Dawei Ma
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Computer Science
Dawei Ma's Degrees
- PhD Computer Science Stanford University
- Masters Computer Science University of California, Berkeley
- Bachelors Computer Science Tsinghua University
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(Suggest an Edit or Addition)Dawei Ma's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Copper/amino acid catalyzed cross-couplings of aryl and vinyl halides with nucleophiles. (2008) (833)
- A Selective Inhibitor of eIF2α Dephosphorylation Protects Cells from ER Stress (2005) (806)
- A selective inhibitor of eIF2alpha dephosphorylation protects cells from ER stress. (2005) (708)
- Beclin1 Controls the Levels of p53 by Regulating the Deubiquitination Activity of USP10 and USP13 (2011) (640)
- Design of Wide-Spectrum Inhibitors Targeting Coronavirus Main Proteases (2005) (556)
- Amino acid promoted CuI-catalyzed C-N bond formation between aryl halides and amines or N-containing heterocycles. (2005) (525)
- Small molecule regulators of autophagy identified by an image-based high-throughput screen (2007) (457)
- Selected Copper-Based Reactions for C-N, C-O, C-S, and C-C Bond Formation. (2017) (355)
- Andrographolide Attenuates Inflammation by Inhibition of NF-κB Activation through Covalent Modification of Reduced Cysteine 62 of p501 (2004) (350)
- N,N-dimethyl glycine-promoted Ullmann coupling reaction of phenols and aryl halides. (2003) (318)
- Mild method for Ullmann coupling reaction of amines and aryl halides. (2003) (297)
- Synthesis of 1,2-disubstituted benzimidazoles by a Cu-catalyzed cascade aryl amination/condensation process. (2007) (245)
- Intramolecular dearomative oxidative coupling of indoles: a unified strategy for the total synthesis of indoline alkaloids. (2015) (243)
- Synthesis of aryl azides and vinyl azides via proline-promoted CuI-catalyzed coupling reactions. (2004) (215)
- Efficient and economical access to substituted benzothiazoles: copper-catalyzed coupling of 2-haloanilides with metal sulfides and subsequent condensation. (2009) (210)
- Synthesis of aryl sulfones via L-proline-promoted CuI-catalyzed coupling reaction of aryl halides with sulfinic acid salts. (2005) (206)
- Highly efficient catalytic system for enantioselective Michael addition of aldehydes to nitroalkenes in water. (2008) (200)
- Highly enantioselective bromocyclization of tryptamines and its application in the synthesis of (-)-chimonanthine. (2013) (174)
- CuI-catalyzed coupling reaction of beta-amino acids or esters with aryl halides at temperature lower than that employed in the normal Ullmann reaction. Facile synthesis of SB-214857. (2001) (172)
- Control of basal autophagy by calpain1 mediated cleavage of ATG5 (2010) (166)
- Asymmetric, protecting-group-free total synthesis of (-)-englerin A. (2010) (165)
- MYB Repressors as Regulators of Phenylpropanoid Metabolism in Plants. (2019) (163)
- Mild Ullmann-type biaryl ether formation reaction by combination of ortho-substituent and ligand effects. (2006) (160)
- Total synthesis and absolute stereochemical assignment of (-)-communesin F. (2010) (156)
- CuI/N,N-dimethylglycine-catalyzed coupling of vinyl halides with amides or carbamates. (2004) (155)
- A general and efficient approach to aryl thiols: CuI-catalyzed coupling of aryl iodides with sulfur and subsequent reduction. (2009) (151)
- Assembly of conjugated enynes and substituted indoles via CuI/amino acid-catalyzed coupling of 1-alkynes with vinyl iodides and 2-bromotrifluoroacetanilides. (2007) (150)
- The MYB182 Protein Down-Regulates Proanthocyanidin and Anthocyanin Biosynthesis in Poplar by Repressing Both Structural and Regulatory Flavonoid Genes1[OPEN] (2015) (142)
- CuI/Oxalic Diamide Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amines. (2015) (141)
- Synthesis of 3-substituted and 2,3-disubstituted quinazolinones via Cu-catalyzed aryl amidation. (2012) (134)
- Enantioselective addition of activated terminal alkynes to 1-acylpyridinium salts catalyzed by Cu-Bis(oxazoline) complexes. (2007) (134)
- Enantioselective arylation of 2-methylacetoacetates catalyzed by CuI/trans-4-hydroxy-L-proline at low reaction temperatures. (2006) (133)
- Elaboration of 2-(trifluoromethyl)indoles via a cascade coupling/condensation/deacylation process. (2008) (131)
- CuI/4-hydro-L-proline as a more effective catalytic system for coupling of aryl bromides with N-boc hydrazine and aqueous ammonia. (2009) (130)
- CuI-catalyzed coupling reaction of aryl halides with terminal alkynes in the absence of palladium and phosphine. (2004) (129)
- Formation of arylboronates by a CuI-catalyzed coupling reaction of pinacolborane with aryl iodides at room temperature (2006) (128)
- Total synthesis of Akuammiline alkaloid (-)-vincorine via intramolecular oxidative coupling. (2012) (128)
- Organocatalytic Michael addition of aldehydes to protected 2-amino-1-nitroethenes: the practical syntheses of oseltamivir (Tamiflu) and substituted 3-aminopyrrolidines. (2010) (126)
- Palladium-catalyzed direct functionalization of 2-aminobutanoic acid derivatives: application of a convenient and versatile auxiliary. (2013) (126)
- Domino condensation/S-arylation/heterocyclization reactions: copper-catalyzed three-component synthesis of 2-N-substituted benzothiazoles. (2011) (122)
- Rhodium-Catalyzed Regioselective C7-Functionalization of N-Pivaloylindoles. (2016) (120)
- Assembly of substituted phenothiazines by a sequentially controlled CuI/ L-proline-catalyzed cascade C-S and C-N bond formation. (2010) (117)
- Assembly of substituted 3-methyleneisoindolin-1-ones via a CuI/l-proline-catalyzed domino reaction process of 2-bromobenzamides and terminal alkynes. (2009) (116)
- l-Proline Promoted Ullmann-Type Coupling Reactions of Aryl Iodides with Indoles, Pyrroles, Imidazoles or Pyrazoles (2004) (113)
- CuI-catalyzed domino process to 2,3-disubstituted benzofurans from 1-bromo-2-iodobenzenes and beta-keto esters. (2007) (111)
- CuI/L-proline-catalyzed coupling reactions of aryl halides with activated methylene compounds. (2005) (109)
- Assembly of isoquinolines via CuI-catalyzed coupling of beta-keto esters and 2-halobenzylamines. (2008) (108)
- Enantioselective total syntheses of communesins A and B. (2011) (107)
- Co-recycling of MT1-MMP and MT3-MMP through the Trans-Golgi Network (2004) (105)
- Copper-Catalyzed Hydroxylation of (Hetero)aryl Halides under Mild Conditions. (2016) (103)
- Beclin 1 Controls the Levels of p 53 by Regulating the Deubiquitination Activity of USP 10 and USP 13 (2011) (102)
- Assembly of substituted 1H-benzimidazoles and 1,3-dihydrobenzimidazol-2-ones via CuI/L-proline catalyzed coupling of aqueous ammonia with 2-iodoacetanilides and 2-iodophenylcarbamates. (2009) (98)
- Assembly of N,N-disubstituted hydrazines and 1-aryl-1H-indazoles via copper-catalyzed coupling reactions. (2012) (94)
- Total synthesis of the monoterpenoid indole alkaloid (±)-aspidophylline A. (2014) (93)
- CuI/DMPAO-catalyzed N-arylation of acyclic secondary amines. (2012) (92)
- Enantioselective assembly of substituted dihydropyrones via organocatalytic reaction in water media. (2008) (90)
- First total synthesis of martinellic acid, a naturally occurring bradykinin receptor antagonist. (2001) (89)
- Aromatic nucleophilic substitution or CuI-catalyzed coupling route to martinellic acid. (2003) (89)
- Two R2R3-MYB proteins are broad repressors of flavonoid and phenylpropanoid metabolism in poplar. (2018) (88)
