry generation of a chitinase inhibitor (2013) (20)
- Preparation of 5‐Substituted 1H‐Tetrazoles from Nitriles in Water. (2002) (20)
- Biological demethylation of 4,4-dimethyl sterols, Evidence for enzymic epimerization of the 4beta-methyl group prior to its oxidative removal. (1969) (20)
- The Osmium-Catalyzed Asymmetric Dihydroxylation: A New Ligand Class and a Process Improvement. (2010) (19)
- Dioxomolybdenum(VI)-substituted 2,6-pyridinedimethanol complexes: new five-coordinate species (1986) (19)
- Nucleophilic substitution by grignard reagents on sulfur mustards. (2004) (19)
- Asymmetric dihydroxylation of α-substituted styrene derivatives (1993) (19)
- A comparison of ligands proposed for the asymmetric dihydroxylation (1994) (19)
- Chemistry ‘On Water’ – Organic Synthesis in Aqueous Suspension (2007) (19)
- Rapid 'sar' via click chemistry : An alkyne-bearing spiramycin is fused with diverse azides to yield new triazole-antibacterial candidates (2006) (19)
- Molecular basis of interactions of cholinesterases with tight binding inhibitors. (2005) (18)
- Synthesis and Crystal Structure of a Chiral C3‐Symmetric Monophosphane (1988) (18)
- A short route to a moshe'rs acid precursor via catalytic asymmetric dihydroxylation (AD) (1994) (18)
- The asymmetric epoxidation of tert-butyl substituted allylic alcohols (1985) (18)
- Reversal of Tabun Toxicity Enabled by a Triazole-Annulated Oxime Library-Reactivators of Acetylcholinesterase. (2019) (18)
- Enzymic cyclization of 15-norsqualene 2,3-oxide (1968) (17)
- Direct deoxygenation of vicinal diols with tungsten(IV). A new olefin synthesis (1972) (17)
- Synthesis of 1,4-triazole linked zanamivir dimers as highly potent inhibitors of influenza A and B (2013) (17)
- Synthesis of optically active secondary allylic alcohols from allylsilanes via successive asymmetric dihydroxylation (AD) and Peterson olefination reactions (1993) (16)
- Oxidation of acetylenes with tert-butyl hydroperoxide catalyzed by selenium dioxide. .alpha.,.alpha.'-Dioxygenation of internal alkynes (1979) (16)
- Selenium dioxide oxidation of d-limonene. Reinvestigation (1975) (16)
- Terpene terminal epoxides. Skeletal rearrangement accompanying bicyclization of squalene 2,3-oxide (1969) (15)
- Assessment of ionizable, zwitterionic oximes as reactivating antidotal agents for organophosphate exposure. (2019) (15)
- Enantioselective Synthesis of Juvenile Hormone III in Three Steps from Methyl Farnesoate (1993) (14)
- IMPROVED PROCEDURE FOR THE OXYAMINATION OF OLEFINS WITH TRIOXO(TERT-BUTYLIMIDO)OSMIUM(VIII) (1980) (14)
- Antiviral Stilbene 1,2-Diamines Prevent Initiation of Hepatitis C Virus RNA Replication at the Outset of Infection (2011) (14)
- REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION TO α,ß-UNSATURATED KETONES. (2008) (14)
- Rapid separation of organic mixtures by formation of metal complexes (1975) (14)
- NH-1,2,3-Triazoles from Azidomethyl Pivalate and Carbamates: Base-Labile N-Protecting Groups (2005) (14)
- The reactions of olefins with permanganate, ruthenium tetroxide, and osmium tetroxide; dependence of rate on degree of substitution (1975) (13)
- Evaluation of high-affinity phenyltetrahydroisoquinoline aldoximes, linked through anti-triazoles, as reactivators of phosphylated cholinesterases. (2019) (13)
- Mechanism of decomposition of sulfonium betaines to epoxides (1972) (13)
- Asymmetric dihydroxylation (AD)/cyclization of N-diBoc allylic and homoallylic amines: Selective differentiation of the hydroxyl groups. (1993) (13)
- First practical synthesis of formamidine ureas and derivatives. (2003) (13)
