Horst Kessler
#63,424
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German chemist
Horst Kessler's AcademicInfluence.com Rankings
Horst Kesslerchemistry Degrees
Chemistry
#841
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#1382
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Organic Chemistry
#88
World Rank
#121
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Chemistry
Why Is Horst Kessler Influential?
(Suggest an Edit or Addition)According to Wikipedia, Horst Kessler is a German chemist and emeritus Professor of Excellence at the Institute for Advanced Study at the Technical University of Munich . Kessler works in the area of bioorganic chemistry, in particular peptide synthesis, and nuclear magnetic resonance spectroscopy. He also made contributions to magnetic resonance imaging.
Horst Kessler's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- RGD modified polymers: biomaterials for stimulated cell adhesion and beyond. (2003) (2235)
- Activation of integrin function by nanopatterned adhesive interfaces. (2004) (1083)
- Cell spreading and focal adhesion dynamics are regulated by spacing of integrin ligands. (2007) (838)
- N-methylated cyclic RGD peptides as highly active and selective αvβ3 integrin antagonists (1999) (713)
- Conformation and Biological Activity of Cyclic Peptides (1982) (711)
- Noninvasive Imaging of αvβ3 Integrin Expression Using 18F-labeled RGD-containing Glycopeptide and Positron Emission Tomography (2001) (546)
- Structural and Functional Aspects of RGD-Containing Cyclic Pentapeptides as Highly Potent and Selective Integrin αVβ3 Antagonists (1996) (538)
- Cilengitide: The First Anti-Angiogenic Small Molecule Drug Candidate. Design, Synthesis and Clinical Evaluation (2010) (526)
- Assignment of carbonyl carbons and sequence analysis in peptides by heteronuclear shift correlation via small coupling constants with broadband decoupling in t1 (COLOC) (1984) (519)
- Arg‐Gly‐Asp constrained within cyclic pentapoptides Strong and selective inhibitors of cell adhesion to vitronectin and laminin fragment P1 (1991) (506)
- Noninvasive Visualization of the Activated αvβ3 Integrin in Cancer Patients by Positron Emission Tomography and [18F]Galacto-RGD (2005) (494)
- Impact of order and disorder in RGD nanopatterns on cell adhesion. (2009) (481)
- Selective recognition of cyclic RGD peptides of NMR defined conformation by alpha IIb beta 3, alpha V beta 3, and alpha 5 beta 1 integrins. (1994) (439)
- Detection of Hindered Rotation and Inversion by NMR Spectroscopy (1970) (433)
- Glycosylated RGD-containing peptides: tracer for tumor targeting and angiogenesis imaging with improved biokinetics. (2001) (409)
- Nachweis gehinderter Rotationen und Inversionen durch NMR‐Spektroskopie (1970) (384)
- Perspectives on NMR in drug discovery: a technique comes of age (2008) (362)
- Stereoisomeric Peptide Libraries and Peptidomimetics for Designing Selective Inhibitors of the αvβ3 Integrin for a New Cancer Therapy (1997) (358)
- A conserved spider silk domain acts as a molecular switch that controls fibre assembly (2010) (357)
- Radiolabeled αvβ3 Integrin Antagonists: A New Class of Tracers for Tumor Targeting (1999) (355)
- A Comprehensive Evaluation of the Activity and Selectivity Profile of Ligands for RGD-binding Integrins (2017) (349)
- Two‐Dimensional NMR Spectroscopy: Background and Overview of the Experiments [New Analytical Methods (36)] (1988) (346)
- N-methylation of peptides: a new perspective in medicinal chemistry. (2008) (334)
- Carbohydrate-based mimetics in drug design: sugar amino acids and carbohydrate scaffolds. (2002) (327)
- Lateral spacing of integrin ligands influences cell spreading and focal adhesion assembly. (2006) (326)
- N-methylation of peptides and proteins: an important element for modulating biological functions. (2013) (324)
- [18F]Galacto-RGD: synthesis, radiolabeling, metabolic stability, and radiation dose estimates. (2004) (306)
- Positron Emission Tomography Using [18F]Galacto-RGD Identifies the Level of Integrin αvβ3 Expression in Man (2006) (303)
- Surface Coating with Cyclic RGD Peptides Stimulates Osteoblast Adhesion and Proliferation as well as Bone Formation (2000) (302)
- Separation of cross-relaxation and J cross-peaks in 2D rotating-frame NMR spectroscopy (1987) (300)
- Peptide conformations. Part 31. The conformation of cyclosporin a in the crystal and in solution (1985) (298)
- Conformation/activity studies of rationally designed potent anti-adhesive RGD peptides. (1992) (290)
- Induction of cell polarization and migration by a gradient of nanoscale variations in adhesive ligand spacing. (2008) (286)
- Transformation of homonuclear two-dimensional NMR techniques into one-dimensional techniques using Gaussian pulses (1986) (286)
- Exploring the Role of RGD-Recognizing Integrins in Cancer (2017) (281)
- Improving oral bioavailability of peptides by multiple N-methylation: somatostatin analogues. (2008) (281)
- Targeting RGD recognizing integrins: drug development, biomaterial research, tumor imaging and targeting. (2006) (267)
- Ligands for mapping alphavbeta3-integrin expression in vivo. (2009) (259)
- Multimeric cyclic RGD peptides as potential tools for tumor targeting: solid-phase peptide synthesis and chemoselective oxime ligation. (2003) (258)
- WT p53, but Not Tumor-derived Mutants, Bind to Bcl2 via the DNA Binding Domain and Induce Mitochondrial Permeabilization* (2006) (243)
- The N-terminal domain of p53 is natively unfolded. (2003) (239)
- Asymmetric activation of the hsp90 dimer by its cochaperone aha1. (2010) (230)
- Two-step methodology for high-yield routine radiohalogenation of peptides: (18)F-labeled RGD and octreotide analogs. (2004) (228)
- Radiolabelled RGD peptides for imaging and therapy (2012) (211)
- The architecture of functional modules in the Hsp90 co‐chaperone Sti1/Hop (2012) (209)
