Gary H. Posner
#56,057
Most Influential Person Now
American chemist
Gary H. Posner's AcademicInfluence.com Rankings
Gary H. Posnerchemistry Degrees
Chemistry
#654
World Rank
#1114
Historical Rank
#292
USA Rank
Organic Chemistry
#111
World Rank
#147
Historical Rank
#44
USA Rank
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Chemistry
Gary H. Posner's Degrees
- PhD Chemistry University of California, Berkeley
- Bachelors Chemistry University of California, Berkeley
Why Is Gary H. Posner Influential?
(Suggest an Edit or Addition)According to Wikipedia, Gary H. Posner was Scowe Professor of Chemistry at Johns Hopkins University in Baltimore, Maryland. Posner is known for his pioneering research in organocopper chemistry, including his involvement in the development of the Corey–House–Posner–Whitesides reaction.
Gary H. Posner's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- A major inducer of anticarcinogenic protective enzymes from broccoli: isolation and elucidation of structure. (1992) (1593)
- Anticarcinogenic activities of sulforaphane and structurally related synthetic norbornyl isothiocyanates. (1994) (703)
- A medicinal chemistry perspective on artemisinin and related endoperoxides. (2004) (422)
- Multicomponent one-pot annulations forming 3 to 6 bonds (1986) (391)
- Organic Reactions at Alumina Surfaces (1978) (257)
- Diels-Alder cycloadditions of 2-pyrones and 2-pyridones (1993) (215)
- Organic reactions at alumina surfaces. Mild and selective opening of epoxides by alcohols, thiols, benzeneselenol, amines, and acetic acid (1977) (207)
- Antimalarial activity of artemisinin (qinghaosu) and related trioxanes: mechanism(s) of action. (1997) (202)
- New stereospecific synthesis of trisubstituted olefins. Stereospecific synthesis of farnesol (1967) (193)
- Knowledge of the proposed chemical mechanism of action and cytochrome p450 metabolism of antimalarial trioxanes like artemisinin allows rational design of new antimalarial peroxides. (2004) (186)
- Selective formation of carbon-carbon bonds between unlike groups using organocopper reagents (1967) (186)
- New class of mixed cuprate(I) reagents, lithium hetero(alkyl) cuprate(I), which allow selective alkyl group transfer (1973) (176)
- A convenient, one-step, high-yield replacement of an anomeric hydroxyl group by a fluorine atom using dast. Preparation of glycosyl fluorides. (1985) (160)
- An Introduction to Synthesis Using Organocopper Reagents (1980) (158)
- Mechanism-based design, synthesis, and in vitro antimalarial testing of new 4-methylated trioxanes structurally related to artemisinin: the importance of a carbon-centered radical for antimalarial activity. (1994) (154)
- Regiospecifically oxygen-18 labeled 1,2,4-trioxane: a simple chemical model system to probe the mechanism(s) for the antimalarial activity of artemisinin (qinghaosu). (1992) (151)
- Design and synthesis of bifunctional isothiocyanate analogs of sulforaphane: correlation between structure and potency as inducers of anticarcinogenic detoxication enzymes. (1994) (145)
- Spectroscopic quantitation of organic isothiocyanates by cyclocondensation with vicinal dithiols. (1992) (140)
- Accumulation of artemisinin trioxane derivatives within neutral lipids of Plasmodium falciparum malaria parasites is endoperoxide-dependent. (2009) (138)
- Orally active, antimalarial, anticancer, artemisinin-derived trioxane dimers with high stability and efficacy. (2003) (136)
- Evidence for Fe(IV):O in the Molecular Mechanism of Action of the Trioxane Antimalarial Artemisinin (1995) (135)
- Vitamin D and vitamin D analogs as cancer chemopreventive agents. (2003) (131)
- Carbon-carbon bond formation by selective coupling of n-alkylcopper reagents with organic halides (1968) (125)
- Asymmetric synthesis of carbon-carbon bonds using sulfinyl cycloalkenones, alkenolides, and pyrones (1987) (120)
- Antimalarial, antiproliferative, and antitumor activities of artemisinin-derived, chemically robust, trioxane dimers. (1999) (119)
- Further evidence supporting the importance of and the restrictions on a carbon-centered radical for high antimalarial activity of 1,2,4-trioxanes like artemisinin. (1995) (116)
- Anticancer and antimalarial efficacy and safety of artemisinin-derived trioxane dimers in rodents. (2004) (112)
- Cancer chemoprevention using natural vitamin D and synthetic analogs. (2003) (111)
- 1,25-Dihydroxyvitamin D and three low-calcemic analogs decrease UV-induced DNA damage via the rapid response pathway (2004) (105)
- Second generation, orally active, antimalarial, artemisinin-derived trioxane dimers with high stability, efficacy, and anticancer activity. (2006) (105)
- Alkylation of enolate ions generated regiospecifically via organocopper reactions. Synthesis of decalin sesquiterpene valerane and of prostaglandin model systems. (1975) (104)
- Antimalarial chemotherapeutic peroxides: artemisinin, yingzhaosu A and related compounds. (2002) (102)
- Physiological Importance of the 1,25(OH)2D3 Membrane Receptor and Evidence for a Membrane Receptor Specific for 24,25(OH)2D3 (1999) (101)
- Extraordinarily potent antimalarial compounds: new, structurally simple, easily synthesized, tricyclic 1,2,4-trioxanes. (1992) (98)
- Antimalarial peroxides: advances in drug discovery and design (2012) (97)
- Organocopper chemistry. Halo-, cyano-, and carbonyl-substituted ketones from the corresponding acyl chlorides and organocopper reagents (1972) (97)
- Antimalarial and antitumor evaluation of novel C-10 non-acetal dimers of 10beta-(2-hydroxyethyl)deoxoartemisinin. (2004) (94)
- In Vitro Inhibition of Toxoplasma gondii by Four New Derivatives of Artemisinin (2006) (91)
- Effect of artemisinins and other endoperoxides on nitric oxide-related signaling pathway in RAW 264.7 mouse macrophage cells. (2008) (87)
- 1,25-(OH)2D3 modulates growth plate chondrocytes via membrane receptor-mediated protein kinase C by a mechanism that involves changes in phospholipid metabolism and the action of arachidonic acid and PGE2 (1999) (87)
- Potent, Selective and Low-Calcemic Inhibitors of CYP24 Hydroxylase: 24-Sulfoximine Analogues of the Hormone 1α,25-Dihydroxyvitamin D3 (2004) (87)
- A directing effect of neighboring aromatic groups on the regiochemistry of formation and stereochemistry of alkylation and bromination of ketone lithium enolates. Evidence for lithium-arene coordination and dramatic effect of copper(I) in controlling stereochemistry and limiting polyalkylation (1979) (84)
- Second-generation antimalarial endoperoxides. (1996) (81)
- Orally active, hydrolytically stable, semisynthetic, antimalarial trioxanes in the artemisinin family. (1999) (79)
- Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin. (2001) (78)
- Organic Chemistry of Vitamin D Analogues (Deltanoids) (2003) (72)
- EVIDENCE FOR THE IMPORTANCE OF HIGH-VALENT FE=O AND OF A DIKETONE IN THE MOLECULAR MECHANISM OF ACTION OF ANTIMALARIAL TRIOXANE ANALOGS OF ARTEMISININ (1996) (71)
- Organic reactions at alumina surfaces. 6. Isopropyl alcohol and diisopropylcarbinol on dehydrated alumina as reagents for very selective carbonyl reductions (1977) (69)
- Artemisinin derivatives inhibit Toxoplasma gondii in vitro at multiple steps in the lytic cycle. (2009) (69)
- Lewis Acid-Promoted, Stereocontrolled, Gram Scale, Diels-Alder Cycloadditions of Electronically Matched 2-Pyrones and Vinyl Ethers: The Critical Importance of Molecular Sieves and the Temperature of Titanium Coordination with the Pyrone. (1996) (69)
- Vitamin D3 analogs stimulate calcium currents in rat osteosarcoma cells. (1994) (68)
- Malaria-infected mice are cured by a single oral dose of new dimeric trioxane sulfones which are also selectively and powerfully cytotoxic to cancer cells. (2009) (67)
- High asymmetric induction during organometallic .beta.-addition to .alpha.,.beta.-ethylenic sulfoxides. Synthesis of optically active .beta.-alkylcarboxylic acids, .beta.-substituted cyclopentanones, and steroidal 11-oxoequilenin methyl ether (1981) (67)
