Amnon Albeck
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Most Influential Person Now
Israeli chemist
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Chemistry
Amnon Albeck's Degrees
- PhD Chemistry Technion – Israel Institute of Technology
- Bachelors Chemistry Technion – Israel Institute of Technology
Why Is Amnon Albeck Influential?
(Suggest an Edit or Addition)According to Wikipedia, Amnon Albeck is an organic and bioorganic chemist. Biography Amnon Albeck was born in Jerusalem, Israel, to Michael and Shulamit Albeck on August 1, 1958. Amnon's father is the chemist Prof. Michael Albeck, the fifth president of Bar Ilan University and former president of The Israel Chemical Society . His grandfather, Hanoch Albeck was a professor of Talmud at the Hebrew University of Jerusalem who was one of the founders of the scientific approach to the study of the Mishna.
Amnon Albeck's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Tellurium Compounds: Selective Inhibition of Cysteine Proteases and Model Reaction with Thiols (1998) (88)
- Multifunctional tellurium molecule protects and restores dopaminergic neurons in Parkinson's disease models (2007) (64)
- Synthesis, biological studies and molecular dynamics of new anticancer RGD-based peptide conjugates for targeted drug delivery. (2016) (42)
- Improved stereocontrolled synthesis of threo peptidyl epoxides (1994) (38)
- Stereocontrolled synthesis of erythro N-protected α-amino epoxides and peptidyl epoxides (1994) (36)
- Dual‐drug RGD conjugates provide enhanced cytotoxicity to melanoma and non‐small lung cancer cells (2016) (33)
- IOOC Route to Substituted Chiral Pyrrolidines. Potential Glycosidase Inhibitors (1999) (33)
- Utilization of L-serine in an oxime olefin cycloaddition route to a functionalized asymmetric pyrrolidine, a selective α-glucosidase inhibitor☆ (1994) (28)
- The synthetic tellurium compound, AS101, is a novel inhibitor of IL-1beta converting enzyme. (2007) (28)
- Beta-carotene as a novel therapy for the treatment of “Autistic like behavior” in animal models of Autism (2017) (25)
- Octa‐O‐bis‐(R,R)‐Tartarate Ditellurane (SAS)—a Novel Bioactive Organotellurium(IV) Compound: Synthesis, Characterization, and Protease Inhibitory Activity (2007) (23)
- Peptidyl Epoxides: Novel Selective Inactivators of Cysteine Proteases1 (1996) (23)
- Challenging a paradigm: Theoretical calculations of the protonation state of the Cys25‐His159 catalytic diad in free papain (2009) (23)
- Is there a weak H‐bond → LBHB transition on tetrahedral complex formation in serine proteases? (2004) (23)
- The mechanism of papain inhibition by peptidyl aldehydes (2011) (23)
- Mechanism of cysteine protease inactivation by peptidyl epoxides. (1997) (21)
- "Switch off/switch on" regulation of drug cytotoxicity by conjugation to a cell targeting peptide. (2014) (20)
- The Anticancer Activity of Organotelluranes: Potential Role in Integrin Inactivation (2016) (20)
- Neutral and positively charged thiols synergize the effect of the immunomodulator AS101 as a growth inhibitor of Jurkat cells, by increasing its uptake. (2007) (16)
- Factors determining the relative stability of anionic tetrahedral complexes in serine protease catalysis and inhibition (2000) (16)
- Differentiating Serine and Cysteine Protease Mechanisms by New Covalent QSAR Descriptors (2011) (15)
- Optically Active N‐ and C‐Terminal Building Blocks for the Synthesis of Peptidyl Olefin Peptidomimetics (2010) (14)
- Functionalized erythro N-protected α-amino epoxides. Stereocontrolled synthesis and biological activity (1997) (14)
- Stepwise Versus Concerted Mechanisms in General-Base Catalysis by Serine Proteases. (2016) (13)
- Epoxidation of Peptidyl Olefin Isosteres. Stereochemical Induction Effect of Chiral Centers at Four Adjacent Cα Positions (2000) (12)
- Chloroketone hydrolysis by chymotrypsin and N-methylhistidyl-57-chymotrypsin: implications for the mechanism of chymotrypsin inactivation by chloroketones. (1994) (12)