- The RGD motif in fibronectin is essential for development but dispensable for fibril assembly (2007) (208)
- An unfolded CH1 domain controls the assembly and secretion of IgG antibodies. (2009) (203)
- N-Methylated cyclic RGD peptides as highly active and selective alpha(V)beta(3) integrin antagonists. (1999) (203)
- Cell adhesion strength is controlled by intermolecular spacing of adhesion receptors. (2010) (193)
- Tumor Targeting via Integrin Ligands (2013) (193)
- Noninvasive imaging of alpha(v)beta3 integrin expression using 18F-labeled RGD-containing glycopeptide and positron emission tomography. (2001) (188)
- Protein repellent properties of covalently attached PEG coatings on nanostructured SiO(2)-based interfaces. (2007) (187)
- Photoswitched cell adhesion on surfaces with RGD peptides. (2005) (186)
- CONFORMATIONAL DYNAMICS DETECTED BY NUCLEAR MAGNETIC-RESONANCE NOE VALUES AND J-COUPLING CONSTANTS (1988) (184)
- PET of CXCR4 Expression by a 68Ga-Labeled Highly Specific Targeted Contrast Agent (2011) (183)
- Cell adhesion and proliferation on RGD-modified recombinant spider silk proteins. (2012) (183)
- Imaging of integrin alpha(v)beta(3) expression in patients with malignant glioma by [18F] Galacto-RGD positron emission tomography. (2009) (181)
- The Kinetic and Mechanistic Evaluation of NMR Spectra. New analytical methods (18) (1980) (176)
- The CLIP/CLAP-HSQC: pure absorptive spectra for the measurement of one-bond couplings. (2008) (175)
- Nanomolar Small Molecule Inhibitors for αvβ6, αvβ5, and αvβ3 Integrins (2002) (165)
- Hsp90 is regulated by a switch point in the C‐terminal domain (2009) (162)
- Zweidimensionale NMR‐Spektroskopie, Grundlagen und Übersicht über die Experimente (1988) (160)
- Cell interactions with hierarchically structured nano-patterned adhesive surfaces. (2009) (159)
- Hsp12 is an intrinsically unstructured stress protein that folds upon membrane association and modulates membrane function. (2010) (158)
- The structures of integrins and integrin-ligand complexes: implications for drug design and signal transduction. (2002) (157)
- Disclosing the CXCR4 Expression in Lymphoproliferative Diseases by Targeted Molecular Imaging (2015) (155)
- Intestinal permeability of cyclic peptides: common key backbone motifs identified. (2012) (154)
- Peptide conformations. Part 30. Assignment of the 1H‐, 13C‐, and 15N‐NMR spectra of cyclosporin A in CDCl3 and C6D6 by a combination of homo‐ and heteronuclear two‐dimensional techniques (1985) (148)
- PET Imaging of CXCR4 Receptors in Cancer by a New Optimized Ligand (2011) (143)
- PET/CT imaging of integrin αvβ3 expression in human carotid atherosclerosis. (2014) (139)
- Synthesis and Conformational Analysis of Linear and Cyclic Peptides Containing Sugar Amino Acids (1996) (138)
- Impact of local versus global ligand density on cellular adhesion. (2011) (138)
- Multi‐dimensional NMR experiments using selective pulses (1991) (130)
- Peptide conformations. 28. Relayed heteronuclear correlation spectroscopy and conformational analysis of cyclic hexapeptides containing the active sequence of somatostatin (1983) (129)
- Radiolabeled alpha(v)beta3 integrin antagonists: a new class of tracers for tumor targeting. (1999) (127)
- Mimicking cellular environments by nanostructured soft interfaces. (2007) (123)
- The urokinase plasminogen activator system as a novel target for tumour therapy (2000) (122)
- PET Imaging of Integrin αVβ3 Expression (2011) (120)
- RGD-peptides for tissue engineering of articular cartilage. (2002) (120)
- Measurement of fast proton exchange rates in isotopically labeled compounds (1993) (120)
- The effect of multiple N-methylation on intestinal permeability of cyclic hexapeptides. (2011) (120)
- pH-dependent dimerization and salt-dependent stabilization of the N-terminal domain of spider dragline silk--implications for fiber formation. (2011) (120)
- Assessment of alphavbeta3 integrin expression after myocardial infarction by positron emission tomography. (2008) (118)
- Selective RGD-Mediated Adhesion of Osteoblasts at Surfaces of Implants. (1999) (118)
- Positron emission tomography using [18F]Galacto-RGD identifies the level of integrin alpha(v)beta3 expression in man. (2006) (117)
- Scalar Coupling Constants—Their Analysis and Their Application for the Elucidation of Structures (1995) (116)
- Stretched poly(dimethylsiloxane) gels as NMR alignment media for apolar and weakly polar organic solvents: an ideal tool for measuring RDCs at low molecular concentrations. (2004) (114)
- N-methylated cyclic pentaalanine peptides as template structures. (2006) (114)
- Cooperativity in adhesion cluster formation during initial cell adhesion. (2008) (113)
- Cyclic RGD Peptides Containing β-Turn Mimetics (1996) (112)
- The Redox Potential of Selenocystine in Unconstrained Cyclic Peptides (1997) (112)
- Structural analysis of the interaction between Hsp90 and the tumor suppressor protein p53 (2011) (111)
- Applications of NMR in drug discovery. (2001) (111)
- An easy and scalable method for the partial alignment of organic molecules for measuring residual dipolar couplings. (2004) (111)
- HETLOC, an Efficient Method for Determining Heteronuclear Long‐Range Couplings with Heteronuclei in Natural Abundance (1991) (111)
- Cyclic RGD peptides ameliorate ischemic acute renal failure in rats. (1994) (110)
- Peptide conformations. 46. Conformational analysis of a superpotent cytoprotective cyclic somatostatin analog (1988) (110)
- N‐Methylation of Peptides: A New Perspective in Medicinal Chemistry (2009) (107)
- Carbohydrate Derivatives for Use in Drug Design: Cyclicαv-Selective RGD Peptides (2000) (106)
- Improving oral bioavailability of cyclic peptides by N-methylation. (2017) (105)
- Reinvestigation of the Conformation of Cyclosporin A in Chloroform (1990) (104)
- Titanium Implant Materials with Improved Biocompatibility through Coating with Phosphonate‐Anchored Cyclic RGD Peptides (2005) (104)
