Gunda Georg
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Professor of Chemistry, University of Minnesota
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Chemistry
Gunda Georg's Degrees
- PhD Chemistry University of Hamburg
Why Is Gunda Georg Influential?
(Suggest an Edit or Addition)According to Wikipedia, Gunda I. Georg is a chemist who is currently the Professor and Head of the Department of Medicinal Chemistry, Regents Professor, McKnight Presidential Chair, Robert Vince Endowed Chair at University of Minnesota and a former Co-Editor-in-Chief of American Chemical Society's Journal of Medicinal Chemistry. Her research interests are total synthesis and semisynthesis as well as evaluating biologically active agents. A cited expert in her field, she was elected to the American Association for the Advancement of Science in 1996 and inducted in the Medicinal Chemistry Hall of Fame in 2017. In 2019, she was announced as the 2020 winner and first woman to receive the Alfred Burger Award in Medicinal Chemistry . She along with chemists, Shameem Syeda and Gustavo Blanco, are leading researchers in male contraception. Dr Georg also works with her research groups to conduct research on Alzheimer's disease, epilepsy and cancer experimental therapeutics.
Gunda Georg's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Taxol®: science and applications. (1995) (361)
- The Organic chemistry of β-lactams (1993) (285)
- A Preclinical Evaluation of Minnelide as a Therapeutic Agent Against Pancreatic Cancer (2012) (203)
- Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors (2014) (184)
- A convenient method for the efficient removal of ruthenium byproducts generated during olefin metathesis reactions. (2001) (149)
- Mild and selective hydrozirconation of amides to aldehydes using Cp2Zr(H)Cl: scope and mechanistic insight. (2007) (147)
- Efficient and practical asymmetric synthesis of the taxol C-13 side chain, N-benzoyl-(2R,3S)-3-phenylisoserine, and its analogs via chiral 3-hydroxy-4-aryl-.beta.-lactams through chiral ester enolate-imine cyclocondensation (1991) (143)
- Discovery of a potential allosteric ligand binding site in CDK2. (2011) (143)
- Palladium(II)-catalyzed direct arylation of enaminones using organotrifluoroborates. (2008) (138)
- Epothilone and paclitaxel: unexpected differences in promoting the assembly and stabilization of yeast microtubules. (2002) (132)
- Cyclin-dependent kinase inhibitor dinaciclib interacts with the acetyl-lysine recognition site of bromodomains. (2013) (131)
- Hydrophobic collapse of taxol and taxotere solution conformations in mixtures of water and organic solvent (1993) (120)
- Understanding tubulin–Taxol interactions: Mutations that impart Taxol binding to yeast tubulin (2003) (103)
- A Novel and Expeditious Reduction of Tertiary Amides to Aldehydes Using Cp2Zr(H)Cl (2000) (103)
- Asymmetric synthesis of (1′R,3R,4R)-4-acetoxy-3-(1′-((tert-butyldimethylsilyl)oxy)ethyl)-2- azetidinone and other 3-(1′-Hydroxyethyl)-2-azetidinones from (S)-(+)-Ethyl 3-hydroxybutanoate: Formal total synthesis of (+)-thienamycin (1987) (100)
- Palladium(II)-catalyzed dehydrogenative alkenylation of cyclic enaminones via the Fujiwara-Moritani reaction. (2011) (99)
- β-Amyloid-Induced Neurodegeneration and Protection by Structurally Diverse Microtubule-Stabilizing Agents (2005) (96)
- Chemical modification of paclitaxel (Taxol) reduces P-glycoprotein interactions and increases permeation across the blood-brain barrier in vitro and in situ. (2005) (88)
- Gamendazole, an orally active indazole carboxylic acid male contraceptive agent, targets HSP90AB1 (HSP90BETA) and EEF1A1 (eEF1A), and stimulates Il1a transcription in rat Sertoli cells. (2008) (86)
- A novel potent indazole carboxylic acid derivative blocks spermatogenesis and is contraceptive in rats after a single oral dose. (2008) (83)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (83)
- Synthesis of biologically active taxol analogues with modified phenylisoserine side chains. (1992) (80)
- The cryptophycins: Their synthesis and anticancer activity (2002) (76)
- Stabilization of the cyclin‐dependent kinase 5 activator, p35, by paclitaxel decreases β‐amyloid toxicity in cortical neurons (2003) (72)
- Development of highly potent and selective diaminothiazole inhibitors of cyclin-dependent kinases. (2013) (66)
- Epothilones, a new class of microtubule-stabilizing agents with a taxol-like mechanism of action (1998) (65)
- Amino acid-derived enaminones: a study in ring formation providing valuable asymmetric synthons. (2006) (63)
- Interaction of cryptophycin 1 with tubulin and microtubules (1995) (61)
- Direct Hiyama cross-coupling of enaminones with triethoxy(aryl)silanes and dimethylphenylsilanol. (2011) (58)
- Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors. (2017) (56)
- Synthesis of tylocrebrine and related phenanthroindolizidines by VOF3-mediated oxidative aryl-alkene coupling. (2011) (56)
- [Bis(2-methoxyethyl)amino]sulfur trifluoride, the Deoxo-Fluor reagent: application toward one-flask transformations of carboxylic acids to amides. (2004) (54)
- Total syntheses of arylindolizidine alkaloids (+)-ipalbidine and (+)-antofine. (2010) (54)
- Polymer-bound triphenylphosphine as traceless reagent for mitsunobu reactions in combinatorial chemistry: Synthesis of aryl ethers from phenols and alcohols (1998) (54)
- The Ecstasy and Agony of Assay Interference Compounds (2017) (53)
- Phosphonooxymethyl Prodrug of Triptolide: Synthesis, Physicochemical Characterization, and Efficacy in Human Colon Adenocarcinoma and Ovarian Cancer Xenografts (2015) (52)
