Andreas Bernkop-Schnürch
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Austrian university teacher
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Andreas Bernkop-Schnürch's Degrees
- PhD Pharmaceutical Sciences University of Innsbruck
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(Suggest an Edit or Addition)According to Wikipedia, Andreas Bernkop-Schnürch is an Austrian pharmaceutical technologist, scientist, pharmacist, entrepreneur, inventor and professor at the Institute of Pharmacy, University of Innsbruck. His research centers on the areas of pharmaceutical sciences, drug delivery, controlled release, bionanotechnology and polymer engineering. He is the inventor of various technologies such as thiolated polymers for that he coined the name thiomers in 2000 and phosphatase triggered charge converting nanoparticles for mucosal drug delivery. From 2016 to 2018 he served as a member of the Scientific Committee of the Innovative Medicines Initiative of the European Union in Brussels giving advice on scientific priorities to be included in the Strategic Research Agenda for Horizon 2020. Since 2014 he is on the scientific advisory board of the Nicotine Science Center, Denmark. Andreas Bernkop-Schnürch is the founder of Mucobiomer Biotechnologische Forschungs- und Entwicklungs GmbH , Thiomatrix Forschungs- und Beratungs GmbH and Green River Polymers Forschungs und Entwicklungs GmbH. He is listed as a Highly Cited Researcher of the Institute of Scientific Information.
Andreas Bernkop-Schnürch's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Chitosan-based drug delivery systems. (2012) (597)
- Strategies to improve plasma half life time of peptide and protein drugs (2006) (553)
- Thiomers: a new generation of mucoadhesive polymers. (2005) (436)
- Thiolated polymers--thiomers: development and in vitro evaluation of chitosan-thioglycolic acid conjugates. (2001) (416)
- Comparison of the mucoadhesive properties of various polymers. (2005) (401)
- Thiolated polymers--thiomers: synthesis and in vitro evaluation of chitosan-2-iminothiolane conjugates. (2003) (383)
- Thiolated polymers: evidence for the formation of disulphide bonds with mucus glycoproteins. (2003) (348)
- Polymers with Thiol Groups: A New Generation of Mucoadhesive Polymers? (1999) (307)
- The use of inhibitory agents to overcome the enzymatic barrier to perorally administered therapeutic peptides and proteins. (1998) (290)
- Mucoadhesive thiolated chitosans as platforms for oral controlled drug delivery: synthesis and in vitro evaluation. (2004) (286)
- Chitosan and its derivatives: potential excipients for peroral peptide delivery systems. (2000) (242)
- Permeation enhancing polymers in oral delivery of hydrophilic macromolecules: thiomer/GSH systems. (2003) (231)
- Improvement in the mucoadhesive properties of alginate by the covalent attachment of cysteine. (2001) (226)
- Synthesis and characterisation of mucoadhesive thiolated polymers. (2000) (222)
- Mucoadhesive polymers as platforms for peroral peptide delivery and absorption: synthesis and evaluation of different chitosan-EDTA conjugates. (1998) (207)
- Thiolated chitosans: development and in vitro evaluation of a mucoadhesive, permeation enhancing oral drug delivery system. (2004) (204)
- Mucoadhesive vs. mucopenetrating particulate drug delivery. (2016) (202)
- Review articleThiolated chitosans (2004) (178)
- Successful oral delivery of poorly water-soluble drugs both depends on the intraluminal behavior of drugs and of appropriate advanced drug delivery systems. (2019) (176)
- Mucoadhesive ocular insert based on thiolated poly(acrylic acid): development and in vivo evaluation in humans. (2003) (170)
- In vitro evaluation of the viscoelastic properties of chitosan-thioglycolic acid conjugates. (2003) (169)
- Oral insulin delivery: the potential of thiolated chitosan-insulin tablets on non-diabetic rats. (2004) (167)
- The Role of Glutathione in the Permeation Enhancing Effect of Thiolated Polymers (2002) (166)
- Design and in vitro evaluation of a novel bioadhesive vaginal drug delivery system for clotrimazole. (2002) (164)
- Preactivated thiomers as mucoadhesive polymers for drug delivery (2012) (160)
- Thiolated polymers: self-crosslinking properties of thiolated 450 kDa poly(acrylic acid) and their influence on mucoadhesion. (2002) (158)
- Development and evaluation of a novel mucus diffusion test system approved by self-nanoemulsifying drug delivery systems. (2013) (141)
- Nano-carrier systems: Strategies to overcome the mucus gel barrier. (2015) (138)
- Synthesis and in vitro evaluation of a novel thiolated chitosan. (2005) (137)
- Development of controlled drug release systems based on thiolated polymers. (2000) (136)
- In vivo evidence of oral vaccination with PLGA nanoparticles containing the immunostimulant monophosphoryl lipid A. (2011) (133)
- Thiomers: potential excipients for non-invasive peptide delivery systems. (2004) (126)
- Mucoadhesive systems in oral drug delivery. (2005) (123)
- Oral peptide drug delivery: polymer-inhibitor conjugates protecting insulin from enzymatic degradation in vitro. (2000) (122)
- Mucoadhesive and cohesive properties of poly(acrylic acid)-cysteine conjugates with regard to their molecular mass. (2003) (120)
- Development and in vivo evaluation of an oral insulin-PEG delivery system. (2004) (118)
- In vivo evaluation of an oral self-microemulsifying drug delivery system (SMEDDS) for leuprorelin. (2014) (114)
- Synthesis and in vitro evaluation of thiolated hyaluronic acid for mucoadhesive drug delivery. (2007) (114)
- In vivo evaluation of an oral delivery system for P-gp substrates based on thiolated chitosan. (2006) (114)
- Modified chitosans for oral drug delivery. (2009) (113)
- In vitro evaluation of the permeation-enhancing effect of thiolated polycarbophil. (2000) (112)
- Thiomers: preparation and in vitro evaluation of a mucoadhesive nanoparticulate drug delivery system. (2006) (110)
- Thiolated chitosan microparticles: a vehicle for nasal peptide drug delivery. (2006) (108)
- Liposomes coated with thiolated chitosan enhance oral peptide delivery to rats☆ (2013) (108)
- Strategies to prolong the intravaginal residence time of drug delivery systems. (2009) (107)
- Nanoparticle diffusion within intestinal mucus: Three-dimensional response analysis dissecting the impact of particle surface charge, size and heterogeneity across polyelectrolyte, pegylated and viral particles. (2015) (106)
- Design and In Vivo Evaluation of An Oral Delivery System for Insulin (2000) (105)
- Chitosan-thioglycolic acid conjugate: a new scaffold material for tissue engineering? (2003) (100)
- Thiomers--from bench to market. (2014) (100)
- Thiolated chitosan nanoparticles for the nasal administration of leuprolide: bioavailability and pharmacokinetic characterization. (2012) (98)
- Distribution of thiolated mucoadhesive nanoparticles on intestinal mucosa. (2011) (98)
- Mucus permeating carriers: formulation and characterization of highly densely charged nanoparticles. (2015) (97)
- Synthesis and in Vitro Evaluation of a Novel Chitosan–Glutathione Conjugate (2005) (97)
- Synthesis and characterization of a chitosan-N-acetyl cysteine conjugate. (2008) (96)
- Preparation and characterization of mucus-penetrating papain/poly(acrylic acid) nanoparticles for oral drug delivery applications (2012) (95)
- Nanoparticles decorated with proteolytic enzymes, a promising strategy to overcome the mucus barrier. (2015) (95)
- Hydrophobic ion pairing: Key to highly payloaded self-emulsifying peptide drug delivery systems. (2017) (93)
- Systemic peptide delivery via the stomach: in vivo evaluation of an oral dosage form for salmon calcitonin. (2003) (93)
- Development and in vitro evaluation of a mucoadhesive vaginal delivery system for progesterone. (2001) (92)
- In situ gelling properties of chitosan-thioglycolic acid conjugate in the presence of oxidizing agents. (2009) (92)