- 2,6-Dichloro-9-thiabicyclo[3.3.1]nonane: multigram display of azide and cyanide components on a versatile scaffold. (2006) (13)
- Transformations of hydroxy cyclic sulfates: stereospecific conversion into 2,3,5-trisubstituted tetrahydrofurans. (1993) (13)
- Vicinal acetoxychlorination of olefins by chromyl chloride in acetyl chloride (1977) (12)
- Biological activities of some terminally modified squalene and squalene 2, 3-oxide analogs. (1967) (12)
- Asymmetric Oxidations and Related Reactions: Catalytic Asymmetric Dihydroxylation—Discovery and Development (2005) (12)
- Threo-N,N'-Bis(.alpha.-methylbenzyl)sulfamide: a readily available chiral ligand for asymmetric lithium aluminum hydride reductions (1984) (12)
- Facile synthesis of enantiopure trans-2,3-diphenyl-1,4-diazabicyclo[2.2.2]octane (1991) (12)
- From Styrenes to Enantiopure α-Arylglycines in Two Steps. (1998) (12)
- Identification of simple arylfluorosulfates as potent agents against resistant bacteria (2021) (12)
- CATALYTIC AMINOHYDROXYLATION USING ADENINE-DERIVATIVES AS THE NITROGEN SOURCE (1998) (12)
- Asymmetric Epoxidation of Allyl Alcohol: Efficient Routes to Homochiral β‐Adrenergic Blocking Agents. (1987) (11)
- NH‐1,2,3‐Triazoles from Azidomethyl Pivalate and Carbamates: Base‐Labile N‐Protecting Groups. (2006) (11)
- Synthesis of erythro-18,19-dihydroxysqualene 2,3-oxide and other internally oxidized squalene derivatives (1970) (11)
- Catalytic Asymmetric Dihydroxylation of cis-Disubstituted Olefins. (2010) (10)
- Multivalent, Bifunctional Dendrimers Prepared by Click Chemistry (2006) (10)
- Bromine-Catalyzed Aziridination of Olefins. A Rare Example of Atom-Transfer Redox Catalysis by a Main Group Element. (1998) (10)
- Titelbild: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. 21/2005) (2005) (10)
- Catalytic Asymmetric Dihydroxylation — Discovery and Development (2001) (9)
- NH-1,2,3-Triazole Inhibitors of the VIM-2 Metallo-β-Lactamase (2010) (9)
- Regioselective Nucleophilic Opening of erythro-and threo-2,3-Epoxy Alcohols (1987) (9)
- NEW TRANSFORMATIONS OF 2,3-EPOXY ALCOHOLS AND RELATED DERIVATIVES. EASY ROUTES TO HOMOCHIRAL SUBSTANCES (1984) (9)
- A simple route to enantiomerically enriched oxazolidin-2-ones (1993) (9)
- The Banert Cascade: A Synthetic Sequence to Polyfunctional NH‐1,2,3‐triazoles. (2005) (9)
- Cover Picture: Efficiency and Fidelity in a Click‐Chemistry Route to Triazole Dendrimers by the Copper(I)‐Catalyzed Ligation of Azides and Alkynes (Angew. Chem. Int. Ed. 30/2004) (2004) (9)
- The Banert Cascade: A Synthetic Sequence to Polyfunctional NH-1,2,3-Triazoles (2005) (8)
- Enzymic transformation of an acyclic sesterterpene terminal epoxide into a lanosterol analogue (1969) (8)
- Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase (2019) (8)
- 3‐[(1S)‐1,2‐Dihydroxyethyl]‐1,5‐Dihydro‐3H‐2,4‐Benzodioxepine (2003) (8)
- Structural insights into conformational flexibility at the peripheral site and within the active center gorge of AChE, Chem Biol Interact. 157-158, 159-65. (2004) (7)
- A Stepwise Huisgen Cycloaddition Process: Copper(I)‐Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes. (2002) (7)
- Selective Transformations of 2,3-Epoxy Alcohols and Related Derivatives. (1986) (7)
- In Situ Click Chemistry for the Identification of a Potent D-Amino Acid Oxidase Inhibitor. (2016) (7)
- Stereochemistry of organic and bioorganic transformations : proceedings of the Seventeenth workshop conference Hoechst, Schloß Reisensburg, 8-11 October 1986 (1987) (6)
- Chapter 2.6. Asymmetric Aminohydroxylation (2008) (6)