- Novel prodrug approach for tertiary amines: synthesis and preliminary evaluation of N-phosphonooxymethyl prodrugs. (1999) (51)
- Synthesis of 6- and 7-membered cyclic enaminones: scope and mechanism. (2010) (50)
- Synthesis of amino acid derived enaminones via Wolff rearrangement using vinylogous amides as carbon nucleophiles. (2010) (50)
- A Facile One-Flask Conversion of Aldehydes and Ketones to N-Sulfonyl Imines (1995) (48)
- Asymmetric synthesis of α-alkylated α-amino acids via Schmidt rearrangement of α,α-bisalkylated β-keto esters (1988) (45)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (44)
- Discovery and development of the covalent hydrates of trifluoromethylated pyrazoles as riboflavin synthase inhibitors with antibiotic activity against Mycobacterium tuberculosis. (2009) (44)
- Chemoenzymatic synthesis of cryptophycin/arenastatin natural products. (2005) (42)
- Overcoming the blood-brain barrier to taxane delivery for neurodegenerative diseases and brain tumors (2007) (40)
- Schotten-Baumann acylation of N-debenzoyltaxol; an efficient route to N-acyl taxol analogues and their biological evaluation (1994) (39)
- An improved method for the stereoselective synthesis of β-lactams from carboxylic acids and imines (1991) (39)
- Stereocontrolled synthesis of N-vinyl-N-(1'-propenyl)-, and N-unsubstituted-β-lactams from 2-aza-1,3-butadienes via the Staudinger reaction (1993) (38)
- Artificial Intelligence in Drug Discovery: Into the Great Wide Open. (2020) (38)
- Structural Basis of ALDH1A2 Inhibition by Irreversible and Reversible Small Molecule Inhibitors. (2018) (38)
- Revisiting microtubule targeting agents: α-Tubulin and the pironetin binding site as unexplored targets for cancer therapeutics. (2019) (36)
- Palladium-catalyzed direct C-H arylation of cyclic enaminones with aryl iodides. (2013) (36)
- Synthesis, Conformational Analysis, and Biological Evaluation of Heteroaromatic Taxanes. (1996) (36)
- Synthesis and evaluation of eight- and four-membered iminosugar analogues as inhibitors of testicular ceramide-specific glucosyltransferase, testicular β-glucosidase 2, and other glycosidases. (2012) (36)
- Copper-assisted palladium(II)-catalyzed direct arylation of cyclic enaminones with arylboronic acids. (2012) (36)
- A one-flask synthesis of Weinreb amides from chiral and achiral carboxylic acids using the deoxo-fluor fluorinating reagent. (2000) (35)
- Butitaxel analogues: synthesis and structure-activity relationships. (1997) (35)
- Novel cytotoxic 3'-(tert-butyl) 3'-dephenyl analogs of paclitaxel and docetaxel. (1995) (34)
- The effect of the aromatic rings of taxol on biological activity and solution conformation: synthesis and evaluation of saturated taxol and taxotere analogues. (1994) (34)
- Total synthesis of cryptophycin-24 (Arenastatin A) amenable to structural modifications in the C16 side chain. (2000) (33)
- One-step facile synthesis of deuterium labeled aldehydes from tertiary amides using Cp2Zr(D)Cl (2004) (33)
- Protection against beta-amyloid toxicity in primary neurons by paclitaxel (Taxol). (1998) (33)
- Conformationally restricted paclitaxel analogues: macrocyclic mimics of the "hydrophobic collapse" conformation. (1999) (33)
- Structure-activity studies of antitumor taxanes: synthesis of novel C-13 side chain homologated taxol and taxotere analogs. (1994) (32)
- An asymmetric synthesis of carbapenem antibiotic (+)-PS-5 from ethyl 3-hydroxybutanoate (1988) (32)
- Asymmetric synthesis of β-lactams and n-benzoyl-3-phenylisoserines via the staudinger reaction (1991) (32)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (32)
- Overview Oncologic, Metabolic & Endocrine: Taxol: a novel antitumour agent (1994) (31)
- Design, Synthesis, and in Vitro and in Vivo Evaluation of Ouabain Analogues as Potent and Selective Na,K-ATPase α4 Isoform Inhibitors for Male Contraception (2018) (31)
- Samarium diiodide-mediated deoxygenation of taxol: A one-step synthesis of 10-deacetoxytaxol (1994) (31)
- Total Syntheses and Cytotoxicity of (R)- and (S)-Boehmeriasin A. (2011) (31)
- Site-specifically traced drug release and biodistribution of a paclitaxel-antibody conjugate toward improvement of the linker structure. (2004) (31)
- Design, synthesis, and antiproliferative and CDK2-cyclin a inhibitory activity of novel flavopiridol analogues. (2007) (31)
- Transition Metal‐Free Direct Trifluoromethylation of 2,3‐Dihydropyridin‐4(1H)‐ones at Room Temperature (2014) (31)
- BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen. (2017) (31)
- A systematic SAR study of C10 modified paclitaxel analogues using a combinatorial approach. (2002) (30)
- Stereoselective synthesis of 3-(1-Hydroxyethyl)-2-azetidinonesfrom 3-hydroxybutyrates (1984) (30)
- Synthesis of skeletally diverse and stereochemically complex library templates derived from isosteviol and steviol. (2013) (30)
- The Future of Drug Repositioning: Old Drugs, New Opportunities (2011) (30)
- Dehydrogenative alkenylation of uracils via palladium-catalyzed regioselective C-H activation. (2013) (30)
- An efficient semisynthesis of taxol from (3R,4S)-N-Benzoyl-3-[(t-butyldimethylsilyl)oxy]-4-phenyl-2-azetidinone and 7-(Triethylsilyl)baccatin III (1993) (29)
- Synthesis of docetaxel and butitaxel analogues through kinetic resolution of racemic beta-lactams with 7-O-triethylsilylbaccatin III. (2007) (29)
- Synthesis of a photoaffinity taxol analogue and its use in labeling tubulin. (1994) (29)
- Interaction of a fluorescent paclitaxel analogue with tubulin. (1995) (28)
- Boron–Heck Reaction of Cyclic Enaminones: Regioselective Direct Arylation via Oxidative Palladium(II) Catalysis (2014) (28)
- N-vinyl and N-unsubstituted β-lactams from 1-substituted 2-aza-1, 3-butadienes (1990) (28)
