Claus Braestrup
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Biology
Why Is Claus Braestrup Influential?
(Suggest an Edit or Addition)Claus Braestrup's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Benzodiazepine receptors in rat brain (1977) (1392)
- International Union of Pharmacology. XV. Subtypes of gamma-aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function. (1998) (1321)
- Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding. (1977) (1104)
- SEVERE ANXIETY INDUCED BY FG 7142, A β-CARBOLINE LIGAND FOR BENZODIAZEPINE RECEPTORS (1983) (571)
- Interaction of convulsive ligands with benzodiazepine receptors. (1982) (529)
- Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors. (1980) (495)
- Some properties of brain specific benzodiazepine receptors: New evidence for multiple receptors (1979) (399)
- High densities of benzodiazepine receptors in human cortical areas (1977) (399)
- Pharmacological characterization of benzodiazepine receptors in the brain. (1978) (273)
- Escitalopram versus citalopram: the surprising role of the R-enantiomer (2004) (236)
- Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitor. (1991) (222)
- Benzodiazepine receptor ligands with positive and negative efficacy (1983) (214)
- (R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake Carrier (1990) (213)
- Evidence for a late evolutionary appearance of brain-specific benzodiazepine receptors: an investigation of 18 vertebrate and 5 invertebrate species (1978) (185)
- Cocaine: Discussion on the Role of Dopamine in the Biochemical Mechanism of Action (1977) (164)
- Benzodiazepine receptors. (1985) (162)
- Audiogenic seizures in DBA/2 mice discriminate sensitively between low efficacy benzodiazepine receptor agonists and inverse agonists. (1983) (153)
- Ontogenetic development of benzodiazepine receptors in the rat brain (1978) (151)
- Ligands for benzodiazepine receptors with positive and negative efficacy. (1984) (148)
- Partial agonists for brain GABA/benzodiazepine receptor complex (1979) (138)
- Biochemical differentiation of amphetamine vs methylphenidate and nomifensine in rats (1977) (137)
- The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (tiagabine) as an anticonvulsant drug candidate. (1993) (136)
- Biologically active peptide-containing fractions in schizophrenia and childhood autism. (1981) (121)
- GABA reduces binding of 3H-methyl β-carboline-3-carboxylate to brain benzodiazepine receptors (1981) (119)
- Methylphenidate-like effects of the new antidepressant drug nomifensine (HOE 984). (1976) (109)
- Multiple benzodiazepine receptors (1980) (106)
- No changes in rat benzodiazepine receptors after withdrawal from continuous treatment with lorazepam and diazepam. (1979) (105)
- Evidence for Different States of the Dopamine Dl Receptor: Clozapine and Fluperlapine May Preferentially Label an Adenylate Cyclase‐Coupled State of the Dl Receptor (1986) (103)
- Does the reversal of the anticonflict effect of phenobarbital by beta-CCE and FG 7142 indicate benzodiazepine receptor-mediated anxiogenic properties? (1982) (103)
- In Vivo Measurement of Dopamine Receptors in Human Brain by Positron Emission Tomography Age and Sex Differences a (1988) (97)
- NNC-112, NNC-687 and NNC-756, new selective and highly potent dopamine D1 receptor antagonists. (1992) (95)
- Some atypical neuroleptics inhibit [3H]SCH 23390 binding in vivo. (1986) (93)
- High affinity of the naturally-occurring biflavonoid, amentoflavon, to brain benzodiazepine receptors in vitro. (1988) (90)
- Effects of the β-carboline, FG 7142, in the social interaction test of anxiety and the holeboard: Correlations between behaviour and plasma concentrations (1985) (85)