- Docking studies on αvβ3 integrin ligands: Pharmacophore refinement and implications for drug design (2003) (103)
- p53--a natural cancer killer: structural insights and therapeutic concepts. (2006) (102)
- Stereoisomerism and Biological Activity of the Selective and Superactive αvβ3 Integrin Inhibitor cyclo(-RGDfV-) and Its Retro-Inverso Peptide (1997) (101)
- Stretched gelatin gels as chiral alignment media for the discrimination of enantiomers by NMR spectroscopy. (2005) (101)
- Design, synthesis, and NMR structure of linear and cyclic oligomers containing novel furanoid sugar amino acids. (2002) (101)
- 3-Substituted indolizine-1-carbonitrile derivatives as phosphatase inhibitors. (2006) (101)
- Die kinetische und mechanistische Auswertung von NMR-Spektren. Neue analytische Methoden (18)† (1980) (100)
- Optimized selective N‐methylation of peptides on solid support (2006) (99)
- Structure refinement using time-averaged J-coupling constant restraints (1993) (99)
- Automated backbone assignment of labeled proteins using the threshold accepting algorithm (1998) (98)
- 68Ga-NODAGA-RGD is a suitable substitute for (18)F-Galacto-RGD and can be produced with high specific activity in a cGMP/GRP compliant automated process. (2012) (98)
- Residual dipolar coupling constants: An elementary derivation of key equations (2004) (97)
- Introducing lasso peptides as molecular scaffolds for drug design: engineering of an integrin antagonist. (2011) (97)
- First 18F-Labeled Tracer Suitable for Routine Clinical Imaging of sst Receptor-Expressing Tumors Using Positron Emission Tomography (2004) (96)
- Synthesis of N-methylated cyclic peptides (2012) (95)
- Peptide conformations. 42. Conformation of side chains in peptides using heteronuclear coupling constants obtained by two-dimensional NMR spectroscopy (1987) (95)
- Design, synthesis, and functionalization of dimeric peptides targeting chemokine receptor CXCR4. (2011) (93)
- A Sugar Amino Acid as a Novel Peptidomimetic (1994) (91)
- Multiple N-methylation of MT-II backbone amide bonds leads to melanocortin receptor subtype hMC1R selectivity: pharmacological and conformational studies. (2010) (90)
- Cellular unbinding forces of initial adhesion processes on nanopatterned surfaces probed with magnetic tweezers. (2006) (89)
- NMR investigation of the multidrug transporter EmrE, an integral membrane protein. (1998) (89)
- An efficient strategy for assignment of cross-peaks in 3D heteronuclear NOESY experiments (1999) (88)
- Probing Integrin Selectivity: Rational Design of Highly Active and Selective Ligands for the α5β1 and αvβ3 Integrin Receptor (2007) (87)
- αvβ3- or α5β1-Integrin-Selective Peptidomimetics for Surface Coating. (2016) (85)
- Hsp90 regulates the dynamics of its cochaperone Sti1 and the transfer of Hsp70 between modules (2015) (85)
- The solution structure and dynamics of human neutrophil gelatinase-associated lipocalin. (1999) (85)
- First poly(2-oxazoline)s with pendant amino groups (2006) (84)
- Telethonin Deficiency Is Associated With Maladaptation to Biomechanical Stress in the Mammalian Heart (2011) (84)
- NMR Spectroscopy Reveals the Solution Dimerization Interface of p53 Core Domains Bound to Their Consensus DNA* (2001) (84)
- Chemoselective pre-conjugate radiohalogenation of unprotected mono- and multimeric peptides via oxime formation (2004) (84)
- Cell adhesion and polarisation on molecularly defined spacing gradient surfaces of cyclic RGDfK peptide patches. (2008) (84)
- New evidence for a membrane-bound pathway in hormone receptor binding. (1993) (83)
- Design and chemical synthesis of integrin ligands. (2007) (83)
- Transmembrane signal transduction of the αIIbβ3 integrin (2002) (82)
- Solid-Phase Synthesis of a Nonpeptide RGD Mimetic Library: New Selective αvβ3 Integrin Antagonists (2001) (82)
- Stretched poly(vinyl acetate) gels as NMR alignment media for the measurement of residual dipolar couplings in polar organic solvents. (2005) (81)
- Thiocyclosporins: Preparation, Solution and Crystal Structure, and Immunosuppressive Activity (1991) (80)
- βVI Turns in peptides and proteins: A model peptide mimicry (1993) (80)
- Structure Refinement of Cyclosporin A in Chloroform by Using RDCs Measured in a Stretched PDMS‐Gel (2005) (80)
- Peptide flexibility and calculations of an ensemble of molecules (1994) (79)
- Functionalizing αvβ3- or α5β1-selective integrin antagonists for surface coating: a method to discriminate integrin subtypes in vitro. (2013) (78)
- NMR Chemical Shift Perturbation Study of the N‐Terminal Domain of Hsp90 upon Binding of ADP, AMP‐PNP, Geldanamycin, and Radicicol (2003) (77)
- Novel backbone conformation of cyclosporin A: the complex with lithium chloride (1992) (77)
- Convenient synthesis of N-methylamino acids compatible with Fmoc solid-phase peptide synthesis. (2005) (77)
- Conformation of cyclic peptides. Principle concepts and the design of selectivity and superactivity in bioactive sequences by 'spatial screening' (1996) (76)
- Mimicking bone extracellular matrix: integrin-binding peptidomimetics enhance osteoblast-like cells adhesion, proliferation, and differentiation on titanium. (2015) (76)
- NMR-based screening: a powerful tool in fragment-based drug discovery. (2006) (76)
- Konformation und biologische Wirkung von cyclischen Peptiden (2006) (76)
- Epitope-mapped monoclonal antibodies as tools for functional and morphological analyses of the human urokinase receptor in tumor tissue. (1997) (75)
- Urokinase-type plasminogen activator (uPA) and its receptor (uPAR): development of antagonists of uPA/uPAR interaction and their effects in vitro and in vivo. (2003) (73)
- Conformational control of integrin-subtype selectivity in isoDGR peptide motifs: a biological switch. (2010) (73)
