Anders Hallberg
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Swedish chemist
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Anders Hallbergchemistry Degrees
Chemistry
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Organic Chemistry
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Chemistry
Anders Hallberg's Degrees
- Bachelors Chemistry Stockholm University
- Masters Chemistry Uppsala University
- PhD Chemistry Lund University
Why Is Anders Hallberg Influential?
(Suggest an Edit or Addition)According to Wikipedia, Anders Hallberg is a Swedish pharmaceutical researcher, professor in medicinal chemistry and 2006-2011 Rector Magnificus and Vice Chancellor at Uppsala University. Biography Hallberg completed his basic education at Lund University, where he obtained a Master of Science in chemistry and physics in 1969. The following year he attended the School of Education in Malmö obtained a BScEd and worked thereafter as a teacher in the junior high school from 1970-1973.
Anders Hallberg's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Microwave-accelerated homogeneous catalysis in organic chemistry. (2002) (574)
- Correlation of human jejunal permeability (in vivo) of drugs with experimentally and theoretically derived parameters. A multivariate data analysis approach. (1998) (399)
- Microwave-assisted high-speed chemistry: a new technique in drug discovery. (2001) (365)
- Design, synthesis, and biological evaluation of the first selective nonpeptide AT2 receptor agonist. (2004) (317)
- Angiotensin II Type 2 Receptor Stimulation: A Novel Option of Therapeutic Interference With the Renin-Angiotensin System in Myocardial Infarction? (2008) (249)
- Microwave-Promoted Palladium-Catalyzed Coupling Reactions (1996) (221)
- Dimethylformamide as a carbon monoxide source in fast palladium-catalyzed aminocarbonylations of aryl bromides. (2002) (215)
- Increased activity of L-type Ca2+ channels exposed to serum from patients with type I diabetes. (1993) (198)
- Direct Angiotensin II Type 2 Receptor Stimulation Acts Anti-Inflammatory Through Epoxyeicosatrienoic Acid and Inhibition of Nuclear Factor &kgr;B (2010) (194)
- 1,2-Additions to heteroatom-substituted olefins by organopalladium reagents (1989) (182)
- Plasmepsins as potential targets for new antimalarial therapy (2006) (160)
- Expedient synthesis of ebselen and related compounds (1989) (147)
- Stimulation of angiotensin AT2 receptors by the non‐peptide agonist, Compound 21, evokes vasodepressor effects in conscious spontaneously hypertensive rats (2010) (143)
- APR-246 overcomes resistance to cisplatin and doxorubicin in ovarian cancer cells (2015) (137)
- Rapid microwave-assisted Suzuki coupling on solid-phase (1996) (136)
- Cyclic HIV-1 protease inhibitors derived from mannitol: synthesis, inhibitory potencies, and computational predictions of binding affinities. (1997) (135)
- Relationships between structure and interaction kinetics for HIV-1 protease inhibitors. (2002) (134)
- In situ generation of carbon monoxide from solid molybdenum hexacarbonyl. A convenient and fast route to palladium-catalyzed carbonylation reactions. (2002) (130)
- Demonstration of GAD-65 as the main immunogenic isoform of glutamate decarboxylase in type 1 diabetes and determination of autoantibodies using a radioligand produced by eukaryotic expression. (1993) (130)
- High-speed heck reactions in ionic liquid with controlled microwave heating. (2002) (129)
- Unexpected binding mode of a cyclic sulfamide HIV-1 protease inhibitor. (1997) (121)
- Stimulation of AT2 receptor exerts beneficial effects in stroke-prone rats: focus on renal damage (2009) (119)
- Non-peptide AT2-receptor agonists. (2011) (110)
- Synthesis of (E)-(2-arylethenyl)silanes by palladium-catalyzed arylation of vinylsilanes in the presence of silver nitrate (1986) (110)
- The effect of added silver nitrate on the palladium-catalyzed arylation of allyltrimethylsilanes (1985) (105)
- Metabolism of N-acetyl-L-cysteine. Some structural requirements for the deacetylation and consequences for the oral bioavailability. (1989) (103)
- High-Glucose Stimulation of 64,000-Mr Islet Cell Autoantigen Expression (1989) (103)
- Highly regioselective, sequential, and multiple palladium-catalyzed arylations of vinyl ethers carrying a coordinating auxiliary: an example of a Heck triarylation process. (2001) (103)
- Synthesis and comparative molecular field analysis (CoMFA) of symmetric and nonsymmetric cyclic sulfamide HIV-1 protease inhibitors. (2001) (97)
- Palladium/phosphinated polystyrene as a catalyst in the Heck arylation. A comparative study (1985) (97)
- Potent inhibitors of the Plasmodium falciparum enzymes plasmepsin I and II devoid of cathepsin D inhibitory activity. (2004) (95)