- Regulation in the central norepinephrine neurotransmission induced in vivo by alpha adrenoceptor active drugs. (1976) (75)
- Oxadiazoles as bioisosteric transformations of carboxylic functionalities. II (1996) (73)
- Evidence that the anticonflict effect of midazolam in amygdala is mediated by the specific benzodiazepine receptors (1985) (72)
- Noradrenergic influence on the stereotyped behaviour induced by amphetamine, phenethylamine and apomorphine (1976) (71)
- ACCUMULATION AND DISAPPEARANCE OF NORADRENALINE AND ITS MAJOR METABOLITES SYNTHESIZED FROM INTRAVENTRICULARLY INJECTED [3H]DOPAMINE IN THE RAT BRAIN (1974) (70)
- Radiation inactivation of brain [35S]t-butylbicyclophosphorothionate binding sites reveals complicated molecular arrangements of the GABA/benzodiazepine receptor chloride channel complex. (1985) (67)
- Differential pharmacological effects of benzodiazepine receptor inverse agonists. (1983) (65)
- Some properties of 3H-diazepam displacing activity from human urine. (1979) (63)
- Effects of phenoxybenzamine, aceperone and clonidine on the level of 3‐methoxy‐4‐hydroxyphenylglycol (MOPEG) in rat brain (1974) (62)
- CHARACTERISTICS AND REGIONAL DISTRIBUTIONS OF TWO DISTINCT [3H]NALOXONE BINDING SITES IN THE RAT BRAIN (1978) (59)
- Specific benzodiazepine receptors in rat brain characterized by high-affinity [ 3 H ] diazepam binding ( affinity binding / diazepam / anxiolytic activity / brain membranes / regional distribution ) (51)
- Binding of [3H]DMCM, a Convulsive Benzodiazepine Ligand, to Rat Brain Membranes: Preliminary Studies (1983) (51)
- Decreased spiroperidol and LSD binding in rat brain after continuous amphetamine. (1980) (47)
- Evaluation of the β-carboline ZK 93 426 as a benzodiazepine receptor antagonist (2004) (42)
- Anticonvulsant action in the photosensitive baboon, Papio papio, of a novel beta-carboline derivative, ZK 91296. (1983) (41)
- Intra‐ and extraneuronal formation of the two major noradrenaline metabolites in the cns of rats (1975) (39)
- Lack of brain specific benzodiazepine receptors on mouse primary astroglial cultures (1978) (39)
- New productOxadiazoles as bioisosteric transformations of carboxylic functionalities. Part I (1994) (38)
- gamma-Aminobutyric acid regulation of the benzodiazepine receptor: biochemical evidence for pharmacologically different effects of benzodiazepines and propyl beta-carboline-3-carboxylate. (1981) (38)
- Searching for endogenous benzodiazepine receptor ligands (1980) (38)
- Neuronal localisation of benzodiazepine receptors in cerebellum (1979) (37)
- The effects of FG 7142 and RO 15-1788 on the release of punished responding produced by chlordiazepoxide and ethanol in the rat (2004) (36)
- Identification of free and conjugated 3-methoxy-4-hydroxyphenylglycol (MOPEG) in rat brain by gas chromatography and mass fragmentography. (1973) (35)
- Effects of Heavy Metal Cations and Other Sulfhydryl Reagents on Brain Dopamine D1 Receptors: Evidence for Involvement of a Thiol Group in the Conformation of the Active Site (1987) (33)
- A METHOD FOR THE ASSAY OF CONJUGATED 3,4‐DIHYDROXYPHENYLGLYCOL, A MAJOR NORADRENALINE METABOLITE IN THE RAT BRAIN (1976) (32)
- Discriminative stimulus properties of methyl 6,7-dimethoxy-4-ethyl-beta-carboline-3-carboxylate (DMCM), an inverse agonist at benzodiazepine receptors. (1985) (31)
- ZK 91296, a partial agonist at benzodiazepine receptors (2004) (29)
- Benzodiazepine receptor ligands with positive and negative efficacy. (1983) (29)
- Glycine Antagonists Structurally Related to 4,5,6,7‐Tetrahydroisoxazolo[5,4‐c]pyridin‐3‐ol Inhibit Binding of [3H]Strychnine to Rat Brain Membranes (1986) (28)
- The benzodiazepine/GABA receptor complex during severe ethanol intoxication and withdrawal in the rat (1982) (27)