- Galactose-Imines in the staudinger reaction (1992) (26)
- Rapid entry into the cryptophycin core via an acyl-beta-lactam macrolactonization: total synthesis of cryptophycin-24. (2001) (26)
- A high-throughput screen utilizing the fluorescence of riboflavin for identification of lumazine synthase inhibitors. (2005) (25)
- An investigation of (R)-(+)-1-(1-naphthyl)ethylimines and (R)-(+)-1-(phenyl)ethylimines as chiral templates in the staudinger reaction (1994) (25)
- Formal total synthesis of (+)-salicylihalamides A and B: a combined chiral pool and RCM strategy. (2003) (25)
- Novel endotoxin-sequestering compounds with terephthalaldehyde-bis-guanylhydrazone scaffolds. (2006) (25)
- Novel d-seco paclitaxel analogues: synthesis, biological evaluation, and model testing. (2001) (24)
- Paclitaxel succinate analogs: Anionic and amide introduction as a strategy to impart blood-brain barrier permeability. (2008) (24)
- Three-component synthesis of cyclic enaminones via ketene cyclization. (2011) (24)
- Inducing Protein Degradation as a Therapeutic Strategy. (2016) (23)
- Heme Binding Biguanides Target Cytochrome P450-Dependent Cancer Cell Mitochondria. (2017) (23)
- Formal syntheses of cryptophycin A and arenastatin A (1997) (23)
- Amyloid peptide toxicity and microtubule-stabilizing drugs (2002) (22)
- Endocrine disruption by indole-3-carbinol and tamoxifen: blockage of ovulation. (2002) (21)
- Synthesis, modeling, and anti-tubulin activity of a D-seco paclitaxel analogue. (2004) (21)
- Probing the environment of tubulin-bound paclitaxel using fluorescent paclitaxel analogues. (1997) (21)
- Ultra-High-Throughput Screening of Natural Product Extracts to Identify Proapoptotic Inhibitors of Bcl-2 Family Proteins (2014) (20)
- Synthesis of a quinolone library from ynones. (2009) (20)
- Discovery and development of a small molecule library with lumazine synthase inhibitory activity. (2009) (20)
- A novel lumazine synthase inhibitor derived from oxidation of 1,3,6,8-tetrahydroxy-2,7-naphthyridine to a tetraazaperylenehexaone derivative. (2007) (20)
- 2,3-Dihydropyridin-4(1H)-ones and 3-Aminocyclohex-2-enones: Synthesis, Functionalization, and Applications to Alkaloid Synthesis (2014) (20)
- Novel Biologically Active Taxol Analogues: Baccatin III 13-(N-(p-chlorobenzoyl)-(2′R,3′S)-3′-phenylisoserinate ) and Baccatin III 13-(N-benzoyl-(2′R,3′S)-3′-(p-chlorophenyl)isoserinate ) (1992) (19)
- The oxetane conformational lock of paclitaxel: structural analysis of D-secopaclitaxel. (1999) (19)
- Preparation and physicochemical characterization of a novel water-soluble prodrug of carbamazepine. (2010) (19)
- 2-aza-1,3-dienes as novel precursors for the synthesis of N-unsubstituted β-lactams. A three step synthesis of 4-acetoxy-3-phenoxy-2-azeridinone (1988) (19)
- RCM approach for the total synthesis of cryptophycin-24 (Arenastatin A) (2004) (19)
- Synthesis and evaluation of the anti-proliferative and NF-κB activities of a library of simplified tylophorine analogs. (2012) (19)
- Synthesis of fused bicyclic systems with nitrogen atom at the bridgehead, including indolizidines and quinolizidines. (2011) (18)
- Efficient synthesis of the 3'-phenolic metabolite of paclitaxel. (2001) (18)
- A reinvestigation of the taxol content of himalayan taxus wallichiana zucc. and a revision of the structure of brevifoliol. (1993) (18)
- Halohydrin analogues of cryptophycin 1: synthesis and biological activity. (1998) (18)
- Characterizing the Epothilone Binding Site on β-Tubulin by Photoaffinity Labeling: Identification of β-Tubulin Peptides TARGSQQY and TSRGSQQY as Targets of an Epothilone Photoprobe for Polymerized Tubulin. (2016) (17)
- Selective C-2 and C-4 deacylation and acylation of taxol: The first synthesis of a C-4 substituted taxol analogue (1994) (17)
- Microwave-assisted Suzuki-Miyaura couplings on α-iodoenaminones. (2007) (17)
- SELECTIVE DEESTERIFICATION STUDIES ON TAXANES : SIMPLE AND EFFICIENT HYDRAZINOLYSIS OF C-10 AND C-13 ESTER FUNCTIONALITIES (1995) (16)
- 3-(1′-hydroxyethyl)-2-azetidinones from 3-hydroxybutyrates and n-arylaldimines☆ (1985) (16)
- Epigenetics: Novel Therapeutics Targeting Epigenetics. (2015) (16)
- Synthesis, in vitro and in vivo cytotoxicity of 6,7-diaryl-2,3,8,8a-tetrahydroindolizin-5(1H)-ones. (2007) (16)
- High-Throughput Screening for Growth Inhibitors Using a Yeast Model of Familial Paraganglioma (2013) (16)
- Practical syntheses of the C12–C21 epothilone subunit via catalytic asymmetric reductions: Itsuno–Corey oxazaborolidine reduction and asymmetric Noyori hydrogenation (2004) (16)
- Synthesis and anti-tubulin activity of a 3'-(4-azidophenyl)-3'-dephenylpaclitaxel photoaffinity probe. (2004) (16)
- Relative stereochemistry and solution conformation of the novel paclitaxel-like antimitotic agent epothilone A (1996) (16)
- Ongoing in vivo studies with cytoskeletal drugs in tau transgenic mice. (2006) (15)
- The anti-parasitic agent suramin and several of its analogues are inhibitors of the DNA binding protein Mcm10 (2019) (15)
- Synthesis of Cryptophycins via an N-Acyl-β-lactam Macrolactonization (2003) (15)
- Recent advances in the chemistry and biology of -lactams and -lactam antibiotics (1993) (15)
- 4-Deacetyltaxol and 10-acetyl-4-deacetyltaxotere: synthesis and biological evaluation. (1994) (15)
- Pharmacological activity of retinoic acid receptor alpha-selective antagonists in vitro and in vivo. (2013) (15)
- Taxol photoaffinity labels 2. Synthesis and biological evaluation of N-(4-azidobenzoyl)-N-debenzoyltaxol, N-(4-azido-2,3,5,6-tetrafluorobenzoyl)-N-debenzoyltaxol, and 7-(4-azido-2,3,5,6-tetrafluorobenzoyl)taxol (1994) (15)