- Facile access to polysubstituted indoles via a cascade Cu-catalyzed arylation-condensation process. (2007) (87)
- Cyclodepsipeptide toxin promotes the degradation of Hsp90 client proteins through chaperone-mediated autophagy (2009) (84)
- Total synthesis of the cyclodepsipeptide apratoxin A and its analogues and assessment of their biological activities. (2006) (83)
- Crystal structure of SARS-CoV-2 main protease in complex with protease inhibitor PF-07321332 (2021) (82)
- Assembly of Primary (Hetero)Arylamines via CuI/Oxalic Diamide-Catalyzed Coupling of Aryl Chlorides and Ammonia. (2015) (78)
- Oxalic Diamides and tert-Butoxide: Two Types of Ligands Enabling Practical Access to Alkyl Aryl Ethers via Cu-Catalyzed Coupling Reaction. (2019) (77)
- Palladium catalyzed synthesis of annelated indoles (1991) (74)
- A one-pot coupling/hydrolysis/condensation process to pyrrolo[1,2-a]quinoxaline. (2008) (73)
- CuI/Oxalamide Catalyzed Couplings of (Hetero)aryl Chlorides and Phenols for Diaryl Ether Formation. (2016) (69)
- Discovery of N-(Naphthalen-1-yl)-N'-alkyl Oxalamide Ligands Enables Cu-Catalyzed Aryl Amination with High Turnovers. (2017) (69)
- Highly asymmetric bromocyclization of tryptophol: unexpected accelerating effect of DABCO-derived bromine complex. (2014) (68)
- Mild and nonracemizing conditions for Ullmann-type diaryl ether formation between aryl iodides and tyrosine derivatives. (2006) (67)
- Cascade coupling/cyclization process to N-substituted 1,3-dihydrobenzimidazol-2-ones. (2007) (67)
- Poplar MYB115 and MYB134 Transcription Factors Regulate Proanthocyanidin Synthesis and Structure1[OPEN] (2017) (64)
- Enantioselective organocatalytic Michael addition of malonates to α,β-unsaturated aldehydes in water (2008) (63)
- Assembly of 3-acyloxindoles via cui/L-proline-catalyzed intramolecular arylation of beta-keto amides. (2006) (63)
- N,N -dimethylglycine -promoted ullmann-type coupling reactions of aryl iodides with aliphatic alcohols (2007) (63)
- L ‐Proline‐Promoted CuI‐Catalyzed C‐S Bond Formation between Aryl Iodides and Thiols (2007) (62)
- Modeling, chemistry, and biology of the benzolactam analogues of indolactam V (ILV). 2. Identification of the binding site of the benzolactams in the CRD2 activator-binding domain of PKCdelta and discovery of an ILV analogue of improved isozyme selectivity. (1997) (62)
- Correction: Design of Wide-Spectrum Inhibitors Targeting Coronavirus Main Proteases (2005) (62)
- Total synthesis of (±)-martinelline (2002) (60)
- Iridium pentahydride complex catalyzed dehydrogenation of alcohols in the absence of a hydrogen acceptor (1987) (60)
- Enantioselective synthesis of functionalized α-amino acids via a chiral guanidine catalyzed Michael addition reaction (1999) (59)
- Synthesis of 2-thio-substituted benzothiazoles via a domino condensation/S-arylation/heterocyclization process. (2011) (59)
- Total synthesis of microsclerodermin E. (2003) (57)
- Total synthesis of the indole alkaloid (±)- and (+)-methyl N-decarbomethoxychanofruticosinate. (2013) (55)
- Synthesis and biology of a 7-nitro-2,1,3-benzoxadiazol-4-yl derivative of 2-phenylindole-3-acetamide: a fluorescent probe for the peripheral-type benzodiazepine receptor. (1997) (54)
- AN IMPROVED PROCEDURE TO HOMOCHIRAL CYCLIC STATINES (1996) (54)
- PIM Kinase Inhibitors Downregulate STAT3Tyr705 Phosphorylation (2010) (53)
- A pharmacoproteomic approach implicates eukaryotic elongation factor 2 kinase in ER stress-induced cell death (2008) (52)
- Organocatalytic approach to polysubstituted piperidines and tetrahydropyrans. (2011) (52)
- A Unified Approach for the Assembly of Atisine- and Hetidine-type Diterpenoid Alkaloids: Total Syntheses of Azitine and the Proposed Structure of Navirine C. (2018) (50)
- Highly stereoselective isomerization of ynones to conjugated dienones catalyzed by transition metal complexes (1989) (50)
- Total synthesis and structure assignment of papuamide B, a potent marine cyclodepsipeptide with anti-HIV properties. (2008) (50)
- A Novel Small Molecule Regulator of Guanine Nucleotide Exchange Activity of the ADP-ribosylation Factor and Golgi Membrane Trafficking* (2008) (50)
- Oxidative coupling strategies for the synthesis of indole alkaloids. (2018) (49)
- Enantioselective synthesis of polysubstituted cyclopentanones by organocatalytic double Michael addition reactions. (2010) (48)
- A novel stereoselective synthesis of conjugated dienones (1988) (47)
- A simple and stereospecfic route to 2,6-disubstituted 4-hydroxypiperidines. Synthesis of dendrobate alkaloid (+)-241D and formal synthesis of (-)-indolizidine 167B. (2000) (47)
- Copper-Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amides. (2017) (46)
- Synthesis of an oxazoline analogue of apratoxin A. (2003) (46)
- Total synthesis of halipeptin A: a potent antiinflammatory cyclic depsipeptide. (2005) (46)
- Total synthesis and cytotoxicity studies of a cyclic depsipeptide with proposed structure of palau'amide. (2005) (45)
- Total synthesis of cyclic tetrapeptide FR235222, a potent immunosuppressant that inhibits mammalian histone deacetylases. (2005) (45)
- Construction of polycyclic spiro-indolines via an intramolecular oxidative coupling/cyclization cascade reaction process. (2012) (44)
- Highly convergent route to cyclopeptide alkaloids: total synthesis of ziziphine N. (2007) (43)
- Diastereoselective aldol reaction of N,N-dibenzyl-alpha-amino aldehydes with ketones catalyzed by proline. (2004) (42)
- CuI/N,N-Dimethylglycine-Catalyzed Cross-Coupling Reaction of Vinyl Halides with Phenols and its Application to the Assembly of Substituted Benzofurans (2005) (41)
- Cyclobutane derivatives as novel nonpeptidic small molecule agonists of glucagon-like peptide-1 receptor. (2012) (41)
- Organocatalytic Michael addition of aldehydes to gamma-keto-alpha,beta-unsaturated esters. an efficient entry to versatile chiral building blocks. (2008) (40)
- A convergent route to the Galbulimima alkaloids (-)-GB 13 and (+)-GB 16. (2010) (40)
- Isomerization of propargylic alcohols catalyzed by an iridium complex (1989) (40)
- Iridium(III)-Catalyzed Regioselective C7-Amination of N-Pivaloylindoles with Sulfonoazides. (2016) (40)
- Convergent Route to ent-Kaurane Diterpenoids: Total Synthesis of Lungshengenin D and 1α,6α-Diacetoxy-ent-kaura-9(11),16-dien-12,15-dione. (2017) (40)
- General route to 2,4,5-trisubstituted piperidines from enantiopure beta-amino esters. Total synthesis of pseudodistomin B triacetate and pseudodistomin F. (2000) (40)
- Synthesis of 1,5-benzothiazepine dipeptide mimetics via two CuI-catalyzed cross coupling reactions. (2009) (38)
- Synthesis of enantiopure substituted dihydrofurans via the reaction of (S)-glyceraldehyde acetonide- or Garner aldehyde acetonide-derived enones with sulfonium ylides (2002) (37)
- Asymmetric Strecker-Type Reaction of alpha-Aryl Ketones. Synthesis of (S)-alphaM4CPG, (S)-MPPG, (S)-AIDA, and (S)-APICA, the Antagonists of Metabotropic Glutamate Receptors. (1999) (37)
- Asymmetric, Regioselective Bromohydroxylation of 2-Aryl-2-propen-1-ols Catalyzed by Quinine-Derived Catalysts (2013) (36)
- Two-component method to enantiopure quinolizidinones and Indolizidinones. Total synthesis of (-)-lasubine II. (2001) (35)
- Structure-activity relationship studies of salubrinal lead to its active biotinylated derivative. (2005) (34)
- Effect of alteration of the heterocyclic nucleus of ILV on its isoform selectivity for PKC. Palladium catalyzed route to benzofuran analogues of ILV (1995) (34)