- Vinyl sulfide cyclized analogues of angiotensin II with high affinity and full agonist activity at the AT(1) receptor. (2002) (92)
- Hydrogen bonding descriptors in the prediction of human in vivo intestinal permeability. (2003) (92)
- Angiotensin type 2 receptor (AT2R) and receptor Mas: a complex liaison. (2015) (90)
- Acyl sulfonamides as potent protease inhibitors of the hepatitis C virus full-Length NS3 (protease-helicase/NTPase): a comparative study of different C-terminals. (2003) (87)
- AT2-receptor stimulation enhances axonal plasticity after spinal cord injury by upregulating BDNF expression (2013) (81)
- Rapid Fluorous Stille Coupling Reactions Conducted under Microwave Irradiation (1997) (81)
- Design, synthesis, computational prediction, and biological evaluation of ester soft drugs as inhibitors of dihydrofolate reductase from Pneumocystis carinii. (2001) (81)
- Direct Angiotensin AT2 Receptor Stimulation Using a Novel AT2 Receptor Agonist, Compound 21, Evokes Neuroprotection in Conscious Hypertensive Rats (2014) (78)
- Selective terminal heck arylation of vinyl ethers with aryl chlorides: a combined experimental-computational approach including synthesis of betaxolol. (2006) (76)
- Design and synthesis of plasmepsin I and plasmepsin II inhibitors with activity in Plasmodium falciparum-infected cultured human erythrocytes. (2003) (75)
- Rapid palladium-catalyzed synthesis of esters from aryl halides utilizing Mo(CO)(6) as a solid carbon monoxide source. (2003) (74)
- Characterization of the inositol 1,4,5-trisphosphate-induced Ca2+ release in pancreatic beta-cells. (1987) (72)
- High-Speed, Highly Fluorous Organic Reactions (1999) (71)
- Regiochemistry of palladium-catalyzed arylation reactions of enol ethers. Electronic control of selection for .alpha.- or .beta.-arylation (1987) (70)
- Angiotensin Type 2 Receptor Stimulation Ameliorates Left Ventricular Fibrosis and Dysfunction via Regulation of Tissue Inhibitor of Matrix Metalloproteinase 1/Matrix Metalloproteinase 9 Axis and Transforming Growth Factor &bgr;1 in the Rat Heart (2014) (67)
- Advances in the development of pharmaceutical antioxidants (1996) (64)
- A new highly asymmetric chelation-controlled heck arylation. (2003) (64)
- Synthesis of 1-trimethylsilyl 1,3-dienes by the palladium-catalyzed reaction of trimethylvinylsilane with vinyl iodides/silver nitrate or vinyl triflates (1988) (62)
- Formamide as a combined ammonia synthon and carbon monoxide source in fast palladium-catalyzed aminocarbonylations of aryl halides. (2003) (62)
- Design, synthesis, and biological activities of four angiotensin II receptor ligands with gamma-turn mimetics replacing amino acid residues 3-5. (1997) (61)
- Alpha-(phenylselenenyl)acetophenone derivatives with glutathione peroxidase-like activity. A comparison with ebselen. (1992) (61)
- Glutathione peroxidase-like activity of diaryl tellurides. (1993) (61)
- Intramolecular Enantioselective Palladium-Catalyzed Heck Arylation of Cyclic Enamides. (1997) (60)
- Extracellular ATP increases cytoplasmic free Ca2+ concentration in clonal insulin-producing RINm5F cells. A mechanism involving direct interaction with both release and refilling of the inositol 1,4,5-trisphosphate-sensitive Ca2+ pool. (1990) (60)
- A new regioselective Heck vinylation with enamides. Synthesis and investigation of fluorous-tagged bidentate ligands for fast separation. (2003) (59)
- Synthesis of .beta.-arylvinyl ethers by palladium-catalyzed reaction of aroyl chlorides with vinyl ethers (1988) (59)
- Chelation-controlled, palladium-catalyzed vinylic substitution reactions of vinyl ethers. 2-Arylethanal equivalents from aryl halides (1990) (59)
- Aqueous DMF-potassium carbonate as a substitute for thallium and silver additives in the palladium-catalyzed conversion of aryl bromides to acetyl arenes. (2001) (57)
- Design and synthesis of new potent C2-symmetric HIV-1 protease inhibitors. Use of L-mannaric acid as a peptidomimetic scaffold. (1998) (57)
- Computational inhibitor design against malaria plasmepsins (2007) (56)
- Computation of affinity and selectivity: Binding of 2,4-diaminopteridine and 2,4-diaminoquinazoline inhibitors to dihydrofolate reductases (1998) (56)
- Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP). (2010) (54)
- Synthesis of malarial plasmepsin inhibitors and prediction of binding modes by molecular dynamics simulations. (2005) (53)
- A selective AT2 receptor ligand with a gamma-turn-like mimetic replacing the amino acid residues 4-5 of angiotensin II. (2004) (51)
- Chelation-controlled, palladium-catalyzed arylation of enol ethers with aryl triflates. Ligand control of selection for α- or β-arylation of [2-(dimethylamino)ethoxy]ethene (1994) (51)