- Integrin αvβ3/Vitronectin Interaction Affects Expression of the Urokinase System in Human Ovarian Cancer Cells* (2001) (73)
- Solid-phase-assisted synthesis of targeting peptide-PEG-oligo(ethane amino)amides for receptor-mediated gene delivery. (2012) (73)
- STEREOSELECTIVE SYNTHESIS OF A C-GLYCOSIDIC ANALOG OF N-GLUCOASPARAGINE (1997) (72)
- Peptoids—A New Approach to the Development of Pharmaceuticals (1993) (72)
- Combined Approach of NMR and Molecular Dynamics within a biphasic Membrane Mimetic: Conformation and Orientation of the Bradykinin Antagonist Hoe 140 (1994) (72)
- Multiple N-methylation by a designed approach enhances receptor selectivity. (2007) (71)
- The solution structure of VAT-N reveals a ‘missing link’ in the evolution of complex enzymes from a simple βαββ element (1999) (71)
- Recognition of NMR proton spin systems of cyclosporin A via heteronuclear proton-carbon long-range couplings (1985) (71)
- Mediating specific cell adhesion to low-adhesive diblock copolymers by instant modification with cyclic RGD peptides. (2005) (70)
- BclxL Changes Conformation upon Binding to Wild-type but Not Mutant p53 DNA Binding Domain* (2009) (70)
- Nachweis innermolekularer beweglichkeit durch NMR-spektroskopie—XV : Untersuchungen zur inversion am doppelt gebundenen stickstoffatom am beispiel der tetramethylguanidine (1970) (69)
- Novel Solid-Phase Synthesis of Azapeptides and Azapeptoides via Fmoc-Strategy and Its Application in the Synthesis of RGD-Mimetics (1999) (69)
- Rational Design of Highly Active and Selective Ligands for the α5β1 Integrin Receptor (2008) (69)
- Molecular targeting with peptides or peptide-polymer conjugates: just a question of size? (2005) (69)
- Systematic mutational analysis of the receptor-binding region of the human urokinase-type plasminogen activator. (1996) (69)
- Ligand Binding Analysis for Human α5β1 Integrin: Strategies for Designing New α5β1 Integrin Antagonists (2005) (68)
- Determination of Connectivities via Small Proton‐Carbon Couplings with a New Two‐Dimensional NMR Technique (1984) (68)
- The Structure of the Polycyclic Nonadecapeptide Ro 09-0198† (1988) (67)
- Thermal isomerization about double bonds: Rotation and inversion (1974) (67)
- Intrinsic Inhibition of the Hsp90 ATPase Activity* (2006) (67)
- Modified somatostatins as inhibitors of a multispecific transport system for bile acids and phallotoxins in isolated hepatocytes. (1985) (67)
- Orally Active Peptides: Is There a Magic Bullet? (2018) (67)
- Urokinase induces proliferation of human ovarian cancer cells: characterization of structural elements required for growth factor function (1998) (67)
- Improvement of NMR experiments by employing semiselective half-Gaussian-shaped pulses (1989) (66)
- Implementation of the DEPT sequence in inverse shift correlation; the DEPT-HMQC (1989) (66)
- Polymeric substrates with tunable elasticity and nanoscopically controlled biomolecule presentation. (2010) (66)
- Two‐Dimensional NMR Spectroscopy: Background and Overview of the Experiments (1988) (66)
- Complete Sequence Determination and Localisation of One Imino and Three Sulfide Bridges of the Nonadecapeptide Ro 09–0198 by Homonuclear 2D-NMR Spectroscopy. The DQF-RELAYED-NOESY-Experiment† (1987) (66)
- Integrin modulators: a patent review (2013) (66)
- Molecular dynamics with dimethyl sulfoxide as a solvent. Conformation of a cyclic hexapeptide (1991) (65)
- Cyclic homooligomers from sugar amino acids: synthesis, conformational analysis, and significance. (2001) (65)
- Diffusion NMR Spectroscopy: Folding and Aggregation of Domains in p53 (2005) (64)
- Orientational properties of stretched polystyrene gels in organic solvents and the suppression of their residual 1H NMR signals. (2005) (63)
- Nanomolar small molecule inhibitors for alphav(beta)6, alphav(beta)5, and alphav(beta)3 integrins. (2002) (63)
- Inhibition of the Interaction of Urokinase-Type Plasminogen Activator (uPA) with Its Receptor (uPAR) by Synthetic Peptides (1997) (62)
- Biselectivity of isoDGR peptides for fibronectin binding integrin subtypes α5β1 and αvβ6: conformational control through flanking amino acids. (2013) (62)
- The solution structure of the N-terminal domain of riboflavin synthase. (2001) (61)
- Nomenclature for Intramolecular Exchange Processes (1971) (61)
- Conformational Prerequisites for the in vitro Inhibition of Cholate Uptake in Hepatocytes by Cyclic Analogues of Antamanide and Somatostatin (1986) (60)
- Dynamic force spectroscopy to probe adhesion strength of living cells. (2002) (60)
- Synthesis of novel 1,4,7,10-tetraazacyclodecane-1,4,7,10-tetraacetic acid (DOTA) derivatives for chemoselective attachment to unprotected polyfunctionalized compounds. (2007) (60)
- NMR-based screening technologies. (2003) (59)
- High‐affinity urokinase‐derived cyclic peptides inhibiting urokinase/urokinase receptor‐interaction: effects on tumor growth and spread (2002) (59)
- A computational model of transmembrane integrin clustering. (2004) (59)
- Nachweis innermolekularer beweglichkeit durch NMR-spektroskopie XVI : Lösungsmitteleinflüsse auf die stickstoffinversion in guanidinen-rotationen um CN-einfach- und CN-doppelbindungen in guanidiniumsalzen (1969) (59)
- Nachweis innermolekularer Beweglichkeit durch NMR‐Spektroskopie, VI. Konformation und gehinderte Rotation in Disulfiden und Diseleniden (1968) (58)
- Induced tissue integration of bone implants by coating with bone selective RGD-peptides in vitro and in vivo studies (1999) (58)
- Hydrogel Micropillars with Integrin Selective Peptidomimetic Functionalized Nanopatterned Tops: A New Tool for the Measurement of Cell Traction Forces Transmitted through αvβ3- or α5β1-Integrins (2013) (58)
- Rational improvement of the affinity and selectivity of integrin binding of grafted lasso peptides. (2014) (58)
- Conformational preference and potential templates of N-methylated cyclic pentaalanine peptides. (2008) (58)