- Diastereoselective Henry reactions of N,N-dibenzyl α-amino aldehydes with nitromethane catalyzed by enantiopure guanidines (2002) (34)
- Total synthesis of kaitocephalin, the first naturally occurring AMPA/KA receptor antagonist. (2001) (34)
- Total synthesis of piperazimycin A: a cytotoxic cyclic hexadepsipeptide. (2009) (33)
- Design, synthesis, and evaluation of potent, nonpeptidic mimetics of second mitochondria-derived activator of caspases. (2009) (33)
- Copper(I) Oxide/N,N′‐Bis[(2‐furyl)methyl]oxalamide‐Catalyzed Coupling of (Hetero)aryl Halides and Nitrogen Heterocycles at Low Catalytic Loading (2017) (32)
- Thiourea-Catalyzed Asymmetric Michael Addition of Carbazolones to 2-Chloroacrylonitrile: Total Synthesis of 5,22-Dioxokopsane, Kopsinidine C, and Demethoxycarbonylkopsin. (2018) (32)
- Asymmetric total synthesis of (-)-alkaloid 223A and its 6-epimer. (2003) (32)
- Total synthesis of lepadins B, d, e, and h; determination of the configuration of the latter three alkaloids. (2004) (31)
- Synthesis of (S)-α-Cyclopropyl-4- phosphonophenylglycine (2001) (31)
- Total synthesis of antimicrobial and antitumor cyclic depsipeptides. (2010) (31)
- Synthesis of chiral N-aryl-α-amino acids by PdCu catalyzed couplings of chiral α-amino acids with aryl halides (1996) (31)
- The N-aryl aminocarbonyl ortho-substituent effect in Cu-catalyzed aryl amination and its application in the synthesis of 5-substituted 11-oxo-dibenzodiazepines. (2011) (31)
- Assembly of indoline-2-carboxylate-embodied dipeptides via Pd-catalyzed C(sp2)-H bond direct functionalization. (2015) (31)
- A formal [3+2] cycloaddition process with nonactivated aziridines to polysubstituted indolizidines. (2005) (30)
- Total synthesis of leucosceptroids A and B. (2015) (30)
- A Scalable Total Synthesis of the Antitumor Agents Et-743 and Lurbinectedin. (2019) (30)
- Synthesis of symmetrical and unsymmetrical N,N'-diaryl guanidines via copper/N-methylglycine-catalyzed arylation of guanidine nitrate. (2012) (29)
- Tetrahydroisoquinoline based sulfonamide hydroxamates as potent matrix metalloproteinase inhibitors. (2004) (29)
- Synthesis of the biaryl moiety of the proteasome inhibitors TMC-95 via a ligandless Pd(OAc)2-catalyzed Suzuki-coupling reaction (2001) (29)
- Organocatalytic approach for the syntheses of corynantheidol, dihydrocorynantheol, protoemetinol, protoemetine, and mitragynine. (2011) (29)
- Synthesis and biological activity of cyclic analogues of MPPG and MCPG as metabotropic glutamate receptor antagonists (1997) (28)
- Synthesis of Aryl Carbamates via Copper‐Catalyzed Coupling of Aryl Halides with Potassium Cyanate (2012) (28)
- A one-pot formal [4 + 2] cycloaddition approach to substituted piperidines, indolizidines, and quinolizidines. total synthesis of indolizidine (-)-209I. (2005) (28)
- Structural basis of RasGRP binding to high-affinity PKC ligands. (2002) (28)
- Synthetic Studies toward Communesins (2011) (28)
- A simple route to α,β-unsaturated aldehydes from prop-2-ynols (1989) (28)
- Total synthesis of salinamide A: a potent anti-inflammatory bicyclic depsipeptide. (2008) (27)
- The MYB182 protein downregulates proanthocyanidin and anthocyanin biosynthesis in poplar by repressing both structural and regulatory flavonoid genes Authors: (2015) (27)
- Stereospecific route to enantiopure all cis-2,3,6-trisubstituted piperidines. Facile synthesis of (-)-deoxocassine and (+)-azimic acid (2003) (27)
- Synthesis, molecular modeling, 2-D NMR, and biological evaluation of ILV mimics as potential modulators of protein kinase C (1993) (27)
- Potentially biomimetic total synthesis and relative stereochemical assignment of (±)-gracilamine. (2012) (26)
- A Class of Amide Ligands Enable Cu-Catalyzed Coupling of (Hetero)aryl Halides with Sulfinic Acid Salts under Mild Conditions. (2018) (26)
- Cu(I)/L-proline-catalyzed coupling of substituted 3-iodoprop-2-en-1-ols with 1-alkynes and subsequent cyclization: a convenient approach for synthesizing polysubstituted furans. (2010) (26)
- Facile synthesis of 1,4-benzodiazepin-3-ones from o-bromobenzylamines and amino acids via a cascade coupling/condensation process (2009) (26)
- Asymmetric total syntheses of marine cyclic depsipeptide halipeptins A-D. (2006) (26)
- Enantioselective construction of the oxidized tryptophan fragment of proteasome inhibitors TMC-95A and TMC-95B (2000) (25)
- Facile entry to substituted decahydroquinoline alkaloids. Total synthesis of lepadins A-E and H. (2006) (25)
- Total syntheses of (±)-spiroquinazoline, (-)-alantryphenone, (+)-lapatin A, and (-)-quinadoline B. (2013) (25)
- Synthesis and protein kinase C binding activity of benzolactam-V7. (1999) (25)
- CuI‐Catalyzed Hydroxylation of Aryl Bromides under the Assistance of 5‐Bromo‐2‐(1H‐imidazol‐2‐yl)pyridine and Related Ligands. (2011) (24)
- Copper-Catalyzed Diaryl Ether Formation from (Hetero)aryl Halides at Low Catalytic Loadings. (2017) (24)
- A new methodology to key intermediates for synthesizing polyene compounds (1990) (24)
- Cu/N,N'-Dibenzyloxalamide-Catalyzed N-Arylation of Heteroanilines. (2019) (24)
- Total Synthesis of Lapidilectine B Enabled by Manganese(III)-Mediated Oxidative Cyclization of Indoles. (2018) (24)
- Pd-Catalyzed Dimethylation of Tyrosine-Derived Picolinamide for Synthesis of (S)-N-Boc-2,6-dimethyltyrosine and Its Analogues. (2017) (24)
- N,N'-Bisoxalamides Enhance the Catalytic Activity in Cu-Catalyzed Coupling of (Hetero)Aryl Bromides with Anilines and Secondary Amines. (2017) (23)
- Synthesis of 7-substituted benzolactam-V8s and their selectivity for protein kinase C isozymes. (2002) (23)
- Identification, biochemical and structural evaluation of species-specific inhibitors against type I methionine aminopeptidases. (2013) (23)
- Asymmetric synthesis of (−)-deoxoprosophylline (2003) (23)
- Prepartion of syn-δ-Hydroxy-β-amino esters via an intramolecular hydrogen bond directed diastereoselective hydrogenation. Total synthesis of (3S,4aS,6R,8S)-hyperaspine (2003) (23)
- An Efficient Synthesis of Phenol via CuI/8-Hydroxyquinoline-Catalyzed Hydroxylation of Aryl Halides and Potassium Hydroxide (2010) (22)
- Organocatalytic approach to 3,5,6-trisubstituted and 4,6-disubstituted tetrahydropyran-2-ones (2010) (22)
- Cascade annulation of malonic diamides: a concise synthesis of polycyclic pyrroloindolines. (2012) (22)
- Amination and Formation of sp2 C-N Bonds (2013) (21)
- Recent advances in the discovery of protein kinase C modulators based on the structures of natural protein kinase C activators. (2001) (21)
- Preparation of N‐Aryl Compounds by Amino Acid‐Promoted Ullmann‐Type Coupling Reactions. (2005) (21)
- Cu-Mediated Ullmann-Type Cross-Coupling and Industrial Applications in Route Design, Process Development, and Scale-up of Pharmaceutical and Agrochemical Processes (2022) (21)
- Total synthesis and stereochemistry assignment of 15-membered peptide alkaloids abyssenine B and mucronine E (2007) (21)
- Synthesis and Biological Evaluation of 1,3,3,4‐Tetrasubstituted Pyrrolidine CCR5 Receptor Antagonists. Discovery of a Potent and Orally Bioavailable Anti‐HIV Agent (2007) (21)
- CuI/N,N-dimethylglycine-catalyzed synthesis of N-aryloxazolidinones from aryl bromides (2012) (21)
- Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers. (2011) (21)
- Selective inhibition of matrix metalloproteinase isozymes and in vivo protection against emphysema by substituted gamma-keto carboxylic acids. (2006) (21)