- Chain-Growth Sulfur(VI) Fluoride Exchange Polycondensation: Molecular Weight Control and Synthesis of Degradable Polysulfates (2021) (6)
- SELENIUM DIOXIDE OXIDATION OF KETONES AND ALDEHYDES. EVIDENCE FOR THE INTERMEDIACY OF β-KETOSELENINIC (1976) (6)
- Enantioselective Synthesis of Both Enantiomers of 7,7-Dimethyl-6,8-dioxa-bicyclo[3.2.1]octane via Regioselective Asymmetric Dihydroxylation (1993) (6)
- Probing gorge dimensions of cholinesterases by freeze-frame click chemistry. (2008) (6)
- Click chemistry-facilitated comprehensive identification of proteins adducted by antimicrobial 5-nitroimidazoles for discovery of alternative drug targets against giardiasis (2020) (6)
- A new approach to osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins. (2002) (6)
- An Expedient Route to the Tetrazole Analogues of α‐Amino Acids. (2002) (5)
- Osmium-Catalyzed Dihydroxylation of Olefins in Acidic Media: Old Process, New Tricks. (2002) (5)
- Some aspects of substrate specificity in biological demethylation at C4 of steroids (1975) (5)
- Asymmetric dihydroxylation affords enantiomerically pure C12 building blocks from traps, traps, cis-1,5,9-cyclododecatriene (1995) (5)
- Vicinal Diol Cyclic Sulfates: Like Epoxides Only More Reactive. (1989) (5)
- Regioselective Azide Opening of 2,3-Epoxy Alcohols by (Ti(O-i-Pr)2(N3)2): Synthesis of α-Amino Acids. (1989) (5)
- Selective Transformations of threo‐2,3‐Dihydroxy Esters. (1991) (5)
- ELECTROPHILIC ORGANOSELENIUM REAGENTS, A NEW ROUTE TO ALLYLIC ACETATES AND ETHERS (1974) (5)
- Reinvestigation of the infrared spectra of oxoosmium(VI) esters by isotopic labeling (1993) (5)
- Rapid “SAR” via Click Chemistry: An Alkyne‐Bearing Spiramycin Is Fused with Diverse Azides to Yield New Triazole‐Antibacterial Candidates. (2007) (5)
- Copper‐Catalyzed Synthesis of N‐Sulfonyl‐1,2,3‐triazoles: Controlling Selectivity. (2007) (4)
- Diols via Catalytic Dihydroxylation (2003) (4)
- Arenesulfonate Derivatives of Homochiral Glycidol: Versatile Chiral Building Blocks for Organic Synthesis. (1989) (4)
- Selective Asymmetric Dihydroxylation of Dienes. (2010) (4)
- Asymmetric Oxidations and Related Reactions: Catalytic Asymmetric Epoxidation of Allylic Alcohols (2005) (4)
- Titelbild: Efficiency and Fidelity in a Click-Chemistry Route to Triazole Dendrimers by the Copper(I)-Catalyzed Ligation of Azides and Alkynes (Angew. Chem. 30/2004) (2004) (4)
- Click Chemistry-Facilitated Structural Diversification of Nitrothiazoles, Nitrofurans, and Nitropyrroles Enhances Antimicrobial Activity against Giardia lamblia (2017) (4)
- Catalytic Asymmetric Aminohydroxylation of Olefins. (1996) (4)
- New Ligands and Improved Enantioselectivities for the Asymmetric Dihydroxylation of Olefins. (1995) (4)
- AN IMPROVED PROCEDURE FOR THE DIRECT OXIDATION OF OLEFINS TO ALPHA-DIKETONES BY POTASSIUM PERMANGANATE IN ACETIC ANHYDRIDE (1974) (4)
- The first d0 metallooxaziridines. Amination of olefins (1979) (4)
- Cover Picture: Angew. Chem. Int. Ed. 6/2002 (2002) (4)
- Palladium‐Catalyzed, Ligand‐Free Suzuki Reaction in Water Using Aryl Fluorosulfates. (2015) (4)
- Comparison of Amine Additives Most Effective in the New Methyltrioxorhenium‐Catalyzed Epoxidation Process. (1999) (4)
- Dioxomolybdenum(VI)-Substituted 2,6-Pyridinedimethanol Complexes: New Five- Coordinate Species. (1986) (4)
- Asymmetric Dihydroxylation of Olefins Containing Sulfur: Chemoselective Oxidation of C-C Double Bonds in the Presence of Sulfides, 1,3-Dithianes, and Disulfides. (1994) (3)
- Deoxygenation of Epoxides with Lower Valent Tungsten Halides: trans‐Cyclododecene (2003) (3)