- Asymmetric induction during organometallic conjugate addition to enantiomerically pure 2-(arylsulfinyl)-2-cyclopentenones (1982) (67)
- Organic reactions at alumina surfaces. Mild and selective opening of arene and related oxides by weak oxygen and nitrogen nucleophiles (1977) (67)
- A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides. (2003) (65)
- Total synthesis of natural estrone and estradiol methyl ethers in extremely high enantiomeric purity via an asymmetric Michael addition to an unsaturated sulfoxide (1986) (65)
- Noncalcemic, antiproliferative, transcriptionally active, 24-fluorinated hybrid analogues of the hormone 1alpha, 25-dihydroxyvitamin D3. Synthesis and preliminary biological evaluation. (1998) (64)
- Thiazole, oxadiazole, and carboxamide derivatives of artemisinin are highly selective and potent inhibitors of Toxoplasma gondii. (2010) (62)
- Synthetic Approaches to Vitamin D (2010) (62)
- Effects of the sulforaphane analog compound 30, indole-3-carbinol, D-limonene or relafen on glutathione S-transferases and glutathione peroxidase of the rat digestive tract. (1998) (61)
- A Medicinal Chemistry Perspective on Artemisinin and Related Endoperoxides (2004) (59)
- An Artemisinin-Derived Dimer Has Highly Potent Anti-Cytomegalovirus (CMV) and Anti-Cancer Activities (2011) (58)
- Malaria-infected mice are cured by a single dose of novel artemisinin derivatives. (2007) (57)
- New vitamin D3 derivatives with unexpected antiproliferative activity: 1-(hydroxymethyl)-25-hydroxyvitamin D3 homologs. (1992) (57)
- Antiproliferative Hybrid Analogs of the Hormone 1alpha,25-Dihydroxyvitamin D(3): Design, Synthesis, and Preliminary Biological Evaluation. (1997) (57)
- Estrogenic activity of glabridin and glabrene from licorice roots on human osteoblasts and prepubertal rat skeletal tissues (2004) (57)
- Asymmetric total synthesis of an A-ring precursor to hormonally active 1.alpha.,25-dihydroxyvitamin D3 (1990) (57)
- Reaction of .alpha.,.alpha.'-dibromo ketones with organocopper reagents. New method for .alpha. alkylation of ketones (1973) (56)
- Conceptually new deltanoids (vitamin D analogs) inhibit multistage skin tumorigenesis. (2000) (55)
- Biological mechanisms of action of novel C-10 non-acetal trioxane dimers in prostate cancer cell lines. (2006) (54)
- Highly stereocontrolled synthesis of some trioxygenated cyclohexenes: an asymmetric total synthesis of (-)-methyl triacetyl-4-epishikimate (1986) (53)
- Stereocontrolled preparation of chiral (E)-1-alkenyl sulfoxides. Efficient reduction of alkenyl sulfoxides to the corresponding alkenyl sulfides (1978) (52)
- Enantiomeric 1,2,4‐Trioxanes Display Equivalent in vitro Antimalarial Activity Versus Plasmodium falciparum Malaria Parasites: Implications for the Molecular Mechanism of Action of the Artemisinins (2005) (52)
- Reaction of .alpha.,.beta.-ethylenic sulfur compounds with organocopper reagents (1973) (52)
- Artemisinin-Derived Dimers Have Greatly Improved Anti-Cytomegalovirus Activity Compared to Artemisinin Monomers (2010) (52)
- Orally active antimalarial 3-substituted trioxanes: new synthetic methodology and biological evaluation. (1998) (51)
- Phenoxide-directed ortho lithiation (1985) (50)
- In Vitro Combination of Anti-Cytomegalovirus Compounds Acting through Different Targets: Role of the Slope Parameter and Insights into Mechanisms of Action (2013) (50)
- Asymmetric Michael additions of ester enolates to enantiomerically pure vinylic sulfoxides: synthesis of 3-substituted glutarate esters in high enantiomeric purity (1986) (50)
- Organic reactions at alumina surfaces. An extremely simple, convenient and selective method for acetylating primary alcohols in the presence of secondary alcohols. (1981) (49)
- Conversion of glycosyl fluorides into C-glycosides using organoaluminum reagents. Stereospecific alkylation at C-6 of a pyranose sugar (1985) (49)
- Design, synthesis, derivatization, and structure-activity relationships of simplified, tricyclic, 1,2,4-trioxane alcohol analogues of the antimalarial artemisinin. (1998) (49)
- Diels-Alder cycloadditions using nucleophilic 3-(p-tolylthio)-2-pyrone. Regiocontrolled and stereocontrolled synthesis of unsaturated, bridged, bicyclic lactones (1992) (47)
- Antimalarial cyclic peroxy ketals. (1998) (47)
- Highly stereocontrolled synthesis of some polyfunctionalized cyclohexenes. A short formal total synthesis of (±)-chorismic acid (1987) (47)
- 5-Bromo-2-pyrone: An easily prepared ambiphilic diene and a synthetic equivalent of 2-pyrone in mild, thermal, Diels-Alder cycloadditions (1992) (46)
- Apc(MIN) modulation of vitamin D secosteroid growth control. (2010) (46)
- Differential use of transcription activation function 2 domain of the vitamin D receptor by 1,25-dihydroxyvitamin D3 and its A ring-modified analogs. (1998) (46)
- Structure-activity relationships of lactone ring-opened analogs of the antimalarial 1,2,4-trioxane artemisinin. (1995) (45)
- Enantiocontrolled synthesis of quaternary carbon centers. 3,3-disubstituted cyclopentanones. (+)-α-cuparenone (1984) (45)
- Asymmetric Diels-Alder cycloadditions using chiral alkyl vinyl ethers and a dienyl sulfone (1986) (44)
- Malaria-infected mice are cured by oral administration of new artemisinin derivatives. (2008) (44)
- Vitamin D analogues targeting CYP24 in chronic kidney disease (2010) (43)
- Trioxane dimers have potent antimalarial, antiproliferative and antitumor activities in vitro. (1997) (43)
- Synthesis and antimalarial activity of heteroatom-containing bicyclic endoperoxides (1997) (43)
- .alpha.,.beta.-Ethylenic sulfones from sulfonomethylphosphonate carbanions and aldehydes and ketones (1972) (43)
- Vitamin D metabolites and analogs induce lipoxygenase mRNA expression and activity as well as reactive oxygen species (ROS) production in human bone cell line (2011) (42)
- Mechanism-based design of simple, symmetrical, easily prepared, potent antimalarial endoperoxides (1996) (42)
- BF3.OEt2 promotes fast, mild, clean and regioselective dehydration of tertiary alcohols (1991) (42)
- One-pot, four-component annulations: flexible and simple syntheses of unsaturated macrolides and of substituted aromatics and heteroaromatics (1988) (42)
- Antimalarial simplified 3-aryltrioxanes: synthesis and preclinical efficacy/toxicity testing in rodents. (2001) (41)
- Direct and Convenient Preparation of Lithium Phenylthio(alkyl)cuprate Reagents (1974) (41)
- New chemical and biological aspects of artemisinin-derived trioxane dimers. (2002) (41)
- 3-bromo-2-pyrone: an easily prepared chameleon diene and a synthetic equivalent of 2-pyrone in thermal diels-alder cycloadditions (1991) (40)
- Synthesis and antimalarial efficacy of two-carbon-linked, artemisinin-derived trioxane dimers in combination with known antimalarial drugs. (2013) (40)
- Potent, low-calcemic, selective inhibitors of CYP24 hydroxylase: 24-sulfone analogs of the hormone 1α,25-dihydroxyvitamin D3 (2004) (39)
- A short, asymmetric synthesis of natural (-)-methyl jasmonate (1985) (39)
- An efficient method for dibromomethylenation and isopropylidenation of ketones (). Synthesis of a selinadiene sesquiterpene. (1975) (38)
- Stereocontrolled total synthesis of an .alpha.-methylene guaianolide in the 4,5-epoxyosmitopsin family (1980) (38)
- S)-(+)-2-(p-tolylsulfinyl)-2-buten-4-olide: an enantiomerically pure Michael acceptor for asymmetric synthesis of 3-substituted 4-butanolides. (—)-podorhizon. (1984) (38)
- Formation of olefins via pyrolysis of sulfonate esters (1989) (38)
- A Thiazole Derivative of Artemisinin Moderately Reduces Toxoplasma gondii Cyst Burden in Infected Mice (2014) (37)
- Antimalarial sulfone trioxanes (1998) (37)
- Methyl and -alkyl ketones from carboxylic acid chlorides and organocopper reagents (1970) (37)
- A CARBONYL OXIDE ROUTE TO ANTIMALARIAL YINGZHAOSU A ANALOGUES : SYNTHESIS AND ANTIMALARIAL ACTIVITY (1998) (37)
- Asymmetric synthesis using enantiomerically pure 2-(p-anisylsulfinyl)-2-cycloalkenones (1984) (37)