- Strychnine as a potent inhibitor of the brain GABA/benzodiazepine receptor complex (1980) (26)
- Modulation of GABA binding to rat brain membranes by alkyl beta-carboline-3-carboxylate esters. (1982) (25)
- Benzodiazepine Receptors (1980) (25)
- Barbiturate shift as a tool for determination of efficacy of benzodiazepine-receptor ligands. (1984) (25)
- Benzodiazepine receptors in the brain as affected by different experimental stresses: The changes are small and not undirectional (1979) (24)
- GABA-dopamine interaction in substantia nigra and nucleus accumbens--relevance to behavioral stimulation and stereotyped behavior. (1978) (18)
- Enhanced binding of the convulsive ligand DMCM to high-energy irradiated benzodiazepine receptors; evidence of complex receptor structure. (1983) (18)
- The molecular target size of brain TBPS binding sites. (1983) (18)
- The apparent target size of rat brain benzodiazepine receptor, acetylcholinesterase, and pyruvate kinase is highly influenced by experimental conditions. (1988) (18)
- Interaction of pitrazepin with the GABA/benzodiazepine receptor complex and with glycine receptors. (1985) (18)
- Evaluation of the beta-carboline ZK 93 426 as a benzodiazepine receptor antagonist. (1984) (18)
- Benzodiazepine receptor ligands with negative efficacy: chloride channel coupling. (1983) (17)
- A study on benzodiazepine receptor binding in audiogenic seizure-susceptible rats. (2009) (17)
- Bidirectional effects on anxiety of ß-carbolines acting as benzodiazepine receptor ligands (1984) (16)
- Absence of brain specific benzodiazepine receptors in cyclostomes and elasmobranchs. (1979) (16)
- beta-Carboline-3-carboxylates and benzodiazepine receptors. (1981) (15)
- Two or more conformations of benzodiazepine receptors depending on GABA receptors and other variables. (1980) (15)
- In vivo labeling of the central GABA uptake carrier with 3H-Tiagabine. (1992) (13)
- Development of 123I-labelled NNC 13-8241 as a radioligand for SPECT visualization of benzodiazepine receptor binding. (1996) (12)
- 3‐METHOXY‐4‐HYDROXYPHENYLETHANOL IN THE RAT BRAIN (1973) (12)
- Synthesis, GABA Agonist Activity and Effects on GABA and Diazepam Binding of Some N-Substituted Analogues of GABA. (1986) (11)
- Gas chromatographic evidence for the presence of 3-methoxy-4-hydroxyphenylethanol in rat brain. (1972) (10)
- Discovery of β-Carboline Ligands for Benzodiazepine Receptors (1993) (10)
- Binding of3H-DMCM to benzodiazepine receptors; chloride dependent allosteric regulation mechanisms (2005) (9)
- MODULATION OF BENZODIAZEPINE RECEPTORS (1981) (8)
- The Case for Involvement of Dopamine in Depression and Mania (1979) (7)
- MOLECULAR INTERACTIONS IN THE GABA/BENZODIAZEPINE RECEPTOR, CHLORIDE CHANNEL COMPLEX. HIGH ENERGY RADIATION INACTIVATION STUDIES (1984) (5)
- New developments in the search for central benzodiazepine endogenous ligand(s) (1988) (5)
- beta-Carbolines and benzodiazepine receptors. (1982) (4)
- Changes in drug-induced stereotyped behavior after 6-OHDA lesions in noradrenaline neurons. (1977) (4)
- Specific 3H-DMCM binding to a non-benzodiazepine binding site after silver ion treatment of rat brain membranes. (1984) (4)
- Reduction of 3H-spiroperidol binding in rat striatum and frontal cortex by chronic amphetamine: Dose response, time course and role of sustained dopamine release (2004) (4)
- Discovery of beta-carboline ligands for benzodiazepine receptors. (1993) (3)
- Oxadiazoles as Bioisosteric Transformations of Carboxylic Functionalities. Part 1. (1994) (3)
- Differentiation of Cl−/Ca2+-dependent and sodium dependent3H-glutamate binding to cortical membranes from rat brain by high energy radiation inactivation analysis (2005) (2)