- Diaryl tellurides as inhibitors of lipid peroxidation in biological and chemical systems. (1994) (51)
- Angiotensin II type 2 receptor promotes adipocyte differentiation and restores adipocyte size in high-fat/high-fructose diet-induced insulin resistance in rats. (2013) (50)
- First reported nonpeptide AT1 receptor agonist (L-162,313) acts as an AT2 receptor agonist in vivo. (2004) (50)
- Regiochemical Control and Suppression of Double Bond Isomerization in the Heck Arylation of 1-(Methoxycarbonyl)-2,5-dihydropyrrole. (1996) (49)
- Presentation of a structurally diverse and commercially available drug data set for correlation and benchmarking studies. (2006) (49)
- Regioselective palladium-catalyzed synthesis of beta-arylated primary allylamine equivalents by an efficient Pd-N coordination. (2001) (49)
- Design and fast synthesis of C-terminal duplicated potent C(2)-symmetric P1/P1'-modified HIV-1 protease inhibitors. (1999) (49)
- Differential Sensitivity to β-Cell Secretagogues in Cultured Rat Pancreatic Islets Exposed to Human Interleukin-1β* (1989) (48)
- Exploration of acyl sulfonamides as carboxylic acid replacements in protease inhibitors of the hepatitis C virus full-length NS3. (2006) (46)
- Two-carbon-elongated HIV-1 protease inhibitors with a tertiary-alcohol-containing transition-state mimic. (2008) (45)
- Inhibitors of the C(2)-symmetric HIV-1 protease: nonsymmetric binding of a symmetric cyclic sulfamide with ketoxime groups in the P2/P2' side chains. (1999) (43)
- Design and synthesis of potent inhibitors of the malaria aspartyl proteases plasmepsin I and II. Use of solid-phase synthesis to explore novel statine motifs. (2004) (42)
- Highly Regioselective Palladium-Catalyzed Internal Arylation of Allyltrimethylsilane with Aryl Triflates (1998) (42)
- Evidence for a common selenolate intermediate in the glutathione peroxidase-like catalysis of α-(phenylselenenyl) ketones and diphenyl diselenide (1994) (41)
- Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors. (2003) (41)
- Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'. (2005) (41)
- Coexpression of the platelet-derived growth factor (PDGF) B chain and the PDGF beta receptor in isolated pancreatic islet cells stimulates DNA synthesis. (1990) (41)
- Antioxidant activity of some diarylselenides in biological systems. (1994) (41)
- New selective AT2 receptor ligands encompassing a gamma-turn mimetic replacing the amino acid residues 4-5 of angiotensin II act as agonists. (2005) (41)
- C2-symmetric inhibitors of Plasmodium falciparum plasmepsin II: synthesis and theoretical predictions. (2003) (41)
- Potent macrocyclic inhibitors of insulin-regulated aminopeptidase (IRAP) by olefin ring-closing metathesis. (2011) (40)
- Controlled Double-Bond Migration in Palladium-Catalyzed Intramolecular Arylation of Enamidines. (1996) (40)
- From the first selective non-peptide AT(2) receptor agonist to structurally related antagonists. (2012) (39)
- Angiotensin AT2-receptor stimulation improves survival and neurological outcome after experimental stroke in mice (2016) (39)
- Microwave-accelerated synthesis of P1'-extended HIV-1 protease inhibitors encompassing a tertiary alcohol in the transition-state mimicking scaffold. (2006) (39)
- A new class of HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold. (2005) (39)
- Scope, Mechanism and Other Fundamental Aspects of the Intermolecular Heck Reaction (2003) (39)
- STYRENE DERIVATIVES VIA PALLADIUM-CATALYZED VINYLATION OF ARYL IODIDES (1982) (38)
- Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II. (2005) (38)
- Direct angiotensin type 2 receptor (AT2R) stimulation attenuates T-cell and microglia activation and prevents demyelination in experimental autoimmune encephalomyelitis in mice. (2015) (38)
- Regioselective palladium-catalyzed tandem .alpha.-arylation/isomerization of cyclic enamides (1990) (37)
- Human immunodeficiency virus type 1 proteinase resistance to symmetric cyclic urea inhibitor analogs (1997) (37)
- Design, synthesis, and incorporation of a beta-turn mimetic in angiotensin II forming novel pseudopeptides with affinity for AT1 and AT2 receptors. (2006) (37)
- Characterization of a Set of HIV-1 Protease Inhibitors Using Binding Kinetics Data from a Biosensor-Based Screen (2000) (36)
- Fast, Convenient, and Efficient Molybdenum‐Catalyzed Asymmetric Allylic Alkylation under Noninert Conditions: An Example of Microwave‐Promoted Fast Chemistry (2000) (36)
- Palladium-catalysed arylation of vinyltrimethylsilane in the presence of silver nitrate (1985) (36)
- Long-term effects of cyclosporin A on cultured mouse pancreatic islets (1984) (36)