- Single-site chemical modification at C10 of the baccatin III core of paclitaxel and Taxol C reduces P-glycoprotein interactions in bovine brain microvessel endothelial cells. (2006) (14)
- A one-step transformation of aromatic aldehydes to nitriles, using S,S-Dimethylsulfurdiimide as iminating agent. Isolation of dithiatetrazocines as reaction intermediates. (1985) (14)
- Stereocontrolled Ketene‐Imine Cycloaddition Reactions (1994) (14)
- Synthesis and evaluation of paclitaxel C7 derivatives: solution phase synthesis of combinatorial libraries. (1998) (14)
- Heteroaromatic taxol analogues : the chemistry and biological activities of 3'-furyl and 3'-pyridyl substituted taxanes (1994) (14)
- A convenient method to remove ruthenium byproducts from olefin metathesis reactions using polymer-bound triphenylphosphine oxide (TPPO) (2005) (14)
- Heme Binding Biguanides Target Cytochrome P450-Dependent Cancer Cell Mitochondria. (2017) (14)
- Topliss approach to the synthesis of biologically active substituted N-benzoyl taxol analogues (1994) (14)
- Synthesis of oximidine II by a copper-mediated reductive ene-yne macrocyclization. (2011) (13)
- Cryptophycin affinity labels: synthesis and biological activity of a benzophenone analogue of cryptophycin-24. (2003) (13)
- Support Vector Machines in HTS Data Mining: Type I MetAPs Inhibition Study (2006) (13)
- Rapid Delivery of Diazepam from Supersaturated Solutions Prepared Using Prodrug/Enzyme Mixtures: Toward Intranasal Treatment of Seizure Emergencies (2014) (13)
- Synthesis of biologically active 2-benzoyl paclitaxel analogues (1995) (13)
- The Na+ and K+ transport system of sperm (ATP1A4) is essential for male fertility and an attractive target for male contraception† (2020) (13)
- Short and efficient chiral pool and RCM approach towards the synthesis of the macrocyclic core of the salicylihalamides (2001) (13)
- Synthesis of 2-O-heteroaroyl taxanes: evaluation of microtubule assembly promotion and cytotoxicity (1995) (13)
- Absolute Quantitative 1H NMR Spectroscopy for Compound Purity Determination (2014) (13)
- Studies toward the synthesis of oximidines I and II. (2003) (13)
- N-methylation of the c3' amide of taxanes: synthesis of N-methyltaxol C and N-methylpaclitaxel. (2008) (13)
- Human Adenine Nucleotide Translocase (ANT) Modulators Identified by High-Throughput Screening of Transgenic Yeast (2016) (12)
- Identification of the Metabolic Profile of the α-Tubulin-Binding Natural Product (-)-Pironetin. (2019) (12)
- Water-soluble benzodiazepine prodrug/enzyme combinations for intranasal rescue therapies (2015) (12)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (12)
- Scalable syntheses of the BET bromodomain inhibitor JQ1. (2015) (12)
- Stability of the Human Hsp90-p50Cdc37 Chaperone Complex against Nucleotides and Hsp90 Inhibitors, and the Influence of Phosphorylation by Casein Kinase 2 (2015) (12)
- Enantiospecific formal total syntheses of (-)-salicylihalamides A and B from D-glucose and L-rhamnose. (2003) (12)
- Potent Pyrimidine and Pyrrolopyrimidine Inhibitors of Testis‐Specific Serine/Threonine Kinase 2 (TSSK2) (2017) (12)
- Epigenetics: novel therapeutics targeting epigenetics. (2015) (12)
- Studies towards the synthesis of methionine aminopeptidase inhibitors: diversification utilizing a ROMP-derived coupling reagent. (2008) (12)
- Synthesis of Strained 1,3-Diene Macrocycles via Copper-Mediated Castro-Stephens Coupling/Alkyne Reduction Tandem Reactions. (2015) (11)
- Thermal, three-carbon + two-atom cycloaddition of cyclopropenone ketals with carbon-heteroatom double bonds: Butenolide, furan, and γ-keto ester preparation. (1984) (11)
- From Dioxin to Drug Lead—The Development of 2,3,7,8‐Tetrachlorophenothiazine (2007) (11)
- Synthesis of 13-epi-Taxol via a Transannular Delivery of a Borohydride Reagent (1995) (11)
- Targeting Protein-Protein Interactions by Small Molecules (2018) (11)
- Enantiospecific synthesis and cytotoxicity of 7-(4-methoxyphenyl)-6-phenyl-2,3,8,8a-tetrahydroindolizin-5(1H)-one enantiomers. (2008) (11)
- Formal total syntheses of the (-)-salicylihalamides A and B from D-glucose and L-rhamnose. (2005) (11)
- Artificial Neural Network—Based Analysis of High-Throughput Screening Data for Improved Prediction of Active Compounds (2009) (11)
- Biomimetic Aerobic C-H Olefination of Cyclic Enaminones at Room Temperature: Development toward the Synthesis of 1,3,5-Trisubstituted Benzenes. (2014) (11)
- A concise formal total synthesis of lactimidomycin. (2015) (10)
- Structure–Activity Studies of N‐Butyl‐1‐deoxynojirimycin (NB‐DNJ) Analogues: Discovery of Potent and Selective Aminocyclopentitol Inhibitors of GBA1 and GBA2 (2017) (10)
- Reformulating Tylocrebrine in Epidermal Growth Factor Receptor Targeted Polymeric Nanoparticles Improves Its Therapeutic Index (2015) (10)
- Enantioselective synthesis of a 3'-dephenylcryptophycin synthon. (1998) (10)
- Asymmetric synthesis of α-alkylated α-amino acids: azepane-2-carboxylic acids (1991) (10)
- SYNTHESIS AND BIOLOGY OF SUBSTITUTED 3'-PHENYL TAXOL ANALOGUES (1994) (10)
- Semisynthesis and biological evaluation of brevifoliol 13-[N-benzoyl-(-2′R,3′S)-3′-phenylisoserinate] (1993) (10)
- Synthesis and Spectral Properties of 8-Anilinonaphthalene-1-sulfonic Acid (ANS) Derivatives Prepared by Microwave-Assisted Copper(0)-Catalyzed Ullmann Reaction (2019) (10)
- Synthetic studies with 13-deoxybaccatin III. (2002) (10)
- THE CHEMISTRY OF THE TAXANE DITERPENE : STEREOSELECTIVE REDUCTIONS OF TAXANES (1998) (10)
- The first synthesis of a C-9 carbonyl modified baccatin III derivative and its conversion to novel taxol® and taxotere® analogues (1994) (10)