- Self-emulsifying peptide drug delivery systems: How to make them highly mucus permeating. (2018) (91)
- Thiolated Chitosans: Design and In Vivo Evaluation of a Mucoadhesive Buccal Peptide Drug Delivery System (2006) (91)
- Thiolated chitosans. (2004) (91)
- Methods to determine the interactions of micro- and nanoparticles with mucus. (2015) (91)
- In Vivo Evaluation of an Oral Salmon Calcitonin-Delivery System Based on a Thiolated Chitosan Carrier Matrix (2003) (90)
- Combining two technologies: multifunctional polymers and self-nanoemulsifying drug delivery system (SNEDDS) for oral insulin administration. (2013) (88)
- Multifunctional matrices for oral peptide delivery. (2001) (86)
- SEDDS: A game changing approach for the oral administration of hydrophilic macromolecular drugs. (2019) (86)
- Development and in Vivo Evaluation of an Oral Delivery System for Low Molecular Weight Heparin Based on Thiolated Polycarbophil (2003) (86)
- In vivo evaluation of an oral self‐emulsifying drug delivery system (SEDDS) for exenatide (2018) (85)
- Lipids and polymers in pharmaceutical technology: Lifelong companions (2019) (85)
- Development and in vivo evaluation of papain-functionalized nanoparticles. (2014) (85)
- Nanocarrier systems for oral drug delivery: do we really need them? (2013) (84)
- Nasal delivery of human growth hormone: in vitro and in vivo evaluation of a thiomer/glutathione microparticulate delivery system. (2004) (83)
- Chitosan-thioglycolic acid conjugate: an alternative carrier for oral nonviral gene delivery? (2007) (83)
- The potential of cystine-knot microproteins as novel pharmacophoric scaffolds in oral peptide drug delivery (2006) (81)
- S-protected thiolated chitosan for oral delivery of hydrophilic macromolecules: evaluation of permeation enhancing and efflux pump inhibitory properties. (2012) (81)
- Development of buccal drug delivery systems based on a thiolated polymer. (2003) (81)
- Development and in vitro evaluation of zeta potential changing self-emulsifying drug delivery systems for enhanced mucus permeation. (2016) (79)
- Strategies to overcome the polycation dilemma in drug delivery (2018) (79)
- Thiolation of polycarbophil enhances its inhibition of intestinal brush border membrane bound aminopeptidase N. (2001) (78)
- Do drug release studies from SEDDS make any sense? (2018) (78)
- Strategies for improving mucosal drug delivery. (2013) (78)
- Thiolated polymers: synthesis and in vitro evaluation of polymer-cysteamine conjugates. (2001) (78)
- Development and in vitro evaluation of a thiomer-based nanoparticulate gene delivery system. (2007) (77)
- Thiolated chitosans: useful excipients for oral drug delivery (2008) (76)
- Chemically modified chitosans as enzyme inhibitors. (2001) (76)
- Novel pectin-4-aminothiophenole conjugate microparticles for colon-specific drug delivery. (2010) (72)
- Development of a mucoadhesive nanoparticulate drug delivery system for a targeted drug release in the bladder. (2011) (72)
- Mucus permeating thiomer nanoparticles. (2015) (70)
- Development, in vitro and in vivo evaluation of a self-emulsifying drug delivery system (SEDDS) for oral enoxaparin administration. (2016) (70)
- Basic studies on bioadhesive delivery systems for peptide and protein drugs (1998) (70)
- In vivo comparison of various polymeric and low molecular mass inhibitors of intestinal P-glycoprotein. (2006) (70)
- Development and in vitro evaluation of slippery nanoparticles for enhanced diffusion through native mucus. (2014) (69)
- Improvement in the in situ gelling properties of deacetylated gellan gum by the immobilization of thiol groups. (2003) (68)
- Pre-systemic metabolism of orally administered drugs and strategies to overcome it. (2014) (68)
- Comparative in vivo mucoadhesion studies of thiomer formulations using magnetic resonance imaging and fluorescence detection. (2006) (68)
- Elaboration and characterization of thiolated chitosan-coated acrylic nanoparticles. (2006) (67)
- Thiolated polymers: Bioinspired polymers utilizing one of the most important bridging structures in nature. (2019) (66)
- Self-emulsifying drug delivery systems in oral (poly)peptide drug delivery (2015) (66)
- Chitosan‐EDTA Conjugate: A Novel Polymer for Topical Gels (1998) (65)
- Synthesis, characterization, mucoadhesion and biocompatibility of thiolated carboxymethyl dextran-cysteine conjugate. (2010) (64)
- Inhibition of malarial topoisomerase II in Plasmodium falciparum by antisense nanoparticles. (2006) (63)
- Novel insulin thiomer nanoparticles: in vivo evaluation of an oral drug delivery system. (2008) (63)
- Synthesis and in vitro characterization of entirely S-protected thiolated pectin for drug delivery. (2013) (63)
- S-protected thiolated chitosan: Synthesis and in vitro characterization (2012) (62)
- Polycarbophil-cysteine conjugates as platforms for oral polypeptide delivery systems. (2000) (62)
- Novel Bioadhesive Chitosan-EDTA Conjugate Protects Leucine Enkephalin from Degradation by Aminopeptidase N (1997) (61)
- Thiolated chitosan: development and in vitro evaluation of an oral delivery system for acyclovir. (2008) (61)
- Comparative evaluation of cytotoxicity of a glucosamine-TBA conjugate and a chitosan-TBA conjugate. (2004) (61)
- Development and in vitro characterisation of an oral self-emulsifying delivery system for daptomycin. (2016) (60)
- Development and In Vitro Evaluation of Surface Modified Poly(lactide-co-glycolide) Nanoparticles with Chitosan-4-Thiobutylamidine (2007) (60)
- Current challenges and future perspectives in oral absorption research: An opinion of the UNGAP network. (2021) (59)
- Development and in vitro evaluation of an oral SEDDS for desmopressin (2016) (59)
- Development and in vivo evaluation of an oral drug delivery system for paclitaxel. (2011) (59)
- Thiomers: forms, functions and applications to nanomedicine. (2007) (59)
- Investigations into the Diffusion Behaviour of Polypeptides in Native Intestinal Mucus with Regard to their Peroral Administration (1996) (58)
- Polyethylene imine-6-phosphogluconic acid nanoparticles--a novel zeta potential changing system. (2015) (58)
- Self-nanoemulsifying drug delivery systems as novel approach for pDNA drug delivery. (2015) (58)
- Improved synthesis and in vitro characterization of chitosan-thioethylamidine conjugate. (2006) (57)
- In situ gelling and mucoadhesive polymers: why do they need each other? (2018) (56)
- An adhesive drug delivery system based on K99-fimbriae (1995) (54)
- Thiolated carboxymethylcellulose: in vitro evaluation of its permeation enhancing effect on peptide drugs. (2001) (54)
- Thiolated chitosans: development and in vitro evaluation of an oral tobramycin sulphate delivery system. (2008) (54)
- Oral delivery of non‐viral nucleic acid‐based therapeutics ‐ do we have the guts for this? (2019) (54)
- In vivo evaluation of a nasal insulin delivery system based on thiolated chitosan. (2006) (54)
- Correlation of in vitro and in vivo models for the oral absorption of peptide drugs (2008) (53)
- Thiolated chitosan: development and in vivo evaluation of an oral delivery system for leuprolide. (2012) (52)
- Mucoadhesive polymers: strategies, achievements and future challenges. (2005) (52)
- In vitro evaluation of natural and methylated cyclodextrins as buccal permeation enhancing system for omeprazole delivery. (2009) (52)
- Thiomers: development and in vitro evaluation of a peroral microparticulate peptide delivery system. (2004) (52)
- Thiomers for oral delivery of hydrophilic macromolecular drugs (2004) (52)
- Comparison of the protective effect of self-emulsifying peptide drug delivery systems towards intestinal proteases and glutathione. (2017) (52)
- Evaluation and improvement of the properties of the novel cystine-knot microprotein McoEeTI for oral administration. (2007) (52)
- Deoxycholate-hydrogels: novel drug carrier systems for topical use. (1999) (52)
- Matrix tablets based on thiolated poly(acrylic acid): pH-dependent variation in disintegration and mucoadhesion. (2004) (52)