- Anticancer activity of artemisinin-derived trioxanes (2006) (37)
- Recombinant luciferase-expressing human cytomegalovirus (CMV) for evaluation of CMV inhibitors (2011) (36)
- Tandem michael-michael-ring closure (mimirc) reactions: One-pot steroid total synthesis-(±)-9,11-dehydroestrones (1981) (36)
- Enantiocontrolled synthesis of (S)-3-substituted cycloalkanones from (s)-2-(p-tolylsulfinyl)-2-cycloalkenones and diorganomagnesium reagents. (1984) (36)
- Cyanocuprates convert carboxylic acids directly into ketones. (2011) (36)
- Photochemical deoxygenation of aryl sulfoxides (1973) (36)
- Inhibition of Human Cytomegalovirus Replication by Artemisinins: Effects Mediated through Cell Cycle Modulation (2015) (35)
- Olefin oxidative cleavage and dioxetane formation using triethylsilyl hydrotrioxide: Applications to preparation of potent antimalarial 1,2,4-trioxanes (1991) (35)
- Synthesis and in vitro antimalarial activity of sulfone endoperoxides. (1998) (35)
- A Rationale for Treatment of Hereditary Vitamin D-resistant Rickets with Analogs of 1α,25-Dihydroxyvitamin D3 * (2001) (35)
- Artemisinin-Derived Dimer Diphenyl Phosphate Is an Irreversible Inhibitor of Human Cytomegalovirus Replication (2012) (34)
- Orally active, water-soluble antimalarial 3-aryltrioxanes: short synthesis and preclinical efficacy testing in rodents. (2002) (34)
- Mild, asymmetric Diels-Alder cycloadditions of electronically matched 2-pyrones and vinyl ethers (1994) (34)
- An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes (2002) (34)
- Three-component, one-flask synthesis of rhodanines (thiazolidinones). (2011) (33)
- An asymmetric total synthesis of fragrant spiro[4.5]decane sesquiterpene (-)-.beta.-vetivone via an enantiomerically pure vinylic sulfoxide (1988) (33)
- Artemisinin-derived dimer phosphate esters as potent anti-cytomegalovirus (anti-CMV) and anti-cancer agents: a structure-activity study. (2013) (32)
- Short, simple, stereocontrolled, steroid synthesis: (.+-.)-11-oxoequilenin methyl ether and a new 9,11-seco-13-ethyl steroid (1979) (32)
- 2-Fluoroalkyl A-Ring Analogs of 1,25-Dihydroxyvitamin D3. Stereocontrolled Total Synthesis via Intramolecular and Intermolecular Diels-Alder Cycloadditions. Preliminary Biological Testing (1995) (32)
- Antimalarial sulfide, sulfone, and sulfonamide trioxanes. (2000) (32)
- Complete Asymmetric Induction in Synthesis of Enantiomerically Pure Steroid Intermediates of Natural Configuration (1981) (32)
- Vitamin D receptor modulates the neoplastic phenotype through antagonistic growth regulatory signals (2009) (32)
- A 20‐epi side chain restores growth‐regulatory and transcriptional activities of an A ring‐modified hybrid analog of 1α,25‐dihydroxyvitamin D3 without increasing its affinity to the vitamin D receptor (1996) (32)
- Antimalarial artemisinin analogs. Synthesis via chemoselective CC bond formation and preliminary biological evaluation (1999) (32)
- Titanium-promoted stereoselective synthesis of hydroindolones from p-quinamines by domino conjugate additions. (2002) (31)
- A chemiluminescent probe specific for singlet oxygen. (1984) (31)
- Diels-Alder cycloadditions using nucleophilic 2-pyridones. Regiocontrolled and stereocontrolled synthesis of unsaturated, bridged, bicyclic lactams (1992) (31)
- Stereocontrolled synthesis of highly functionalized cyclohexenes. A short synthesis of a chorismic acid precursor (1990) (31)
- Membranal effects of phytoestrogens and carboxy derivatives of phytoestrogens on human vascular and bone cells: New insights based on studies with carboxy-biochanin A (2005) (30)
- Stereocontrolled Total Synthesis of Calcitriol Derivatives: 1,25-Dihydroxy-2-(4'-hydroxybutyl)vitamin D3 Analogs of an Osteoporosis Drug (1994) (30)
- Vitamin D side chain triazole analogs via cycloaddition `click' chemistry (2004) (30)
- Conceptually new sulfone analogues of the hormone 1alpha, 25-dihydroxyvitamin D(3): synthesis and preliminary biological evaluation. (1999) (30)
- Low-calcemic, efficacious, 1α,25-dihydroxyvitamin D3 analog QW-1624F2-2: calcemic dose–response determination, preclinical genotoxicity testing, and revision of A-ring stereochemistry (2004) (30)
- A new and efficient asymmetric synthesis of an A-ring precursor to physiologically active 1.alpha.-hydroxyvitamin D3 steroids (1992) (29)
- Sequential Michael-Michael-aldol additions for easy, one-pot, 2 + 2 + 2 construction of polyfunctionalized cyclohexanols. (1986) (29)
- Malaria-infected mice live until at least day 30 after a new monomeric trioxane combined with mefloquine are administered together in a single low oral dose. (2009) (29)
- 3-Cuprio-2-pyrone: an extraordinary organocopper reagent (1985) (29)
- A study of cross coupling reactions between halides and anionic manganese, iron, and cobalt alkyls (1970) (28)
- Unique and Highly Selective Anticytomegalovirus Activities of Artemisinin-Derived Dimer Diphenyl Phosphate Stem from Combination of Dimer Unit and a Diphenyl Phosphate Moiety (2013) (28)
- New silicon-mediated, sequential ring expansions of n-sized 2-cycloalkenones into hydroxyolefinic n + m + p medium-sized lactones: short synthesis of (-)-phoracantholide-J. (2005) (28)
- Direct conversion of pyranose anomeric OH→F→R in the artemisinin family of antimalarial trioxanes (1998) (28)
- Chemiluminescence mechanism and quantum yield of synthetic vinylpyrene analogues of benzo[a]pyrene-7,8-dihydrobiol (1986) (28)
- Organic reactions at alumina surfaces. Displacement reactions effected by alcohols, thiols, and acetic acid on dehydrated alumina. (1975) (28)
- Biological effects of 1alpha-hydroxy- and 1beta-(hydroxymethyl)-vitamin D compounds relevant for potential colorectal cancer therapy. (1999) (28)
- Anticancer effects of the novel 1α, 25‐dihydroxyvitamin D3 hybrid analog QW1624F2‐2 in human neuroblastoma (2006) (28)
- 1 alpha,25-dihydroxyvitamin D3 analogs featuring aromatic and heteroaromatic rings: design, synthesis, and preliminary biological testing. (1995) (27)
- Substitution and conjugate addition reactions using new lithium -butoxy-alkylcuprate(I) reagents (1973) (27)
- Additive Pummerer rearrangements. Asymmetric synthesis of (–)-methyl jasmonate (1985) (27)
- Antimalarially potent, easily prepared, fluorinated endoperoxides (1996) (27)
- Interrupted polymerization of acrylates: sequential Michael-Michael-Dieckmann cyclizations for easy, one-pot, 2 + 2 + 2 construction of polyfunctionalized cyclohexanones (1989) (27)
- [3,3]-sigmatropic rearrangements: short, stereocontrolled syntheses of functionalized vitamin D3 side-chain units (2002) (26)
- Malaria-infected mice are completely cured by one 6 mg/kg oral dose of a new monomeric trioxane sulfide combined with mefloquine. (2012) (26)
- Artemisinin-derived dimer ART-838 potently inhibited human acute leukemias, persisted in vivo, and synergized with antileukemic drugs (2016) (26)
- An extremely efficient method for one-pot, three-component, 2+2+2 construction of functionalized cyclohexenes (1985) (26)
- Organic reactions at alumina surfaces. A mechanistic and synthetic study of sulfonate ester elimination reactions effected by chromatographic alumina (1977) (25)
- Antimalarial peroxides in the qinghaosu (artemisinin) and yingzhaosu families (1998) (25)
- A mechanistic and synthetic study of organocopper substitution reactions with some homoallylic and cyclopropylcarbinyl substrates : Application to isoprenoid synthesis (1976) (24)
- Synthesis and antimalarial activities of structurally simplified 1,2,4‐trioxanes related to artemisinin (1995) (24)
- Stereocontrolled synthesis of a trihydroxylated A ring as an immediate precursor to 1.alpha.,2.alpha.,25-trihydroxyvitamin D3 (1991) (24)
- 2,2-Disubstituted analogues of the natural hormone 1α,25-dihydroxyvitamin D3: Chemistry and biology (2002) (24)
- Iron(II)-induced degradation of antimalarial beta-sulfonyl endoperoxides: evidence for the generation of potentially cytotoxic carbocations. (2001) (24)
- One-flask, regiospecific conversions of allylic alcohols into 2-carbon-extended, conjugated dienoate esters. Use of a new sulfinyl orthoester (1991) (24)