- Assembly of substituted 3-aminoindazoles from 2-bromobenzonitrile via a CuBr-catalyzed coupling/condensation cascade process. (2013) (21)
- General and Stereospecific Route to 9-Substituted, 8,9-Disubstituted, and 9,10-Disubstituted Analogues of Benzolactam-V8 (1999) (21)
- Synthesis of enantiopure alpha,alpha-disubstituted amino acids from the asymmetric Strecker reaction products of aldehydes. (2000) (20)
- Organocatalytic and scalable synthesis of the anti-influenza drugs zanamivir, laninamivir, and CS-8958. (2014) (20)
- Stereoselective synthesis of (S)-MPPG, (S)-MTPG and (S)-(+)-αM4CPG from (R)-4-hydroxyphenylglycine (1997) (20)
- Organocatalytic Michael addition of aldehydes to trisubstituted nitroolefins (2012) (20)
- Enantioselective Organocatalytic Conjugate Addition of Aldehydes to α,β-Unsaturated Thiol Esters (2009) (20)
- Amino acid-promoted Ullmann-type coupling reactions and their applications in organic synthesis (2009) (20)
- Total Synthesis of (2S,3S,4R)-Plakoridine A. (2000) (19)
- Divergent Entry to Gelsedine-Type Alkaloids: Total Syntheses of (-)-Gelsedilam, (-)-Gelsenicine, (-)-Gelsedine, and (-)-Gelsemoxonine. (2018) (19)
- A sequential reaction process to assemble polysubstituted indolizidines, quinolizidines and quinolizidine analogues (2006) (19)
- A xanthone and a polyketide derivative from the leaves of Cassia obtusifolia (Leguminosae) (2008) (19)
- STEREOSPECIFIC SYNTHESIS OF (1S,3R)-1-AMINOCYCLOPENTANE-1,3-DICARBOXYLIC ACID, A SELECTIVE AGONIST OF METABOTROPIC GLUTAMATE RECEPTORS (1997) (19)
- CuI/8‐Hydroxyquinalidine Promoted N‐Arylation of Indole and Azoles (2012) (19)
- Asymmetric Strecker reaction of γ-keto acids. Facile entry to α-substituted and α,γ-disubstituted glutamic acids (2004) (18)
- Assembly of α-(Hetero)aryl Nitriles via Cu-Catalyzed Coupling Reactions with (Hetero)aryl Chlorides and Bromides. (2020) (18)
- Diastereoselective synthesis of 2,4,5-trisubstituted piperidines from enantiopure β-amino esters (1999) (18)
- Chiral Guanidine Catalyzed Annulation to the Core Structure of (‐)‐Huperzine A (2010) (18)
- An efficient sequential reaction process to polysubstituted indolizidines and quinolizidines and its application to the total synthesis of indolizidine 223A. (2005) (18)
- ENANTIOSELECTIVE SYNTHESES OF TUSSILAGINE AND ISOTUSSILAGINE (1998) (17)
- Metal-catalyzed derivatization of C(alpha)-tetrasubstituted amino acids and their use in the synthesis of cyclic peptides. (2009) (17)
- Synthesis of 7,8-disubstituted benzolactam-V8 and its binding to protein kinase C. (2001) (16)
- 6-Methylenebicyclo[3.2.1]oct-1-en-3-one: A twisted olefin as Diels-Alder dienophile for expedite syntheses of four kaurane diterpenoids. (2019) (16)
- Polyfunctionalized pyrrolidinones via the coupling of N,N- disubstituted β-amino esters with ethyl glyoxalate (1998) (16)
- Synthesis of N-(Hetero)aryl Carbamates via CuI/MNAO Catalyzed Cross-Coupling of (Hetero)aryl Halides with Potassium Cyanate in Alcohols. (2018) (16)
- Facile synthesis of (2S,1'S,2'S)-2-(Carboxycyclopropyl) glycine, an isotype-selective agonist of metabotropic glutamate receptors (1997) (16)
- Facile synthesis of (2E,4E)-dienoic esters via stereoselective isomerization of 2-ynoic esters (1989) (16)
- Assembly of N-substituted pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones via copper catalyzed aryl amination (2010) (16)
- Asymmetric synthesis of (S)-1-aminoindan-1,5-dicarboxylic acid and related analogues via intramolecular acylation of enantiopure α,α-disubstituted amino acids (2002) (16)
- Oxidation of benzylic methylene compounds to ketones with m-chloroperoxybenzoic acid and oxygen (1999) (16)
- Copper-catalyzed coupling of aryl iodides and tert-butyl β-keto esters: efficient access to α-aryl ketones and α-arylacetic acid tert-butyl esters (2014) (16)
- Small-molecule PD-L1 inhibitor BMS1166 abrogates the function of PD-L1 by blocking its ER export (2020) (15)
- Total synthesis of clavepictines A and B and pictamine. (2006) (15)
- Synthesis and antitumor activity of cyclodepsipeptide zygosporamide and its analogues. (2008) (15)
- Total synthesis and cytotoxicity of bisebromoamide and its analogues (2011) (15)
- Stereospecific total synthesis of (−)-8-epi-hyperaspine (2003) (15)
- In Pursuit of Synthetic Efficiency: Convergent Approaches. (2021) (15)
- Stereocontrolled cyclopropanation of Garner's aldehyde derived enones (2000) (14)
- A flexible route to immunosuppressive agent FR252921. Asymmetric total synthesis of its (13R,14R,19R)-isomer (2006) (14)
- Diastereoselective construction of continuous all-carbon quaternary centers via intramolecular oxidative coupling reaction (2013) (14)
- Assembly of 4‐Substituted 3‐Nitro‐1,2,3,4‐tetrahydropyridines via Organocatalytic Michael Addition (2012) (14)
- Stereoselective synthesis of (S)-(+)-αM4CPG, a selective antagonist of metabotropic glutamate receptors (1996) (14)
- Total synthesis of kopsinitarine E. (2020) (14)
- Efficient formal synthesis of the dendrobatid alkaloid, indolizidine (−)-209B (2002) (14)
- A concise route to the proposed structure of lydiamycin B, an antimycobacterial depsipeptide. (2009) (14)
- Reinvestigation on total synthesis of kaitocephalin and its isomers (2011) (14)
- A copper-catalyzed coupling reaction of vinyl halides and carbazates: application in the assembly of polysubstituted pyrroles. (2014) (14)
- Conformationally Constrained Analogues ofL-Glutamate as Subtype-Selective Modulators of Metabotropic Glutamate Receptors (1999) (13)
- Pyridinylquinazolines selectively inhibit human methionine aminopeptidase-1 in cells. (2013) (13)
- Trypanocidal labdane diterpenoids from the seeds of Aframomum aulacocarpos (Zingiberaceae) (2007) (13)
- A new three-carbon homologating agent for synthesis of α- keto aldehydes (1991) (12)
- Synthesis of Aryl Hydrazines via CuI/BMPO Catalyzed Cross-Coupling of Aryl Halides with Hydrazine Hydrate in Water (2018) (12)
- Cu((i))/amino acid catalyzed coupling reactions of aryl halides and nucleophiles: applications in large-scale production. (2011) (12)
- Novel reactions catalyzed by iridium pentahydride complex (1988) (12)
- A New Class of Amide Ligands Enable Cu‐Catalyzed Coupling of Sodium Methanesulfinate with (Hetero)aryl Chlorides (2017) (12)
- Enantioselective syntheses of α-substituted glutamic acids and α,γ-disubstituted glutamic acids by an asymmetric Strecker reaction (1999) (12)
- β-Amino ester route to tussilagine, isotussilagine and (–)-petasinecine (1999) (12)
- Copper‐Catalyzed Ligand Promoted Ullmann‐Type Coupling Reactions (2010) (12)
- Synthesis of (2S,1′ S,2′ S)-2-methyl-2-(carboxycyclopropyl)glycine and (S)-2-amino-2-methyl-4-phosphonobutyric acid from l-alanine (1997) (12)
- Asymmetric synthesis of α,α-disubstituted amino acids by diastereoselective functionalization of enantiopure phenyloxazinones, derivatives of asymmetric Strecker reaction products of aldehydes (2001) (11)
- Pd/Cu-catalyzed couplings of β-amino esters with aryl bromides. Synthesis of chiral 1,2,3,4-tetrahydro-4-oxo-2-alkyl-1-quinolines (1998) (11)
- A short synthesis of the HIV-protease inhibitor nelfinavir via a diastereoselective addition of ammonia to the α,β-unsaturated sulfoxide derived from (R)-glyceraldehyde acetonide (2002) (11)
- Selective cconversion of pinane into β-pinene catalyzed by an iridium pentahydride complex (1987) (11)
- Synthesis of polysubstituted 1,2-dihydroisoquinolines via a CuI-catalyzed arylation/condensation cascade process (2009) (11)