- ADAM15 decreases integrin αvβ3/vitronectin-mediated ovarian cancer cell adhesion and motility in an RGD-dependent fashion (2005) (57)
- Improvement of drug-like properties of peptides: the somatostatin paradigm (2010) (57)
- Structure and dynamics of synthetic O-glycosylated cyclopeptide in solution determined by NMR spectroscopy and MD calculations (1992) (57)
- Two novel probes reveal tubular and vascular Arg-Gly-Asp (RGD) binding sites in the ischemic rat kidney. (1997) (57)
- Interface Immobilization Chemistry of cRGD-based Peptides Regulates Integrin Mediated Cell Adhesion (2013) (56)
- Behavior of primary human osteoblasts on trimmed and sandblasted Ti6Al4V surfaces functionalized with integrin αvβ3-selective cyclic RGD peptides. (2013) (56)
- Does a Molecule have the Same Conformation in the Crystalline State and in Solution? Comparison of NMR Results for the Solid State and Solution with those of the X‐ray Structural Determination (1981) (55)
- Spatial Screening for the Identification of the Bioactive Conformation of Integrin Ligands (2006) (55)
- Introduction of functional groups into peptides via N-alkylation. (2008) (55)
- Mesomere Kationen: III—13C‐Fourier‐Transform‐NMR‐Spektren von Harnstoffen, Thioharnstoffen und Guanidinen (1974) (54)
- Synthesis of C-Glycopeptides via Free Radical Addition of Glycosyl Bromides to Dehydroalanine Derivatives†‡ (1992) (54)
- Selective adhesion of endothelial cells to artificial membranes with a synthetic RGD-lipopeptide. (2001) (53)
- Guiding plant virus particles to integrin-displaying cells. (2012) (53)
- Stereoselective Synthesis of C‐Glycoside with a Glycosyl Dianion (1993) (52)
- C‐Glycoside Analogues of N4‐(2‐Acetamido‐2‐deoxy‐β‐D‐glucopyranosyl)‐L‐asparagine: Synthesis and conformational analysis of a cyclic C‐glycopeptide (1996) (52)
- A backbone-cyclic, receptor 5-selective somatostatin analogue: synthesis, bioactivity, and nuclear magnetic resonance conformational analysis. (1998) (52)
- Eine Nomenklatur für intramolekulare Austauschprozesse (1971) (52)
- Solution structure of the IIB domain of the glucose transporter of Escherichia coli. (1996) (52)
- A molecular toolkit for the functionalization of titanium-based biomaterials that selectively control integrin-mediated cell adhesion. (2013) (52)
- Nachweis innermolekularer Beweglichkeit durch NMR‐Spektroskopie, XVII. Lineare Hammett‐Korrelation von Aktivierungsbarrieren der Rotation um CC‐Dopple‐und‐Einfachbindungen und CN‐Einfachbindungen in Ketenaminalen (1970) (51)
- Increasing αvβ3 selectivity of the anti-angiogenic drug cilengitide by N-methylation. (2011) (51)
- Conformational Analysis of a Cyclic RGD Peptide Containing a .psi.[CH2-NH] Bond: A Positional Shift in Backbone Structure Caused by a Single Dipeptide Mimetic (1994) (51)
- N‐Methylierung von Peptiden und Proteinen: ein wichtiges Element für die Regulation biologischer Funktionen (2013) (51)
- Cooperative binding of p53 to DNA: regulation by protein-protein interactions through a double salt bridge. (2005) (51)
- Improved Resolution in Proton-Detected Heteronuclear Long-Range Correlation (1990) (50)
- An unexpected cis peptide bond in the minor conformation of a cyclic hexapeptide containing only secondary amide bonds (1990) (50)
- Can N‐methylated amino acids serve as substitutes for prolines in conformational design of cyclic pentapeptides? (2009) (50)
- Stable Peptides Instead of Stapled Peptides: Highly Potent αvβ6-Selective Integrin Ligands. (2016) (50)
- Comparison of cyclic RGD peptides for αvβ3 integrin detection in a rat model of myocardial infarction (2013) (50)
- Molecular dynamics simulations of cyclosporin A: The crystal structure and dynamic modelling of a structure in apolar solution based on NMR data (1987) (49)
- Substrate engagement of integrins α5β1 and αvβ3 is necessary, but not sufficient, for high directional persistence in migration on fibronectin (2016) (49)
- A conformationally frozen peptoid boosts CXCR4 affinity and anti-HIV activity. (2012) (49)
- Sugar amino acid containing somatostatin analogues that induce apoptosis in both drug-sensitive and multidrug-resistant tumor cells. (2001) (48)
- Design of selective peptidomimetic agonists for the human orphan receptor BRS-3. (2003) (48)
- Benefits of NOPO as chelator in gallium-68 peptides, exemplified by preclinical characterization of (68)Ga-NOPO-c(RGDfK). (2014) (47)
- J-Spectroscopy in the presence of residual dipolar couplings: determination of one-bond coupling constants and scalable resolution (2007) (47)
- Peptide conformation. 17. cyclo-(L-Pro-L-Pro-D-Pro). Conformational analysis by 270- and 500-MHZ one- and two-dimensional proton NMR spectroscopy (1982) (46)
- Reversible backbone protection enables combinatorial solid-phase ring-closing metathesis reaction (RCM) in peptides. (2002) (46)
- Conformational Analysis of Furanoid ε-Sugar Amino Acid Containing Cyclic Peptides by NMR Spectroscopy, Molecular Dynamics Simulation, and X-ray Crystallography: Evidence for a Novel Turn Structure (2003) (46)
- Specific integrin labeling in living cells using functionalized nanocrystals. (2007) (46)
- Conformational Analysis of the cis‐ and trans‐Isomers of FK506 by NMR and Molecular Dynamics (1991) (46)
- The structure of a folding intermediate provides insight into differences in immunoglobulin amyloidogenicity (2008) (45)
- Korrelation der 13C‐NMR‐chemischen Verschiebungen von Carbonyl‐ und Thiocarbonyl‐Gruppen (1974) (45)
- Isothiocyanate-functionalized RGD peptides for tailoring cell-adhesive surface patterns. (2008) (45)
- Peptide conformations. 20. Conformational analysis of proline rings from proton spin-spin coupling constants and force-field calculations: application to three cyclic tripeptides (1983) (45)
- Intervesicle cross-linking with integrin alpha IIb beta 3 and cyclic-RGD-lipopeptide. A model of cell-adhesion processes. (2000) (44)