- Asymmetric, organocatalytic, three-step synthesis of alpha-hydroxy-(E)-beta,gamma-unsaturated esters. (2010) (23)
- Potent, selective and low-calcemic inhibitors of CYP24 hydroxylase: 24-sulfoximine analogues of the hormone 1alpha,25-dihydroxyvitamin D(3). (2004) (23)
- 1-(hydroxyalkyl)-25-hydroxyvitamin D3 analogs of calcitriol. 1. Synthesis (1993) (23)
- Cyclopentanone ring expansion leading to functionalized delta-lactams: short synthesis of simple sedum alkaloids. (2007) (23)
- Mild, fast, and stereoselective epoxide opening by ketone enolate anions. Application to synthesis of the norlignan curculigine. (2003) (23)
- Vitamin D analogs as anti-carcinogenic agents. (2006) (23)
- A new synthetic approach to pseudoguaianes. (1978) (23)
- A‐ring analogues of 1,25‐(OH)2D3 with low affinity for the vitamin D receptor modulate chondrocytes via membrane effects that are dependent on cell maturation (1997) (23)
- Enantiocontrolled Synthesis of (R)-3-Substituted Cyclohexanones Using (S)-2-(p-Tolylsulfinyl)-2-cyclohexenone and Various Organometallic Reagents in 2,5-Dimethyltetrahydrofuran (1984) (22)
- Asymmetric synthesis using organometallic reagents and optically pure vinylic sulfoxides (1981) (22)
- A non-calcemic sulfone version of the vitamin D(3) analogue seocalcitol (EB 1089): chemical synthesis, biological evaluation and potency enhancement of the anticancer drug adriamycin. (2001) (22)
- Antitumor Effects of Two Less-Calcemic Vitamin D Analogs (Paricalcitol and QW-1624F2-2) in Squamous Cell Carcinoma Cells (2007) (21)
- One-flask, consecutive [3,3]- and [2,3]-sigmatropic rearrangements for conversions of propargylic alcohols into 2-carbon-extended 4-oxo-2-alkenoate esters. Use of a new 1-chloro-1-ethoxy-2-sulfinylethylene (1991) (21)
- Alkylation of enolate ions generated regiospecifically via organocopper conjugate addition reactions. Synthesis of decalin sesquiterpene valerane and of a prostaglandin model system (1974) (20)
- Treatment with non-hypercalcemic analogs of 1,25-dihydroxyvitamin D3 increases responsiveness to 17β-estradiol, dihydrotestosterone or raloxifene in primary human osteoblasts (2004) (20)
- Malaria: new chemotherapeutic peroxide drugs. (2002) (20)
- Asymmetric total synthesis, x-ray crystallography, and preliminary biological evaluation of 1-(1'-hydroxyethyl)-25-hydroxyvitamin D3 analogs of natural calcitriol (1993) (20)
- A single, low, oral dose of a 5-carbon-linked trioxane dimer orthoester plus mefloquine cures malaria-infected mice. (2011) (20)
- Reaction of lithium dialkylcuprates with β-alkoxy and β-alkylthio αβ-unsaturated carbonyl compounds (1973) (20)
- 8 – Addition of Organometallic Reagents to Chiral Vinylic Sulfoxides (1983) (19)
- Nitroolefins in one-flask, tandem. A+B+C coupling reactions producing heterocycles (1990) (19)
- Generation and reactions of 1-(arylsulfinyl)alkenyllithium reagents. Terminal allenes from 2-alkenyl aryl sulfoxides. (1978) (19)
- A one-flask multicomponent annulation reaction as the key step in a total synthesis of spirobicyclic (±)-β-vetivone (1992) (19)
- A 24-Phenylsulfone Analog of Vitamin D Inhibits 1α,25-Dihydroxyvitamin D3 Degradation in Vitamin D Metabolism-Competent Cells (2007) (19)
- Asymmetric, organocatalytic, three-step synthesis of gamma-hydroxy-(E)-alpha,beta-unsaturated sulfones and esters. (2008) (19)
- Binaphthol-titanium-promoted, highly enantiocontrolled, Diels-Alder cycloadditions of electronically matched 2-pyrones and vinyl ethers: Streamlined asymmetric synthesis of an A-ring precursor to physiologically active 1α-hydroxyvitamin D3 steroids (1994) (19)
- Lewis acid-catalyzed, high pressure, stereospecific, regiospecific, Diels-Alder cycloaddition of unsubstituted 2-pyrone: Short synthesis of a racemic A-ring precursor to physiologically active 1-hydroxyvitamin D3 steroids (1994) (19)
- Antimalarial chemotherapy: artemisinin-derived dimer carbonates and thiocarbonates. (2014) (18)
- AN IMPROVED PREPARATION OF 3-BROMO-2(H)-PYRAN-2-ONE : AN AMBIPHILIC DIENE FOR DIELS-ALDER CYCLOADDITIONS : (2H-PYRAN-2-ONE, 3-BROMO-) (1996) (18)
- Vitamin D analogs as modulators of vitamin D receptor action. (2003) (18)
- Ground state oxygen in synthesis of cyclic peroxides. Part 1: Benzo fused ketals (2006) (18)
- Conceptually new 20-epi-22-oxa sulfone analogues of the hormone 1alpha,25-dihydroxyvitamin D(3): synthesis and biological evaluation. (2000) (18)
- One-pot, four-different-component annulations: flexible and efficient conversion of n-sized cycloalkenones into n+4 alkenolides (1987) (18)
- Sequential Michael-Michael-Michael-ring closure reactions for high-yield, one-pot, 4-component coupling (1986) (18)
- Molecular sieves promote stereocontrolled αα-disaccharide formation via direct dimerization of free sugars (1996) (17)
- Differentiation-inducing potency of the seco-steroid JK-1624F2-2 can be increased by combination with an antioxidant and a p38MAPK inhibitor which upregulates the JNK pathway (2007) (16)
- Vitamin D analogs induce lipoxygenase mRNA expression and activity as well as reactive oxygen species (ROS) production in human bone cells (2010) (16)
- Antiproliferative, low-calcemic, fluorinated sulfone analogs of 1alpha,25-dihydroxyvitamin D3: chemical synthesis and biological evaluation. (2007) (16)
- 1α,25-dihydroxyvitamin D3 hybrid analogs with structural changes at both the A-ring and the C,D-ring side-chain (1994) (16)
- Reductive Elimination of Bromine from 1,2-Dibromoalkanes Using Organometallic Reagents (1973) (16)
- Diels-Alder cycloadditions using electrophilic sulfonyl pyridones (1987) (16)
- Three-different-component [1+2+n]-annulation reactions: ionic and radical cyclizations (1990) (16)
- Examination of structurally selective derivatization of vitamin D(3) analogues by electrospray mass spectrometry. (2001) (16)
- Malaria-infected mice live until at least day 30 after a new artemisinin-derived thioacetal thiocarbonate combined with mefloquine are administered together in a single, low, oral dose. (2012) (15)
- Conceptually new low-calcemic oxime analogues of the hormone 1 alpha,25-dihydroxyvitamin D(3): synthesis and biological testing. (2002) (15)
- Antimalarial Endoperoxides that are Potent and Easily Synthesized (1997) (15)
- Diels–Alder cycloadditions using alkenyl sulphoxides (1985) (15)
- ASYMMETRIC SYNTHESES OF ENANTIOMERIC 3-P-FLUOROPHENYL 1,2,4-TRIOXANE ANALOGUES OF THE ANTIMALARIAL ARTEMISININ (1999) (15)
- Modulation of response to estrogens in cultured human female bone cells by a non-calcemic Vitamin D analog: changes in nuclear and membranal binding (2004) (15)
- Asymmetric Conjugate Additions of an Hydroxymethyl Carbanion Equivalent. Synthesis of (+)-A Factor (1987) (15)
- A non-calcemic Vitamin D analog modulates both nuclear and putative membranal estrogen receptors in cultured human vascular smooth muscle cells (2004) (15)
- Chemiluminescent probes for singlet oxygen in biological reactions. (1986) (15)
- QW-1624F2-2, a synthetic analogue of 1,25-dihydroxyvitamin D3, enhances the response to other deltanoids and suppresses the invasiveness of human metastatic breast tumor cells (2006) (15)
- New silicon-mediated ring expansion of n-sized conjugated cycloalkenones into homoallylic n+3 lactones (2003) (15)
- The survival times of malaria-infected mice are prolonged more by several new two-carbon-linked artemisinin-derived dimer carbamates than by the trioxane antimalarial drug artemether. (2014) (15)
- A non-calcemic analog of 1α,25 dihydroxy vitamin D3 (JKF) upregulates the induction of creatine kinase B by 17β estradiol in osteoblast-like ROS 17/2.8 cells and in rat diaphysis (2001) (14)
- Multicomponent One-Pot Annulations Forming Three to Six Bonds (1987) (14)
- CHAPTER 80 – Overview: Rational Design of 1α,25-Dihydroxyvitamin D3 Analogs (Deltanoids) (2005) (14)
- 1.5 – Alkylations of Nonstabilized Carbanions (1991) (14)