- Internal Nucleophile Assisted Selective Deesterification Studies on Baccatin III. Synthesis of 2-Debenzoyl- and 4-Deacetylbaccatin III Analogs (1994) (10)
- Synthesis and Cytotoxicity Evaluation of C4‐ and C5‐Modified Analogues of the α,β‐Unsaturated Lactone of Pironetin (2017) (10)
- Preparation of phenolic paclitaxel metabolites. (1996) (9)
- Total synthesis and anti-tubulin activity of epi-c3 analogues of cryptophycin-24. (2004) (9)
- Metal directed stereoselective synthesis of 3-(1'-hydroxyethyl)-2-azetidinones from ethyl 3-hydroxybutyrate (1990) (9)
- Total synthesis and antitubulin activity of c10 analogues of cryptophycin-24. (2004) (9)
- Reaction of 4-(iodomethyl)azetidin-2-ones with tetracarbonylferrate(II) (1983) (9)
- Synthesis and interactions of 7-deoxy-, 10-deacetoxy, and 10-deacetoxy-7-deoxypaclitaxel with NCI/ADR-RES cancer cells and bovine brain microvessel endothelial cells. (2006) (8)
- Digital chemistry in the Journal of Medicinal Chemistry. (2014) (8)
- Recombinant production of enzymatically active male contraceptive drug target hTSSK2 - Localization of the TSKS domain phosphorylated by TSSK2. (2016) (8)
- Syntheses of novel C-9 and C-10 modified bioactive taxanes (1995) (8)
- Ionic immobilization, diversification, and release: application to the generation of a library of methionine aminopeptidase inhibitors. (2008) (8)
- Erratum: Heme Binding Biguanides Target Cytochrome P450-Dependent Cancer Cell Mitochondria (Cell Chemical Biology (2017) 24(10) (1259–1275.e6) (S2451945617302830)(10.1016/j.chembiol.2017.08.009)) (2017) (8)
- Review of rationale and progress toward targeting cyclin-dependent kinase 2 (CDK2) for male contraception† (2020) (8)
- (3R,5S,7as)-(3,5-Bis(4-fluorophenyl)tetrahydro-1H-oxazolo[3,4-c]oxazol-7a-yl)methanol, a novel neuroprotective agent. (2009) (7)
- The chemistry of the taxane diterpene: Stereoselective synthesis of 10-deacetoxy-11,12-epoxypaclitaxel (1995) (7)
- The Fungal Sexual Pheromone Sirenin Activates the Human CatSper Channel Complex (2015) (7)
- Total synthesis and evaluation of C26-hydroxyepothilone D derivatives for photoaffinity labeling of beta-tubulin. (2010) (7)
- Intranasal Coadministration of a Diazepam Prodrug with a Converting Enzyme Results in Rapid Absorption of Diazepam in Rats (2019) (7)
- Stereoselective synthesis of 9β-hydroxytaxanes via reduction with samarium diiodide (1995) (7)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (7)
- Syntheses of PDE3A inhibitor ORG9935 and determination of the absolute stereochemistries of its enantiomers by X-ray crystallography. (2018) (7)
- Paclitaxel and docetaxel photoaffinity labels (1995) (7)
- Cooperativity Between Orthosteric Inhibitors and Allosteric Inhibitor 8-Anilino-1-Naphthalene Sulfonic Acid (ANS) in Cyclin-Dependent Kinase 2. (2020) (7)
- Synthesis and evaluation of C2 functionalized analogs of the α-tubulin-binding natural product pironetin. (2017) (7)
- Synthesis and evaluation of a β-lactam-containing dipeptide analog as a protease inhibitor (1996) (7)
- Enantioselective Synthesis of 3,4-Dihydro-1,2-oxazepin-5(2H)-ones and 2,3-Dihydropyridin-4(1H)-ones from β-Substituted β-Hydroxyaminoaldehydes (2014) (7)
- The Ecstasy and Agony of Assay Interference Compounds. (2017) (6)
- Women in Medicinal Chemistry Special Issue Call for Papers. (2019) (6)
- The use of polymer-bound triphenylphosphine in the stereochemical inversion of secondary alcohols. (2000) (6)
- Stereo- and enantio-controlled synthesis of chiral intermediates for the total synthesis of thienamycin and related β-lactam antibiotics from 3-hydroxybutyrates (1985) (6)
- Discovery and Characterization of Multiple Classes of Human CatSper Blockers (2022) (6)
- Transition in leadership: opportunities and challenges. (2012) (6)
- Chirally Pure Prodrugs and Their Converting Enzymes Lead to High Supersaturation and Rapid Transcellular Permeation of Benzodiazepines. (2016) (6)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (6)
- Retinoic acid receptor antagonists for male contraception: current status† (2020) (6)
- Confronting Racism in Chemistry Journals. (2020) (6)
- 7-O-acylpaclitaxel analogues: potential probes to map the paclitaxel binding site (1997) (5)
- Design, Synthesis, and Characterization of a Fluorescence Polarization Pan-BET Bromodomain Probe. (2018) (5)
- From HTS to Phase I: the Institute for Therapeutics Discovery and Development at the University of Minnesota. (2014) (5)
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- BRDT Inhibitors for Male Contraceptive Drug Discovery: Current Status (2018) (2)
- Enantiospecific Synthesis and Cytotoxicity Evaluation of Oximidine II Analogues (2016) (2)
- Investigation of 3'-debenzoyl-3'-(3-([¹²⁴I]-iodobenzoyl))paclitaxel analog as a radio-tracer to study multidrug resistance in vivo. (2012) (2)
- Synthesis, tubulin assembly, and antiproliferative activity against MCF7 and NCI/ADR-RES cancer cells of 10-O-acetyl-5'-hydroxybutitaxel. (2008) (2)
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- A ONE-STEP TRANSFORMATION OF AROMATIC ALDEHYDES TO NITRILES, USING S,S-DIMETHYLSULFURDIIMIDE AS IMINATING AGENT. ISOLATION OF DITHIATETRAZOCINES AS REACTION INTERMEDIATES (1985) (1)
- Anti-Spermatogenic Efficacy of Nonhormonal Male Contraceptive Agent, H2-Gamendazole, in Mice, Rats, Rabbits, and Nonhuman Primates (Rhesus), and a Multiple Low Dose Oral Regimen That Gives 100% Infertility with Complete Reversibility. (2011) (1)
- Formal Syntheses of Cryptophycin A and Arenastatin A. (1997) (1)
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- Confronting Racism in Chemistry Journals. (2020) (1)