- Roles of monoamines, particularly dopamine, in clinical depression and in the regulation of mood (1977) (2)
- Future directions in anxiety research. (1988) (1)
- INTERACTION OF -CARBOLINES WITH BENZODIAZEPINE RECEPTORS: (1984) (1)
- 2053 – DOES GABA ANTAGONIZE THE NIGRO-STRIATAL SYSTEM? (1978) (1)
- Receptor subtypes and endogenous ligands: rational tools in the search for psychotropic drugs? (1989) (1)
- Urinary and brain f 3-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors ( f-carboline / endogenous ligand / urine ) (1)
- Foerfarande Foer framstaellning of carboline-3-karboxylsyraderivat. (1984) (0)
- Different States of the Dopamine D1 Receptor: Fact or Fantasy? (1988) (0)
- Foerfarande Foer framstaellning of pharmacologically active five-alkoxi- carboline-3-karboxylsyraderivat. (1984) (0)
- Urinary and brain 3-carboline-3-ca brain benzodiazepine receptors (/-carboline/endogenous ligand/urine) (2016) (0)
- Analogifremgangsmaade for the preparation of beta-carboline-3-carboxylic acid derivatives (1983) (0)
- Ss-carboline, processes for their preparation and pharmaceutical compositions containing them (1982) (0)
- -karboliner, foerfarande Foer deras framstaellning Science innehaollande of pharmaceutical industry preparat (1983) (0)
- Benzodiazepinreceptoraktive compounds and methods for preparing the same (1982) (0)
- Beta-carbon line-3-carboxylic acid derivatives and processes for preparing the same (1980) (0)
- β-Carboline-3-carboxylic acid Derivatives and Brain Benzodiazepine Receptors (1984) (0)
- Foerfarande Foer framstaellning of pharmacologically active 2,3,4,5-tetrahydro-1H-3-benzazepinderivat. (1986) (0)
- 3-substituted beta-carboline derivatives, process for preparing them as well as drug containing the same (1984) (0)
- 5-substituted 2,3,4,5-tetrahydro-1H-3-benzazepines. (1986) (0)
- New (beta) carbolines, methods for their manufacture and their use as pharmaceuticals (h) (1983) (0)
- Beta-carboline-3-karboxylsyraderivat Science foerfaranden Foer framstaellning of dem (1980) (0)
- Analogifremgangsmaade for preparing oxadiazolylimidazo-oe1,4aa-benzodiazepine derivatives (1982) (0)
- Beta-carbolines, method for preparing the same and pharmaceutical composition containing the same (1983) (0)
- ANXIETY (1982) (0)
- Endogenous benzodiazepine receptor agonists? (1979) (0)
- New ss-carboline, process for their production and their use as drug (s) (1983) (0)
- Peripheral metabolism of beta-carboline-carboxylic acid esters. (1982) (0)
- Oxadiazoles as Bioisosteric Transformations of Carboxylic Functionalities. Part 2. (2010) (0)
- Beta-carboline-3-carboxylic acid derivatives and process for obtaining same (1983) (0)
- Beta-carbolines, a process for preparing the same and pharmaceutical composition containing the same (1983) (0)
- 2,3,4,5-tetrahydro-1H-3-benzazepine derivatives and pharmaceutical compositions containing them (1986) (0)
- Foerfarande Foer framstaellning psykofaramaka anvaendbarabeta of the i-carboline-3-karboxylsyraderivat (1980) (0)
- 3-substituted beta-carboline derivatives, process for preparing them as well as drug on the basis of the same (1984) (0)
- [Research on receptors and their psychiatric perspectives]. (1983) (0)
- Introductory comments: a brief history of the development of paroxetine. (1992) (0)
- Substituted ss-carboline, process for their production and their use as medicines (1983) (0)
- Neurotransmitter receptors, Part 1: Amino acids, peptides and benzodiazepines: edited by S.J. Enna and H.I. Yamamura, Chapman & Hall, 1980. £15.00 (xi + 212 pages) ISBN 0 412 16250 4 (1982) (0)
- Beta-carboline derivatives, procedure for their production and pharmaceutical product containing the same (1984) (0)
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