- Vitamin D less-calcemic analog modulates the expression of estrogen receptors, vitamin D receptor and 1α-hydroxylase 25-hydroxy vitamin D in human thyroid cancer cell lines (2013) (14)
- Sequential Michael-Michael-Ring Closure reactions for 3-different-component, one-pot, 2+2+2 construction of acylcyclohexenes and an acylcyclohexanol (1986) (13)
- Antimalarial preclinical drug development: a single oral dose of a 5‐carbon‐linked trioxane dimer plus mefloquine cures malaria‐infected mice (2010) (13)
- Differential photoprotective effects of 1,25-dihydroxyvitamin D3 and a low calcaemic deltanoid. (2012) (13)
- New, antimalarial, tricyclic 1,2,4-trioxanes: evaluations in mice and monkeys. (1994) (13)
- Alkyl and aryl isothiocyanates as masked primary amines (1992) (13)
- A new oxidizing reagent: triethylsilyl hydrotrioxide (1989) (13)
- Scope of [1+2+3] annulations using aminonitriles as Michael donors (1993) (13)
- Noncalcemic, Antiproliferative, Transcriptionally Active, 24-Fluorinated Hybrid Analogues of the Hormone 1α,25-Dihydroxyvitamin D3. Synthesis and Preliminary Biological Evaluation. (1998) (13)
- A furoxan-amodiaquine hybrid as a potential therapeutic for three parasitic diseases(). (2012) (13)
- Specificity of chemiluminescence in the metabolism of benzo[a]pyrene to its carcinogenic diol epoxide. (1981) (13)
- ORGANIC REACTIONS AT ALUMINA SURFACES: AN EXTREMELY SIMPLE, MILD AND CONVENIENT METHOD FOR ACETYLATING PRIMARY ALCOHOLS (1981) (12)
- Highly antiproliferative, low-calcemic, side-chain ketone analogs of the hormone 1alpha,25-dihydroxyvitamin D3. (2005) (12)
- Antimalarial chemotherapy: orally curative artemisinin-derived trioxane dimer esters. (2015) (12)
- Alumina-promoted Opening of Medium Ring Epoxides: cis-Cyclooctene Oxide - trans-2-Acetoxycyclooctanol (1981) (12)
- Organic reactions at alumina surfaces. V. Highly selective alcohol and diol oxidation reactions on alumina (1976) (12)
- Microsomal chemiluminescence of benzo[a]pyrene-7,8-dihydrodiol and its synthetic analogues trans- and cis-1-methoxyvinylpyrene. (1986) (12)
- Organocopper chemistry. reaction of benzal and other benzylic chlorides with lithium dimethylcopper (1972) (11)
- Inhibition of P-glycoprotein by two artemisinin derivatives (2012) (11)
- New synthetic methodology for ring expansion of n-sized conjugated cycloalkenones into homoallylic n+3 lactones: 3-step synthesis of fragrant phoracantholide ☆ (2000) (11)
- Organic reactions at alumina surfaces. Elimination reactions effected by dehydrated chromatographic alumina (1976) (11)
- Alumina-accelerated methanolysis and hydrolysis of acyl and phosphoryl fluorides (1981) (11)
- Highly stereocontrolled and regiocontrolled syntheses of polyoxygenated [2.2.2]oxabicyclic synthons (2013) (11)
- α-Chloro-β,γ-ethylenic esters: enantiocontrolled synthesis and substitutions. (2010) (11)
- A-ring hydroxymethyl 19-nor analogs of the natural hormone 1alpha,25-dihydroxyvitamin D(3): synthesis and preliminary biological evaluation. (2005) (11)
- Organic reactions at alumina surfaces. chemospecific oxidation of β-hydroxy sulfides and selenides into the corresponding β-keto sulfides and selenides using chloral on activated alumina. (1977) (11)
- Low-calcemic vitamin D analogs (deltanoids) for human cancer prevention. (2002) (11)
- New synthetic methodology using organosulfur compounds (1990) (10)
- Low-calcemic, highly antiproliferative, 1-difluoromethyl hybrid analogs of the natural hormone 1alpha,25-dihydroxyvitamin D3: design, synthesis, and preliminary biological evaluation. (2006) (10)
- Inhibition of prostate cancer-meditated osteoblastic bone lesions by the low-calcemic analog 1α-hydroxymethyl-16-ene-26,27-bishomo-25-hydroxy vitamin D3 (2005) (10)
- Metabolites and analogs of 1α,25-dihydroxyvitamin D3: evaluation of actions in bone (2001) (10)
- Novel A-ring analogs of the hormone 1alpha,25-dihydroxyvitamin D3: synthesis and preliminary biological evaluation. (2005) (10)
- Chemiluminescence Mechanism and Quantum Yield of Synthetic Vinylpyrene Analogues of Benzo[a]pyrene‐7,8‐dihydrodiol. (1986) (10)
- Less calcemic Vitamin D analogs enhance creatine kinase specific activity and modulate responsiveness to gonadal steroids in the vasculature (2006) (9)
- 'Novel alkyl side chain sulfone 1alpha,25-dihydroxyvitamin D3 analogs: a comparison of in vitro antiproliferative activities and in vivo calcemic activities'. (2009) (9)
- A new approach to the bicyclo[3.2.1]octane ring system: Intramolecular michael and aldol reactions of 3-(5-oxohexyl)-2-cyclopentenones (1978) (9)
- Organocopper chemistry. Reaction of α,β-ethylenic sulfones with lithium dialkylcuprates (1973) (9)
- A useful method for α-methylation of γ-butyrolactones (1972) (9)
- AN ANTIMALARIALLY ACTIVE CYCLIC PEROXY KETAL (1998) (9)
- A surprising effect of a 3-phenyl group on the stereochemistry of cyclopentanone enolate alkylation. Highly stereoselective organocopper 2,3-dialkylation of 2-cyclopentenones. Synthesis of sesquiterpene hydrocarbon (±)-laurene (1977) (9)
- The effects of native and synthetic estrogenic compounds as well as vitamin D less-calcemic analogs on adipocytes content in rat bone marrow. (2011) (9)
- Lewis acid catalysed rearrangements of unsaturated bicyclic [2.2.n] endoperoxides in the presence of vinyl silanes; access to novel Fenozan BO-7 analogues (2005) (9)
- Artemisinins target the intermediate filament protein vimentin for human cytomegalovirus inhibition (2020) (9)
- NEW ORGANOCOPPER SYNTHETIC METHODS. α,β‐DIALKYLATION OF α,β‐ETHYLENIC KETONES: SYNTHESIS OF SESQUITERPENES * (1977) (8)
- 1,2-Dioxetanes from vinyl aromatics (1987) (8)
- 1-(hydroxyalkyl)-25-hydroxyvitamin D3 analogs of calcitriol. 2. Preliminary biological evaluation (1993) (8)
- Copper and silicon mediated, HMPA-free, n+3 ring expansions for the construction of medium sized lactones and lactams: short synthesis of (+)-cis-lauthisan (2016) (8)
- A chemiluminescence assay specific for the microsomal metabolite, benzo[a]pyrene-7,8-dihydrodiol. (1983) (8)
- Responsiveness to phytoestrogens in primary human osteoblasts is modulated differentially by a “less-calcemic” analog of 1,25 dihydroxyvitamin D3: JK 1624F2-2 (JKF) (2006) (8)
- Low-calcemic, highly antiproliferative, 23-oxa ether analogs of the natural hormone 1 alpha,25-dihydroxyvitamin D3: design, synthesis, and preliminary biological evaluation. (2007) (8)
- Highly antiproliferative, low-calcemic, side-chain amide and hydroxamate analogs of the hormone 1alpha,25-dihydroxyvitamin D3. (2006) (8)
- Antiproliferative Hybrid Analogues of the Hormone 1α,25‐ Dihydroxyvitamin D3: Design, Synthesis, and Preliminary Biological Evaluation. (1997) (7)
- Antimalarial 1,2,4-Trioxanes Related to Artemisinin: Rules for Assignment of Relative Stereochemistry in Diversely Substituted Analogs (1997) (7)
- Design, Synthesis, Derivatization, and Structure—Activity Relationships of Simplified, Tricyclic, 1,2,4-Trioxane Alcohol Analogues of the Antimalarial Artemisinin. (1998) (7)
- A short, simple, stereocontrolled, steroid total synthesis: (±)-11-oxoequilenin methyl ether (1978) (7)
- 2-Fluoroalkyl A-Ring Analogues of 1,25-Dihydroxyvitamin D3. Stereocontrolled Total Synthesis via Intramolecular and Intermolecular Diels-Alder Cycloadditions. Preliminary Biological Testing. (1995) (7)
- Unexpected steric effects of remote alkyl groups on the rate of conjugate additions to alkyl α/β-ethylenic sulfones, sulfoxides, and esters (2007) (7)
- Regiocontrolled and Stereocontrolled Diels-Alder Cycloadditions of 2-Pyrones and Unactivated, Unbranched 1-Alkenes (1997) (7)
- Short nonannelation approach to synthesis of oxygenated eudesmane sesquiterpenes (1973) (7)
- Conjugate Addition Reactions of Organocopper Reagents (2011) (7)
- Mutual interaction of special phytoestrogenic compounds, their synthetic carboxy-derivatives and the less-calcemic vitamin D analog activities in human derived female cultured osteoblasts (2011) (7)
- Substitution Reactions Using Organocopper Reagents (2011) (7)
- A mechanistic study of organocopper substitution reactions with some ethylenic p-toluenesulfonate esters (1974) (7)