- Thiomer-coated liposomes harbor permeation enhancing and efflux pump inhibitory properties (2013) (51)
- Development and in vitro evaluation of a mucoadhesive vaginal delivery system for nystatin. (2009) (51)
- Thiolated chitosan micelles: Highly mucoadhesive drug carriers. (2017) (51)
- Synthesis and In Vitro Evaluation of Chitosan-Thioglycolic Acid Conjugates (2001) (51)
- The use of thiolated polymers as carrier matrix in oral peptide delivery--proof of concept. (2005) (51)
- Chitosan solutions and particles: evaluation of their permeation enhancing potential on MDCK cells used as blood brain barrier model. (2009) (50)
- Oral gene delivery: Strategies to improve stability of pDNA towards intestinal digestion (2006) (50)
- Evidence for the interpenetration of mucoadhesive polymers into the mucous gel layer (2003) (50)
- The Impact of Vehicles on the Mucoadhesive Properties of Orally Administrated Nanoparticles: a Case Study with Chitosan-4-Thiobutylamidine Conjugate (2010) (50)
- Impact of lipases on the protective effect of SEDDS for incorporated peptide drugs towards intestinal peptidases. (2016) (49)
- Insulin loaded mucus permeating nanoparticles: Addressing the surface characteristics as feature to improve mucus permeation. (2016) (49)
- Design and synthesis of a novel cationic thiolated polymer. (2011) (48)
- Thiolated polymeric hydrogels for biomedical application: Cross-linking mechanisms. (2020) (48)
- Impact of different hydrophobic ion pairs of octreotide on its oral bioavailability in pigs (2018) (48)
- In vitro evaluation of polymeric excipients protecting calcitonin against degradation by intestinal serine proteases. (2003) (48)
- Chemical coupling of thiolated chitosan to preformed liposomes improves mucoadhesive properties (2012) (48)
- Thiomers: promising platform for macromolecular drug delivery. (2012) (48)
- In vitro evaluation of chitosan-EDTA conjugate polyplexes as a nanoparticulate gene delivery system (2006) (48)
- Thiomers in noninvasive polypeptide delivery: in vitro and in vivo characterization of a polycarbophil-cysteine/glutathione gel formulation for human growth hormone. (2004) (47)
- Preactivated hyaluronic acid: A potential mucoadhesive polymer for vaginal delivery. (2015) (47)
- Advanced formulations for intranasal delivery of biologics (2018) (47)
- Development of a nasal spray containing xylometazoline hydrochloride and iota-carrageenan for the symptomatic relief of nasal congestion caused by rhinitis and sinusitis (2018) (47)
- Development and in vitro characterization of a papain loaded mucolytic self-emulsifying drug delivery system (SEDDS). (2017) (47)
- Strategies to prolong the residence time of drug delivery systems on ocular surface. (2020) (45)
- Thiolated Chitosans: A Multi-talented Class of Polymers for Various Applications (2020) (45)
- In vitro evaluation of the permeation enhancing effect of polycarbophil-cysteine conjugates on the cornea of rabbits. (2002) (44)
- Role of sulfhydryl groups in transfection? A case study with chitosan-NAC nanoparticles. (2007) (44)
- In vivo evaluation of an oral drug delivery system for peptides based on S-protected thiolated chitosan. (2012) (44)
- Preparation of Thiomer Microparticles and In Vitro Evaluation of Parameters Influencing Their Mucoadhesive Properties (2006) (43)
- Self‐emulsifying drug delivery systems: Impact of stability of hydrophobic ion pairs on drug release (2019) (43)
- Design and in vitro evaluation of a novel polymeric P-glycoprotein (P-gp) inhibitor. (2010) (43)
- Thiolated Hyaluronic Acid as Versatile Mucoadhesive Polymer: From the Chemistry Behind to Product Developments—What Are the Capabilities? (2018) (42)
- Thiolated hydroxyethyl cellulose: design and in vitro evaluation of mucoadhesive and permeation enhancing nanoparticles. (2013) (42)
- Peptidase activity on the surface of the porcine buccal mucosa. (2002) (42)
- Cell-penetrating self-nanoemulsifying drug delivery systems (SNEDDS) for oral gene delivery (2016) (42)
- Presystemic metabolism of orally administered peptide drugs and strategies to overcome it. (2007) (42)
- Development of phosphorylated nanoparticles as zeta potential inverting systems. (2015) (41)
- Design and evaluation of an intravesical delivery system for superficial bladder cancer: preparation of gemcitabine HCl-loaded chitosan–thioglycolic acid nanoparticles and comparison of chitosan/poloxamer gels as carriers (2015) (41)
- Intravaginal drug delivery systems (2003) (41)
- Direct compressible polymethacrylic acid-starch compositions for site-specific drug delivery. (2001) (41)
- Mucus permeating thiolated self-emulsifying drug delivery systems. (2016) (41)
- Enzyme decorated drug carriers: Targeted swords to cleave and overcome the mucus barrier☆ (2017) (41)
- Lipophilic peptide character - What oral barriers fear the most. (2017) (40)
- Synthesis and In Vitro Evaluation of Chitosan-EDTA-Protease-Inhibitor Conjugates Which Might Be Useful in Oral Delivery of Peptides and Proteins (1998) (40)
- Thiolated particles as effective intravesical drug delivery systems for treatment of bladder-related diseases. (2013) (40)
- Mucoadhesive drug delivery systems. (2010) (39)
- Viscoelastic Properties of a New in situ Gelling Thiolated Chitosan Conjugate (2005) (39)
- In vivo evaluation of thiolated chitosan tablets for oral insulin delivery. (2014) (39)
- In vitro cytotoxicity testing of non-thiolated and thiolated chitosan nanoparticles for oral gene delivery (2007) (39)
- Preactivated thiomers: Permeation enhancing properties (2012) (39)
- Preparation and in vitro characterization of poly(acrylic acid)-cysteine microparticles. (2003) (39)
- Enzymatic degradation of thiolated chitosan (2013) (39)
- Synergistic effects of conjugating cell penetrating peptides and thiomers on non-viral transfection efficiency. (2012) (38)
- Zeta potential changing self‐emulsifying drug delivery systems containing phosphorylated polysaccharides (2017) (38)
- Design and in vivo evaluation of a patch delivery system for insulin based on thiolated polymers. (2008) (38)
- Preparation and in vitro evaluation of thiolated chitosan microparticles (2005) (38)
- Chitosan-graft-6-mercaptonicotinic acid: synthesis, characterization, and biocompatibility. (2009) (38)
- Synthesis and characterization of thiolated β-cyclodextrin as a novel mucoadhesive excipient for intra-oral drug delivery. (2015) (38)
- Pectin‐cysteine conjugate: synthesis and in‐vitro evaluation of its potential for drug delivery (2006) (38)
- In vivo determination of the time and location of mucoadhesive drug delivery systems disintegration in the gastrointestinal tract. (2008) (37)
- Preactivated thiomers: their role in drug delivery (2015) (37)
- Thiolated hydroxyethylcellulose: synthesis and in vitro evaluation. (2010) (37)
- Hydrophobic ion-pairs and lipid-based nanocarrier systems: The perfect match for delivery of BCS class 3 drugs. (2019) (37)
- Preactivated thiomers: evaluation of gastroretentive minitablets. (2013) (36)
- Preactivated thiolated glycogen as mucoadhesive polymer for drug delivery (2017) (36)
- In Vitro Evaluation of Various Buccal Permeation Enhancing Systems for PACAP (Pituitary Adenylate Cyclase-Activating Polypeptide) (2005) (36)
- Self‐emulsifying drug delivery systems and cationic surfactants: do they potentiate each other in cytotoxicity? (2018) (36)
- Thiolated chitosans: influence of various sulfhydryl ligands on permeation-enhancing and P-gp inhibitory properties (2011) (35)
- Development and in vitro evaluation of a drug delivery system protecting from trypsinic degradation (1997) (35)
- The Antistaphylococcal Effect of Nisin in a Suitable Vehicle: A Potential Therapy for Atopic Dermatitis in Man (1996) (35)
- S-protected gellan gum: Decisive approach towards mucoadhesive antimicrobial vaginal films. (2019) (35)
- The use of chitosan-6-mercaptonicotinic acid nanoparticles for oral peptide drug delivery (2011) (35)