- Synthesis of Vicinal Diamines from Cyclic Sulfates. (1996) (3)
- “Sleeping Beauty” Phenomenon: SuFEx-Enabled Discovery of Selective Covalent Inhibitors of Human Neutrophil Elastase (2019) (3)
- Synthesis of Carbohydrates via Tandem Use of the Osmium‐Catalyzed Asymmetric Dihydroxylation and Enzyme‐Catalyzed Aldol Addition Reactions. (1994) (3)
- Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors (2022) (3)
- Asymmetric Dihydroxylation of Aryl Allyl Ethers. (1993) (3)
- α-Hydroxy Ketones in High Enantiomeric Purity from Asymmetric Dihydroxylation of Enol Ethers. (1993) (3)
- Improved Enantioselectivity in Asymmetric Dihydroxylations of Terminal Olefins Using Pyrimidine Ligands. (1993) (3)
- Enantioselective Epoxidation of Allylic Alcohols: (2S,3S)‐3‐Propyloxiranemethanol (2003) (3)
- Osmium‐Catalyzed Asymmetric Dihydroxylation of Cyclic cis‐ Disubstituted Olefins. (1995) (3)
- Short and Practical Syntheses of (R)‐(‐)‐Carnitine and (R)‐(‐)‐γ‐ Amino‐β‐hydroxybutyric Acid (GABOB). (1993) (3)
- Ligand design for human acetylcholinesterase and nicotinic acetylcholine receptors, extending beyond the conventional and canonical (2021) (2)
- Homogeneous Selective Oxidation (1977) (2)
- A Practical Route to Enantiopure 1,2-Amino Alcohols. (1996) (2)
- Applications of Aziridinium Ions. Selective Syntheses of β‐Aryl‐α,β‐diamino Esters. (2000) (2)
- TOTAL SYNTHESIS OF THE LHEXOSES (1990) (2)
- STEREO AND REGIOSELECTIVE OPENINGS OF CHIRAL 2,3‐EPOXY ALCOHOLS. VERSATILE ROUTES TO OPTICALLY PURE NATURAL PRODUCTS AND DRUGS. UNUSUAL KINETIC RESOLUTIONS (1983) (2)
- [18F]SuFEx Click Chemistry Enabled Ultrafast Late-stage Radiosynthesis (2020) (2)
- Procedure for the Catalytic Asymmetric Epoxidation of Allylic Alcohols in the Presence of Molecular Sieves. (1986) (2)
- PL-01The secret life of enzymes (2008) (2)
- Study of the Regio- and Enantioselectivity of the Reactions of Osmium Tetroxide with Allylic Alcohols and Allylic Sulfonamides. (1994) (2)
- A New Approach to Osmium‐Catalyzed Asymmetric Dihydroxylation and Aminohydroxylation of Olefins. (2002) (2)
- IMPROVED PROCEDURE FOR THE TUNGSTATE-CATALYZED EPOXIDATION OF α,β-UNSATURATED ACIDS (1985) (2)
- High-performing polysulfate dielectrics for electrostatic energy storage under harsh conditions. (2023) (2)
- Enantioselective Synthesis of Juvenile Hormone III in Three Steps from Methyl Farnesoate. (1994) (2)
- A Ligand Structure-Enantioselectivity Relationship for the Osmium- Catalyzed Asymmetric Dihydroxylation of Olefins. (1992) (2)
- Asymmetric Dihydroxylation of Enynes. (1992) (2)
- Rücktitelbild: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF 4 )‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. 24/2019) (2019) (2)
- 2,6‐Dichloro‐9‐thiabicyclo[3.3.1]nonane: A Privileged, Bivalent Scaffold for the Display of Nucleophilic Components. (2001) (2)
- A new rearrangement of N-arylhydroxamic acids catalyzed by seleninic acids and phenylselenenyl chloride (1978) (2)
- A General Approach to γ-Lactones via Osmium-Catalyzed Asymmetric Dihydroxylation. Synthesis of (-)- and (+)-Muricatacin. (1993) (2)
- Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines. (2021) (2)
- Click Chemistry Expedited Radiosynthesis: Sulfur [18F]fluoride Exchange of Aryl Fluorosulfates (2019) (1)
- Asymmetric Synthesis of γ-Hydroxy α,β-Unsaturated Amides via an AD-Elimination Process. Synthesis of (+)-Coriolic Acid. (1993) (1)
- A New Ligand Class for the Asymmetric Dihydroxylation of Olefins. (1996) (1)
- RUTHENIUM-CATALYZED OXIDATION OF ALCOHOLS TO ALDEHYDES AND KETONES BY AMINE-N-OXIDES (1976) (1)