- Stereoselective palladium-catalyzed synthesis of (Z)-trimethyl(2-arylethenyl)silanes by arylation of (E)-1,2-bis(trimethylsilyl)ethylene. Effects of added halides compared to silver salts (1989) (36)
- Fast synthesis of aryl triflates with controlled microwave heating. (2002) (36)
- Tetrapeptides as potent protease inhibitors of Hepatitis C Virus full-length NS3 (protease-helicase/NTPase). (2002) (36)
- Synthesis and enzymatic hydrolysis of esters, constituting simple models of soft drugs. (1998) (36)
- RAPID MICROWAVE-INDUCED PALLADIUM-CATALYZED ASYMMETRIC ALLYLIC ALKYLATION (1999) (36)
- Design and synthesis of potent inhibitors of plasmepsin I and II: X-ray crystal structure of inhibitor in complex with plasmepsin II. (2005) (36)
- Enhanced stimulus-secretion coupling in polyamine-depleted rat insulinoma cells. An effect involving increased cytoplasmic Ca2+, inositol phosphate generation, and phorbol ester sensitivity. (1993) (35)
- Inhibition of hepatitis C virus NS3 protease activity by product-based peptides is dependent on helicase domain. (2001) (35)
- Angiotensin II, a Neuropeptide at the Frontier between Endocrinology and Neuroscience: Is There a Link between the Angiotensin II Type 2 Receptor and Alzheimer’s Disease? (2011) (35)
- HIV-1 protease inhibitors with a transition-state mimic comprising a tertiary alcohol: improved antiviral activity in cells. (2010) (34)
- Macrocyclic inhibitors of the malarial aspartic proteases plasmepsin I, II, and IV. (2006) (34)
- P1/P1' modified HIV protease inhibitors as tools in two new sensitive surface plasmon resonance biosensor screening assays. (2001) (34)
- Synthesis of two conformationally constrained analogues of the minor tobacco alkaloid anabasine. (2000) (33)
- Effects of long‐term chloroquine exposure on the phospholipid metabolism in retina and pigment epithelium of the mouse (1990) (33)
- DIRECT SYNTHESIS OF CYCLIC KETALS OF ACETOPHENONES BY PALLADIUM-CATALYZED ARYLATION OF HYDROXYALKYL VINYL ETHERS (1997) (33)
- Rapid and stereoselective C-C, C-O, C-N and C-S couplings via microwave accelerated palladium-catalyzed allylic substitutions (2000) (32)
- Design, synthesis and SAR of potent statine-based BACE-1 inhibitors: exploration of P1 phenoxy and benzyloxy residues. (2008) (31)
- Angiotensin II pseudopeptides containing 1,3,5-trisubstituted benzene scaffolds with high AT2 receptor affinity. (2005) (31)
- Small‐molecule AT2 receptor agonists (2018) (30)
- Microwave-Accelerated Homogeneous Catalysis in Organic Chemistry (2002) (30)
- Regioselective palladium-catalyzed arylation of vinyl ethers with 4-nitrophenyl triflate. Control by addition of halide ions (1988) (30)
- Selective angiotensin II AT2 receptor agonists: Benzamide structure-activity relationships. (2008) (30)
- Palladium-catalyzed aroylation of alkyl vinyl ethers. An entry to monoprotected 1-aryl-1,3-dicarbonyl equivalents (1988) (30)
- Palladium-catalyzed vinylation of alkyl vinyl ethers with enol triflates. A convenient synthesis of 2-alkoxy 1,3-dienes (1989) (29)
- Palladium-catalyzed arylation of methyl vinyl ether (1981) (29)
- Comparative functional properties of two structurally similar selective nonpeptide drug-like ligands for the angiotensin II type-2 (AT(2)) receptor. Effects on neurite outgrowth in NG108-15 cells. (2013) (29)
- Effects of N-acetylcysteine stereoisomers on oxygen-induced lung injury in rats. (1995) (29)
- High-speed synthesis of potent C2-symmetric HIV-1 protease inhibitors by in-situ aminocarbonylations. (2005) (28)
- HIV-1 protease inhibitors based on acyclic carbohydrates (1998) (28)
- An improved procedure for N- to C-directed (Inverse) solid-phase peptide synthesis. (2000) (27)
- Inhibitor binding to the plasmepsin IV aspartic protease from Plasmodium falciparum. (2006) (27)
- Synthesis, receptor binding affinities and conformational properties of cyclic methylenedithioether analogues of angiotensin II. (2001) (26)
- Design and synthesis of potent and selective BACE-1 inhibitors. (2010) (26)
- Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: use of cyclopentane and cyclopentene P2-motifs. (2007) (25)
- New potent C2-symmetric malaria plasmepsin I and II inhibitors. (2003) (25)
- Selective angiotensin II AT(2) receptor agonists with reduced CYP 450 inhibition. (2010) (25)
- AT2-selective angiotensin II analogues containing tyrosine-functionalized 5,5-bicyclic thiazabicycloalkane dipeptide mimetics. (2004) (25)
- Synthesis and AT2 receptor-binding properties of angiotensin II analogues. (2004) (25)
- The Enåsen gold deposit, central Sweden (1994) (25)
- Bicyclic tripeptide mimetics with reverse turn inducing properties. (1999) (24)
- Masked 3-aminoindan-1-ones by a palladium-catalyzed three-component annulation reaction. (2005) (24)