- Oral heparin delivery: design and in vivo evaluation of a stomach-targeted mucoadhesive delivery system. (2005) (35)
- Anionic Mucoadhesive Polymers as Auxiliary Agents for the Peroral Administration of (Poly)Peptide Drugs: Influence of the Gastric Juice (2000) (35)
- Preparation and evaluation of microparticles from thiolated polymers via air jet milling. (2008) (34)
- Uptake of phenothiazines by the harvested chylomicrons ex vivo model: influence of self-nanoemulsifying formulation design. (2011) (34)
- Self‐emulsifying drug delivery systems: Design of a novel vaginal delivery system for curcumin (2017) (34)
- S-protected thiolated cyclodextrins as mucoadhesive oligomers for drug delivery. (2018) (34)
- Improved paracellular uptake by the combination of different types of permeation enhancers. (2005) (34)
- Mucoadhesive hydrogels for buccal drug delivery: In vitro- in vivo correlation study. (2019) (34)
- Development of a novel method for the preparation of submicron particles based on thiolated chitosan. (2006) (34)
- Chitosan-4-mercaptobenzoic acid: synthesis and characterization of a novel thiolated chitosan (2010) (33)
- Chitosan–gum arabic polyelectrolyte complex films: physicochemical, mechanical and mucoadhesive properties (2016) (33)
- Preactivated thiomers for vaginal drug delivery vehicles. (2013) (33)
- Thiolated and S-protected hydrophobically modified cross-linked poly(acrylic acid)--a new generation of multifunctional polymers. (2014) (32)
- Evaluation of functional characteristics of preactivated thiolated chitosan as potential therapeutic agent for dry mouth syndrome. (2015) (32)
- Cationic starch derivatives as mucoadhesive and soluble excipients in drug delivery. (2019) (32)
- Nasal drug delivery: Design of a novel mucoadhesive and in situ gelling polymer. (2017) (32)
- Novel bioadhesive drug delivery system protecting (poly)peptides from gastric enzymatic degradation (1996) (31)
- Mucoadhesive self-emulsifying delivery systems for ocular administration of econazole. (2018) (31)
- Thiolated polymers: evaluation of the influence of the amount of covalently attached L-cysteine to poly(acrylic acid). (2007) (31)
- Zeta Potential Changing Polyphosphate Nanoparticles: A Promising Approach To Overcome the Mucus and Epithelial Barrier. (2019) (31)
- In vitro and ex vivo evaluation of an intestinal permeation enhancing self-microemulsifying drug delivery system (SMEDDS) (2013) (31)
- Arginine-based cationic surfactants: Biodegradable auxiliary agents for the formation of hydrophobic ion pairs with hydrophilic macromolecular drugs. (2019) (30)
- Preactivated thiolated nanoparticles: A novel mucoadhesive dosage form. (2016) (30)
- Synthesis and characterization of pH tolerant and mucoadhesive (thiol-polyethylene glycol) chitosan graft polymer for drug delivery. (2014) (30)
- Mucoadhesive micro-composites: Chitosan coated halloysite nanotubes for sustained drug delivery. (2019) (30)
- Polymer-cysteamine conjugates: new mucoadhesive excipients for drug delivery? (2002) (30)
- Mucoadhesive polymers in the treatment of dry X syndrome. (2016) (30)
- Non-Clinical Safety Evaluation of Intranasal Iota-Carrageenan (2015) (29)
- Influence of the molecular mass on the permeation enhancing effect of different poly(acrylates) (2002) (29)
- Poly(acrylic acid)-cysteine for oral vitamin B12 delivery. (2012) (29)
- Synthesis and In Vitro Characterization of a Poly(Acrylic Acid)‐Homocysteine Conjugate (2004) (29)
- Chitosan and Thiolated Chitosan (2011) (29)
- Development of a Novel Method for the Preparation of Thiolated Polyacrylic Acid Nanoparticles (2006) (29)
- Thiolated silicone oil: Synthesis, gelling and mucoadhesive properties (2015) (29)
- Chitosan based micelle with zeta potential changing property for effective mucosal drug delivery. (2019) (29)
- Papain: An Effective Permeation Enhancer for Orally Administered Low Molecular Weight Heparin (2007) (29)
- Zeta potential changing self-emulsifying drug delivery systems utilizing a novel Janus-headed surfactant: A promising strategy for enhanced mucus permeation (2019) (29)
- Evaluation of the potential of air jet milling of solid protein-poly(acrylate) complexes for microparticle preparation. (2006) (28)
- In vivo evaluation of thiolated poly(acrylic acid) as a drug absorption modulator for MRP2 efflux pump substrates. (2009) (28)
- Thiolated nanocarriers for oral delivery of hydrophilic macromolecular drugs. (2015) (28)
- Trypsin decorated self-emulsifying drug delivery systems (SEDDS): Key to enhanced mucus permeation. (2018) (28)
- Entirely S-protected chitosan: A promising mucoadhesive excipient for metronidazole vaginal tablets. (2017) (28)
- Insulin-loaded poly(acrylic acid)-cysteine nanoparticles: Stability studies towards digestive enzymes of the intestine (2009) (28)
- Zeta potential changing self-emulsifying drug delivery systems: A promising strategy to sequentially overcome mucus and epithelial barrier. (2019) (27)
- Improvement of the intestinal membrane permeability of low molecular weight heparin by complexation with stem bromelain. (2006) (27)
- Development of a Sustained Release Dosage Form for α‐Lipoic Acid. II. Evaluation in Human Volunteers (2004) (27)
- Highly mucus permeating and zeta potential changing self‐emulsifying drug delivery systems: A potent gene delivery model for causal treatment of cystic fibrosis (2019) (27)
- Improved mucoadhesive properties of self-nanoemulsifying drug delivery systems (SNEDDS) by introducing acyl chitosan. (2017) (27)
- Analysis of some Malaysian dart poisons. (1992) (27)
- Chitosan-N-Acetyl Cysteine Conjugates: In Vitro Evaluation of Permeation Enhancing and P-Glycoprotein Inhibiting Properties (2008) (27)
- Novel bioadhesive polymers as intra-articular agents: Chondroitin sulfate-cysteine conjugates. (2016) (27)
- Mucus permeating self-emulsifying drug delivery systems (SEDDS): About the impact of mucolytic enzymes. (2018) (27)
- S-protected thiolated hyaluronic acid: In-situ crosslinking hydrogels for 3D cell culture scaffold. (2020) (27)
- S‐preactivated thiolated glycol chitosan useful to combine mucoadhesion and drug delivery (2018) (27)
- Enhanced transport of P-glycoprotein substrate saquinavir in presence of thiolated chitosan (2007) (26)
- Phosphorothioate Oligonucleotide Quantification by μ-Liquid Chromatography-Mass Spectrometry (2012) (26)
- Development and in vitro evaluation of a self‐emulsifying drug delivery system (SEDDS) for oral vancomycin administration (2019) (26)
- Thiolated α-Cyclodextrin: The Invisible Choice to Prolong Ocular Drug Residence Time. (2016) (26)
- Polymeric efflux pump inhibitors in oral drug delivery (2006) (26)
- Development and in vivo bioavailability study of an oral fondaparinux delivery system. (2010) (26)
- Intestinal peptide and protein delivery: novel bioadhesive drug-carrier matrix shielding from enzymatic attack. (1998) (25)
- Development of oral self nano-emulsifying delivery system(s) of lanreotide with improved stability against presystemic thiol-disulfide exchange reactions (2016) (25)
- Synthesis and evaluation of lysozyme derivatives exhibiting an enhanced antimicrobial action. (1998) (25)
- Zeta potential changing nanoemulsions based on a simple zwitterion. (2020) (25)
- Preparation and characterisation of thiolated poly(methacrylic acid)-starch compositions. (2004) (25)
- Multifunctional adhesive polymers: Preactivated thiolated chitosan‐EDTA conjugates (2017) (25)
- Thiolated graphene oxide as promising mucoadhesive carrier for hydrophobic drugs. (2016) (25)
- Design and in vitro evaluation of a novel polymeric excipient for buccal applications. (2013) (25)
- Development of a mucoadhesive and permeation enhancing buccal delivery system for PACAP (pituitary adenylate cyclase-activating polypeptide). (2005) (25)
- Thiomer nanoparticles: Stabilization via covalent cross-linking (2011) (24)
- Improvement of the enzymatic stability of a cytotoxic T-lymphocyte-epitope model peptide for its oral administration (2002) (24)