- The orally active male contraceptive agent H2‐gamendazole interacts with organic anion transporting polypeptides expressed in human hepatocytes (1064.18) (2014) (1)
- Introduction: Drug Metabolism and Toxicology Special Issue. (2020) (1)
- Dehydrogenative Alkenylation of Uracils via Palladium-Catalyzed Regioselective C—H Activation. (2013) (1)
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- A convenient preparation of 2‐[15N]‐amino‐4,6‐dimethoxypyrimidine (1990) (1)
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- Effect of H2-Gamendazole and Other Indazole Carboxylic Acid (ICA) Analogs on Primary Rat Sertoli Cells Cytoskeletal Structure and Elongation Factor 1 Alpha (EEF1A1) Expression and Function. (2011) (1)
- Diversity-Oriented Library Synthesis from Steviol and Isosteviol-Derived Scaffolds. (2020) (1)
- In Vitro Versus In Vivo Effects of NB-DGJ and NB-DNJ as Lead Compounds for Development of Non-Hormonal Reversible Oral Male Contraceptives. (2010) (1)
- Screening through Lead Optimization of High Affinity, Allosteric Cyclin-Dependent Kinase 2 (CDK2) Inhibitors as Male Contraceptives That Reduce Sperm Counts in Mice. (2023) (1)
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- Steroidal Antagonists of Progesterone- and Prostaglandin E1-Induced Activation of the Cation Channel of Sperm (2021) (1)
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- N,O‐Dimethylhydroxylamine (2006) (1)
- α-Arylation of Enaminones Using Organotrifluoroborates (2008) (1)
- Advances toward COVID-19 Therapies Special Issue Call for Papers. (2020) (1)
- Synthesis of Arylazide‐ and Diazirine‐Containing CrAsH‐EDT2 Photoaffinity Probes (2016) (1)
- Abstract 2689: Breast cancer inhibition by a novel and potent biguanide, N1-hexyl-N5-benzyl-biguanide (2014) (1)
- The non-mevalonate pathway for isoprenoid biosynthesis: New opportunities for drug design (2000) (1)
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- Novel methods for the synthesis of N-trichloroacetyl- and N-formyl-S,S-diarylsulfilimines (1984) (1)
- Oxidation of Baccatin III at C14: A Facile Rearrangement of the Baccatin III Core. (2007) (1)
- Synthesis and Evaluation of Heteroaromatic 6,7‐Diaryl‐2,3,8,8a‐tetrahydroindolizin‐5(1H)‐ones for Cytotoxicity Against the HCT‐116 Colon Cancer Cell Line. (2008) (1)
- Asymmetric Synthesis of α‐Alkylated α‐Amino Acids: Azocane‐2‐carboxylic Acids. (1992) (1)
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- Epigenetics 2.0: Special Issue on Epigenetics-Call for Papers. (2020) (1)
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- Rapid Entry into the Cryptophycin Core via an Acyl-β-lactam Macrolactonization: Total Synthesis of Cryptophycin-24. (2001) (1)
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- Total synthesis and evaluation of 22-( 3-azidobenzoyloxy ) methyl epothilone C for photoaffinity labeling of β-tubulin (2010) (0)
- A one-step synthesis of a deuterated paclitaxel analogue: 10-deacetoxy-(10alpha-2H)paclitaxel. (1999) (0)
- Stereocontrolled Synthesis of N-Vinyl-, N-(1′-Propenyl)-, and N- Unsubstituted β-Lactams from 2-Aza-1,3-butadienes via the Staudinger Reaction. (1994) (0)
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- Probing the Paclitaxel-microtubule Binding Site and Interactions: Design, Synthesis and Evaluation of New Photoaffinity Taxoids (2000) (0)
- Effect of Gamendazole on Expression of Heat Shock Proteins HSP70 and HSP90 in Rat Testis and Primary Sertoli Cells. (2009) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Pharmaco Chemistry Library, Vol. 22. The Chemistry and Pharmacology of Taxol® and its Derivatives By Vittorio Farina, Boehringer-Ingelheim Pharmaceuticals. Elsevier Science, Tarrytown, NY. 1995. ix + 339 pp. 16.5 × 24 cm. $350.00. ISBN 0-444-81771-9. (1998) (0)
- Stereoselective syn-Aldol Reaction of the Lithium Ester Enolate of Ethyl N,N-Dimethylglycine in the Presence of Triethylborane. (1992) (0)
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- Correction to BET Bromodomain Inhibitors with One-Step Synthesis Discovered from Virtual Screen. (2017) (0)
- Development of allosteric, selective cyclin-dependent kinase 2 (CDK2) inhibitors that are negatively cooperative with cyclin binding and show potential as contraceptive agents (2022) (0)
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- Stereoselective Synthesis of 9β-Hydroxytaxanes via Reduction with Samarium Diiodide. (1995) (0)
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- Asymmetric Synthesis of β‐Lactams (III) and N‐Benzoyl‐3‐ phenylisoserines (VI) via the Staudinger Reaction. (1992) (0)
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- Enhancing the Visibility of Women in the ACS Division of Medicinal Chemistry (ACS MEDI). (2023) (0)
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- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Synthesis of 2-O-Heteroaroyl Taxanes: Evaluation of Microtubule Assembly Promotion and Cytotoxicity. (2010) (0)
- Hepatitis C virus (HCV) therapies special thematic issue: call for papers. (2013) (0)
- Cover Picture: Enantiospecific Synthesis and Cytotoxicity Evaluation of Oximidine II Analogues (ChemMedChem 15/2016) (2016) (0)
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- Short and Efficient Chiral Pool and RCM Approach Towards the Synthesis of the Macrocyclic Core of the Salicylihalamides. (2001) (0)
- Editorial Confronting Racism in Chemistry Journals (2020) (0)
- Formal Total Synthesis of (+)‐Salicylihalamides A (Ia) and B (Ib): A Combined Chiral Pool and RCM Strategy. (2004) (0)