- Direct observation of recombination barriers of ion pairs by dynamic NMR spectroscopy (1982) (44)
- Cyclopropane-derived peptidomimetics. Design, synthesis, evaluation, and structure of novel HIV-1 protease inhibitors. (1998) (44)
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- Dynamic NMR Measurements of Boc-amino Esters with Application of Lanthanoid Shift Reagents†‡ (1973) (8)
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- Gestreckte Gelatine als chirales Orientierungsmedium zur Unterscheidung von Enantiomeren durch NMR-Spektroskopie† (2005) (8)
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- Novel synthesis of a Phe-Gly E-alkene dipeptide isostere (1996) (7)
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- A Spin System Labeled and Highly Resolved ed-H(CCO)NH-TOCSY Experiment for the Facilitated Assignment of Proton Side Chains in Partially Deuterated Samples (1998) (6)
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- uPA-Silica-Particles (SP-uPA): A Novel Analytical System to Investigate uPA-uPAR Interaction and to Test Synthetic uPAR Antagonists as Potential Cancer Therapeutics (2002) (5)
- Oral aktive Peptide: Gibt es ein Patentrezept? (2018) (5)
- Assessment of a v b 3 integrin expression after myocardial infarction by positron emission tomography (2008) (5)
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- KONFORMATION GESCHUETZTER AMINOSAEUREN 4. MITT. NMR- UND IR-UNTERSUCHUNGEN VON BOC-OMEGA-AMINOSAEUREN (1975) (0)
- 184 Inhibition of uPA/uPAR-interaction by cyclic uPA-derived peptides (1997) (0)
- NMR SPECTROSCOPIC STUDIES ON THE KINETICS AND THERMODYNAMICS OF REVERSIBLE DISSOCIATION REACTIONS. 3. IONIZATION BARRIERS OF TRITYL CHLORIDE IN SULFUR DIOXIDE (1977) (0)
- SYNTHESIS OF THE STREPTOGRAMIN B ANALOG CYCLODEPSIPEPTIDE CYCLO(-(BOC)SER-D-ABU-PRO-(ME)PHE-PIP-PHG-O-) (1983) (0)
- Die Beschlagnahmung jüdischer Kunstsammlungen 1938/39 in München: Das Beispiel Anna Caspari (2012) (0)
- NACHWEIS INNERMOLEKULARER BEWEGLICHKEIT DURCH NMR-SPEKTROSKOPIE 17. MITT. LINEARE HAMMET-KORRELATION VON AKTIVIERUNGSBARRIEREN DER ROTATION UM C=C-DOPPEL- UND EINFACHBINDUNGEN UND C-N-EINFACHBINDUNGEN IN KETENAMINALEN (1970) (0)
- Modification and Functionalization of the Guanidine Group by Tailor-made Precursors. (2017) (0)
- Cyclopentapeptid-Derivate und deren Verwendungen (2010) (0)
- PEPTIDE CONFORMATIONS. XXII. CYCLOENKEPHALIN ‐ SYNTHESIS AND CONFORMATIONAL STUDIES (1982) (0)
- Rücktitelbild: Selektive Bildgebung der angiogenetisch relevanten Integrine α5β1 und αvβ3 (Angew. Chem. 44/2013) (2013) (0)
- NACHWEIS INNERMOLEKULARER BEWEGLICHKEIT DURCH NMR‐SPEKTROSKOPIE 22. MITT. SYN‐ANTI‐ISOMERIE AN DER KOHLENSTOFF‐SCHWEFEL‐DOPPELBINDUNG IN ISOTHIURONIUMSALZEN (1970) (0)
- NMR-Untersuchungen zur Rotation und Inversion an Doppelbindungen (1969) (0)
- Design, Synthesis, and Biological Evaluation of alpha(4)beta(1) Integrin Antagonists Based on beta-D-Mannose as Rigid Scaffold. (2001) (0)
- NACHWEIS INNERMOLEKULARER BEWEGLICHKEIT DURCH NMR-SPEKTROSKOPIE 18. MITT. VERGLEICH DER INVERSIONSGESCHWINDIGKEITEN AM DOPPELT GEBUNDENEN STICKSTOFF BEI GUANIDINEN UND IMIDAZOLIDINIMINEN (1970) (0)
- UNGEWOEHNLICHER VERLAUF EINER ACETALHYDROLYSE BEI EINER HOMOTROPILIDEN-SYNTHESE (1974) (0)
- Stereoselektive ätherbildung durch dehydratisierung von diolen (1968) (0)
- Transmembranstruktur von Integrin aIIb3 - Bedeutung fr die Signalbertragung (2009) (0)
- PEPTIDE CONFORMATION, IX. CONFORMATIONAL STUDIES ON CYCLOTRIPEPTIDES CONTAINING N-BENZYL-GLYCINE (1980) (0)
- Development of urokinase-derived peptide analogues as potential therapeutic agents to block tumor invasion and metastasis (2007) (0)
- Hsp90 Delta24-N210 mutant (2006) (0)
- Der Kunsthändler als Opportunist. Karl Haberstock im "Dritten Reich" (2010) (0)
- Peptidic Inhibitors of Protein–Protein Interactions for Cell Adhesion Receptors: RGD Peptides and Beyond (2013) (0)
- Funktionalisierte RGD-Peptidmimetika und deren Herstellung sowie Implantat mit einer Beschichtung, die solche funktionalisierte RGD-Peptidmimetika enthält (2011) (0)
- Use of D-glucopyranuronsäuren and its derivatives for incorporation into pharmacologically active peptides and salts thereof (1993) (0)
- NACHWEIS INNERMOLEKULARER BEWEGLICHKEIT DURCH NMR‐SPEKTROSKOPIE 13. MITT. NACHWEIS GEHINDERTER ROTATIONEN UND INVERSIONEN DURCH NMR‐SPEKTROSKOPIE (1970) (0)
- Cellular solid-phase binding assay and mass spectrometry for screening of alpha 4 beta 7 integrin antagonists. (2001) (0)
- Application of Homonuclear and Heteronuclear Two-Dimensional NMR Spectroscopy to Cyclolinopeptide A (1) (1983) (0)
- Stereoselective Syntheses of Retro‐Isomers of N‐Glucoasparagine. (1996) (0)
- Are we curing one evil with another? A translational approach targeting the role of neoatherosclerosis in late stent failure (2020) (0)
- Peptidic Inhibitors for Protein-Protein Interactions at Cell Surfaces (2001) (0)
- Synthesis and conformational analysis of C - and N -glycopeptides (2002) (0)
- Clip to Fit: the Nucleotide Binding Mode in the Prokaryotic Kdp-ATPase Studied by NMR-Spectroscopy (2005) (0)
- NACHWEIS INNERMOLEKULARER BEWEGLICHKEIT DURCH NMR-SPEKTROSKOPIE 15. MITT. INVERSION AM DOPPELT GEBUNDENEN STICKSTOFFATOM AM BEISPIEL DER TETRAMETHYLGUANIDINE (1970) (0)
- 溶液中のα‐アミラーゼ阻害剤テンダミスタット(HOE467)の15種の環状ヘキサペプチド類似体の構造,動力学および生物活性 (1995) (0)
- NEW ANALYTICAL METHODS. 18. KINETIC AND MECHANISTIC EVALUATION OF NMR SPECTRA (1980) (0)
- Berichtigung zu dem Beitrag Peptidkonformationen, 50. - Synthese und Konformationsanalyse von cyclischen Alanin-Analogen des Thymopoietins durch NMR-Spektroskopie und Molecular-Dynamics-Rechnungen im Vakuum und in Lösung (1989) (0)
- Surface Co-Presentation of BMP-2 and Integrin Selective Ligands at the Nanoscale Favors β1 Integrin Adhesion (2019) (0)
- Peptide and peptide mimetics derivatives having properties integrininhibitor-II (2001) (0)