- Preactivated thiolated poly(methacrylic acid-co-ethyl acrylate): synthesis and evaluation of mucoadhesive potential. (2014) (24)
- Efficient MRI labeling of endothelial progenitor cells: design of thiolated surface stabilized superparamagnetic iron oxide nanoparticles. (2013) (24)
- Totally S-protected hyaluronic acid: Evaluation of stability and mucoadhesive properties as liquid dosage form. (2016) (24)
- Oral self-emulsifying delivery systems for systemic administration of therapeutic proteins: science fiction? (2019) (24)
- Hydrophobic Thiolation of Pectin with 4-Aminothiophenol: Synthesis and In Vitro Characterization (2010) (24)
- Development and in vitro evaluation of a buccal drug delivery system based on preactivated thiolated pectin (2014) (24)
- Modified mucoadhesive polymers for the peroral administration of mainly elastase degradable therapeutic (poly)peptides (1997) (24)
- Comparative in vitro study of different chitosan-complexing agent conjugates. (1999) (23)
- Degradation of teriparatide by gastro-intestinal proteolytic enzymes (2006) (23)
- Thiolated polycarbophil as an adjuvant for permeation enhancement in nasal delivery of antisense oligonucleotides. (2010) (23)
- Development and in vivo evaluation of a new oral nanoparticulate dosage form for leuprolide based on polyacrylic acid (2011) (23)
- Self‐emulsifying drug delivery systems (SEDDS): Proof‐of‐concept how to make them mucoadhesive (2017) (23)
- Oral self-nanoemulsifying peptide drug delivery systems: impact of lipase on drug release (2015) (23)
- Thinking continuously: a microreactor for the production and scale-up of biodegradable, self-assembled nanoparticles (2013) (23)
- Thiomers: Inhibition of cytochrome P450 activity. (2011) (23)
- Zeta potential changing phosphorylated nanocomplexes for pDNA delivery. (2016) (23)
- Synthesis and evaluation of a modified mucoadhesive polymer protecting from α-chymotrypsinic degradation (1997) (22)
- Thiolated chitosans: Are Cys-Cys ligands key to the next generation? (2020) (22)
- Biomembrane permeability of peptides: strategies to improve their mucosal uptake. (2002) (22)
- Characterisation of the thiol–disulphide chemistry of desmopressin by LC, μ-LC, LC-ESI-MS and Maldi-Tof (2006) (22)
- Development of self‐emulsifying drug delivery systems (SEDDS) for ciprofloxacin with improved mucus permeating properties (2018) (22)
- Development of a Sustained Release Dosage Form for α‐Lipoic Acid. I. Design and In Vitro Evaluation (2004) (22)
- Development and in vivo characterization of a novel peptide drug delivery system providing extended plasma half life. (2012) (22)
- Thiolated hydroxypropyl-β-cyclodextrin as mucoadhesive excipient for oral delivery of budesonide in liquid paediatric formulation. (2019) (22)
- Synthesis and in vitro characterization of a novel S-protected thiolated alginate. (2015) (21)
- Development and analysis of a polymer protecting from luminal enzymatic degradation caused by α-chymotrypsin (1997) (21)
- Absorption and Metabolism of Resveratrol Carboxyesters and Methanesulfonate by Explanted Rat Intestinal Segments (2009) (21)
- Controlled Drug Delivery Systems Based on Thiolated Chitosan Microspheres (2005) (21)
- Hydrophobic ion pairing of a GLP-1 analogue for incorporating into lipid nanocarriers designed for oral delivery. (2020) (21)
- Polymer/inhibitor conjugates a promising strategy to overcome the enzymatic barrier to perorally administered (poly)peptide drugs? (1999) (21)
- An in-vitro exploration of permeation enhancement by novel polysulfonate thiomers. (2015) (21)
- Thiolated Polymers: Stability of Thiol Moieties under Different Storage Conditions (2002) (21)
- Lysozyme-caffeic acid conjugates: possible novel preservatives for dermal formulations (1998) (21)
- Thiopyrazole preactivated chitosan: combining mucoadhesion and drug delivery. (2013) (21)
- Development and in vitro characterization of self-emulsifying drug delivery system (SEDDS) for oral opioid peptide delivery (2017) (21)
- Nanoparticular delivery system for a secretoneurin derivative induces angiogenesis in a hind limb ischemia model (2017) (20)
- Surface phosphorylation of nanoparticles by hexokinase: A powerful tool for cellular uptake improvement. (2018) (20)
- Evaluation of the inhibition effect of thiolated poly(acrylates) on vaginal membrane bound aminopeptidase N and release of the model drug LH‐RH (2002) (20)
- Thiomers and thiomer-based nanoparticles in protein and DNA drug delivery (2012) (20)
- Characterisation of the barrier caused by luminally secreted gastro-intestinal proteolytic enzymes for two novel cystine-knot microproteins (2008) (20)
- Thiolated cyclodextrins: Mucoadhesive and permeation enhancing excipients for ocular drug delivery. (2021) (20)
- About the impact of water movement on the permeation behaviour of nanoparticles in mucus. (2017) (19)
- Phosphorylated PEG-emulsifier: Powerful tool for development of zeta potential changing self-emulsifying drug delivery systems (SEDDS). (2020) (19)
- Oral peptide delivery: in‐vitro evaluation of thiolated alginate/poly(acrylic acid) microparticles (2007) (19)
- Self‐emulsifying drug delivery systems changing their zeta potential via a flip‐flop mechanism (2018) (19)
- Zeta-potential-changing nanoparticles conjugated with cell-penetrating peptides for enhanced transfection efficiency. (2017) (19)
- Development and in vivo evaluation of an oral vitamin B12 delivery system. (2013) (18)
- In vitro characterization of insulin containing thiomeric microparticles as nasal drug delivery system. (2016) (18)
- In situ gelling properties of anionic thiomers (2012) (18)
- Oral Delivery of Macromolecular Drugs (2009) (18)
- Safety assessment of thiolated polymers: effect on ciliary beat frequency in human nasal epithelial cells (2011) (18)
- Zeta potential changing nanoemulsions: Impact of PEG-corona on phosphate cleavage. (2020) (18)
- Transport Characteristics of a Beta Sheet Breaker Peptide Across Excised Bovine Nasal Mucosa (2007) (18)
- Nanocarriers protecting toward an intestinal pre-uptake metabolism. (2017) (18)
- Zeta potential changing nanoemulsions based on phosphate moiety cleavage of a PEGylated surfactant (2020) (18)
- Bioadhesive properties of poly(anhydride) nanoparticles coated with different molecular weights chitosan (2011) (18)
- Natural dendrimers: Synthesis and in vitro characterization of glycogen‐cysteamine conjugates (2017) (17)
- Solubilizing agents in nasal formulations and their effect on ciliary beat frequency. (2012) (17)
- ζ potential changing nanoparticles as cystic fibrosis transmembrane conductance regulator gene delivery system: an in vitro evaluation. (2017) (17)
- Development of pre-activated α-cyclodextrin as a mucoadhesive excipient for intra-vesical drug delivery. (2017) (17)
- Evaluation of In Vitro Enzymatic Degradation of Various Thiomers and Cross-Linked Thiomers (2007) (17)
- Thiolated Cyclodextrin: Development of a Mucoadhesive Vaginal Delivery System for Acyclovir. (2016) (17)
- Intestinal enzyme delivery: Chitosan/tripolyphosphate nanoparticles providing a targeted release behind the mucus gel barrier. (2019) (17)
- 2,2'Dithiodinicotinyl ligands: Key to more reactive thiomers. (2016) (17)
- Thiolated polyacrylic acid-modified iron oxide nanoparticles for in vitro labeling and MRI of stem cells (2011) (17)
- Chitosan: The One and Only? Aminated Cellulose as an Innovative Option for Primary Amino Groups Containing Polymers. (2018) (17)
- Tetradeca-thiolated cyclodextrins: Highly mucoadhesive and in-situ gelling oligomers with prolonged mucosal adhesion. (2020) (17)
- Non-ionic thiolated cyclodextrins – the next generation (2018) (17)
- Bioinert, Stealth or Interactive: How Surface Chemistry of Nanocarriers Determines Their Fate In Vivo (2021) (17)
- Enhancing the efficiency of thiomers: Utilizing a highly mucoadhesive polymer as backbone for thiolation and preactivation (2017) (17)