- Total Synthesis of Cryptophycin‐24 (Arenastatin A) (III) Amenable to Structural Modifications in the C16 Side Chain. (2001) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Enhancing the Visibility of Women in the ACS Division of Medicinal Chemistry (ACS MEDI). (2023) (0)
- Direct Hiyama Cross‐Coupling of Enaminones with Triethoxy(aryl)silanes and Dimethylphenylsilanol. (2012) (0)
- Preparation and Three‐Carbon + Two‐Carbon Cycloaddition of Cyclopropenone 1,3‐propanediol ketal: 5,5‐Dicyano‐4‐phenyl‐2‐cyclopenten‐1‐one 1,3‐propanediol ketal (2003) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
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- STEREOSELECTIVE SYNTHESIS OF 3-(1-HYDROXYETHYL)-2-AZETIDINONES FROM 3-HYDROXYBUTYRATES (1985) (0)
- Targeting carrier-mediated transport to improve the blood-brain barrier permeation of paclitaxel (2006) (0)
- 2-Aza-1,3-dienes as Novel Precursors for the Synthesis of N-Unsubstituted β-Lactams. A Three Step Synthesis of 4-Acetoxy-3-phenoxy-2-azetidinone. (1988) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Formal Total Syntheses of the (-)-Salicylihalamides A (Ia) and B (Ib) from D-Glucose and L-Rhamnose. (2006) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- A Novel and Expeditious Reduction of Tertiary Amides to Aldehydes Using Cp2Zr(H)Cl. (2001) (0)
- Synthese d'epothilones (2000) (0)
- Experiences in Academic and Industry Partnerships – Forging a Path to Translational Drug Discovery (2021) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- 1,4‐Dihydropyridinebutyrolactone‐derived ring‐opened ester and amide analogs targeting BET bromodomains (2022) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities—April 2020 (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Efficient and Practical Asymmetric Synthesis of the Taxol C‐13 Side Chain, N‐Benzoyl‐(2R,3S)‐3‐phenylisoserine, and Its Analogues via Chiral 3‐Hydroxy‐4‐aryl‐β‐lactams Through Chiral Ester Enolate. (1991) (0)
- An Efficient Gram‐Scale Synthesis of (+)‐Discodermolide (2000) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- An Improved Method for the Stereoselective Synthesis of β‐Lactams from Carboxylic Acids and Imines. (1991) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Abstract 3568: CYP3A4 epoxygenase activity mediates ER+ mammary tumor growth and angiogenesis, in part, through EET biosynthesis and is inhibited by biguanides (2015) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- CatSper as a Target for Male Contraception (2016) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities - April 2020 (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals (2020) (0)
- Synthesis of cryptophycins via an N-acyl-beta-lactam macrolactonization. (2003) (0)
- Topliss Approach to the Synthesis of Biologically Active Substituted N- Benzoyl Taxol Analogues. (1995) (0)
- Rapid Delivery of Diazepam from Supersaturated Solutions Prepared Using Prodrug/Enzyme Mixtures: Toward Intranasal Treatment of Seizure Emergencies (2014) (0)
- Synthesis of 6‐ and 7‐Membered Cyclic Enaminones: Scope and Mechanism. (2011) (0)
- Transition Metal-Free Direct Trifluoromethylation of 2,3-Dihydropyridin-4(1H)-ones at Room Temperature. (2015) (0)
- Drug Metabolism and Toxicology Special Issue Call for Papers. (2019) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Exploiting the Potential of Iminosugars as Novel Reversible Non-Hormonal Male Contraceptive. (2008) (0)
- Taxol Photoaffinity Labels. Part 2. Synthesis and Biological Evaluation of N-(4-Azidobenzoyl)-N-debenzoyltaxol, N-(4-Azido-2,3,5,6- tetrafluorobenzoyl)-N-debenzoyltaxol, and 7-(4-Azido-2,3,5,6- tetrafluorobenzoyl)taxol. (1994) (0)
- Asymmetric Synthesis of α‐Alkylated α‐Amino Acids: Azepane‐2‐carboxylic Acids. (2010) (0)
- Pancreatic Cancer A Preclinical Evaluation of Minnelide as a Therapeutic Agent Against (2012) (0)
- Dihydropyridine Lactam Analogs Targeting BET Bromodomains (2021) (0)
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- Synthesis and Biology of Substituted 3′-Phenyl Taxol Analogues. (1995) (0)
- Drug Metabolism and Toxicology Special Issue Call for Papers. (2019) (0)
- Cover Picture: Biomimetic Aerobic CH Olefination of Cyclic Enaminones at Room Temperature: Development toward the Synthesis of 1,3,5‐Trisubstituted Benzenes (Adv. Synth. Catal. 6/2014) (2014) (0)
- Asymmetric Synthesis of α-Alkylated α-Amino Acids (IV) and (V) via Schmidt Rearrangement of α,α-Bisalkylated β-Keto Esters (I). (1988) (0)
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- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Samarium Diiodide Mediated Deoxygenation of Taxol: A One-Step Synthesis of 10-Deacetoxytaxol (IIa). (1995) (0)
- Allosteric Modulators of Drug Targets Special Issue. (2018) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Effect of H2-Gamendazole on Rapid HSF1 Expression and Interaction with Heat Shock Proteins in Rat Testis In Vivo and Primary Sertoli Cells. (2010) (0)
- Stereo‐ and Enantio‐Controlled Synthesis of Chiral Intermediates for the Total Synthesis of Thienamycin and Related β‐Lactam Antibiotics fromh 3‐Hydroxybutyrates. (1986) (0)
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- Synthesis of Dihydropyridin-4(1H)-onesvia Wolff Rearrangement (2011) (0)
- The lonidamine derivative H2-gamendazole reduces cyst formation in polycystic kidney disease (2020) (0)
- Confronting Racism in Chemistry Journals (2020) (0)
- Erratum: Asymmetric synthesis of (1′R,3R,4R)-4-acetoxy-3-(1′-((tert-butyldimethylsilyl)oxy)ethyl)-2- azetidinone and other 3-(1′-hydroxyethyl)-2-azetidinones from (S)-(+)-ethyl 3-hydroxybutanoate: Formal total synthesis of (+)-thienamycin (Journal of the American Chemical Society (1987) 109 (1129-11 (1987) (0)