- Recent Advances in Diels—Alder Cycloadditions of 2-Pyrones (1999) (6)
- A rationale for treatment of hereditary vitamin D-resistant rickets with analogs of 1 alpha,25-dihydroxyvitamin D(3). (2001) (6)
- Organic reactions at alumina surfaces II. 2-propanol on dehydrated alumina as a reagent for selective reduction of aldehydes (1975) (6)
- Electronically stabilized versions of the antimalarial acetal trioxanes artemether and artesunate. (2008) (6)
- A covalent fluorescence probe based on excited-state proton transfer. (1979) (6)
- Conformationally restricted hybrid analogues of the hormone 1 alpha,25-dihydroxyvitamin D(3): design, synthesis, and biological evaluation. (2001) (6)
- Modulation of the response to estradiol-17β of rat vascular tissues by a non calcemic vitamin D analog (2004) (6)
- Some unusual aspect aspects of organocopper chemistry: lithium organocuprate reaction with some neopentylic p-tosylate esters (1979) (6)
- Less-calcemic vitamin D analogs enhance creatine kinase specific activity and modulate responsiveness to gonadal steroids in rat skeletal tissues (2007) (5)
- Nucleophilic opening of a polycyclic aromatic K-region epoxide (1984) (5)
- Metabolites and analogs of 1alpha,25-dihydroxyvitamin D(3): evaluation of actions in bone. (2001) (5)
- Highly stereocontrolled and regiocontrolled syntheses of 2,3,4-trisubstituted alkanoates and lactones. (2011) (5)
- ORGANIC REACTIONS AT ALUMINA SURFACES. MILD, SELECTIVE, AND HIGH-YIELD OXIDATION OF CYCLOBUTANOL TO CYCLOBUTANONE (1977) (5)
- Stereocontrolled Total Synthesis of Calcitriol Derivatives: 1,25- Dihydroxy-2-(4′-hydroxybutyl)vitamin D3 Analogues of an Osteoporosis Drug. (1995) (5)
- a-Fluorination of -keto sulfoxides (1985) (4)
- An organometallic route to (±)-3-p-toluenesulfinyl-2-pyrone (1985) (4)
- SHORT, SIMPLE, STEREOCONTROLLED, STEROID SYNTHESIS: (.+‐.)‐11‐OXOEQUILENIN METHYL ETHER AND A NEW 9,11‐SECO‐13‐ETHYL STEROID (1980) (4)
- Studies of protonated and anionic artemisinin in the gas-phase by infrared multi-photon dissociation and by negative ion photoelectron spectroscopies (2007) (4)
- Quantitation of isothiocyanates by cyclocondensation with 1,2-benzenedithiol (1993) (4)
- Malaria-Infected Mice Are Cured by a Single Low Dose of a New Silylamide Trioxane Plus Mefloquine (2009) (4)
- Alumina-catalyzed opening of cyclohexene oxide by alcohols, acetic acid, and aniline (1980) (4)
- New A-ring analogs of the hormone 1α,25-dihydroxyvitamin D3: (2′-hydroxymethyl)tetrahydrofuro[1,2-a]-25-hydroxyvitamin D3 (2009) (4)
- An Efficient Synthesis of Bridged-Bicyclic Peroxides Structurally Related to Antimalarial Yingzhaosu A Based on Radical Co-Oxygenation of Thiols and Monoterpenes. (2002) (4)
- Iron(II)-Induced Degradation of Antimalarial β-Sulfonyl Endoperoxides. Evidence for the Generation of Potentially Cytotoxic Carbocations. (2002) (4)
- New vitamin D analogues. (1996) (4)
- Alkyl and Aryl Isothiocyanates as Masked Primary Amines. (1992) (4)
- An Asymmetric Total Synthesis of Fragrant Spiro(4.5)decane Sesquiterpene (-)-β-Vetivone via an Enantiomerically Pure Vinylic Sulfoxide. (1989) (3)
- Synthesis and characterization of two stereoisomeric hydroazulenones. Versatile precursors to guaianolides. (1978) (3)
- Synthesis and Antimalarial Activities of Structurally Simplified 1,2,4‐ Trioxanes Related to Artemisinin. (1995) (3)
- Difluoromethyl analogs of the natural hormone 1α,25-dihydroxyvitamin D3: Design, synthesis, and preliminary biological evaluation (2007) (3)
- Highly regiocontrolled and stereocontrolled syntheses of polysubstituted aminocyclohexanes: mild inverse-electron-demand Diels–Alder cycloadditions of electrophilic 2-pyridones (2016) (3)
- Syntheses and Iron(II) Induced Reactions of Phenyl-Substituted 1,2,4-Trioxanes. (1998) (3)
- Asymmetric Total Synthesis, X-Ray Crystallography, and Preliminary Biological Evaluation of 1-(1′-Hydroxyethyl)-25-hydroxyvitamin D3 Analogues of Natural Calcitriol. (1994) (3)
- Asymmetric Carbon-Carbon Bond Formation Using Enantiomerically Pure Vinylic Sulfoxides (1982) (3)
- Stereochemistry of hydrolysis and elimination reaction of toluene-p-sulphonate esters on alumina (1972) (3)
- Three‐Component, One‐Flask Synthesis of Rhodanines (Thiazolidinones). (2012) (3)
- Modern Organocopper Chemistry Edited by Norbert Krause (University of Dortmund). Wiley VCH: Weinheim. 2002. xiv + 378 pp. $125.00. ISBN 3-527-29773-1. (2002) (3)
- 2,2-Disubstituted analogues of the natural hormone 1 alpha,25-dihydroxyvitamin D(3): chemistry and biology. (2002) (2)
- A Short Synthesis of 6,9-Desmethyldeoxoartemisinin and Its Isomer. (1997) (2)
- Antimalarial Artemisinin Analogues. Synthesis via Chemoselective C—C Bond Formation and Preliminary Biological Evaluation. (1999) (2)
- A surprising effect of 3-aryl groups on the regiochemistry of formation of cyclopentanone lithium enolates. Evidence for lithium-arene π-coordination (1977) (2)
- Recent major advances in the studies on Qinghaosu and related antimalarial agents (1999) (2)
- A non-calcemic analog of 1 alpha,25 dihydroxy vitamin D(3) (JKF) upregulates the induction of creatine kinase B by 17 beta estradiol in osteoblast-like ROS 17/2.8 cells and in rat diaphysis. (2001) (2)
- Asymmetric Syntheses of Enantiomeric 3‐p‐Fluorophenyl 1,2,4‐Trioxane Analogues of the Antimalarial Artemisinin. (2000) (2)
- Age-dependent responsiveness of human female bone cells to vitamin D analog and PTH (2013) (2)
- 1α,25-Dihydroxyvitamin D3 Analogues Featuring Aromatic and Heteroaromatic Rings: Design, Synthesis, and Preliminary Biological Testing. (2010) (2)
- Secondary and Tertiary Alkyl Ketones from Carboxylic Acid Chlorides and Lithium Phenylthio(Alkyl)Cuprate Reagents: tert‐Butyl Phenyl Ketone (2003) (2)
- Stereochemical evidence for a carbonium ion rearrangement during reaction of dimethyltitanium dichloride with a ketone (1983) (2)
- 16 – ALUMINA AND ALUMINA-SUPPORTED REAGENTS (1987) (2)
- A CONVENIENT, ONE-STEP, HIGH-YIELD REPLACEMENT OF AN ANOMERIC HYDROXYL GROUP BY A FLUORINE ATOM USING DAST. PREPARATION OF GLYCOSYL FLUORIDES (1985) (2)
- Nucleophilic Opening of a Polycyclic Aromatic K-Region Epoxide. (1984) (2)
- Systemic treatments with the low‐calcemic 1,25(OH)2D3 analogs JKF or QW increase both the morphological and biochemical responses to estradiol‐17β in rat tibiae (2007) (2)
- A NEW DIRECT METHOD FOR SELECTIVE DEMETHYLATION OF N(+)‐METHYL QUATERNARY AMMONIUM IODIDES (1975) (2)
- Direct conversion of cinnamate esters into β,β-disubstituted ketones mediated by cyano-magnesio cuprates (2016) (2)
- 1‐(Hydroxyalkyl)‐25‐hydroxyvitamin D3 Analogs of Calcitriol. Part 1. Synthesis. (1994) (2)
- The Carroll Rearrangement (2007) (2)
- Asymmetric Intramolecular Diels—Alder Cycloadditions of 2‐Pyrone‐3‐carboxylates and Synthesis of Vitamin D3 A‐Ring Phosphine Oxide. (1999) (2)
- Age-Dependent Responsiveness of Human Female Cultured Bone Cells to Estrogenic Compounds (2011) (2)
- Asymmetric Synthesis Using α‐Sulfinyl Carbanions and β‐Unsaturated Sulfoxides (2006) (2)
- The Response of Creatine Kinase Specific Activity in Rat Pituitary to Estrogenic Compounds and Vitamin D Less-Calcemic Analogs (2009) (2)
- HIGH ASYMMETRIC INDUCTION DURING ORGANOMETALLIC β‐ADDITION TO α,β‐ETHYLENIC SULFOXIDES. SYNTHESIS OF OPTICALLY ACTIVE β‐ALKYLCARBOXYLIC ACIDS, β‐SUBSTITUTED CYCLOPENTANONES, AND STEROIDAL 11‐OXOEQUILENIN METHYL ETHER (1981) (1)
- Dechloroethylation of Chloroethyl Ethers and Amines Using n-Butyllithium (1975) (1)
- Abstract 818: Repurposing Artemisinins for treatment of acute leukemias (2014) (1)
- Stereocontrolled Synthesis of a Trihydroxylated A Ring as an Immediate Precursor to 1α,2α,25‐Trihydroxyvitamin D3. (1991) (1)
- Age- and sex-dependent hormonal modulation of the expression of vitamin D receptor and 25-hydroxyvitamin D 1α hydroxylase in human bone cells (2014) (1)
- Preparation of ring-tritiated and of aldehyde-14C-labelled 1-pyrenecarboxaldehyde (1985) (1)