- Facile synthesis of (+)-α-allokainic acid via Pd-catalyzed hydrogenolysis of allyl acetate derived from trans-4-hydroxy-L-proline (2001) (11)
- CuI-Catalyzed One-Pot Synthesis of Benzothiazolones from 2-Iodoaniline-Derived Carbamates and Sodium Sulfide. (2012) (11)
- Thiourea-Catalyzed Asymmetric Michael Addition of Carbazolones to 2-Chloroacrylonitrile: Total Synthesis of 5,22-Dioxokopsane, Kopsinidine C, and Demethoxycarbonylkopsin (2018) (11)
- Recent progress on the total synthesis of natural products in China. (2006) (10)
- Stereoselective isomerization of acetylenic derivatives as a new methodology in organic synthesis (1990) (10)
- Development of 3‐Phenyl‐N‐(2‐(3‐phenylureido)ethyl)‐thiophene‐2‐sulfonamide Compounds as Inhibitors of Antiapoptotic Bcl‐2 Family Proteins (2014) (10)
- Synthesis of Aryl Azides and Vinyl Azides via Proline‐Promoted CuI‐Catalyzed Coupling Reactions. (2004) (10)
- Amino Acid Promoted/CuI‐Catalyzed C—N Bond Formation Between Aryl Halides and Amines or N‐Containing Heterocycles. (2005) (9)
- Intramolecular Oxidative Coupling: Applications in Synthesis of Complex Indole Akaloid Scaffolds (2013) (9)
- Ring-Opening Reactions of α,β-Epoxy Silanes with Organocopper Reagents: Reaction at Carbon or Silicon? (1996) (9)
- An efficient and tunable route to AG7088, a rhinovirus protease inhibitor (2004) (9)
- Copper/Amino Acid Catalyzed Cross-Couplings of Aryl and Vinyl Halides with Nucleophiles (2009) (9)
- Synthesis of enantiopure N-protected 4,5-disubstituted 3-pyrrolidinones and N-protected 2,5-disubstituted 3-pyrrolidinones via the Dieckmann reaction of dicarbonyl compounds derived from enantiopure β-amino esters (2001) (9)
- Poplar MYB117 promotes anthocyanin synthesis and enhances flavonoid B-ring hydroxylation by upregulating the flavonoid 3',5'-hydroxylase gene. (2021) (9)
- 6‐Methylenebicyclo[3.2.1]oct‐1‐en‐3‐one: A Twisted Olefin as Diels–Alder Dienophile for Expedited Syntheses of Four Kaurane Diterpenoids (2019) (8)
- Stereospecific synthesis of 9-substituted benzolactam-V8 from L-tyrosine via regioselective aromatic nitration (1998) (8)
- Synthesis of 2-alkyl-2-arylcyanoacetates via CuI/sodium picolinate-catalyzed direct arylation of α-substituted cyanoacetates (2013) (8)
- Synthetic Studies toward Plumisclerin A. (2019) (8)
- Synthesis of 1,2,4-Benzotriazines via Copper(I) Iodide/1H-Pyrrole-2-carboxylic Acid Catalyzed Coupling of o-Haloacetanilides and N-Boc Hydrazine (2015) (8)
- Synthesis and biological evaluation of two analogues of (S)- α-methyl -3-carboxyphenylalanine (1998) (8)
- Synthesis of (2S,1′R,2′R,3′R)-2-(2′,3′-Dicarboxycyclopropyl)-glycine via the Stereochemically Controlled Cyclopropanation of (S)-Glyceraldehyde Acetonide-Derived Enones (2000) (8)
- CHAPTER 1:Cu‐Catalyzed Ullmann‐Type C–Heteroatom Bond Formation: The Key Role of Dinucleating Ancillary Ligands (2013) (8)
- Enantioselective Arylation of 2‐Methylacetoacetates Catalyzed by CuI/trans‐4‐Hydroxy‐L‐proline at Low Reaction Temperatures. (2007) (7)
- Total Synthesis of the Indole Alkaloid (.+-.)- and (+)-Methyl N-Decarbomethoxychanofruticosinate. (2014) (7)
- Assembly of N,N-disubstituted-N′-arylureas via a copper-catalyzed one-pot three-component reaction of aryl bromides, potassium cyanate, and secondary amines (2013) (7)
- Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1. (2013) (7)
- Modern Ullmann–Goldberg Chemistry: Arylation of N‐Nucleophiles with Aryl Halides (2013) (7)
- Regioselective acylation at the 5- or 6-position of l-tryptophan derivatives (2002) (7)
- Assembly of N-Containing Heterocycles via Pd- and Cu-Catalyzed C–N Bond Formation Reactions (2013) (7)
- Synthetic studies toward galbulimima alkaloid (-)-GB 13 and (+)-GB 16 and (-)-himgaline. (2011) (7)
- Efficient synthesis of pyrrolo[2,3-d]pyrimidines via a Cu(I)/6-methylpicolinic acid catalyzed coupling reaction (2015) (6)
- Identification of a small molecule activator of novel PKCs for promoting glucose-dependent insulin secretion (2011) (6)
- N,N‐Dimethyl Glycine‐Promoted Ullmann Coupling Reaction of Phenols and Aryl Halides. (2004) (6)
- Sodium Amalgam, a Useful Reducing Reagent for Formation of Amines from Azides Bearing a Variety of Functional Groups (2005) (6)
- An efficient synthesis of isocoumarins via a CuI catalyzed cascade reaction process (2009) (6)
- Efficient Entry to Polysubstituted Pyrrolizidines, Indolizidines and Quinolizidines via a Sequential Reaction Process (2006) (5)
- Samarium iodide-mediated C–C bond formation in the total synthesis of natural products (2022) (5)
- A Convenient Synthesis of 3-(1,3-Alkadienyl)-2-cycloalken-1-ones (1990) (5)
- A Scalable Process to the Key Intermediate of Cilazapril, (S)-1-Benzyloxycarbonylhexahydropyridazine-3-carboxylic Acid, Through a Novel Cascade Course (2013) (5)
- A palladium catalyzed route to a benzofuran analogue of idolactam V (ILV): Effects on PKC isotype selectivity (1994) (5)
- Synthesis of (2-Arylindol-3-yl)acetamides as Probes of Mitochondrial Steroidogenesis—A New Mechanism for GABAA Receptor Modulation† (1992) (5)
- Preparation of (R)‐4‐Cyclohexyl‐2,3‐butadien‐1‐ol (2014) (5)
- Synthesis and Protein Kinase C Binding Activity of Benzolactam‐V7. (1999) (5)
- Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group (2017) (5)
- Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 2: Discovery of highly potent anti-HIV agents. (2010) (5)
- Diphenylbutylpiperidine-based cell autophagy inducers: Design, synthesis and SAR studies (2011) (5)
- Intramolecular Dearomative Oxidative Coupling of Indoles: A Unified Strategy for the Total Synthesis of Indoline Alkaloids (2015) (4)
- A Sequential Reaction Process to Assemble Polysubstituted Indolizidines, Quinolizidines and Quinolizidine Analogues. (2006) (4)
- Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 1: Tuning the N-substituents. (2010) (4)
- Formation of arylboronates by a CuI-catalyzed coupling reaction of pinacolborane with aryl iodides at room temperature. (2006) (4)
- Assembly of 7-carboxylate indoles via the Cu-catalyzed coupling of substituted 2-iodobenzoic acids and substituted hydrazines (2020) (4)
- Recent advances in the synthesis of ent-kaurane diterpenoids. (2021) (4)
- MYB134-RNAi poplars show reduced tannin synthesis in leaves but not roots, and increased susceptibility to oxidative stress. (2020) (4)
- Asymmetric Total Syntheses of Marine Cyclic Depsipeptide Halipeptins A—D. (2006) (3)
- Synthesis of Tetrahydropyrrolo[1,2-a]quinoxalines and Tetrahydropyrido[1,2-a]quinoxalines via a One-PotCuI-Catalyzed Aryl Amination-Hydrolysis-CondensationProcess (2010) (3)
- Synthesis of Chiral N-Aryl-α-amino Acids by Pd-Cu Catalyzed Couplings of Chiral α-Amino Acids with Aryl Halides (1997) (3)
- Accelerating Effect Induced by the Structure of α‐Amino Acid in the Copper‐Catalyzed Coupling Reaction of Aryl Halides with α‐Amino Acids. Synthesis of Benzolactam‐V8. (2010) (3)
- CuI‐Catalyzed Domino Process to 2,3‐Disubstituted Benzofurans from 1‐Bromo‐2‐iodobenzenes and β‐Keto Esters. (2007) (3)
- Total Synthesis of Complex Natural Products via Dearomatization (2016) (3)
- Palladium‐Catalyzed Direct Functionalization of 2‐Aminobutanoic Acid Derivatives: Application of a Convenient and Versatile Auxiliary. (2014) (3)
- Room Temperature Cu-Catalyzed N-Arylation of Oxazolidinones and Amides with (Hetero)Aryl Iodides. (2022) (3)
- Migration of trimethylsilyl groups in enolates of silyl esters (1997) (3)