- Synthesis of a novel pentacoordinate glyoxime-based ligand and preparation of its chlorocobalt(III) complex (2002) (1)
- Bacterial glycosyltransferase-mediated cell-surface chemoenzymatic glycan modification (2019) (1)
- Enhancing Target Tissue Levels and Diminishing Plasma Clearance of Ionizing Zwitterionic Antidotes in Organophosphate Exposures (2021) (1)
- Cyclic Sulfates Containing Acid‐Sensitive Groups and Chemoselective Hydrolysis of Sulfate Esters. (1989) (1)
- Toward an Understanding of the High Enantioselectivity in the Osmium‐ Catalyzed Asymmetric Dihydroxylation (AD). Part 1. Kinetics. (1994) (1)
- Catalytic Osmylation of Conjugated Dienes: A One-Pot Stereoselective Synthesis of Polyols. (1991) (1)
- A Short Route to β-Lactams: Use of Cyclic Sulfites from syn-2,3- Dihydroxy Esters. (1991) (1)
- N‐Bromoacetamide ‐ A New Nitrogen Source for the Catalytic Asymmetric Aminohydroxylation of Olefins. (1997) (1)
- Ligand‐Based Improvement of Enantioselectivity in the Catalytic Asymmetric Dihydroxylation of Dialkyl‐Substituted Olefins. (1991) (1)
- A Short Route to a Mosher′s Acid Precursor (III) via Catalytic Asymmetric Dihydroxylation (AD). (1995) (1)
- Tsutomu Katsuki (1946-2014). (2015) (1)
- ASYMMETRIC EPOXIDATION OF HOMOALLYLIC ALCOHOLS. SYNTHESIS OF (-)-Γ-AMINO-β-(R)-HYDROXYBUTYRIC ACID (GABOB) (1985) (1)
- One-Pot Synthesis of Homochiral Aziridines and Amino Alcohols from Homochiral 1,2-Cyclic Sulfates. (1989) (1)
- (R,R)‐1,2‐Diphenyl‐1,2‐Ethanediol (Stilbene Diol) (2003) (1)
- Type I Intramolecular Cycloadditions of Vinylketenes (1989) (1)
- A simple life—finding function and making connections (2019) (1)
- An expedient route to the tetrazole analogues of alpha-amino acids. (2002) (1)
- The Discovery of Titanium-Catalyzed Asymmetric Epoxidation (1986) (1)
- A Simple Method for the Preparation of N‐Sulfonylsulfilimines from Sulfides. (2001) (1)
- STEREOSELECTIVE EPOXIDATIONS OF ACYCLIC ALLYLIC ALCOHOLS BY TRANSITION METAL-HYDROPEROXIDE REAGENTS, SYNTHESIS OF DL-C18 CECROPIA JUVENILE HORMONE FROM FARNESOL (1974) (1)
- Oxime Reactivation Mechanisms for Organophosphate Conjugated Human Acetylcholinesterase (2016) (1)
- ELECTROPHILIC AND NUCLEOPHILIC ORGANOSELENIUM REAGENTS, NEW ROUTES TO ALPHA,BETA-UNSATURATED CARBONYL COMPOUNDS (1973) (1)
- Applications of aziridinium ions. Selective syntheses of beta-aryl-alpha,beta-diamino esters. (1999) (1)
- A Simple and Efficient Method for the Preparation of Pyridine N‐Oxides. (1998) (1)
- Stereospecific Conversion of Chiral 1,2-Cyclic Sulfates to Chiral Imidazolines. (1991) (0)
- Allylic Amination and 1,2-Diamination with a Modified Diimidoselenium Reagent. (1996) (0)
- Asymmetric Synthesis of Both Enantiomers of Tomoxetine and Fluoxetine. Selective Reduction of 2,3-Epoxycinnamyl Alcohol with Red-Al. (1989) (0)
- Dihydroxylation asymetrique catalytique acceleree par un ligand (1989) (0)
- Applications of Aziridinium Ions: Selective Syntheses of Pyrazolidin‐3‐ones and Pyrazolo[1,2‐a]pyrazoles. (2000) (0)
- PHENYLTETRAHYDROISOQUINOLINE-BASED TRIAZOLE COMPOUNDS ARE HIGH-AFFINITY POTENTIAL REACTIVATORS OF NERVE AGENT-INHIBITED HUMAN ACETYLCHOLINESTERASE (2018) (0)
- Asymmetric Dihydroxylation Affords Enantiomerically Pure C12 Building Blocks from trans,trans,cis-1,5,9-Cyclododecatriene. (2010) (0)
- New Ligands Double the Scope of the Catalytic Asymmetric Dihydroxylation of Olefins. (1991) (0)
- Kinetic Role of the Alkaloid Ligands in Asymmetric Catalytic Dihydroxylation. (1989) (0)
- On the Mechanism of Asymmetric Epoxidation with Titanium-Tartrate (1986) (0)