- Computational predictions of binding affinities to dihydrofolate reductase: synthesis and biological evaluation of methotrexate analogues. (2000) (24)
- Synthesis of a new class of druglike angiotensin II C-terminal mimics with affinity for the AT2 receptor. (2007) (24)
- Aspartic protease inhibitors containing tertiary alcohol transition-state mimics. (2015) (23)
- The En isen gold deposit , central Sweden 1 . A palaeoproterozoic high-sulphidation epithermal gold mineralization (23)
- Synthesis of Amino Acids with Modified Principal Properties. 1. Amino Acids with Fluorinated Side Chains. (1993) (23)
- Microwave-mediated palladium-catalyzed asymmetric allylic alkylation; an example of highly selective fast chemistry (2000) (23)
- A new structural theme in C2-symmetric HIV-1 protease inhibitors: ortho-substituted P1/P1' side chains. (2006) (23)
- Design, synthesis, and computational affinity prediction of ester soft drugs as inhibitors of dihydrofolate reductase from Pneumocystis carinii. (2004) (22)
- Synthesis of potent BACE-1 inhibitors incorporating a hydroxyethylene isostere as central core. (2010) (22)
- Plasma membrane associated ATP as a regulator of the secretory activity of the pancreatic beta-cell. (2009) (22)
- Catalytic effects of glutathione peroxidase mimetics on the thiol reduction of cytochrome c. (1994) (22)
- CHELATION-CONTROLLED, PALLADIUM-CATALYZED ARYLATION OF VINYL ETHERS (1993) (21)
- Terminal Heck Vinylations of Chelating Vinyl Ethers (2004) (21)
- Design and synthesis of potent C(2)-symmetric diol-based HIV-1 protease inhibitors: effects of fluoro substitution. (2001) (21)
- Hydrozirconation--Isomerisation. Reactions of Terminally Functionalised Olefins with Zirconocene Hydrides and General Aspects. (1993) (21)
- Effects of starvation and different culture conditions on the phospholipid content of isolated pancreatic islets. (1984) (21)
- Structure-activity relationships for the selectivity of hepatitis C virus NS3 protease inhibitors. (2004) (21)
- Potent inhibitors of the hepatitis C virus NS3 protease: use of a novel P2 cyclopentane-derived template. (2006) (21)
- New inhibitors of the malaria aspartyl proteases plasmepsin I and II. (2003) (20)
- The correlation of the oxidation potentials of structurally related dibenzo[1,4]dichalcogenines to their antioxidance capacity in biological systems undergoing free radical-induced lipid peroxidation. (1991) (20)
- Heck arylation of 1,2-cyclohexanedione and 2-ethoxy-2-cyclohexenone (1998) (20)
- 3-Substituted pyrazoles and 4-substituted triazoles as inhibitors of human 15-lipoxygenase-1. (2015) (19)
- Synthesis of enantiomerically pure cis and trans 2-aminocyclopentanecarboxylic acids. Use of proline replacements in potential HIV-protease inhibitors (1997) (19)
- Modulation of beta-cell activity and its influence on islet cell antibody (ICA) and islet cell surface antibody (ICSA) reactivity. (1993) (19)
- Short pseudopeptides containing turn scaffolds with high AT2 receptor affinity. (2006) (19)
- Synthesis of 1-propyl-3-(3-hydroxyphenyl)piperidine by regiocontrolled palladium-catalyzed arylation (1992) (19)
- A Simplified Synthesis of 3-Bromoselenophene and Some 3-Bromothiophenes (1981) (19)
- Selectivity and reactivity in asymmetric allylic alkylation (1999) (19)
- Metal sources in the Early Proterozoic Svecofennian terrain of central Sweden: Pb isotope evidence (1989) (18)
- Angiotensin II type 2 receptor stimulation improves fatty acid ovarian uptake and hyperandrogenemia in an obese rat model of polycystic ovary syndrome. (2014) (18)
- Design and synthesis of dihydrofolate reductase inhibitors encompassing a bridging ester group. Evaluation in a mouse colitis model. (2003) (18)
- Transfection of insulin-producing cells with a transforming c-Ha-ras oncogene stimulates phospholipase C activity. (1989) (18)
- A convenient synthesis of 1-(S)-[1′-(S)-(t-butyloxycarbonylamino)-2′-phenylethyl]oxirane. A useful building block in the synthesis of HIV protease inhibitors (1997) (17)
- Hydrozirconation of (E)-3-methoxy-1-phenyl-1-propene and (E)-3-phenyl-2-propenol (1991) (17)
- Variations of the P2 group in HIV-1 protease inhibitors containing a tertiary alcohol in the transition-state mimicking scaffold. (2006) (17)
- Angiotensin II analogues encompassing 5,9- and 5,10-fused thiazabicycloalkane tripeptide mimetics. (1999) (17)
- Symmetric fluoro-substituted diol-based HIV protease inhibitors. Ortho-fluorinated and meta-fluorinated P1/P1'-benzyloxy side groups significantly improve the antiviral activity and preserve binding efficacy. (2004) (16)
- Structural determinants of subtype selectivity and functional activity of angiotensin II receptors. (2016) (16)
- Fast and selective synthesis of novel cyclic sulfamide HIV-1 protease inhibitors under controlled microwave heating (2006) (15)