- Elaboration of the OxazepineRing System via CuI/l-Proline-Catalyzed IntramolecularAryl Amination (2008) (3)
- Synthesis of 7‐Substituted Benzolactam‐V8s and Their Selectivity for Protein Kinase C Isozymes. (2002) (3)
- CuI/4‐Hydro‐L‐proline as a More Effective Catalytic System for Coupling of Aryl Bromides with N‐Boc Hydrazine and Aqueous Ammonia. (2009) (3)
- CuI‐Catalyzed Coupling Reaction of Aryl Halides with Terminal Alkynes in the Absence of Palladium and Phosphine. (2005) (2)
- Facile Access to Polysubstituted Indoles via a Cascade Cu‐Catalyzed Arylation—Condensation Process. (2008) (2)
- Synthesis and biological evaluation of two analogues of (S)-alpha-methyl-3-carboxyphenylalanine. (1998) (2)
- Metal-Catalyzed Derivatization of Cα-Tetrasubstituted Amino Acids and Their Use in the Synthesis of Cyclic Peptides. (2009) (2)
- Asymmetric Strecker‐Type Reaction of α‐Aryl Ketones. Synthesis of (S)‐αM4CPG, (S)‐MPPG, (S)‐AIDA, and (S)‐APICA, the Antagonists of Metabotropic Glutamate Receptors. (1999) (2)
- Cascade Coupling/Cyclization Process to N‐Substituted 1,3‐Dihydrobenzimidazol‐2‐ones. (2008) (2)
- CuI-catalyzed coupling reaction of aryl halides with terminal alkynes in the absence of palladium and phosphine (2004) (2)
- CuI/N,N‐Dimethylglycine‐Catalyzed Synthesis of N‐Aryloxazolidinones from Aryl Bromides. (2012) (2)
- Assembly of α‐(Hetero)aryl Nitriles via Copper‐Catalyzed Coupling Reactions with (Hetero)aryl Chlorides and Bromides (2021) (2)
- CuBr/N,N-Dimethylglycine-Catalyzed Coupling Reaction of 2-Chlorotrifluoroacetanilides with Phenols at Mild Conditions (2010) (2)
- L-Proline Promoted Ullmann-Type Coupling Reactions of Aryl Iodides with Indoles, Pyrroles, Imidazoles or Pyrazoles. (2004) (2)
- The N-aryl aminocarbonyl ortho-substituent effect in Cu-catalyzed aryl amination and its application in the synthesis of 5-substituted 11-oxo-dibenzodiazepines. (2012) (2)
- Synthesis of the benzofuran analogue of ILV, a new protein kinase C(PKC) activator (1994) (2)
- Editorial for the Special Issue on Heterocycles. (2016) (2)
- Highly Convergent Route to Cyclopeptide Alkaloids. Total Synthesis of Ziziphine N. (2007) (2)
- Synthesis of Benzofuran Analogue of Go6976, an Isoform‐Selective Protein Kinase C Inhibitor (2010) (2)
- Iridium Pentahydride Complex Catalyzed Formation of C‐C Bond by C‐H Bond Activation Followed by Olefin Insertion. (1987) (2)
- Transition-metal and organocatalysis in natural product synthesis (2013) (2)
- Divergent Total Syntheses of Napelline-Type C20-Diterpenoid Alkaloids: (-)-Napelline, (+)-Dehydronapelline, (-)-Songorine, (-)-Songoramine, (-)-Acoapetaldine D, and (-)-Liangshanone. (2022) (2)
- Total Synthesis of Salinamide A: A Potent Antiinflammatory Bicyclic Depsipeptide. (2008) (2)
- Effect of alteration of the heterocyclic nucleus of ILV on its isoform selectivity for PKC. Palladium catalyzed route to benzofuran analogues of ILV. (1995) (2)
- The Total Synthesis of ent-Kaurane Diterpenoids (2019) (2)
- Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (—)‐Chimonanthine. (2014) (2)
- Enantioselective Organocatalytic Michael Addition of Malonates to α,β-Unsaturated Aldehydes in Water. (2008) (1)
- Assembly of Conjugated Enynes and Substituted Indoles via CuI/Amino Acid Catalyzed Coupling of 1‐Alkynes with Vinyl Iodides and 2‐Bromotrifluoroacetanilides. (2007) (1)
- Construction of Polycyclic Spiroindolines via an Intramolecular Oxidative Coupling/Cyclization Cascade Reaction Process. (2012) (1)
- Complex Regulation of Proanthocyanidin Biosynthesis in Plants by R2R3 MYB Activators and Repressors (2021) (1)
- Mild and Nonracemizing Conditions for Ullmann‐Type Diaryl Ether Formation Between Aryl Iodides and Tyrosine Derivatives. (2006) (1)
- A Convenient Stereoselective Synthesis of Conjugated Dienoic Esters and Amides. (1990) (1)
- Iridium Pentahydride Complex Catalyzed Dehydrogenation of Alcohols in the Absence of a Hydrogen Acceptor. (1987) (1)
- Assembly of Substituted Homophthalimides via CuI-Catalyzed Coupling of 2-Bromobenzamides with β-Keto Ester. (2009) (1)
- Rhodium‐Catalyzed Regioselective C7‐Functionalization of N‐Pivaloylindoles. (2016) (1)
- Stereocontrolled Cyclopropanation of Garner′s Aldehyde Derived Enones. (2001) (1)
- Synthesis of Tetrahydropyrrolo[1,2-a]quinoxalines and Tetrahydropyrido[1,2-a]quinoxalines via a One-Pot CuI-Catalyzed Aryl Amination—Hydrolysis—Condensation Process. (2011) (1)
- Total Synthesis of the Monoterpenoid Indole Alkaloid (.+-.)-Aspidophylline A. (2014) (1)
- Assembly of Isoquinolines via CuI‐Catalyzed Coupling of β‐Keto Esters and 2‐Halobenzylamines. (2008) (1)
- Selective Conversion of Pinane into β-Pinene Catalyzed by an Iridium Pentahydride Complex. (1987) (1)
- A Novel Small Molecule Regulator of Guanine Nucleotide Exchange Activity of ARF and Golgi Membrane Trafficking (2008) (1)
- L-Proline-Promoted CuI-Catalyzed C—S Bond Formation Between Aryl Iodides and Thiols. (2007) (1)
- Letter to the Editor: 1H, 13C and 15N backbone resonance assignments of matrilysin (MMP7) complexed with a sulfonamide hydroxamate-type inhibitor (2004) (1)
- Clear Evidence for Two Rounds of Vertebrate Genome Duplication (2005) (1)
- N,N-Dimethylglycine-Promoted Ullmann-Type Coupling Reactions of Aryl Iodides with Aliphatic Alcohols. (2007) (1)
- Elaboration of the Oxazepine Ring System via CuI/L‐Proline‐Catalyzed Intramolecular Aryl Amination. (2008) (1)
- Synthesis and Biological Activity of Cyclic Analogues of MPPG and MCPG as Metabotropic Glutamate Receptor Antagonists. (1997) (1)
- An Efficient Synthesis of Phenol via CuI/8‐Hydroxyquinoline‐Catalyzed Hydroxylation of Aryl Halides and Potassium Hydroxide. (2010) (1)
- CuI/Oxalic Diamide Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amines (2016) (1)
- Synthesis of (2‐Arylindol‐3‐yl)acetamides as Probes of Mitochondrial Steroidogenesis. A New Mechanism for GABAA Receptor Modulation. (1992) (1)
- An Efficient and Tunable Route to AG7088, a Rhinovirus Protease Inhibitor. (2005) (1)
- Fibroblast Culture Cells Keep Track of Circadian Rhythms (2005) (1)
- Highly Stereoselective Isomerization of Ynones to Conjugated Dienones Catalyzed by Transition-Metal Complexes. (1989) (1)
- Synthesis of a Cyclic Analogue of Galardin (2010) (1)
- Synthesis of Galbulimima Alkaloid (-)-GB 13 (2006) (1)
- Synthesis of Enantiopure α,α-Disubstituted Amino Acids from the Asymmetric Strecker Reaction Products of Aldehydes. (2000) (1)
- Organocatalytic Michael Addition of Aldehydes to Trisubstituted Nitroolefins. (2013) (1)
- Cascade Annulation of Malonic Diamides: A Concise Synthesis of Polycyclic Pyrroloindolines (2012) (1)
- Synthesis of ortho-Linked Oligo-9,9′-spirobifluorenes (2009) (1)
- General and Stereospecific Route to 9-Substituted, 8,9-Disubstituted, and 9,10-Disubstituted Analogues of Benzolactam-V8. (2000) (1)
- Organocatalytic Michael Addition of Aldehydes to γ-Keto-α,β-Unsaturated Esters. An Efficient Entry to Versatile Chiral Building Blocks. (2009) (1)
- A Scalable Total Synthesis of the Antitumor Agents Et‐743 and Lurbinectedin (2019) (1)
- General Route to 2,4,5‐Trisubstituted Piperidines from Enantiopure β‐Amino Esters. Total Synthesis of Pseudodistomin B Triacetate (X) and Pseudodistomin F (XIII). (2001) (1)
- Cu/ Picolinamides‐Catalyzed Coupling of (Hetero)aryl Halides with Secondary Phosphine Oxides and Phosphite † (2021) (1)
- MicroRNA-939 induces apoptosis in human liver cancer cells by targeting CRKL expression (2020) (0)