- Regioselective Openings of 2,3-Epoxy Acids with Organocuprates. (1986) (0)
- Fluorosulfuryl Isocyanate Enabled SuFEx Ligation of Alcohols and Amines (2021) (0)
- A Comparison of Ligands Proposed for the Asymmetric Dihydroxylation. (1994) (0)
- Mechanism of Asymmetric Epoxidation. Part 2. Catalyst Structure. (1991) (0)
- STEREOSELECTIVE EPOXIDATION OF ACYCLIC ALLYLIC ALCOHOLS. A CORRECTION OF OUR PREVIOUS WORK (1980) (0)
- N‐Chloro‐N‐sodio‐2‐trimethylsilyl Ethyl Carbamate: A New Nitrogen Source for the Catalytic Asymmetric Aminohydroxylation. (1998) (0)
- Serratia marcescens Chitinase B, tetragonal form (2013) (0)
- Large‐Scale and Highly Enantioselective Synthesis of the Taxol C‐13 Side Chain (VII) Through Asymmetric Dihydroxylation. (1995) (0)
- Special Products: Sections 3.3.1–3.3.4 (2008) (0)
- Serratia marcescens Chitinase B complexed with syn-triazole inhibitor (2013) (0)
- Catalytic Asymmetric Di hydroxylation (2001) (0)
- Serratia marcescens Chitinase B complexed with azide inhibitor (2013) (0)
- Asymmetric Dihydroxylation of Tertiary Allylic Alcohols. (2010) (0)
- Preclusion of the “Second Cycle” in the Osmium-Catalyzed Asymmetric Dihydroxylation of Olefins Leads to a Superior Process. (1991) (0)
- Chain-Growth SuFEx Polycondensation: Molecular Weight Control and Synthesis of Degradable Polysulfates (2021) (0)
- Asymmetric Dihydroxylation of Primary Allylic Halides and a Concise Synthesis of (‐)‐Diepoxybutane. (1994) (0)
- Enantioselective Synthesis of Both Enantiomers of 7,7-Dimethyl-6,8- dioxabicyclo(3.2.1)octane via Regioselective Asymmetric Dihydroxylation. (1994) (0)
- Syntheses and Crystal Structures of the Cinchona Alkaloid Derivatives Used as Ligands in the Osmium‐Catalyzed Asymmetric Dihydroxylation of Olefins, e.g. (I). Used as Ligands in the Osmium‐Catalyzed Asymmetric Dihydroxylation of Olefines. (1994) (0)
- Structure-Reactivity Relationships in "Special" 2nd Cycle Osmium Catalyzed Amino Hydroxylation (2003) (0)
- HIGH STEREO- AND REGIOSELECTIVITIES IN THE TRANSITION METAL CATALYZED EPOXIDATIONS OF OLEFINIC ALCOHOLS BY TERT.-BUTYL HYDROPEROXIDE (1973) (0)
- IONIZABLE, ZWITTERIONIC OXIMES AS COUNTERMEASURES TO VOLATILE ORGANOPHOSPHATE (OP) EXPOSURE (2018) (0)
- Synthesis and Structure of a Chiral, C3‐Symmetric Monophosphane. (1988) (0)
- Dihydroxylation of Polyenes Using Narasaka′s Modification of the Upjohn Procedure. (1999) (0)
- Regioselective Nucleophilic Opening of erythro- and threo-2,3-Epoxy Alcohols. (1987) (0)
- An Efficient Synthesis of Enantiomerically Pure trans‐2‐ Phenylcyclohexanol. (1994) (0)
- A Highly Efficient Aminohydroxylation Process. (1998) (0)
- Patent Number : 45 ) Date of Patent : 5 , 126 , 494 Jun (2017) (0)
- A Convenient Synthesis of Sulfinate Esters from Sulfonyl Chlorides. (1987) (0)
- A Concept for the Regioselective Synthesis of 1,2,3-Triazoles (2006) (0)
- Enantioselective Hydrogenation of Allylic and Homoallylic Alcohols. (1989) (0)
- The Osmium‐Catalyzed Aminohydroxylation of Baylis—Hillman Olefins. (1999) (0)
- Synthesis of Resin Acid Intermediates. 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9,3,4-hexahydronaphthalone-2 and 8α,10β-Dimethyl-8β-carbomethoxy-Δ1,9-octalone-2 (1964) (0)
- Synthesis of a C3‐Symmetric Phospha(2.2.2)cyclophane. (1989) (0)
- Smaller Substituents on Nitrogen Facilitate the Osmium-Catalyzed Asymmetric Aminohydroxylation. (1997) (0)
- A Simple Route to Enantiomerically Enriched Oxazolidin‐2‐ones. (1993) (0)
- Pharmacokinetic Analysis of Ionizable Zwitterionic Oximes: Antidotes to Organophosphate Exposure. (2020) (0)