- AM Flo 7 Compact Electro-Optic Modulator on Silicon-on-Insulator Platform (2004) (0)
- Inhibitors of cyclic adhesion. (1993) (0)
- Highly N-Methylated Somatostatin Analogs: Synthesis, Biological Activity and Structure-Activity Relationship Studies (2006) (0)
- Subject Index Vol. 10, 2005 (2006) (0)
- Simple modifications of MD force fields for determination of peptide structures from NMR data (1993) (0)
- Synthesis and NMR structure of peptidomimetic alpha4beta7-integrin antagonists. (2002) (0)
- Facile Synthesis of a β(1-3)-Linked gal-galactal Disaccharide and Its Use in N-Iodosuccinimide-Activated O-Glycopeptide Synthesis. (1990) (0)
- Assignments of the Carbon Resonances in tert-Butylated 2-Naphthols by the Two-Dimensional C-Relayed H,C-COSY Technique. (1986) (0)
- Structure of the Lichen Macrolide (+)‐Aspicilin (1986) (0)
- Diacyl hydrazine derivatives as integrin inhibitors. (1999) (0)
- Peptide Conformations. Part 42. Conformation of Side Chains in Peptides Using Heteronuclear Coupling Constants Obtained by Two-Dimensional NMR Spectroscopy. (1988) (0)
- Diacylhydrazinderivater as integrin (1999) (0)
- NMR SPECTROSCOPIC INVESTIGATIONS OF KINETIC AND THERMODYNAMIC REVERSIBLE DISSOCIATION REACTIONS. II. CHLOROTROPYLIUM CHLORIDE-CHLORO-SUBSTITUTED 7-CHLOROCYCLOHEPTATRIENE- EQUILIBRUM AND HALOGEN MIGRATION (1976) (0)
- Rational drug design via molecular dynamics simulations of HIV-1 protease inhibitor complexes (1991) (0)
- Novel small-molecule Factor VIII affinity ligands and their application in affinity purification (2006) (0)
- Solution structure of the yeast Sti1 DP1 domain (2012) (0)
- Solution Structure of (Me‐L‐Leu7)Didemnin B Determined by NMR Spectroscopy and Refined by MD Calculation. (1990) (0)
- Molecular dynamics simulations of cyclosporin A: The crystal structure and dynamic modelling of a structure in apolar solution based on N M R data (0)
- NMR Spectroscopic Elucidation of Constitutions of Glycopeptides by the COLOC Technique. (1986) (0)
- Peptide Conformations. Part 34. Conformational Analysis of Peptides by Two-Dimensional NMR Spectroscopy (1987) (0)
- Conformational analysis of a cyclic hexapeptide by rotating frame NOE (ROE) evaluation and molecular dynamics (MD) calculations (1988) (0)
- PEPTIDE CONFORMATIONS. 11. CYCLO‐LEU5‐ENKEPHALIN (1981) (0)
- NMR SPECTROSCOPIC STUDIES ON THE KINETICS AND THERMODYNAMICS OF REVERSIBLE DISSOCIATION REACTIONS. VII. DIRECT OBSERVATION OF IONIZATION AND ION RECOMBINATION OF TRITYL CHLORIDE IN SULFUR DIOXIDE (1980) (0)
- Cyclopeptides with immuno-stimulating activity or its salts, their preparation and use as well as precursors thereof and their preparation (1984) (0)
- Biological Evaluation of the Distinct Integrin Subtypes alpha v beta 3 and alpha 5 beta 1 via Surface Coating and PET Imaging (2011) (0)
- HIGH RESOLUTION NMR STRUCTURE OF THE D(GCGTCAGG)R(CCUGACGC) HYBRID, MINIMIZED AVERAGE STRUCTURE (1998) (0)
- DETECTION OF INTRAMOLECULAR MOBILITY BY NMR SPECTROSCOPY. XXIX. CARBON‐13 DNMR INVESTIGATION OF THE MOLECULAR MOBILITY OF α‐TRIPIPERIDEINE (1977) (0)
- Different Function of α5β1 and αVβ3 Integrins: Elucidating their Interactions and Spatial Requirements for Adhesion and Migration (2013) (0)
- PEPTIDE CONFORMATIONS. 28. RELAYED HETERONUCLEAR CORRELATION SPECTROSCOPY AND D CONFORMATIONAL ANALYSIS OF CYCLIC HEXAPEPTIDES CONTAINING THE ACTIVE SEQUENCE OF SOMATOSTATIN (1984) (0)
- Antagonists for integrin alpha¶4¶beta¶7¶ (2001) (0)
- Novel Synthesis of a Phe‐Gly E‐Alkene Dipeptide Isostere. (1996) (0)
- Is a Potent Competitive Antagonist of the Interaction of Urokinase-Type Plasminogen Activator with Its Receptor ( CD 87 ) fragment (2001) (0)
- Conformational differences of cyclic RGD-peptides and their retro-inverso isomers: The effect on antiadhesive activities (1995) (0)
- GLUCOSE PERMEASE (DOMAIN IIB), NMR, 11 STRUCTURES (1996) (0)
- NMR STRUCTURE OF VAT-N: THE N-TERMINAL DOMAIN OF VAT (VCP-LIKE ATPASE OF THERMOPLASMA) (1999) (0)
- Structure-Activity Relationship of Cyclosporin A using Dynamic Forcing (1993) (0)
- Secondary structure of the IIB domain of the Escherichia coli mannose transporter, a new fold in the class of alpha/beta twisted open-sheet structures. (1997) (0)
- Synthesis and Biological Evaluation of Highly Active Nonpeptidic α- vs. β-3 Integrin Antagonists (2004) (0)
- Complementary , Selective PET Imaging of Integrin Subtypes a 5 b 1 and a v b 3 Using 68 Ga-Aquibeprin and 68 Ga-Avebetrin (2016) (0)
- CARBON-13 NMR SPECTROSCOPY OF NORBORNANE DERIVATIVES, II. THE INFLUENCE OF HOMOCONJUGATIVE INTERACTIONS ON THE CARBONYL CHEMICAL SHIFTS IN NORBORNANONES (1978) (0)
- A 68Ga-labelled PET probe for selective imaging of αvβ8-integrin (2019) (0)
- Stereoselective Synthesis of C-Glycosides with a Glycosyl Dianion. (1993) (0)
- NMR-Based Modeling of Protein-Protein Complexes and Interaction of Peptides and Proteins with Anisotropic Solvents (1999) (0)
- Recent progress in the field of αv-integrin antagonists (2002) (0)
- Differences of the conformation in crystal and solution and methods for the determination of the conformation in solution by NMR spectroscopy (1987) (0)
- The HSP90 binding mode of a radicicol-like -oxime from docking, binding free energy estimations, and NMR N chemical shifts (2020) (0)
- Experimental Prototype for automated Beta Sheet Pairing based on NOESY spectra (2005) (0)
- Towards the cell-instructive bactericidal substrate: exploring the combination of nanotopographical features and integrin selective synthetic ligands (2017) (0)
- Short and Efficient Synthesis of Statine and Isostatine Derivatives. (1990) (0)
- Novel peptide-based strategies to install osteointegrative properties on metallic biomaterials (2015) (0)
- Conformational analysis of furanoid epsilon-sugar amino acid containing cyclic peptides by NMR spectroscopy, molecular dynamics simulation, and X-ray crystallography: evidence for a novel turn structure. (2003) (0)