- Synthesis of potent C(2)-symmetric, diol-based hiv-1 protease inhibitors. Investigation of thioalkyl and thioaryl P1/P1' substituents. (2001) (15)
- Palladium on charcoal-catalysed arylation of methyl vinyl ether with 4-bromonitrobenzene (1984) (15)
- Angiotensin Peptides as AT2 Receptor Agonists. (2017) (15)
- Human interleukin 1 beta stimulates islet insulin release by a mechanism not dependent on changes in phospholipase C and protein kinase C activities or Ca2+ handling. (1989) (15)
- Synthesis of novel, potent, diol-based HIV-1 protease inhibitors via intermolecular pinacol homocoupling of (2S)-2-benzyloxymethyl-4-phenylbutanal. (2001) (15)
- Comparison of three γ-turn mimetic scaffolds incorporated into angiotensin II (2000) (15)
- The Enåsen gold deposit, central Sweden (1994) (14)
- Synthesis of a small library of non-symmetric cyclic sulfamide HIV-1 protease inhibitors (2010) (14)
- Microwave-Assisted Enantioselective Heck Reactions: Expediting High Reaction Speed and Preparative Convenience (2002) (14)
- Controlled Microwave Heating as an Enabling Technology: Expedient Synthesis of Protease Inhibitors in Perspective (2007) (14)
- Aryl Radical Endo Cyclization of Enamidines. Selective Preparation of Trans and Cis Fused Octahydrobenzo[f]quinolines. (1998) (13)
- On the reaction of methoxide ion with bromoiodothiophenes (1980) (13)
- A one-pot isomerization-arylation of 2,3-epoxycyclohexanone under controlled microwave heating. (2005) (13)
- Solid-phase library synthesis of reversed-statine type inhibitors of the malarial aspartyl proteases plasmepsin I and II. (2003) (13)
- AT2 Receptor Agonists: Exploiting the Beneficial Arm of Ang II Signaling (2012) (13)
- Discovery of potent BACE-1 inhibitors containing a new hydroxyethylene (HE) scaffold: exploration of P1' alkoxy residues and an aminoethylene (AE) central core. (2010) (13)
- Preparation of N-Formyl- and N-carbomethoxy-2,3-dihydropyrroles by palladium-catalyzed isomerization of the corresponding N-acyl-2,5-dihydropyrrole (1995) (13)
- Microwave-Promoted Palladium-Catalyzed Coupling Reactions. (1997) (13)
- N-Substituted pyrazole-3-carboxamides as inhibitors of human 15-lipoxygenase. (2015) (13)
- Hydrozirconation of 1-arylalkenes (1989) (13)
- Stereoselective synthesis of 3-aminoindan-1-ones and subsequent incorporation into HIV-1 protease inhibitors. (2006) (13)
- Seven days treatment with the angiotensin II type 2 receptor agonist C21 in hospitalized COVID-19 patients; a placebo-controlled randomised multi-centre double-blind phase 2 trial (2021) (12)
- Design and synthesis of HIV-1 protease inhibitors. Novel tetrahydrofuran P2/P2'-groups interacting with Asp29/30 of the HIV-1 protease. Determination of binding from X-ray crystal structure of inhibitor protease complex. (2003) (12)
- Ring-opening reactions. Part 16. Ring-opening of 2,5-dimethoxy-3-thienyl-lithium and some related compounds (1980) (12)
- Effect of 3-5 monocyclizations of angiotensin II and 4-aminoPhe6-Ang II on AT2 receptor affinity. (2003) (12)
- Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides (2018) (12)
- Aspects of the preparation of cyclohexenyl- and menthenylthioenynesviaring-opening of thiophenes: Preparation of Cyclohexenyl- and Menthenylthioenynes (1983) (12)
- Synthesis of Bis(alpha-alkylaminobenzylidene)hydrazines and their Transformation into 4-Alkyl-4H-1,2,4-triazoles. (1991) (12)
- Design and synthesis of P1-P3 macrocyclic tertiary-alcohol-comprising HIV-1 protease inhibitors. (2013) (12)
- Chromatographic resolution, circular dichroism spectra, and absolute configurations of dimers of 5H-indolo[1,7-ab][1]benzazepine and coumarin with C2 symmetry (1989) (12)
- Design and synthesis of novel P2 substituents in diol-based HIV protease inhibitors. (2010) (12)
- Determination of Absolute Configurations of N-Formyl-3,3‘,4,4‘-tetrahydrospiro[naphthalene-1(2H),2‘(1‘H)-pyridine] (2) and N-Formyl-3‘,4‘-dihydrospiro[indan-1,2‘(1‘H)-pyridine] (3) by Analysis of Circular Dichroism Spectra. A Case of Two Compounds with Similar Configuration But Nearly Mirror Image C (1997) (11)
- New synthesis of pentasubstituted benzenes by tandem dimerization-ring opening of 3-halo-2,5-dialkylthiophene 1,1-dioxides (1988) (11)
- A stereoselective synthesis of dialkylaminomethyl substituted halobutadienes via amine induced ring-opening of thiophene-1,1-dioxides (1987) (11)
- Further examples of tandem dimerization ring-opening of substituted 3-bromothiophene 1,1-dioxides. Preparation of trisubstituted benzenes. X-ray structure determination of 3,5-dibromo-7,7a-dimethyl-2,4-diphenyl-cis-3a,7a-dihydrobenzo[b]thiophene 1,1-dioxide (1991) (11)
- Mass spectral fragmentation patterns of heterocycles. VI. Carbazole and 1,8-dideuteriocarbazole† (1984) (11)