- In vivo evaluation of anionic thiolated polymers as oral delivery systems for efflux pump inhibition. (2015) (17)
- Synthesis and In Vitro Evaluation of Thiolated Carrageenan. (2015) (17)
- Reactive keratin derivatives: A promising strategy for covalent binding to hair. (2019) (17)
- Development and in Vitro Evaluation of Systems to Protect Peptide Drugs from Aminopeptidase N (1997) (16)
- Thiolated Polymers: Development and Evaluation of Transdermal Delivery Systems for Progesterone (2001) (16)
- Cellular uptake of self-emulsifying drug-delivery systems: polyethylene glycol versus polyglycerol surface. (2020) (16)
- Reprint of: Nanocarrier systems for oral drug delivery: do we really need them? (2013) (16)
- Thiomers: Influence of molecular mass and thiol group content of poly(acrylic acid) on efflux pump inhibition. (2015) (16)
- Novel in vitro transport method for screening the reversibility of P-glycoprotein inhibitors. (2016) (16)
- Role of sonication pre-treatment and cation valence in the sol-gel transition of nano-cellulose suspensions (2017) (16)
- Protease-functionalized mucus penetrating microparticles: In-vivo evidence for their potential. (2017) (16)
- Comprehensive mucoadhesive study of anionic polymers and their derivate (2017) (16)
- Mucoadhesive polymers: Synthesis and in vitro characterization of thiolated poly(vinyl alcohol). (2016) (16)
- Hydrophobic ion pairing (HIP) of (poly)peptide drugs: Benefits and drawbacks of different preparation methods. (2020) (15)
- Noninvasive delivery systems for peptides and proteins in osteoporosis therapy: a retroperspective (2009) (15)
- Cosolvents in Self-Emulsifying Drug Delivery Systems (SEDDS): Do They Really Solve Our Solubility Problems? (2020) (15)
- Development and in vitro evaluation of a drug delivery system based on chitosan-EDTA BBI conjugate. (1998) (15)
- Per-6-Thiolated Cyclodextrins: A Novel Type of Permeation Enhancing Excipients for BCS Class IV Drugs (2020) (15)
- Evaluation of the impact of multivalent metal ions on the permeation behavior of Dolutegravir sodium (2016) (15)
- Thiomers: influence of molar mass on in situ gelling properties. (2012) (15)
- Synthesis and Characterization of Thiolated PVP-Iodine Complexes: Key to Highly Mucoadhesive Antimicrobial Gels. (2018) (15)
- Synthesis and in vitro characterization of a novel poly(acrylic acid)-glutathione conjugate (2005) (15)
- Auxiliary agents for the peroral administration of peptide and protein drugs: synthesis and evaluation of novel pepstatin analogues. (1998) (15)
- In vitro evaluation of the potential of thiomers for the nasal administration of Leu-enkephalin (2006) (15)
- In vitro evaluation of matrix tablets based on thiolated polycarbophil (2001) (15)
- Synthesis and in vitro characterization of a preactivated thiomer via polymerization reaction. (2012) (15)
- Thiolated silicone oils as adhesive skin protectants for improved barrier function (2016) (14)
- New perspectives of starch: Synthesis and in vitro assessment of novel thiolated mucoadhesive derivatives (2018) (14)
- Thiolated gelatin films: Renaissance of gelatin as sustained intraoral dosage form (2017) (14)
- In Vitro-in Vivo Correlation of Mucoadhesion Studies on Buccal Mucosa. (2019) (14)
- Design and evaluation of SEDDS exhibiting high emulsifying properties (2018) (14)
- Modification of lysozyme with cinnamaldehyde: A strategy for constructing novel preservatives for dermatics (1997) (14)
- Development and in vitro characterization of an oral self-emulsifying delivery system (SEDDS) for rutin fatty ester with high mucus permeating properties. (2019) (14)
- New-generation efflux pump inhibitors (2008) (14)
- Combination of SEDDS and Preactivated Thiomer Technology: Incorporation of a Preactivated Thiolated Amphiphilic Polymer into Self-Emulsifying Delivery Systems (2017) (14)
- Chitosan-N-acetyl cysteine conjugates: in vitro evaluation of permeation enhancing and P-glycoprotein inhibiting properties. (2008) (14)
- Oral peptide delivery: Are there remarkable effects on drugs through sulfhydryl conjugation? (2006) (13)
- Self-Emulsifying Drug Delivery Systems: Hydrophobic Drug Polymer Complexes Provide a Sustained Release in Vitro (2020) (13)
- The efflux pump inhibitory properties of (thiolated) polyallylamines (2009) (13)
- Alkaline Phosphatase: A Reliable Endogenous Partner for Drug Delivery and Diagnostics (2022) (13)
- Diaminated Starch: A Competitor of Chitosan with Highly Mucoadhesive Properties due to Increased Local Cationic Charge Density (2020) (13)
- Enzyme-Functionalized PLGA Nanoparticles with Enhanced Mucus Permeation Rate (2014) (13)
- Thiolated cyclodextrins: New perspectives for old excipients (2020) (13)
- SIZE SHIFTING OF SOLID LIPID NANOPARTICLE SYSTEM TRIGGERED BY ALKALINE PHOSPHATASE FOR SITE SPECIFIC MUCOSAL DRUG DELIVERY. (2021) (13)
- The Effect of Counterions in Hydrophobic Ion Pairs on Oral Bioavailability of Exenatide. (2020) (13)
- Bioadhesion to the intestine by means of E. coli K99-fimbriae: (1997) (13)
- Immobilization of 2-mercaptoethylamine on oxidized chitosan: a substantially mucoadhesive and permeation enhancing polymer (2012) (12)
- Can thiolation render a low molecular weight polymer of just 20-kDa mucoadhesive? (2016) (12)
- A gellan gum derivative as in-situ gelling cationic polymer for nasal drug delivery. (2020) (12)
- Effect of a thiolated polymer on oral paclitaxel absorption and tumor growth in rats (2008) (12)
- Self-emulsifying drug delivery systems (SEDDS) - The splendid comeback of an old technology. (2019) (12)
- Chitosan and Derivatives for Biopharmaceutical Use: Mucoadhesive Properties (2012) (12)
- Hydrophobic H-bond pairing: A novel approach to improve membrane permeability. (2019) (12)
- Thiomers: Impact of in situ cross‐linkers on mucoadhesive properties (2017) (12)
- Thiolated alkyl-modified carbomers: Novel excipients for mucoadhesive emulsions. (2015) (12)
- Synthesis, development and in vitro evaluation of drug delivery systems with protective effect against degradation by pepsin. (1999) (12)
- About the impact of superassociation of hydrophobic ion pairs on membrane permeability. (2020) (12)
- Development of thiolated poly(acrylic acid) microparticles for the nasal administration of exenatide (2014) (12)
- Thiolated polycarbophil/glutathione: Defining its potential as a permeation enhancer for oral drug administration in comparison to sodium caprate (2011) (11)
- Thiolated Hydroxypropyl-β-cyclodextrin: A Potential Multifunctional Excipient for Ocular Drug Delivery (2022) (11)
- Amikacin-containing self-emulsifying delivery systems via pulmonary administration for treatment of bacterial infections of cystic fibrosis patients. (2018) (11)
- Storage Stability of Bivalirudin: Hydrophilic Versus Lipophilic Solutions. (2017) (11)
- In Vitro Investigation of Thiolated Chitosan Derivatives as Mucoadhesive Coating Materials for Solid Lipid Nanoparticles (2021) (11)
- Peroral Polypeptide Delivery (1999) (11)
- Spray-Dried Mucoadhesive Microparticles Based On S-Protected Thiolated Hydroxypropyl- β -Cyclodextrin For Budesonide Nasal Delivery. (2021) (11)
- Design and in vivo evaluation of a patch system based on thiolated polymers. (2009) (11)
- The use of multifunctional polymers for non-invasive peptide and protein application (2000) (11)
- Mucoadhesive S-protected thiolated cyclodextrin-iodine complexes: a promising strategy to prolong mucosal residence time of iodine. (2019) (11)
- Self-emulsifying drug delivery systems: In vivo evaluation of their potential for oral vaccination. (2019) (11)
- S-protected thiolated hydroxyethyl cellulose (HEC): Novel mucoadhesive excipient with improved stability. (2016) (10)
- Nasal delivery of antisense oligonucleotides: in vitro evaluation of a thiomer/glutathione microparticulate delivery system (2010) (10)
- Thiolated polymers: evaluation of their potential as dermoadhesive excipients (2017) (10)