- The Chemistry of the Taxane Diterpene: Stereoselective Synthesis of 10- Deacetoxy-11,12-epoxypaclitaxel. (1996) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Palladium-Catalyzed Direct C—H Arylation of Cyclic Enaminones with Aryl Iodides. (2013) (0)
- P3-192 Parallels between ER-stress and Aβ-induced toxicity in primary neurons: involvement of the cytoskeletal network (2004) (0)
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- 3-(1′-HYDROXYETHYL)-2-AZETIDINONES FROM 3-HYDROXYBUTYRATES AND N-ARYLALDIMINES (1985) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Topics in Medicinal Chemistry (2009) (0)
- Gene Therapy for Rare Diseases : Promise and Challenges February 23 , 2018 11 : 00 AM2 : 30 (2018) (0)
- Abstract A105: Minnelide, a potent chemotherapeutic agent, causes pancreatic tumor regression. (2012) (0)
- Update to Our Reader, Reviewer, and Author Communities—April 2020 (2020) (0)
- KU-AS-272, a Potential Single-Dose Sterilant for Cats and Dogs, Shows Safety and Ability to Block Spermatogenesis in Testis to Sertoli Cells Only after a Single Subcutaneous Injection in Male Rat. (2012) (0)
- Novel D‐Seco Paclitaxel Analogues: Synthesis, Biological Evaluation, and Model Testing. (2001) (0)
- Ongoing in vivo studies with cytoskeletal drugs in tau transgenic mice (Current Alzheimer Research 3, 3, (215-219)) (2009) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Current Medicinal Chemistry Research in India: Progress and Opportunities. (2017) (0)
- Abstract LB078: Hexyl-(cuban-1-yl-methyl)-biguanide (HCB) inhibits hormone therapy resistant breast cancer cells, in part by Inhibiting CYP3A4 arachidonic acid epoxygenase activity (2021) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Editorial preface (1999) (0)
- Abstract 1771: Therapeutic management of pancreatic cancer using a novel drug, Minnelide (2010) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- The First Synthesis of a C‐9 Carbonyl Modified Baccatin III Derivative and Its Conversion to Novel Taxol and Taxotere Analogues. (1995) (0)
- Issue Information (2021) (0)
- Metal Ion-Directed Stereoselective Synthesis of 3-(1′-Hydroxyethyl)-2- azetidinones from Ethyl 3-Hydroxybutyrate. (1991) (0)
- Abstract 44: Hexyl-benzyl-biguanide (HBB) potently and selectively inhibits CYP3A4 epoxygenase activity and inhibits EET stabilization of mitochondrial respiration in ER+HER2- breast cancer cells, inducing glycolysis and pyruvate biosynthesis (2016) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Synthesis of Cryptophycin Affinity Labels and Tubulin Labeling (2005) (0)
- Asymmetric Synthesis of (1′R,3R,4R)-4-Acetoxy-3-(1′-((tert-butyldimethylsilyl)oxy)ethyl)-2-azetidinone and Other 3-(1′-Hydroxyethyl)-2-azetidinones from (S)-(+)-Ethyl 3-Hydroxybutanoate: Formal Total Synthesis of (+)-Thienamycin. (1987) (0)
- Corrigendum: Discovery and Characterization of Multiple Classes of Human CatSper Blockers (2022) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Special Section on Drug Delivery Technologies Intranasal Coadministration of a Diazepam Prodrug with a Converting Enzyme Results in Rapid Absorption of Diazepam in Rats s (2019) (0)
- Alzheimer's disease special thematic issue: call for papers. (2012) (0)
- The NIH COBRE Center for Cancer Experimental Therapeutics at the University of Kansas. (2004) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- DFG-1 Binding: A New Residue for Developing Selective Kinase Inhibitors. (2020) (0)
- The Candidate Male Contraceptive Agent, Gamendazole, Affects Actin Organization and Vinculin Based Focal Contact Distribution in Sertoli Cells In Vitro. (2008) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Investigation of 3 0-debenzoyl-3 0-( 3-( [ 124 I ]-iodobenzoyl ) ) paclitaxel analog as a radio-tracer to study multidrug resistance in vivo (2012) (0)
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- Confronting Racism in Chemistry Journals (2020) (0)
- A Message from the Editors-in-Chief. (2019) (0)
- Boron—Heck Reaction of Cyclic Enaminones: Regioselective Direct Arylation via Oxidative Palladium(II) Catalysis. (2014) (0)
- Construction of Affinity Probes to Study the Epothilone Binding Site on Tubulin (2003) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Enabling Science: Selective Reduction with ZrHCl(Cp)2 (2001) (0)
- Abstract LB102: Hexyl-(cuban-1-yl-methyl)-biguanide (HCB) suppresses N-glycosylation of immune checkpoint proteins B7-H3 and B7-H4, reverses tumor hypoxia, decreases intratumoral regulatory T cells, and increases intratumoral CD8+ T cells in the ovarian dependent ER+HER2- SSM2ucd mammary cancer allo (2023) (0)
- A Facile One-Flask Conversion of Aldehydes and Ketones to N-Sulfonyl Imines. (1996) (0)
- AMIDO- AND AMINO-ALKYLATION OF SULFIMIDES, SULFOXIMIDES, AND SULFODIIMIDES (1979) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- CPNP 2019 Annual Meeting Poster Abstracts (2019) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Syntheses of Novel C-9 and C-10 Modified Bioactive Taxanes. (1995) (0)
- 570 Minnelide as an Emerging Single Therapeutic Agent Against Pancreatic Cancer (2010) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Effective Thermal One-Carbon + Two-Carbon Cycloaddition to Cyclopropenone Ketals with Electron-Deficient Olefins: Cyclopropane Formation. Thermal Three-Carbon + Two-Atom Cycloaddition of Cyclopropenone Ketals with Carbon-Heteroatom Do (1985) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Update to Our Reader, Reviewer, and Author Communities-April 2020. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
- Confronting Racism in Chemistry Journals. (2020) (0)
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