- Microwave spectrum, conformation, intramolecular hydrogen bonding and Ab initio computations for 2,2,3,3-tetrafluoro-1-propanol (1993) (11)
- A Study of Allylboronates as Substrates in Palladium-Mediated Arylation. (1988) (11)
- Glutathione in human melanoma cells. Effects of cysteine, cysteine esters and glutathione isopropyl ester. (1990) (11)
- Impact of the Central Hydroxyl Groups on the Activity of Symmetrical HIV-1 Protease Inhibitors Derived From l-Mannaric Acid (2000) (11)
- Acylations of 1,10-dilithiophenothiazine. A new synthesis of 1-formylphenothiazine (1982) (10)
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- Dimerization reactions of some thiophene 1,1-dioxides. Preparation of benzo[b]thiophene 1,1-dioxides (1991) (9)
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- The Palaeoproterozoic apatite-iron oxide deposite of the Grängesberg areas: Kiruna-type deposits in central Sweden (2010) (7)
- A MODIFIED BISCHLER SYNTHESIS OF SOME TETRACYCLIC INDOLE DERIVATIVES (1982) (7)
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- Mass spectral fragmentation patterns of heterocycles. VII . Reinvestigation of fundamental processes in phenothiazines (1984) (6)
- Resistance Profiles of Cyclic and Linear Inhibitors of HIV-1 Protease (2002) (6)
- Islet cell antibodies: variable immunostaining of pancreatic islet cells and carcinoid tissue (1995) (6)
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- Effects of starvation on phospholipid metabolism of pancreatic islets. (1984) (6)
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- MAIN METALLOGENIC EVENTS IN FENNOSCANDIA: SUMMARY (2012) (6)
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- Novel synthesis of some tricyclic ketones via lithium di-isopropylamidemediated cyclization of 2-o-carboxyphenyl ethenylfurans, thiophens, and selenophens (1983) (5)
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- Fmoc protected peptide mimetic based on a cyclohexane framework and incorporation into angiotensin II (1997) (5)
- Synthesis of C-2 symmetric potential inhibitors of HIV-1 protease from D-mannitol (1996) (5)
- Solid- and liquid-phase photodimerizations of 5H-indolo[1,7-ab][1]benzazepine (1984) (5)
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- INDOLO(1,7-AB)(1)BENZAZEPINE, A NEW 18 Π-ELECTRON HETEROCYCLE (1981) (4)
- Chromatographic enantiomer separation and chiroptical properties of 1-acyl-2-aryl-1,2,3,4-tetrahydropyridines and some analogues (1991) (4)
- Aspects of the hydrozirconation-isomerisation reaction (1989) (4)
- Metallations of 5 H‐dibenz [b, f] azepine and 10,11‐dihydro‐5H‐dibenz [b, f] azepine. Synthesis of 4‐substituted derivatives (1983) (4)
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- The Unexpected Formation of 3,4,7,8-Tetramethyl-1,2,5,6-tetrahydrodicyclobuta[a,e]cyclooctene from a Zirconacyclopentadiene. (1993) (4)
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- Oxygen isotopes and geochemistry of Palaeoproterozoic Kiruna-type deposits in the Bergslagen province, Sweden (2011) (3)
- Unexpected disproportionation of 4,4′-dialkylamino substituted diaryl selenides and tellurides (1995) (3)
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- The synthesis of some novel polycyclic chromans (1993) (3)
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- ASPECTS OF THE PREPARATION OF CYCLOHEXENYL‐ AND MENTHENYLTHIOENYNES VIA RING‐OPENING OF THIOPHENES (1984) (2)
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- The genesis of the Enåsen gold deposit (1993) (1)
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- RING-OPENING REACTIONS. XVII. ON THE REACTION OF 2-CHLORO-5-METHOXYTHIOPHENE AND ITS MONOBROMO DERIVATIVES WITH BUTYLLITHIUM (1980) (1)
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- THE SELECTIVITY OF ARYL RADICALS IN REACTIONS WITH HALIDE IONS. THE KEY STEP IN THE SRN1 MECHANISM (1982) (1)
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- TOTAL ASSIGNMENT OF THE CARBON-13 NMR SPECTRA OF 5H-INDOLO(1,7-AB)(1)BENZAZEPINE AND 6,7-DIHYDRO-5H-INDOLO(1,7-AB)(1)BENZAZEPINE USING TWO-DIMENSIONAL PROTON-CARBON CHEMICAL SHIFT CORRELATION EXPERIMENTS (1985) (0)
- MASS SPECTRAL FRAGMENTATION PATTERNS OF HETEROCYCLES. VI. CARBAZOLE AND 1,8-DIDEUTERIOCARBAZOLE (1985) (0)
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- ON THE REACTION OF SOME THIENYLLITHIUM DERIVATIVES WITH 1-CHLORO-2-DIMETHYLAMINOETHANE (1981) (0)
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- NOVEL SYNTHESIS OF SOME TRICYCLIC KETONES VIA LITHIUM DIISOPROPYLAMIDE-MEDIATED CYCLIZATION OF 2-(O-CARBOXYPHENYL)ETHENYLFURANS, -THIOPHENES, AND -SELENOPHENES (1983) (0)