- Synthesis of orthogonally protected optically pure ketopiperazine, diketopiperazine, ketodiazepane, and 3-aminopyrrolidone building blocks for peptidomimetic combinatorial chemistry (2009) (12)
- Screening of the active site from water by the incoming ligand triggers catalysis and inhibition in serine proteases (2007) (11)
- Facile Synthesis of Orthogonally Protected Optically Pure Keto- and Diketopiperazine Building Blocks for Combinatorial Chemistry (2008) (11)
- Biolabile peptidyl delivery systems toward sequential drug release (2016) (11)
- Efficient and Stereospecific Synthesis of (z)-Hex-3-Enedioic Acid, a Key Intermediate for Gly-Gly cis Olefin Isostere (2000) (11)
- Synthesis of Antitumor Carbazole‐Amonafide Structural Hybrids (2015) (11)
- The Cooperative Effect Between Active Site Ionized Groups and Water Desolvation Controls the Alteration of Acid/Base Catalysis in Serine Proteases (2007) (11)
- How does the exosite of rhomboid protease affect substrate processing and inhibition? (2017) (10)
- The Catalytic Machinery of Rhomboid Proteases: Combined MD and QM Simulations. (2012) (10)
- One-Pot Synthesis of Novel Antiproliferative 9-Aminoacridines (2011) (10)
- Enzyme Isoselective Inhibitors: Application to Drug Design (2006) (9)
- From Catalytic Mechanism to Rational Design of Reversible Covalent Inhibitors of Serine and Cysteine Hydrolases (2014) (9)
- Identification of protons position in acid–base enzyme catalyzed reactions: The hepatitis C viral NS3 protease (2004) (8)
- Optically Active γ‐Hydroxy Sulfone Julia Reagents for the Synthesis of Peptidyl Olefin Peptidomimetics (2008) (8)
- α-Aminoisobutyric Acid Leads a Fluorescent syn-bimane LASER Probe Across the Blood-brain Barrier. (2016) (8)
- Asymmetric Induction by a Remote Chiral Substituent – Computationally Determined Stereodifferentiation in Michael Additions of α-Lithiated Allyl Sulfones (2007) (8)
- 1,4-Dihydropyridine Cationic Peptidomimetics with Antibacterial Activity (2015) (8)
- Enzyme Isoselective Inhibitors: A Tool for Binding‐Trend Analysis (2006) (8)
- Peptidyl epoxides as selective protease inactivators (2000) (8)
- Beta-Carotene derivatives as novel therapy for the prevention and treatment of autistic symptoms. (2021) (7)
- Structural and spatial considerations in the N,N'-diacyl- and bis(alkoxycarbonyl)bispidinone series. (2008) (7)
- Peptidyl epoxides extended in the P' direction as cysteine protease inhibitors: effect on affinity and mechanism of inhibition. (2008) (7)
- Antimicrobial benzodiazepine‐based short cationic peptidomimetics (2015) (7)
- EMBM - A New Enzyme Mechanism-Based Method for Rational Design of Chemical Sites of Covalent Inhibitors (2010) (7)
- Facile synthesis and antitumor activity of novel N(9) methylated AHMA analogs (2012) (7)
- A New Oxopiperazin‐Based Peptidomimetic Molecule Inhibits Prostatic Acid Phosphatase Secretion and Induces Prostate Cancer Cell Apoptosis (2016) (7)
- Ligand-Substitution Reactions of the Tellurium Compound AS-101 in Physiological Aqueous and Alcoholic Solutions. (2016) (7)
- Design of a new selective cysteine protease inactivator and its mechanistic implications (1995) (7)
- Peptidyl cyclopropenones: Reversible inhibitors, irreversible inhibitors, or substrates of cysteine proteases? (2013) (6)
- Anti-neoplastic activity of 1,3-diaza-2-functionalized-adamantan-6-one compounds against melanoma cells. (2013) (6)
- Synthesis of Novel Protected Nα(ω-Drug) Amino Acid Building Units for Facile Preparation of Anticancer Drug-Conjugates (2016) (6)
- Inactivation of cysteine proteases by peptidyl epoxides: characterization of the alkylation sites on the enzyme and the inactivator. (2000) (5)
- Octa-O-bis-(R,R)-Tartarate Ditellurane (SAS) - A Novel Bioactive Organotellurium(IV) Compound: Synthesis, Characterization, and Protease Inhibitory Activity. (2008) (5)