- Structural And Functional Analysis Of Acetylcholinesterase Complexes With “In Situ Click‐Chemistry” Inhibitors (2016) (0)
- Asymmetric Dihydroxylation (AD) and Drug Synthesis. (1993) (0)
- Metal Catalysis in the Synthesis of Heterocycles (1977) (0)
- Eric Jacobsen@60, a Personal Statement (2020) (0)
- Characterizing the therapeutic efficacy of novel oximes synthesized by click chemistry against organophosphorous compounds poisoning (2010) (0)
- OLEFIN SYNTHESIS, RATE ENHANCEMENT OF THE ELIMINATION OF ALKYL ARYL SELENOXIDES BY ELECTRON-WITHDRAWING SUBSTITUENTS (1975) (0)
- Synthesis of Optically Active Secondary Allylic Alcohols from Allylsilanes via Successive Asymmetric Dihydroxylation (AD) and Peterson Olefination Reactions. (1993) (0)
- Design and evaluation of phenyltetrahydroisoquinoline pyridinium aldoximes as reactivators of nerve-agent-inhibited human cholinesterases (2019) (0)
- Asymmetric Epoxidation Models: An Alkyl Hydroperoxide Dependent Change in Mechanism. (1987) (0)
- Searching for New Reactivity (Nobel Lecture) (2002) (0)
- Back Cover: A New Portal to SuFEx Click Chemistry: A Stable Fluorosulfuryl Imidazolium Salt Emerging as an “F−SO2+” Donor of Unprecedented Reactivity, Selectivity, and Scope (Angew. Chem. Int. Ed. 10/2018) (2018) (0)
- Unexpected Diversity in the Coordination Chemistry of Tartrate Esters with Titanium(IV). (1987) (0)
- Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts. (2017) (0)
- Generation of selective ligands for nicotinic acetylcholine receptors (2012) (0)
- Affinity selection of double-click triazole libraries for rapid discovery of allosteric modulators for GLP-1 receptor. (2023) (0)
- accelerated by a complexing catalytic asymmetric dihydroxylation (1989) (0)
- Synthesizing Selective Agonists for the α 7 Nicotinic Receptor with in situ Click-Chemistry on Acetylcholine Binding Protein Templates (2012) (0)
- A Simplified Procedure for the Stereospecific Transformation of 1,2- Diols into Epoxides. (1993) (0)
- Foreword by K. Barry Sharpless (2000) (0)
- A NEW REACTION, STEREOSPECIFIC VICINAL OXYAMINATION OF OLEFINS BY ALKYL IMIDO OSMIUM COMPOUNDS (1975) (0)
- In situ Opening of Epoxy Alcohols: A Convenient Alternative to the Isolation of Unstable Epoxy Alcohols. (1987) (0)
- Bifluoride Ion Catalyzed Late-Stage SuFEx Trifluoromethylation of Sulfonyl Fluorides and Iminosulfur Oxydifluorides (2018) (0)
- Heterogeneous Catalytic Asymmetric Dihydroxylation: Use of a Polymer- Bound Alkaloid. (1991) (0)
- Back Cover: SuFEx‐Based Polysulfonate Formation from Ethenesulfonyl Fluoride–Amine Adducts (Angew. Chem. Int. Ed. 37/2017) (2017) (0)
- A 60th Birthday (2007) (0)
- Tartrate-Like Ligands in the Asymmetric Epoxidation. (1989) (0)
- Synthesis and Stereochemical Assignments for Goniobutenolides A and B. (1994) (0)
- Catalytic Asymmetric Aminohydroxylation Provides a Short Taxol Side- Chain Synthesis (1996) (0)
- A MAJOR IMPROVEMENT IN THE OSMIUM CATALYZED VICINAL HYDROXYLATION OF OLEFINS BY TERT‐BUTYL HYDROPEROXIDE (2002) (0)
- Structural Characterization of the Pseudoenantiomeric cis-Dioxoosmium(VI) Esters of Chiral Diols with Chinchona Alkaloid Ligands. (1990) (0)
- Documenting the Scope of the Catalytic Asymmetric Dihydroxylation. (1989) (0)
- Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases. (2012) (0)
- Crystal structure of the mouse acetylcholinesterase-TZ2PA6 anti complex (2004) (0)
- THE REACTIONS OF OLEFINS WITH PERMANGANATE, RUTHENIUM TETROXIDE, AND OSMIUM TETROXIDE, DEPENDENCE OF RATE ON DEGREE OF SUBSTITUTION (1975) (0)
- MINIREVIEW Chiral N -Heterocyclic Carbene Ligands Enable Asymmetric CH Bond Functionalization. (2019) (0)