- Vitamin D Side Chain Triazole Analogues via Cycloaddition ′Click′ Chemistry. (2004) (1)
- New Silicon-Mediated Ring Expansion of n-Sized Conjugated Cycloalkenones into Homoallylic [n + 3] Lactones. (2003) (1)
- Knowledge of the Proposed Chemical Mechanism of Action and Cytochrome P450 Metabolism of Antimalarial Trioxanes Like Artemisinin Allows Rational Design of New Antimalarial Peroxides (2004) (1)
- Chemopreventive Efficacy of Natural Vitamin D and Synthetic Analogs (2004) (1)
- Highly Regiocontrolled and Stereocontrolled Syntheses of Polysubstituted Aminocyclohexanes: Mild Inverse‐Electron‐Demand Diels—Alder Cycloadditions of Electrophilic 2‐Pyridones. (2016) (1)
- Asymmetric, Organocatalytic, Three‐Step Synthesis of γ‐Hydroxy‐(E)‐α,β‐Unsaturated Sulfones and Esters. (2009) (1)
- TANDEM MICHAEL-MICHAEL-RING CLOSURE (MIMIRC) REACTIONS. ONE-POT STEROID TOTAL SYNTHESIS. (.+-.)-9,11-DEHYDROESTRONES (1982) (1)
- One-Flask, Regiospecific Conversions of Allylic Alcohols into Two- Carbon-Extended, Conjugated Dienoate Esters. Use of a New Sulfinyl Orthoester. (1992) (1)
- ALKYLATION OF ENOLATE IONS GENERATED REGIOSPECIFICALLY VIA ORGANOCOPPER REACTIONS, SYNTHESIS OF DECALIN SESQUITERPENE VALERANE AND OF PROSTAGLANDIN MODEL SYSTEMS (1975) (1)
- REDUCTIVE ELIMINATION OF BROMINE FROM 1,2-DIBROMOALKANES (1974) (1)
- Design and Synthesis of Bifunctional Isothiocyanate Analogues of Sulforaphane: Correlation Between Structure and Potency as Inducers of Anticarcinogenic Detoxication Enzymes. (1994) (1)
- New Antimalarial Trioxanes and Endoperoxides (2001) (1)
- NEW SYNTHETIC METHODS. 24. ORGANIC REACTIONS ON ALUMINUM OXIDE SURFACES (1978) (1)
- Alumina-Catalyzed Alcoholysis of Cyclohexene Oxide (1979) (1)
- Antimalarial sulfide trioxanes: a revision of mechanism (2008) (1)
- Orally Active Antimalarial 3‐Substituted Trioxanes: New Synthetic Methodology and Biological Evaluation. (1998) (1)
- (S)‐( + )‐2‐(p‐Toluenesulfinyl)‐2‐Cyclopentenone: Precursor for Enantioselective Synthesis of 3‐Substituted Cyclopentanones (2003) (1)
- A MECHANISTIC AND SYNTHETIC STUDY OF ORGANOCOPPER SUBSTITUTION REACTIONS WITH SOME HOMOALLYLIC AND CYCLOPROPYLCARBINYL SUBSTRATES. APPLICATION TO ISOPRENOID SYNTHESIS (1977) (1)
- Cyclopentanone Ring Expansion Leading to Functionalized δ‐Lactams: Short Synthesis of Simple Sedum Alkaloids. (2007) (1)
- Molecular Sieves Promote Stereocontrolled α,α-Disaccharide Formation via Direct Dimerization of Free Sugars. (1996) (1)
- Diels‐Alder Cycloadditions Using Nucleophilic 3‐(p‐Tolylthio)‐2‐pyrone. Regiocontrolled and Stereocontrolled Synthesis of Unsaturated, Bridged, Bicyclic Lactones. (2010) (1)
- Organocopper Reagents, The Practical Approach in Chemistry Series (1995) (1)
- Abstract 2023: Artemisinins enhanced the antileukemic efficacy of BCL2 inhibitors (2017) (1)
- Ground State Oxygen in Synthesis of Cyclic Peroxides. Part 1. Benzo Fused Ketals. (2006) (1)
- Isolation and identification of the principal inducer of anticarcinogenic protective enzymes from broccoli (1993) (1)
- Catalytic and enantioselective ester hydrolysis by a modified polyethylenimine (1986) (0)
- Contents Vol. 70, 2006 (2007) (0)
- Tetrahedron reports on organic chemistry (2007) (0)
- New Silicon‐Mediated, Sequential Ring Expansions of n‐Sized 2‐Cycloalkenones into Hydroxyolefinic n + m + p Medium‐Sized Lactones: Short Synthesis of (‐)‐Phoracantholide‐J. (2006) (0)
- ASYMMETRIC SYNTHESIS OF 1α,25-DIHYDROXYVITAMIN D3 AND ANALOGS. (1988) (0)
- Subject Index Vol. 70, 2006 (2007) (0)
- A New and Efficient Asymmetric Synthesis of an A-Ring Precursor to Physiologically Active 1α-Hydroxyvitamin D3 Steroids. (2010) (0)
- Scope of (1 + 2 + 3)Annulations Using Amino Nitriles as Michael Donors. (1993) (0)
- Binaphthol-Titanium-Promoted, Highly Enantiocontrolled, Diels-Alder Cycloadditions of Electronically Matched 2-Pyrones and Vinyl Ethers: Streamlined Asymmetric Synthesis of an A-Ring Precursor to Physiologically Active 1α-Hydroxyvitamin D3 Steroids. (1995) (0)
- ENANTIOCONTROLLED SYNTHESIS OF (S)-3-SUBSTITUTED CYCLOALKANONES FROM (S)-2-(P-TOLYLSULFINYL)-2-CYCLOALKENONES AND DIORGANOMAGNESIUM REAGENTS (1984) (0)
- Antimalarially Potent, Easily Prepared, Fluorinated Endoperoxides. (1997) (0)
- A SUPRISING EFFECT OF 3-ARYL GROUPS ON THE REGIOCHEMISTRY OF FORMATION OF CYCLOPENTANONE LITHIUM ENOLATES. EVIDENCE FOR LITHIUM-ARENE Π-COORDINATION (1977) (0)
- Highly Stereocontrolled Synthesis of Some Trioxygenated Cyclohexenes: An Asymmetric Total Synthesis of (‐)‐Methyl Triacetyl‐4‐epishikimate. (1987) (0)
- New Chemical and Biological Aspects of Artemisinin‐Derived Trioxane Dimers. (2002) (0)
- ADDITION OF ORGANOMETALLIC REAGENTS TO CHIRAL VINYLIC SULFOXIDES (1984) (0)
- A DIRECTING EFFECT OF NEIGHBORING AROMA (1979) (0)
- A NEW APPROACH TO THE BICYCLO(3.2.1)OCTANE RING SYSTEM: INTRAMOLECULAR MICHAEL AND ALDOL REACTIONS OF 3-(5-OXOHEXYL)-2-CYCLOPENTENONES (1979) (0)
- Chemoselective Reactions of Functionalized Piperidines (1993) (0)
- Stereochemical Evidence for a Carbonium Ion Rearrangement During Reaction of Dimethyltitanium Dichloride with a Ketone. (1984) (0)
- New Sulfone Analogues of the Hormone 1 r , 25-Dihydroxyvitamin D 3 : Synthesis and Preliminary Biological Evaluation (1999) (0)
- ALUMINA-PROMOTED OPENING OF MEDIUM RING EPOXIDES: CIS-CYCLOOCTENE OXIDE → TRANS-2-ACETOXYCYCLOOCTANOL (1982) (0)
- One-Pot, Four-Different-Component Annulations: Flexible and Efficient Conversion of n-Sized Cycloalkenones into n+4 Alkenolides. (1988) (0)
- Nitroolefins in One‐Flask, Tandem, A+B+C Coupling Reactions Producing Heterocycles. (1991) (0)
- 24 sulfoximine compounds vitamin D3 (2003) (0)
- One-pot, three-component, sequential Michael-Michael-ring-closure reactions. Annulation of meta-dicarboxylated aromatic rings. Total synthesis of juncunol (1988) (0)
- ADDITIVE PUMMERER REARRANGEMENTS. ASYMMETRIC SYNTHESIS OF (-)-METHYL JASMONATE (1985) (0)
- ORGANIC REACTIONS AT ALUMINA SURFACES. II. 2-PROPANOL ON DEHYDRATED ALUMINA AS A REAGENT FOR SELECTIVE REDUCTION OF ALDEHYDES (1976) (0)
- Foreword by the Guest Editors of this Issue (1984) (0)
- Asymmetric Conjugate Additions of an Hydroxyethyl Carbanion Equivalent. Synthesis of (+)-A Factor. (1988) (0)
- Highly Stereocontrolled and Regiocontrolled Syntheses of Polyoxygenated [2.2.2]Oxabicyclic Synthons. (2014) (0)
- ORGANIC REACTIONS AT ALUMINA SURFACES. CHEMOSPECIFIC OXIDATION OF β-HYDROXY SULFIDES AND SELENIDES INTO THE CORRESPONDING β-KETO SULFIDES AND SELENIDES USING CHLORAL ON ACTIVATED ALUMINA (1977) (0)
- STEREOCONTROLLED TOTAL SYNTHESIS OF AN α-METHYLENE GUAIANOLIDE IN THE 4,5-EPOXYOSMITOPSIN FAMILY (1981) (0)
- Olefin Oxidative Cleavage and Dioxetane Formation Using Triethylsilyl Hydrotrioxide: Application to Preparation of Potent Antimalarial 1,2,4‐ Trioxanes. (1992) (0)
- Diels-Alder Cycloadditions Using Alkenyl Sulphoxides. (1986) (0)
- ASYMMETRIC SYNTHESIS USING ENANTIOMERICALLY PURE SULFOXIDES (1983) (0)
- Stereocontrolled Synthesis of Conjugated E-Dienoate Esters via Double Alkylation and via Pyrolysis of Methyl Phenylsulfinylacetate. (1995) (0)
- Nephrology Dialysis Transplantation New vitamin D analogues (2005) (0)
- BF3×OEt2 Promotes Fast, Mild, Clean, and Regioselective Dehydration of Tertiary Alcohols, e.g. (I), (IV). (1992) (0)
- An Antimalarially Active Cyclic Peroxy Ketal. (1998) (0)
- Mechanism-Based Design of Simple, Symmetrical, Easily Prepared, Potent Antimalarial Endoperoxides. (1996) (0)
- SYNTHESIS AND CHARACTERIZATION OF TWO STEREOISOMERIC HYDROAZULENONES. VERSATILE PRECURSORS TO GUAIANOLIDES (1979) (0)
- A Short Asymmetric Synthesis of Natural (-)-Methyl Jasmonate. (1986) (0)
- Ovariectomy modulates the effect of phytoestrogens on creatine kinase specific activity in skeletal organs in female rats (2012) (0)
- 3-Cuprio-2-pyrone: An Extraordinary Organocopper Reagent. (1986) (0)
- REACTION OF LITHIUM DIALKYLCUPRATES WITH BETA-ALKOXY AND BETA-ALKYLTHIO ALPHA,BETA-UNSATURATED CARBONYL COMPOUNDS (1974) (0)