- Synthesis of 1,2‐Disubstituted Benzimidazoles by a Cu‐Catalyzed Cascade Aryl Amination/Condensation Process. (2007) (0)
- Sodium Amalgam, a Useful Reducing Reagent for Formation of Amines from Azides Bearing a Variety of Functional Groups. (2006) (0)
- Asymmetric Total Synthesis of (‐)‐Alkaloid 223A (I) and Its 6‐Epimer (II). (2003) (0)
- Total Synthesis of Antimicrobial and Antitumor Cyclic Depsipeptides (2010) (0)
- β‐Amino Ester Route to Tussilagine, Isotussilagine and (‐)‐Petasinecine. (1999) (0)
- Synthesis and Antitumor Activity of Cyclodepsipeptide Zygosporamide (Ia) and Its Analogues. (2008) (0)
- CuI-Catalyzed Coupling of Aryl Iodides with Pinacolborane (2006) (0)
- A Novel Stereoselective Synthesis of Conjugated Dienones. (1988) (0)
- Assembly of N,N-Disubstituted-N′-arylureas via a Copper-Catalyzed One-Pot Three-Component Reaction of Aryl Bromides, Potassium Cyanate, and Secondary Amines. (2013) (0)
- Target Synthesis Directed Methodology Development (2013) (0)
- Regioselective Acylation at the 5- or 6-Position of L-Tryptophan Derivatives. (2010) (0)
- Copper-Catalyzed Coupling of Aryl Iodides and tert-Butyl β-Keto Esters: Efficient Access to α-Aryl Ketones and α-Arylacetic Acid tert-Butyl Esters. (2014) (0)
- CuI/DMPAO‐Catalyzed N‐Arylation of Acyclic Secondary Amines. (2012) (0)
- Synthesis of (-)-Englerin A (2010) (0)
- Asymmetric, Regioselective Bromohydroxylation of 2-Aryl-2-propen-1-ols Catalyzed by Quinine-Derived Catalysts. (2013) (0)
- Stereospecific Synthesis of (1S,3R)-1-Aminocyclopentane-1,3- dicarboxylic Acid, a Selective Agonist of Metabotropic Glutamate Receptors. (1997) (0)
- Synthesis of Enantiopure Substituted Dihydrofurans via the Reaction of (S)-Glyceraldehyde Acetonide- or Garner Aldehyde Acetonide-Derived Enones with Sulfonium Ylides. (2002) (0)
- Enantioselective Organocatalytic Conjugate Addition of Aldehydes to α,β-Unsaturated Thiol Esters. (2010) (0)
- Copper-Catalyzed Asymmetric Synthesis of Dihydropyridines (2007) (0)
- Asymmetric, Protecting-Group-Free Total Synthesis of (-)-Englerin A (I). (2010) (0)
- Synthesis of (-)-Communesin F (2011) (0)
- A Flexible Route to Immunosuppressive Agent FR252921. Asymmetric Total Synthesis of Its (13R,14R,19R)-Isomer. (2007) (0)
- Facile Synthesis of (2E,4E)‐Dienoic Esters (II) via Stereoselective Isomerization of 2‐Ynoic Esters (I). (1989) (0)
- Efficient Entry to Polysubstituted Pyrrolizidines, Indolizidines and Quinolizidines via a Sequential Reaction Process. (2006) (0)
- CuI/L‐Proline‐Catalyzed Coupling of Substituted 3‐Iodoprop‐2‐en‐1‐ols with 1‐Alkynes and Subsequent Cyclization: A Convenient Approach for Synthesizing Polysubstituted Furans. (2010) (0)
- Synthesis of Isoindolin-1-ones via Copper-Catalyzed IntramolecularCyclization (2009) (0)
- Enantioselective Syntheses of Tussilagine and Isotussilagine. (1999) (0)
- Synthesis of (2S,1′R,2′R,3′R)-2-(2′,3′-Dicarboxycyclopropyl)glycine via the Stereochemically Controlled Cyclopropanation of (S)-Glyceraldehyde Acetonide-Derived Enones. (2001) (0)
- Preparation of syn‐δ‐Hydroxy‐β‐amino Esters via an Intramolecular Hydrogen Bond Directed Diastereoselective Hydrogenation. Total Synthesis of (3S,4aS,6R,8S)‐Hyperaspine (I). (2004) (0)
- Pd/Cu-Catalyzed Couplings of β-Amino Esters with Aryl Bromides. Synthesis of Chiral 1,2,3,4-Tetrahydro-4-oxo-2-alkyl-1-quinolines. (1998) (0)
- Total Synthesis of Lepadins B, D, E, and H; Determination of the Configuration of the Latter Three Alkaloids (II). (2004) (0)
- Assembly of Substituted Phenothiazines by a Sequentially Controlled CuI/L-Proline-Catalyzed Cascade C—S and C—N Bond Formation. (2010) (0)
- A Palladium Catalyzed Route to a Benzofuran Analogue of Indolactam V ( ILV): Effects on PKC Isotype Selectivity. (1995) (0)
- Facile Synthesis of 1,4‐Benzodiazepin‐3‐ones from o‐Bromobenzylamines and Amino Acids via Cascade Coupling/Condensation Process. (2010) (0)
- Synthesis of 2-Alkyl-2-arylcyanoacetates via Cul/Sodium Picolinate-Catalyzed Direct Arylation of α-Substituted Cyanoacetates. (2013) (0)
- Synthesis of Symmetrical and Unsymmetrical N,N′‐Diaryl Guanidines via Copper/N‐Methylglycine‐Catalyzed Arylation of Guanidine Nitrate. (2012) (0)
- Achieving Blue Phosphorescence (2007) (0)
- Assembly of 4‐Substituted 3‐Nitro‐1,2,3,4‐tetrahydropyridines via Organocatalytic Michael Addition. (2012) (0)
- Synthesis of Aryl Sulfones via L‐Proline‐Promoted CuI‐Catalyzed Coupling Reaction of Aryl Halides with Sulfinic Acid Salts. (2005) (0)
- Facile Synthesis of (2S,1′S,2′S)-2-(Carboxycyclopropyl)glycine, an Isotype-Selective Agonist of Metabotropic Glutamate Receptors. (1998) (0)
- Enantioselective Addition of Activated Terminal Alkynes to 1‐Acylpyridinium Salts Catalyzed by Cu—Bis(oxazoline) Complexes. (2007) (0)
- A Formal [3 + 2] Cycloaddition Process with Nonactivated Aziridines to Polysubstituted Indolizidines. (2006) (0)
- Synthesis of Salinamide A (2008) (0)
- Assembly of N‐Substituted Pyrrolo[2,1‐c][1,4]benzodiazepine‐5,11‐diones via Copper Catalyzed Aryl Amination. (2010) (0)
- An Improved Procedure to Homochiral Cyclic Statines. (1997) (0)
- Efficient and Economical Access to Substituted Benzothiazoles: Copper‐Catalyzed Coupling of 2‐Haloanilides with Metal Sulfides and Subsequent Condensation. (2009) (0)
- Stereospecific Route to Enantiopure All cis-2,3,6-Trisubstituted Piperidines. Facile Synthesis of (-)-Deoxocassine and (+)-Azimic Acid. (2003) (0)
- Studies on the Synthesis of Biaryl Ether Embodied Cyclopeptides (2007) (0)
- Synthesis of Aryl Carbamates via Copper‐Catalyzed Coupling of Aryl Halides with Potassium Cyanate. (2013) (0)
- Cu/Oxalic Diamide-Catalyzed Coupling of Terminal Alkynes with Aryl Halides. (2023) (0)
- Total Synthesis of Clavepictines A (Ia) and B (Ib) and Pictamine (Ic). (2006) (0)
- Isoform‐Selective Modulators for Metabotropic Glutamate Receptors and Protein Kinase C: Synthesis and Biological Evaluation (1999) (0)
- Domino Condensation/S‐Arylation/Heterocyclization Reactions: Copper‐Catalyzed Three‐Component Synthesis of 2‐N‐Substituted Benzothiazoles. (2011) (0)
- Enantioselective Syntheses of α‐Substituted Glutamic Acids and α,γ‐Disubstituted Glutamic Acids by an Asymmetric Strecker Reaction. (1999) (0)
- Michael Addition of Aldehydes to 2-Amino-1-nitroethenes (2010) (0)
- Facile Synthesis of (+)-α-Allokainic Acid via Pd-Catalyzed Hydrogenolysis of Allyl Acetate Derived from trans-4-Hydroxy-L-proline. (2002) (0)
- Synthesis, Molecular Modeling, 2‐D NMR, and Biological Evaluation of ILV Mimics as Potential Modulators of Protein Kinase C. (1993) (0)
- Recent Progress on the Total Synthesis of Natural Products in China (2007) (0)
- Diastereoselective Synthesis of 2,4,5-Trisubstituted Piperidines from Enantiopure β-Amino Esters. (1999) (0)
- Oxidation of Benzylic Methylene Compounds to Ketones with m-Chloroperoxybenzoic Acid and Oxygen. (2000) (0)
- Palladium-Catalyzed Synthesis of Anellated Indoles. (1992) (0)
- 2‐Methoxyimino Acetic Acid (2016) (0)
- Copper-Catalyzed Enantioselective Arylation of 2-Methylacetoacetates (2007) (0)
- Stereoselective Synthesis of (S)‐(+)‐αM4CPG (XIV), a Selective Antagonist of Metabotropic Glutamate Receptors. (2010) (0)
- Preparation of syn-delta-hydroxy-beta-amino esters via an intramolecular hydrogen bond directed diastereoselective hydrogenation. Total synthesis of (3S,4aS,6R,8S)-hyperaspine. (2003) (0)
- Stereospecific Total Synthesis of (-)-8-epi-Hyperaspine (I). (2004) (0)
- Total Synthesis and Stereochemistry Assignment of 15‐Membered Peptide Alkaloids Abyssenine B (Ia) and Mucronine E (Ib). (2008) (0)