- Free nonimmobilized ligands as a tool for purification of proteins. (2005) (5)
- Phenols-useful templates for the synthesis of bi-functional orthogonally protected dendron building blocks via solid phase Mitsunobu reaction (2010) (5)
- A general approach for antibody purification utilizing [Protein A-catechol:Fe3+] macro-complexes. (2006) (4)
- Exocyclic vinyl ethers of ketofuranosides (2008) (4)
- 12-Substituted-13,14-dihydroretinols designed for affinity labeling of retinol binding- and processing proteins (2004) (3)
- A new method for filtering of reactive "warheads" of transition-state analog protease inhibitors. (2014) (3)
- Gas Phase Bond Formation in Dipeptide Clusters. (2020) (2)
- Efficient and Stereospecific Synthesis of (Z)-Hex-3-enedioic Acid, a Key Intermediate for Gly-Gly cis Olefin Isostere. (2001) (2)
- Bio‐labile peptidyl delivery systems towards sequential drug release (2015) (2)
- Epoxidation of Peptidyl Olefin Isosteres. Stereochemical Induction Effect of Chiral Centers at Four Adjacent Cα Positions. (2000) (1)
- 13-Demethyl-13-substituted-13,14-dihydroretinols as potential affinity labels of retinol-binding proteins: syntheses and stability studies. (2004) (1)
- Application of EMBM to Structure‐Based Design of Warheads for Protease Inhibitors (2014) (1)
- Development and characterisation of SMURF2-targeting modifiers (2021) (1)
- FUNCTIONALIZED ERYTHRO N-PROTECTED ALPHA -AMINO EPOXIDES. STEREOCONTROLLEDSYNTHESIS AND BIOLOGICAL ACTIVITY (1997) (0)
- Optically Active Functionalized Building Blocks for Peptidyl Olefin Peptidomimetics (2021) (0)
- Synthesis of Novel Protected Nα(ω-Drug) Amino Acid Building Units for Facile Preparation of Anticancer Drug-Conjugates (2016) (0)
- Functionalized erythro N-Protected α-Amino Epoxides. Stereocontrolled Synthesis and Biological Activity. (2010) (0)
- Lessons Learned from a Pandemic: One Medical School’s Response to COVID-19 (2020) (0)
- Facile Synthesis and Antitumor Activity of Novel N(9) Methylated AHMA Analogues. (2013) (0)
- Computational, Drug Release and Biological Evaluation of Three New Anti- Cancer Cyclic RGD Peptide Conjugates (2014) (0)
- Poster Session A: Biomaterials 1 Molecular Origin of Biolubrication (2008) (0)
- BAOJ Microbiology (2018) (0)
- Design of a New Selective Cysteine Protease Inactivator and Its Mechanistic Implications. (1995) (0)
- An Unexpected Rearrangement During Mitsunobu Epimerization Reaction of Sugar Derivatives. (2000) (0)
- 1,4-Dihydropyridine Cationic Peptidomimetics with Antibacterial Activity (2015) (0)
- Intact Retinol Polyene Side Chain is Essential for Isomerization, but Not Binding, by RPE65 Isomerohydrolase (2008) (0)
- Ics-Med Chem 2014 (2014) (0)
- Improved Stereocontrolled Synthesis of threo Peptidyl Epoxides (VIII). (1994) (0)
- Publisher Correction: Sourcing Herod the Great’s calcite-alabaster bathtubs by a multi-analytic approach (2022) (0)
- Targeting Necrosis: Elastase-like Protease Inhibitors Curtail Necrotic Cell Death Both In Vitro and in Three In Vivo Disease Models. (2021) (0)
- Stereocontrolled Synthesis of erythro N‐Protected α‐Amino Epoxides and Peptidyl Epoxides. (1994) (0)
- Peptide Bond Formation in Protonated Serine Dimer Following VUV Photon-Induced Excitation. (2023) (0)
- Sourcing Herod the Great's calcite-alabaster bathtubs by a multi-analytic approach (2022) (0)
- Cycloadditions. Part 52. Utilization of L-Serine in an Oxime Olefin Cycloaddition Route to a Functionalized Asymmetric Pyrrolidine, a Selective α-Glucosidase Inhibitor. (1994) (0)
- Lithium Aluminum Hydride Assay Suitable for the Organic Chemistry Laboratory (2016) (0)
- Inside Cover: The Anticancer Activity of Organotelluranes: Potential Role in Integrin Inactivation (ChemBioChem 10/2016) (2016) (0)
- A double heteroatom Mitsunobu coupling with amino hydroxybenzoic acids on solid phase: a novel application of the Mitsunobu reaction to form dendron building blocks (2010) (0)
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