- Polyphosphate coatings: A promising strategy to overcome the polycation dilemma. (2020) (10)
- Thiolated pectins: In vitro and ex vivo evaluation of three generations of thiomers. (2021) (10)
- The inhibitory effect of glutathione on buccal enzymatic degradation of therapeutic peptides (leu-enkephalin, luteinizing hormone-releasing hormone and pituitary adenylate cyclase activating peptide) (2005) (10)
- Preactivated thiolated pullulan as a versatile excipient for mucosal drug targeting. (2016) (10)
- Charge reversal self-emulsifying drug delivery systems: A comparative study among various phosphorylated surfactants. (2021) (10)
- Imine bond formation: A novel concept to incorporate peptide drugs in self-emulsifying drug delivery systems (SEDDS). (2019) (10)
- Covalently binding mucoadhesive polymers: N‐hydroxysuccinimide grafted polyacrylates (2019) (10)
- Synthesis and in vitro characterisation of preactivated thiolated gelatin (2015) (10)
- In vitro evaluation of intravesical mucoadhesive self-emulsifying drug delivery systems. (2019) (10)
- Characterization of an amino acid based biodegradable surfactant facilitating the incorporation of DNA into lipophilic delivery systems. (2020) (10)
- Improved Intestinal Mucus Permeation of Vancomycin via Incorporation Into Nanocarrier Containing Papain-Palmitate. (2019) (10)
- Glyceryl ester surfactants: Promising excipients to enhance the cell permeating properties of SEDDS (2018) (10)
- Lysine-based biodegradable surfactants: Increasing the lipophilicity of insulin by hydrophobic ion paring. (2020) (10)
- Preparation and evaluation of thiomer nanoparticles via high pressure homogenization (2010) (10)
- Solidification of self-emulsifying drug delivery systems (SEDDS): Impact on storage stability of a therapeutic protein. (2020) (10)
- In vitro evaluation of a self-emulsifying drug delivery system (SEDDS) for nasal administration of dimenhydrinate (2019) (10)
- Peroral Administration of Enzymes: Strategies to Improve the Galenic of Dosage Forms for Trypsin and Bromelain (2000) (9)
- Development and In Vitro Evaluation of Stearic Acid Phosphotyrosine Amide as New Excipient for Zeta Potential Changing Self-Emulsifying Drug Delivery Systems (2020) (9)
- Charge changing phosphorylated polymers: Proof of in situ mucoadhesive properties. (2016) (9)
- Nanostructured Lipid Carriers (NLCs) for Oral Peptide Drug Delivery: About the Impact of Surface Decoration (2021) (9)
- P-glycoprotein inhibitors: synthesis and in vitro evaluation of a preactivated thiomer (2016) (9)
- Influence of the spacer on the inhibitory effect of different polycarbophil-protease inhibitor conjugates. (2001) (9)
- Vitamin B₁₂ and derivatives--In vitro permeation studies across Caco-2 cell monolayers and freshly excised rat intestinal mucosa. (2016) (9)
- Evaluation of thiolated silicone oil as advanced mucoadhesive antifoaming agent (2016) (9)
- Composite nanocellulose-based hydrogels with spatially oriented degradation and retarded release of macromolecules. (2020) (9)
- Design and Evaluation of a New Gastrointestinal Mucoadhesive Patch System Containing Chitosan-Glutathione (2007) (9)
- A comprehensive in vitro and in vivo evaluation of thiolated matrix tablets as a gastroretentive delivery system (2011) (8)
- Self-emulsifying drug delivery systems containing hydrophobic ion pairs of polymyxin B and agaric acid: A decisive strategy for enhanced antimicrobial activity (2020) (8)
- Self-emulsifying drug delivery systems comprising chlorhexidine and alkyl-EDTA: A novel approach for augmented antimicrobial activity (2019) (8)
- Mucoadhesive properties of polyacrylates: Structure – Function relationship (2021) (8)
- Preactivated thiomers for intranasal delivery of apomorphine: In vitro and in vivo evaluation. (2016) (8)
- Entirely S-protected silicone oil as second generation mucoadhesive agent (2016) (8)
- Effect of a thiolated polymer on oral paclitaxel absorption and tumor growth in rats. (2008) (8)
- Near infrared spectroscopy compared to liquid chromatography coupled to mass spectrometry and capillary electrophoresis as a detection tool for peptide reaction monitoring (2008) (8)
- Simplified pepstatins: synthesis and evaluation of N-terminally modified analogues. (1999) (7)
- Targeted Self-Emulsifying Drug Delivery Systems to Restore Docetaxel Sensitivity in Resistant Tumors (2022) (7)
- 6-mercaptonicotinamide-functionalized chitosan: a potential excipient for mucoadhesive drug delivery systems (2010) (7)
- Less Reactive Thiol Ligands: Key towards Highly Mucoadhesive Drug Delivery Systems (2020) (7)
- Permeation studies on freshly excised rat gastric mucosa: influence of pH (2011) (7)
- Emerging technologies to increase gastrointestinal transit times of drug delivery systems. (2022) (7)
- N-Hydroxysulfosuccinimide Esters versus Thiomers: A Comparative Study Regarding Mucoadhesiveness. (2019) (7)
- P-glycoprotein inhibitors: synthesis and in vitro evaluation of a preactivated thiomer. (2016) (7)
- Impact of bile salts and a medium chain fatty acid on the physical properties of self-emulsifying drug delivery systems (2020) (7)
- Bacterial adhesins as a drug carrier: covalent attachment of K99 fimbriae to 6-methylprednisolone. (1997) (6)
- Entirely S-Protected Thiolated Silicone: A Novel Hydrophobic Mucoadhesive and Skin Adhesive. (2019) (6)
- S-Protected thiolated nanostructured lipid carriers exhibiting improved mucoadhesive properties. (2020) (6)
- In vivo investigation of thiomer-polyvinylpyrrolidon nanoparticles using magnetic resonance imaging. (2010) (6)
- Inhibitory effect of emulsifiers in sedds on protease activity: Just an illusion? (2017) (6)
- Intestinal enzymatic metabolism of drugs (2011) (6)
- Synthesis and evaluation of sulfosuccinate-based surfactants as counterions for hydrophobic ion pairing. (2022) (6)
- Strategies for improved hair binding: Keratin fractions and the impact of cationic substructures. (2020) (6)
- Lipophilic Arginine Esters: The Gateway to Preservatives without Side Effects (2020) (6)
- Mucoadhesive Polymers: Basics, Strategies, and Future Trends (2013) (6)
- Thiolated Nanoparticles for Biomedical Applications: Mimicking the Workhorses of Our Body (2021) (6)
- Preactivated silicone oil as potential long-term vitreous replacement with nonemulsifying properties. (2017) (5)
- Valaminols, probably the most simplified peptide-analogs acting as pepsin inhibitors (2000) (5)
- Synthesis and in vitro characterization of a preactivated thiolated acrylic acid/acrylamide-methylpropane sulfonic acid copolymer as a mucoadhesive sprayable polymer. (2020) (5)
- Evaluation of dermal adhesive formulations for topical application (2018) (5)
- Mucolytic self-emulsifying drug delivery systems (SEDDS) containing a hydrophobic ion-pair of proteinase. (2020) (5)
- The Use of Auxiliary Agents to Improve the Mucosal Uptake of Peptides (2004) (5)
- Reactive oxygen species (ROS) in colloidal systems: Are "PEG-free" surfactants the answer? (2022) (5)
- Anhydrous thiomers: Strategy for enhanced mucoadhesion (2018) (5)
- Comparison of mucoadhesive and cohesive features of poly(acrylic acid)‐conjugates respective their molecular mass (2017) (5)
- Thiolated chitosans in non-invasive drug delivery (2008) (4)
- Development of nanoparticulate drug delivery systems based on thiolated poly(acrylic acid) (2009) (4)
- In vitro skin permeation studies of the lantibiotic nisin (1996) (4)
- In vitro evaluation of thiomer microparticles for nasal drug delivery (2006) (4)
- Storage stability of proteins in a liquid-based formulation: liquid vs. solid self-emulsifying drug delivery. (2020) (4)
- Development and In Vitro Evaluation of a Mucoadhesive Oral Deliverv System for Antisense Oliaonucleotides (2003) (4)
- In vitro evaluation of tumor targeting ability of a parenteral enoxaparin-coated self-emulsifying drug delivery system (2019) (4)
- Development and In Vitro Characterization of Transferrin-Decorated Nanoemulsion Utilizing Hydrophobic Ion Pairing for Targeted Cellular Uptake (2021) (4)