- New Synthetic Methodology for Ring Expansion of n‐Sized Conjugated Cycloalkenones into Homoallylic [n + 3] Lactones: Three‐Step Synthesis of Fragrant Phoracantholide. (2001) (0)
- SOME UNUSUAL ASPECTS OF ORGANOCOPPER CHEMISTRY: LITHIUM ORGANOCUPRATE REACTION WITH SOME NEOPENTYLIC P-TOSYLATE ESTERS (1980) (0)
- Asymmetric Michael and Diels-Alder Reactions Using Sulfoxides and Sulfones (1987) (0)
- Total Synthesis of Natural Estrone and Estradiol Methyl Ethers in Extremely High Enantiomeric Purity via an Asymmetrie Michael Addition to an Unsaturated Sulfoxide. (1986) (0)
- GENERATION AND REACTIONS OF 1-(ARYLSULFINYL)ALKENYLLITHIUM REAGENTS. TERMINAL ALLENES FROM 2-ALKENYL ARYL SULFOXIDES (1979) (0)
- AN ORGANOMETALLIC ROUTE TO (.+-.)-3-P-TOLUENESULFINYL-2-PYRONE (1985) (0)
- Erratum: Malaria-infected mice are completely cured by one 6 mg/kg oral dose of a new monomeric trioxane sulfide combined with mefloquine (Journal of Medicinal Chemistry (2012) 55 (291-296) DOI: 10.1021/jm201214d) (2012) (0)
- The Unique and Highly-Selective Anti-Cytomegalovirus Activities of Artemisinin-Derived (2013) (0)
- ORGANIC REACTIONS AT ALUMINA SURFACES. AN EXTREMELY SIMPLE, CONVENIENT AND SELECTIVE METHOD FOR ACETYLATING PRIMARY ALCOHOLS IN THE PRESENCE OF SECONDARY ALCOHOLS (1982) (0)
- Oxime analogs of 1-alpha, 25-dihydroxy-vitamin D3 with low effective calcemischer (2002) (0)
- Diels-Alder Cycloadditions Using Electrophilic Sulfonylpyridones. (1987) (0)
- One‐Flask, Consecutive (3,3)‐ and (2,3)Sigmatropic Rearrangements for Conversion of Propargylic Alcohols into Two‐Carbon‐Extended 4‐Oxo‐2‐alkenoate Esters. Use of a New 1‐Chloro‐1‐ethoxy‐2‐sulfinylethylene. (1992) (0)
- A SURPRISING EFFECT OF A 3-PHENYL GROUP ON THE STEREOCHEMISTRY OF CYCLOPENTANONE ENOLATE ALKYLATION. HIGHLY STEREOSELECTIVE ORGANOCOPPER 2,3-DIALKYLATION OF 2-CYCLOPENTENONES. SYNTHESIS OF SESQUITERPENE HYDROCARBON (.+-.)-LAURENE (1977) (0)
- Sequential Michael-Michael Ring Closure Reactions for High-Yield, One- Pot, 4-Component Coupling. (1986) (0)
- A One-Flask Multicomponent Annulation Reaction as the Key Step in a Total Synthesis of Spirobicyclic (.+-.)-β-Vetivone. (1992) (0)
- Formation of Olefins via Pyrolysis of Sulfonate Esters. (1989) (0)
- Mutual modulation of the vitamin D system and estrogen receptors in human bone cells in culture (2007) (0)
- ORGANIC REACTIONS AT ALUMINA SURFACES. DISPLACEMENT REACTIONS EFFECTED BY ALCOHOLS, THIOLS, AND ACETIC ACID ON DEHYDRATED ALUMINA (1976) (0)
- Interrupted Polymerization of Acrylates: Sequential Michael-Michael-Dieckmann Cyclizations for Easy, One-Pot, (2 + 2 + 2)Construction of Polyfunctionalized Cyclohexanones. (1990) (0)
- Sequential Michael-Michael-Aldol Additions for Easy, One-Pot, 2 +2 + 2 Construction of Polyfunctionalized Cyclohexanols. (1986) (0)
- Less-calcemic vitamin D analogs enhance biological responses and modulate responsiveness to gonadal steroids in skeletal tissues (2007) (0)
- Antimalarial Sulfone Trioxanes. (1998) (0)
- AN EFFICIENT METHOD FOR DIBROMOMETHYLENATION AND ISOPROPYLIDENATION OF KETONES (=C=O - =C=BR2 - =C=CME2), SYNTHESIS OF SELINADIENE SESQUITERPENE (1975) (0)
- A SHORT, SIMPLE, STEREOCONTROLLED, STEROID TOTAL SYNTHESIS: (.+-.)-11-OXOEQUILENIN METHYL ETHER (1979) (0)
- Lewis Acid Catalyzed, High Pressure, Stereospecific, Regiospecific, Diels-Alder Cycloaddition of Unsubstituted 2-Pyrone: Short Synthesis of a Racemic A-Ring Precursor (III) to Physiologically Active 1- Hydroxyvitamin D3 Steroids. (2010) (0)
- Regulation de l'aspect de la peau et composition contenant un compose d'analogue de vitamine d3 fluore (2000) (0)
- Stereocontrolled Synthesis of Functionalized Cyclohexenes via Diels- Alder Cycloadditions of 2-Pyrones and 2-Pyridones - Applications to Synthesis of Physiologically Active Compounds (1996) (0)
- Three-Different-Component (1 + 2 + n)Annulation Reactions: Ionic and Radical Cyclizations. (1990) (0)
- 3-Bromo-2-pyrone: An Easily Prepared Chameleon Diene and a Synthetic Equivalent of 2-Pyrone in Thermal Diels-Alder Cycloadditions. (1992) (0)
- One-Pot, Four-Component Annulations: Flexible and Simple Syntheses of Unsaturated Macrolides and of Substituted Aromatics and Heteroaromatics. (1988) (0)
- Unexpected steric effects of "remote" alkyl groups on the rate of conjugate additions to alkyl alpha,beta-ethylenic sulfones, sulfoxides, and esters. (2007) (0)
- Potent anticancer activity of the second generation artemisinin-derived trioxane dimers on pancreatic cancer cells. (2007) (0)
- 5-Bromo-2-pyrone: An Easily Prepared Ambiphilic Diene and a Synthetic Equivalent of 2-Pyrone in Mild, Thermal Diels-Alder Cycloadditions. (1993) (0)
- A NEW SYNTHETIC APPROACH TO PSEUDOGUAIANES (1979) (0)
- Synthesis and Antimalarial Activity of Heteroatom-Containing Bicyclic Endoperoxides. (1997) (0)
- 1,2-Dioxetanes from Vinyl Aromatics. (1987) (0)
- DESIGN AND ASYMMETRIC TOTAL SYNTHESIS OF RING-A ANALOGS OF 1,25- DIHYDROXYVITAMIN D3 (1991) (0)
- A General Method for the Preparation of 9‐, 10‐, and 11‐Membered Unsaturated Macrolides: Synthesis of 8‐Propionyl‐(E)‐5‐Nonenolide (2003) (0)
- AN EXTREMELY EFFICIENT METHOD FOR ONE-POT, THREE-COMPONENT, 2 + 2 + 2 CONSTRUCTION OF FUNCTIONALIZED CYCLOHEXENES (1985) (0)
- Asymmetric Total Synthesis of an A-Ring Precursor to Hormonally Active 1α,25-Dihydroxyvitamin D3. (1990) (0)
- Asymmetric, Organocatalytic, Three‐Step Synthesis of α‐Hydroxy‐(E)‐β,γ‐unsaturated Esters. (2010) (0)
- The 3-Drug Combination Treatment ART838, ABT199 Plus Sorafenib Is Effective Against AML Xenografts, Possibly Via Cooperative Targeting of MCL1 (2018) (0)
- A NEW CLASS OF MIXED CUPRATE(I) REAGENTS, HET(R)CULI, WHICH ALLOW SELECTIVE ALKYL GROUP TRANSFER (1974) (0)
- Stereocontrolled Synthesis of Highly Functionalized Cyclohexenes. A Short Synthesis of a Chorismic Acid Precursor. (1990) (0)
- ALKYLATION OF ENOLATE IONS GENERATED REGIOSPECIFICALLY VIA ORGANOCOPPER CONJUGATE ADDITION REACTIONS, SYNTHESIS OF DECALIN SESQUITERPENE VALERANE AND OF A PROSTAGLANDIN MODEL SYSTEM (1974) (0)
- Asymmetrie Michael Additions of Ester Enolates to Enantiomerically Pure Vinylic Sulfoxides. (1986) (0)
- 24-sulfur-substituted-1-alpha-25-dihydroxy-vitamin D3 analog (2002) (0)
- Sequential Michael‐Michael Ring Closure Reactions for 3‐Different‐Component, One‐Pot, [2+2+2] Construction of Acylcyclohexenes and an Acylcyclohexanol. (1986) (0)
- Direct Conversion of Pyranose Anomeric OH→F→R in the Artemisinin Family of Antimalarial Trioxanes. (1998) (0)
- α‐FLUORINATION OF β‐KETO SULFOXIDES (1985) (0)
- Asymmetric Diels‐Alder Cycloadditions Using Chiral Alkyl Vinyl Ethers and a Dienyl Sulfone. (1986) (0)
- A SHORT NONANNELATION APPROACH TO SYNTHESIS OF OXYGENATED EUDESMANE SESQUITERPENES (1974) (0)
- Mild, Asymmetric Diels-Alder Cycloadditions of Electronically Matched 2-Pyrones and Vinyl Ethers. (1994) (0)
- Direct Conversion of Carboxylic Acids into Ketones (2011) (0)
- (S)-(+)-2-(P-TOLYLSULFINYL)-2-BUTEN-4-OLIDE: AN ENANTIOMERICALLY PURE MICHAEL ACCEPTOR FOR ASYMMETRIC SYNTHESIS OF 3-SUBSTITUTED 4-BUTANOLIDES. (-)-PODORHIZON (1984) (0)
- Analogues de vitamine d¿3? (1993) (0)
- An Improved Preparation of 3‐Bromo‐2H‐Pyran‐2‐one: An Ambiphilic Diene for Diels‐Alder Cycloadditions (2003) (0)
- Diels‐Alder Cycloadditions Using Nucleophilic 2‐Pyridones. Regiocontrolled and Stereocontrolled Synthesis of Unsaturated, Bridged, Bicyclic Lactams. (1992) (0)
- Inhibition of P-glycoprotein by two artemisinin derivatives (2012) (0)
- A New, Direct Method for Selective Demethylation of N+-Methyl Quaternary Ammonium Iodides (1974) (0)
- A New Oxidizing Reagent: Triethylsilyl Hydrotrioxide. (1990) (0)
- Highly Stereocontrolled Synthesis of Some Polyfunctionalized Cyclohexenes. A Short Formal Total Synthesis of (.+-.)-Chorismic Acid. (1988) (0)
- Regiocontrolled and Stereocontrolled Diels‐Alder Cycloadditions of 2‐ Pyrones and Unactivated, Unbranched 1‐Alkenes. (1997) (0)
- Analogs of 1-alpha, 25-dihydroxy vitamin d3 no calcemic, antiproliferative, transcriptionally active sulfur-containing. (2000) (0)
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