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- Palladium‐Catalyzed Vinylation of Alkyl Vinyl Ethers with Enol Triflates. A Convenient Synthesis of 2‐Alkoxy‐1,3‐dienes. (1989) (0)
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- PALLADIUM ON CHARCOAL-CATALYZED ARYLATION OF METHYL VINYL ETHER WITH 4-BROMONITROBENZENE (1984) (0)
- A process for organic reactions (1997) (0)
- Reaction of the Aromatic Olefin 1-(1-Hexenyl)-2-thiomethylbenzene with Cp2Zr(H)Cl. Unexpected Cleavage of the Methyl-Sulfur Bond. (1989) (0)
- Palladium-Catalyzed Aroylation of Alkyl Vinyl Ethers. An Entry to Monoprotected 1-Aryl-1,3-dicarbonyl Equivalents. (1989) (0)
- Investigating the Mimetic Potential of β-Turn Mimetics (2000) (0)
- Synthesis of 3‐Dialkylaminochromans via Thallium(III)‐Induced Cyclization of Allyl Aryl Ethers. (1991) (0)
- ON THE ASSIGNMENT OF THE CARBON-13 NMR SPECTRUM OF PHENOTHIAZINE (1984) (0)
- Reaction of 3‐Bromo‐2,5‐dimethylthiophene 1,1‐Dioxide with Some Grignard Reagents. The Formation of a Heterotricycloheptane Derivative. (1991) (0)
- Reaction of 3,4-Dibromo-2,5-dimethylthiophene-1,1-dioxide with Piperidine. X-Ray Structure Determination of 3-Bromo-2-methyl-4-piperidino-5-piperidinomethyl-cis-4,5-dihydrothiophene-1,1-dioxide. (1987) (0)
- A One-Pot Isomerization—Arylation of 2,3-Epoxycyclohexanone under Controlled Microwave Heating. (2005) (0)
- MASS SPECTRAL FRAGMENTATION PATTERNS OF HETEROCYCLES. V. ELECTRON IMPACT PROMOTED MASS SPECTRAL FRAGMENTATION OF INDOLO(1,7-AB)(1)BENZAZEPINE AND SOME OF ITS DERIVATIVES (1984) (0)
- Rapid and Stereoselective C-C, C-O, C-N and C-S Couplings via Microwave Accelerated Palladium-Catalyzed Allylic Substitutions. (2000) (0)
- 1,2-Additions to Heteroatom-Substituted Olefins by Organo-Palladium Reagents (1990) (0)
- A method for regio-directed bicyclization of peptides. (1998) (0)
- Chromatographic Resolution, CD Spectra, and Absolute Configurations of Dimers of 5H-Indolo(1,7-ab)(1)benzazepine and Coumarin with C2 Symmetry (1989) (0)
- Regioselective Palladium-Catalyzed Tandem α-Arylation/Isomerization of Cyclic Enamides (I). (1990) (0)
- A New Synthesis of Pentasubstituted Benzenes by Tandem Dimerization Ring Opening of 3‐Halo‐2,5‐dialkylthiophene 1,1‐Dioxides. (1988) (0)
- Intramolecular Enantioselective Palladium‐Catalyzed Heck Arylation of Cyclic Enamides. (2010) (0)
- New High Speed New High Speed Regioselective Regioselective Heck Coupling Heck Coupling Reactions Assisted By Reactions Assisted By Microwave Flash Heating (2001) (0)
- Seven Days Treatment With the Angiotensin II Type 2 Receptor Agonist C21 in Hospitalized COVID-19 Patients: A Placebo-Controlled Randomized Phase 2 Trial (2021) (0)
- THE ASSIGNMENT OF THE PROTON NMR AND CARBON‐13 NMR SPECTRA OF 5H‐DIBENZ(B,F)AZEPINE AND 10,11‐DIHYDRO‐5H‐DIBENZ(B,F)AZEPINE (1984) (0)
- Unexpected Disproportionation of 4,4′-Dialkylamino Substituted Diaryl Selenides and Tellurides. (1995) (0)
- P1' Extended HIV-1 Protease Inhibitors Encompassing a Tertiary Alcohol in the Transition-State Mimicking Scaffold (2007) (0)
- Highly Stereo‐ and Regioselective Allylations Catalyzed by Mo—Pyridylamide Complexes: Electronic and Steric Effects of the Ligand. (2000) (0)
- Preparation of Pyrrolo[3,2,1-jk]carbazole by Nickel(0) Mediated Ring Contraction of Pyrrolo[3,2,1-jk]phenothiazine. (1986) (0)
- Cyclic 7-membered sulfamide HIV-1 protease inhibitors (1998) (0)
- New bicyclic agonists angiotensin II (2006) (0)
- Regulation of phospholipid metabolism in isolated pancreatic islets (1984) (0)
- Agonists tricyclic compounds useful as angiotensin ii (2002) (0)
- Thermal and photochemical hydrolysis and water exchange reactions of aqua(1,3-propanediamine) complexes of chromium(III) (1993) (0)
- Synthesis of Enantiomerically Pure cis and trans 2- Aminocyclopentanecarboxylic Acids. Use of Proline Replacements in Potential HIV-Protease Inhibitors. (1997) (0)
- A flexible regioselective method for bicyclization of peptides. (2002) (0)
- Investigation of the possible dopaminergic toxicity of 1-methyl-3-phenyl-1,2,3,6-tetrahydropyridine, an isomer to the neurotoxin MPTP. (1991) (0)
- Potent Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease. Use of Cyclopentane and Cyclopentene Derived P2-Scaffolds (2007) (0)
- Different Types of P1 Residues in Peptide-Based Inhibitors of Hepatitis C Virus Full-Length NS3 Protease (2001) (0)
- Trials with different cutting times in leys combined with conservation and digestibility studies. (1961) (0)
- Peptide-based protease inhibitors of the hepatitis C virus full-length NS3 protein (protease-helicase/NTPase) (2002) (0)
- Microwave-Assisted Enantioselective Heck Reactions: Expediting High Reaction Speed and Preparative Convenience. (2002) (0)
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