- Self-emulsifying drug delivery systems: About the fate of hydrophobic ion pairs on a phospholipid bilayer (2020) (4)
- Gastroretentive particles formulated with thiomers: development and in vitro evaluation (2010) (3)
- Charge converting nanostructured lipid carriers containing a cell-penetrating peptide for enhanced cellular uptake. (2022) (3)
- Imine bond formation as a tool for incorporation of amikacin in self-emulsifying drug delivery systems (SEDDS). (2021) (3)
- Digestion of lipid excipients and lipid-based nanocarriers by pancreatic lipase and pancreatin. (2022) (3)
- Preparation and detailed characterization of the thiomer chitosan-cysteine as a suitable mucoadhesive excipient for nasal powders. (2022) (3)
- Assembly and in vitro characterization of thiomeric nanoparticles (2016) (3)
- Enhanced oral bioavailability of rutin by a self-emulsifying drug delivery system of an extract of calyces from Physalis peruviana (2021) (3)
- Polyaminated pullulan, a new biodegradable and cationic pullulan derivative for mucosal drug delivery. (2022) (3)
- Replacing PEG-surfactants in self-emulsifying drug delivery systems: Surfactants with polyhydroxy head groups for advanced cytosolic drug delivery. (2022) (3)
- Thiolation of non-ionic surfactants for the development of lipid-based mucoadhesive drug delivery systems. (2022) (3)
- [Nisin, a potential preservative for topical preparations]. (1996) (2)
- Overcoming the Mucosal Barrier: Tetraether Lipid‐Stabilized Liposomal Nanocarriers Decorated with Cell‐Penetrating Peptides Enable Oral Delivery of Vancomycin (2021) (2)
- Thiolated Chitosan Conjugated Liposomes for Oral Delivery of Selenium Nanoparticles (2022) (2)
- Development of a dosage form for accelerated release. (2014) (2)
- Grafting of wool fibers through disulfide bonds: An advanced application of S-protected thiolated starch. (2020) (2)
- Nano- and Microparticles in Oral Delivery of Macromolecular Drugs (2009) (2)
- Charge-reversal nanoemulsions: A systematic investigation of phosphorylated PEG-based surfactants. (2021) (2)
- Lipid-based nanoparticles: enhanced cellular uptake via surface thiolation. (2023) (2)
- Mucoadhesive Polymers: Gateway to Innovative Drug Delivery (2021) (2)
- Thiolated 2-Methyl-β-Cyclodextrin as a Mucoadhesive Excipient for Poorly Soluble Drugs: Synthesis and Characterization (2022) (2)
- Synthesis and in vitro characterization of a novel PAA–ATP conjugate (2011) (2)
- Corrigendum to “Inhibition of malarial topoisomerase II in Plasmodium falciparum by antisense nanoparticles” [Int. J. Pharm. 319 (2006) 139–146] (2006) (2)
- Evaluation of peptide drug delivery via skin barrier-impact of permeation enhancers (2017) (2)
- Design of nanostructured lipid carriers and solid lipid nanoparticles for enhanced cellular uptake. (2022) (2)
- Low Molecular Mass Permeation Enhancers in Oral Delivery of Macromolecular Drugs (2009) (2)
- Phosphate decorated lipid-based nanocarriers providing a prolonged mucosal residence time. (2022) (1)
- Surface design of nanocarriers: Key to more efficient oral drug delivery systems. (2023) (1)
- Oral delivery of calcitonin-ion pairs: In vivo proof of concept for a highly lipophilic counterion. (2022) (1)
- Polymer-enzyme inhibitor conjugates: influence of the molecular mass on the inhibition of membrane-bound aminopeptidase N activity (2004) (1)
- Combination of SEDDS and Preactivated Thiomer Technology: Incorporation of a Preactivated Thiolated Amphiphilic Polymer into Self-Emulsifying Delivery Systems (2017) (1)
- Per-thiolated cyclodextrins: Nanosized drug carriers providing a prolonged gastrointestinal residence time. (2022) (1)
- Betaine-modified hydroxyethyl cellulose (HEC): A biodegradable mucoadhesive polysaccharide exhibiting quaternary ammonium substructures. (2022) (1)
- Pharmaceutical Non-Viral Formulations for Gene Vaccines (2012) (1)
- Thiolated Pectins: In vitro and Ex vivo Evaluation of Three Generations of Thiomers (2021) (1)
- Chitosan – Polyphosphate nanoparticles for a targeted drug release at the absorption membrane (2022) (1)
- Biodegradable arginine based steroid-surfactants: cationic green agents for hydrophobic ion-pairing. (2022) (1)
- Corrigendum to “Thiolated silicone oil: Synthesis, gelling and mucoadhesive properties” [Acta Biomater. 16 (2015) 169–177] (2015) (1)
- LDD 02 Non-Invasive Oligonucleotide Delivery System Based on a Thiolated Polymer : Development and In Vitro Evaluation (2010) (0)
- Iminated aminoglycosides in self-emulsifying drug delivery systems: Dual approach to break down the microbial defense. (2022) (0)
- Charge-Converting Nanoemulsions as Promising Retinal Drug and Gene Delivery Systems (2022) (0)
- Development and In Vitro Evaluation of Stearic Acid Phosphotyrosine Amide as New Excipient for Zeta Potential Changing Self-Emulsifying Drug Delivery Systems (2020) (0)
- In Situ Crosslinkable Thiolated Chitosan as Scaffold Material for Tissue Engineering (2012) (0)
- Self-emulsifying drug delivery systems (SEDDS): In vivo-proof of concept for oral delivery of insulin glargine. (2023) (0)
- SEDDS-loaded mucoadhesive fiber patches for advanced oromucosal delivery of poorly soluble drugs. (2022) (0)
- Oral delivery of therapeutic peptides: Barriers and strategies to overcome them (2006) (0)
- Preparation and evaluation of charge reversal solid lipid nanoparticles. (2022) (0)
- Design and in vitro evaluation of a mucoadhesive oral delivery system for a model polypeptide antigen. (2001) (0)
- Role of sonication pre-treatment and cation valence in the sol-gel transition of nano-cellulose suspensions (2017) (0)
- It is containing sustained-release form (derivatives) alpha lipoic acid. (2000) (0)
- Pre-activated thiomer for nasal delivery of Apomorphine: Synthesis and in vitro evaluation (2015) (0)
- In vitro evaluation of a self-emulsifying drug delivery system (SEDDS) for nasal administration of dimenhydrinate (2019) (0)
- Mucoadhesive Polymers: Basics, Strategies, and Trends (2017) (0)
- Hydrophobic Ion Pairing of Small Molecules: How to Minimize Premature Drug Release from SEDDS and Reach the Absorption Membrane in Intact Form (2023) (0)
- Relation Between Scaffold Size and Membrane Bound Enzyme Caused Degradation of Two Novel Cystine Knot Microproteins (2007) (0)
- C3PY20939C 2342..2352 (2013) (0)
- Preparation and Evaluation of Charge Reversal Solid Lipid Nanoparticles (2021) (0)
- Thiomers : A potent tool for the non-invasive administration of efflux pump substrates ? (2006) (0)
- Thiolated cyclodextrins: A comparative study of their mucoadhesive properties. (2023) (0)
- Supplementary data to: Non-ionic thiolated cyclodextrins - The next generation (2018) (0)
- Solidification of self-emulsifying drug delivery systems (SEDDS): Impact on storage stability of a therapeutic protein Journal of Colloid and Interface Science (2020) (0)
- Phosphorothioate Oligonucleotide Quantification by μ-Liquid Chromatography-Mass Spectrometry (2012) (0)
- Entirely S-protected thiolated hydroxyethylcellulose: Design of a dual cross-linking approach for hydrogels. (2022) (0)
- Nanoarchitectonics of Layer-by-Layer (LbL) coated nanostructured lipid carriers (NLCs) for Enzyme-Triggered charge reversal. (2022) (0)
- Biodegradable Cationic and Ionizable Cationic Lipids: A Roadmap for Safer Pharmaceutical Excipients. (2023) (0)
- Per-Thiolated β-Cyclodextrins: Mucoadhesive Excipients Providing a Prolonged Gastrointestinal Residence Time (2022) (0)
- Thiolated PVP-Amphotericin B Complexes: An Innovative Approach toward Highly Mucoadhesive Gels for Mucosal Leishmaniasis Treatment. (2020) (0)
- Non-Invasive Oligonucleotide Delivery System Based on a Thiolated Polymer: Development and In Vitro Evaluation (2010) (0)
- WITHDRAWN: Zeta potential changing nanoemulsions: Impact of PEG-corona on phosphate cleavage (2020) (0)
- DEVELOPMENT AND IN VITRO EVALUATION OF MUCUS INERT NANOPARTICLES FOR MUCOSAL DISEASES (2012) (0)
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