- RS194B pharmacokinetics and antidotal potential in mice exposed to VX and sarin (2018) (0)
- Reversal of Regioselection in the Asymmetric Aminohydroxylation of Cinnamates. (2010) (0)
- Bis(trimethylsilyl) Peroxide Extends the Range of Oxorhenium Catalysts for Olefin Epoxidation. (1998) (0)
- Permeation Across the Mycomembrane in Live Mycobacteria (2022) (0)
- The Asymmetric Dihydroxylation of cis‐Allylic and Homoallylic Alcohols. (1994) (0)
- Catalytic Asymmetric Epoxidation and Kinetic Resolution: Modified Procedures Including in situ Derivatization. (1988) (0)
- Asymmetric Dihydroxylation of α-Substituted Styrene Derivatives ( I), (III). (1994) (0)
- ‘Click Chemistry’ Synthesis of Macrolide Derivatives with Anti-MRSA and Anti-VRE Activity (2008) (0)
- Modified Cinchona Alkaloid Ligands: Improved Selectivities in the Osmium Tetroxide Catalyzed Asymmetric Dihydroxylation (AD) of Terminal Olefins. (1994) (0)
- Ligand design for human nicotinic acetylcholine receptors using in situ freeze‐frame click chemistry (2010) (0)
- Rücktitelbild: SuFEx‐Based Polysulfonate Formation from Ethenesulfonyl Fluoride–Amine Adducts (Angew. Chem. 37/2017) (2017) (0)
- Applications of aziridinium ions. Selective syntheses of alpha, beta-diamino esters, alpha-sulfanyl-beta-amino esters, beta-lactams, and 1,5-benzodiazepin-2-one. (2000) (0)
- p-Nitrobenzoate Esters of Epoxy Alcohols: Convenient Synthons for Water-Soluble Epoxy Alcohols. (1987) (0)
- The “fittest sterol” - origin mysteries still fascinate (2021) (0)
- Catalytic Aminohydroxylation Using Adenine-Derivatives as the Nitrogen Source. (1998) (0)
- Back Cover: Biocompatible SuFEx Click Chemistry: Thionyl Tetrafluoride (SOF 4 )‐Derived Connective Hubs for Bioconjugation to DNA and Proteins (Angew. Chem. Int. Ed. 24/2019) (2019) (0)
- Catalytic Asymmetric Synthesis of New Halogenated Chiral Synthons. (1997) (0)
- Double Diastereoselection in Asymmetric Dihydroxylation. (1993) (0)
- CARBONYL PARTICIPATION IN THE ADDITION OF P-CHLOROPHENYLSELENENYL BROMIDE TO (E)-4-HEXENAL: A NEW ROUTE TO 2,6-DIDEOXYGLYCOSIDES (1979) (0)
- Serratia marcescens Chitinase B complexed with azide inhibitor and quinoline compound (2013) (0)
- New pathways for organic synthesis: Practical applications of transition metals. By H. M. Colquhoun, J. Holton, D. J. Thompson, and M. V. Twigg. Plenum Press, 233 Spring Street, New York, NY 10013. 1984. 454 pp. 16 × 2. cm. $59.50 (1985) (0)
- Cover Picture: Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry (Angew. Chem. Int. Ed. 36/2014) (2014) (0)
- A Simple and Efficient Method for Epoxidation of Terminal Alkenes. (1997) (0)
- Applications of Aziridinium Ions. Selective Syntheses of α,β‐Diamino Esters, α‐Sulfanyl‐β‐amino Esters, β‐Lactams, and 1,5‐Benzodiazepin‐2‐one. (2001) (0)
- New ligands for asymmetric dihydroxylation: cinchona alkaloid multiple devices attached to a central heterocyclic core (1992) (0)
- Asymmetric Dihydroxylation (AD) of α,β-Unsaturated Ketones. (2010) (0)
- Facile Synthesis of Enantiopure trans-2,3-Diphenyl-1,4-diazabicyclo(2. 2.2)octane. (2010) (0)
- Through complex medium accelerated catalytic asymmetric dihydroxylation. (1989) (0)
- Ti(O-i-Pr)4-Mediated Formation of 2,3-Epithio Alcohols from 2,3-Epoxy Alcohols. (1989) (0)
- Asymmetric Dihydroxylation (AD) of N,N-Dialkyl and N-Methoxy-N-methyl . alpha.,β- and β,γ-Unsaturated Amides. (1993) (0)
- Asymmetric Dihydroxylation of Acrolein Acetals: Synthesis of Stable Equivalents of Enantiopure Glyceraldehyde and Glycidaldehyde. (1992) (0)
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