- This Paper Has Been Withdrawn.Highly Convergent Route to Cyclopeptide Alkaloids. Total Synthesis of Ziziphine N (2006) (0)
- SYNTHESIS OF CHIRAL N-ARYL-ALPHA -AMINO ACIDS BY PD-CU CATALYZED COUPLINGSOF CHIRAL ALPHA -AMINO ACIDS WITH ARYL HALIDES (1996) (0)
- Cascade Process from Anilines to Indoles Involving a Copper-Catalyzed Arylation (2008) (0)
- A General and Efficient Approach to Aryl Thiols: CuI‐Catalyzed Coupling of Aryl Iodides with Sulfur and Subsequent Reduction. (2010) (0)
- A Simple and Stereospecific Route to 2,6-Disubstituted 4-Hydroxypiperidines. Synthesis of Dendrobate Alkaloid (+)-241D (XII) and Formal Synthesis of (-)-Indolizidine 167B (XVII). (2000) (0)
- Assembly of Substituted 1H‐Benzimidazoles and 1,3‐Dihydrobenzimidazol‐2‐ones via CuI/L‐Proline Catalyzed Coupling of Aqueous Ammonia with 2‐Iodoacetanilides and 2‐Iodophenylcarbamates. (2010) (0)
- Synthesis of (2S,1′S,2′S)-2-Methyl-2-(carboxycyclopropyl)glycine (XIII) and (S)-2-Amino-2-methyl-4-phosphonobutyric Acid (VII) from L-Alanine. (1997) (0)
- Asymmetric Synthesis of α,α‐Disubstituted Amino Acids by Diastereoselective Functionalization of Enantiopure Phenyloxazinones, Derivatives of Asymmetric Strecker Reaction Products of Aldehydes. (2010) (0)
- Diastereoselective Aldol Reaction of N,N-Dibenzyl-α-amino Aldehydes with Ketones Catalyzed by Proline. (2004) (0)
- Synthesis of Enantiopure N‐Protected 4,5‐Disubstituted 3‐Pyrrolidinones and N‐Protected 2,5‐Disubstituted 3‐Pyrrolidinones via the Dieckmann Reaction of Dicarbonyl Compounds Derived from Enantiopure β‐Amino Esters. (2001) (0)
- A Novel Small Molecule Regulator of Guanine Nucleotide Exchange Activity of ARF and Golgi Membrane Trafficking * 8 / 11 / 2008 (2008) (0)
- A New Methodology to Key Intermediates for Synthesizing Polyene Compounds. (1990) (0)
- Cu-Catalyzed One-Pot Synthesis of 1,2-Disubstituted Benzimidazoles (2007) (0)
- Synthesis and biological activity of l-aminoindan-l,3-dicarboxylic acid, a benzo-analogue of (1S, 3R)-ACPD† (2010) (0)
- Synthesis and Biological Evaluation of 1,3,3,4‐Tetrasubstituted Pyrrolidine CCR5 Receptor Antagonists. Discovery of a Potent and Orally Bioavailable anti‐HIV Agent. (2007) (0)
- CuBr/N,N‐Dimethylglycine‐Catalyzed Coupling Reaction of 2‐Chlorotrifluoroacetanilides with Phenols at Mild Conditions. (2011) (0)
- Efficient Synthesis of Pyrrolo[2,3‐d]pyrimidines via a Cu(I)/6‐Methylpicolinic Acid Catalyzed Coupling Reaction (2015) (0)
- Polyfunctionalized Pyrrolidinones via the Coupling of N,N-Disubstituted β-Amino Esters with Ethyl Glyoxalate. (1998) (0)
- Retraction of "Total Synthesis of Kaitocephalin, the First Naturally Occurring AMPA/KA Receptor Antagonist". (2017) (0)
- A New Three‐Carbon Homologating Agent for Synthesis of γ‐Keto Aldehydes. (1992) (0)
- Synthesis of Zanamivir (2015) (0)
- Facile Entry to Substituted Decahydroquinoline Alkaloids. Total Synthesis of Lepadins A—E and H. (2007) (0)
- Synthesis of (S)‐α‐Cyclopropyl‐4‐phosphonophenylglycine. (2001) (0)
- Synthesis of an Oxazoline Analogue (Ia) of Apratoxin A (Ib). (2004) (0)
- Stereoselective Synthesis of (S)-MPPG, (S)-MTPG, and (S)-(+)-αM4CPG from (R)-4-Hydroxyphenylglycine. (1998) (0)
- Synthesis of (S)-alpha-cyclopropyl-4-phosphonophenylglycine. (2001) (0)
- 2‐((2,6‐Dimethylphenyl)amino)‐2‐oxoacetic Acid (DMPAO) (2016) (0)
- Cu-Catalyzed Coupling Reactions of Sulfonamides with (Hetero)Aryl Chlorides/Bromides. (2022) (0)
- Facile Synthesis of 1,4‐Diketones via Palladium Complex‐Catalyzed Isomerization of Alkynediols. (1992) (0)
- Stereochemically Controlled Cyclopropanation of (S)-Glyceraldehyde Acetonide-Derived Olefins. Synthesis of (2S,1′R,2′R,3′R)-2-(2′,3′-Dicarboxycyclopropyl)glycine. (1999) (0)
- Total Synthesis of Kopsinitarine E (2020) (0)
- Synthetic Studies Toward Two Marine Cyclic Peptides (2005) (0)
- CuI/N,N-Dimethylglycine-Catalyzed Cross-Coupling Reaction of Vinyl Halides with Phenols and Its Application to the Assembly of Substituted Benzofurans. (2005) (0)
- Ligand-Promoted Rosenmund–von Braun Reaction (2022) (0)
- Organocatalytic Approach to 3,5,6‐Trisubstituted and 4,6‐Disubstituted Tetrahydropyran‐2‐ones. (2010) (0)
- Synthesis and Biological Evaluation of Two Analogues of (S)‐α‐Methyl‐3‐carboxyphenylalanine. (1999) (0)
- The Molting Worm Sheds Its Genetic Secrets (2005) (0)
- Synthesis of Polysubstituted 1,2‐Dihydroisoquinolines via a CuI‐Catalyzed Arylation/Condensation Cascade Process. (2009) (0)
- Total Synthesis of (.+‐.)‐Martinelline. (2003) (0)
- A Novel Approach to Predicting Interactions Between Microbes and Hosts (2021) (0)
- A Global View of DNA-Packing Proteins Cracks the Histone Code (2005) (0)
- Comparing Gene Trees and Genome Trees: A Cobweb of Life? (2005) (0)
- Structure—Activity Relationship Studies of Salubrinal Lead to Its Active Biotinylated Derivative. (2005) (0)
- Structure-assisted design of inhibitors targeting coronavirus main proteases (2005) (0)
- CCDC 765298: Experimental Crystal Structure Determination (2010) (0)
- Synthesis of 1,5‐Benzothiazepine Dipeptide Mimetics via Two CuI‐Catalyzed Cross Coupling Reactions. (2009) (0)
- Stereospecific Synthesis of 9-Substituted Benzolactam-V8 from L-Tyrosine via Regioselective Aromatic Nitration. (1998) (0)
- Isomerization of Proparglyic Alcohols Catalyzed by an Iridium Complex. (1989) (0)
- Enantioselective Synthesis of Functionalized α-Amino Acids via a Chiral Guanidine Catalyzed Michael Addition Reaction. (1999) (0)
- Casting a Wide Net to Fight Coronaviruses (2005) (0)
- Title : Transcriptional control of proanthocyanidin synthesis 2 3 4 5 Corresponding (2017) (0)
- Field Tested: Grasslands Won’t Help Buffer Climate Change as CO2 Levels Rise (2005) (0)
- Discovery Kinase Inhibitors Downregulate Ther T 3 Tyr 705 Phosphorylation (2010) (0)
- Complex Cells in the Brain's Vision Center Tune in to Natural Scenes (2005) (0)
- Clues to the Evolution of the Malarial Chromosome (2005) (0)
- Mapping Core Communication Networks in Bacteria (2005) (0)
- A Signaling Pathway at the Heart of Muscle Development (2005) (0)
- Functional characterization of R2R3-MYB activators and repressors as flavonoid transcriptional regulators in poplar (2019) (0)
- A Simple Route to α,β‐Unsaturated Aldehydes from Prop‐2‐ynols. (1989) (0)
- Abstract SY36-03: Development of small-molecule inhibitors of autophagy as anticancer therapy (2012) (0)
- Small molecule “on” and “off” switches for autophagy (2012) (0)
- ENANTIOSELECTIVE SYNTHESES OF ALPHA -SUBSTITUTED GLUTAMIC ACIDS AND ALPHA , GAMMA -DISUBSTITUTED GLUTAMIC ACIDS BY AN ASYMMETRIC STRECKER REACTION (1999) (0)
- A Convenient Synthesis of 3-(1,3-Alkadienyl)-2-cycloalken-1-ones. (1990) (0)
- Copper/l-Proline-CatalyzedSynthesis of Phenothiazines (2010) (0)
- Aromatic Nucleophilic Substitution or CuI‐Catalyzed Coupling Route to Martinellic Acid. (2003) (0)
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What Schools Are Affiliated With Dawei Ma?
Dawei Ma is affiliated with the following schools:
- University of California, Berkeley
- Harbin Institute of Technology
- East China University of Science and Technology
- University of Alberta
- University of Michigan
- China Pharmaceutical University
- Tsinghua University
- University of Toronto
- Shanghai University
- University of the Chinese Academy of Sciences
- Shenyang Pharmaceutical University
- University of Victoria
- Howard University
- Stanford University
- Georgetown University
- Fudan University
- Harvard University