- TMS Triflate-Promoted O-Glycosylation of Amino Acids and Peptides by L- Acosaminal and L-Ristosaminal. (1995) (0)
- CONFORMATION OF PEPTIDES, II. PROTON NMR INVESTIGATION OF THE CONFORMATION OF CYCLO(-PHE3-GLY2-) (1978) (0)
- Nuclear Magnetic Resonance in Drug Discovery (2007) (0)
- NMR Assignment of the C-terminal Domain of yeast Aha-1 (2009) (0)
- SYNTHESIS OF THE CYCLIC PENTAPEPTIDES CONTAINING L-PHENYLALANINE AND GLYCINE (1978) (0)
- β-D-Mannose Based Peptidomimetics in the Design of α4ß1 and α4β7 Antagonists (2001) (0)
- Solvent simulations and internal motions (1994) (0)
- HIGH RESOLUTION NMR STRUCTURE OF THE STEREOREGULAR (ALL-RP)-PHOSPHOROTHIOATE-DNA/RNA HYBRID D (G*PS*C*PS*G*PS*T*PS*C*PS*A*PS*G*PS*G)R(CCUGACGC), MINIMIZED AVERAGE STRUCTURE (1998) (0)
- PEPTIDE CONFORMATIONS. 22. THE CONFORMATION OF CYCLO(PRO2‐(NB)GLY) IN CRYSTAL AND SOLUTION BY X‐RAY ANALYSIS AND ONE‐ AND TWO‐DIMENSIONAL NMR SPECTROSCOPY (1983) (0)
- At last: J-couplings again (1993) (0)
- C‐Glycoside Analogues of N4‐(2‐Acetamido‐2‐deoxy‐β‐D‐ glucopyranosyl)‐L‐asparagine: Synthesis and Conformational Analysis of a Cyclic C‐Glycopeptide. (1996) (0)
- THE STRUCTURE OF 2,6-DIPHENYLHOMOTROPYLIDENE (1980) (0)
- Combinatorial and rational strategies to develop nonpeptidic alpha4beta7-integrin antagonists from cyclic peptides. (2002) (0)
- A process for preparing 2,3,4,6-tetra-O-benzyl-D-glucopyranose and 2,3,4,6-tetra-O-allyl-D-glucopyranose (1995) (0)
- Non-natural peptide modifications using sugars and lipophilic side chains (1999) (0)
- Structure of the C-terminal non-repetitive domain of the spider dragline silk protein ADF-3 (2010) (0)
- Structure and Design of Cyclic Peptides for the Regulation of the Immune System (1993) (0)
- Chain Elongation of Thiodipeptides with Proteases Without Racemization. (1992) (0)
- ANTAGONISTEN FÜR α4-INTEGRINE (2002) (0)
- Cover Picture: Breaking the Dogma of the Metal‐Coordinating Carboxylate Group in Integrin Ligands: Introducing Hydroxamic Acids to the MIDAS To Tune Potency and Selectivity (Angew. Chem. Int. Ed. 24/2009) (2009) (0)
- Synthesis of O‐(α‐Glyco)peptides by the N‐Iodosuccinimide Procedure. (1987) (0)
- Imaging of integrin {alpha}5{beta}1 in post infarct myocardium using 68Ga-FR336 (2014) (0)
- The solution structure of the p63 DNA-binding domain (2008) (0)
- [Structure determination by NMR-spectroscopy. II]. (1969) (0)
- The use of coupling constants in structure refinement of peptides and proteins (1995) (0)
- Scalar Coupling Constants ‐ Their Analysis and Their Application for Elucidation of Structures (1995) (0)
- TPR2AB-domain:pHSP90-complex of yeast Sti1 (2012) (0)
- Chemical shift assignments, 3JHNHA coupling constants, secondary structure and 15N{1H} Heteronuclear NOE values of the N-domain of VAT (VCP like ATPase of Thermoplasma). A group II AAA ATPase. (1999) (0)
- Development of modified cyclic peptides for imaging of CXCR4 receptors (2011) (0)
- NMR SPECTROSCOPIC STUDIES ON KINETICS AND THERMODYNAMICS OF REVERSIBLE DISSOCIATION REACTIONS, IV. TRIS(4-METHOXYPHENYL)METHYL ISOTHIOCYANATE - DIRECT OBSERVATION AND COMPLETE LINE SHAPE ANALYSIS OF IONIZATION AND ION PAIR RECOMBINATI (1978) (0)
- Conformational studies on cyclic tetrapeptides: Hydrophobic cluster formation (1995) (0)
- New Perspectives in Peptide Chemistry by Multiple N‐Methylation (2009) (0)
- The Structure of the Polycyclic Nonadecapeptide Ro 09-0198 (I). (1989) (0)
- Solution structure of Ph1500: a homohexameric protein centered on a 12-bladed beta-propeller (2014) (0)
- Antagonists for integrins alpha¶4¶ (2001) (0)
- Solution structure of the yeast Sti1 DP2 domain (2012) (0)
- Synthesis of S‐α‐Glucosylated L‐Cysteine ‐ A Novel S‐Glycosyl Amino Acid. (1997) (0)
- LIGANDS FOR INTEGRIN αvβ8, SYNTHESIS AND USES THEREOF (2018) (0)
- Chemical shift assignments, 3JHNHA coupling constants and secondary structure of HNGAL (Human Neutrophil Gelatinase-Associated Lipocalin) in its apo form. (2011) (0)
- PEPTIDE CONFORMATIONS. 26. ONE‐ AND TWO‐DIMENSIONAL PROTON NMR STUDIES FOR CONFORMATIONAL ANALYSIS OF THE CYCLIC PENTAPEPTIDES CYCLO(PRO‐PHE‐GLY‐SER‐GLY) AND CYCLO(PRO‐SER‐GLY‐PHE‐GLY) (1983) (0)
- P1-IS-32 Targeted Alpha Therapy for Ovarian Cancer : Development and Characterization of Bismuth-213 (213 Bi) labeled uPAR-selective Radioligands (2007) (0)
- Improved pharmacokinetics of [18F]RGD‐peptides by serine‐conjugation (2001) (0)
- PEPTIDE CONFORMATIONS. 27. CYCLO(L‐PRO‐(BZL)GLY‐D‐PRO). SYNTHESIS AND CONFORMATION IN THE CRYSTAL AND IN SOLUTION (1983) (0)
- Introduction into moderm NMR spectroscopy modern NMR spectroscopy: A guide for chemists: by Jeremy K. M. Sanders and Brian K. Hunter, Oxford University Press, 1987. £35.00 (cloth) (xii + 308 pages) ISBN 0 19 855191 6 (1987) (0)
- CONFORMATION OF PROTECTED AMINO ACIDS. VI. TERT‐BUTOXYCARBONYL‐L‐α‐PHENYLALANINE. CRYSTAL STRUCTURE AND CONFORMATIONAL TRANSFORMATIONS IN SOLUTION (1980) (0)
- Cyclic Heptapeptides Axinastatin 2, 3, and 4: Conformational Analysis and Evaluation of the Biological Potential. (1997) (0)
- SYNTHESES OF ENDO‐EXO‐TETRACYCLO(3,3,1,0(2,4),0(7,8))NONAN‐9‐ONES AND THE UNUSUAL COURSE OF THEIR KETAL HYDROLYSIS (1973) (0)
- Implants coated peptides and processes for their manufacture. (1998) (0)
- 2-(2-PYRIDYL)ETHYL ESTERS. A NEW CARBOXYL PROTECTING GROUP IN PEPTIDE SYNTHESIS (1985) (0)
- First Coating of Titanium with alpha v beta 3 or alpha 5 beta 1 Selective Peptidomimetics: Design, Synthesis and Biological Evaluation (2011) (0)
- Ligands for integrin .alpha.v.beta.6, synthesis and uses thereof (2016) (0)
- HUMAN NEUTROPHIL GELATINASE-ASSOCIATED LIPOCALIN (HNGAL), REGULARISED AVERAGE NMR STRUCTURE (1999) (0)
- The solution structure of the AMP-PNP bound nucleotide binding domain of KdpB (2005) (0)
- Stereochemie: Principles of Organic Stereochemistry. Von B. Teste (Studies in Organic Chemistry). Marcel Dekker, Inc., New York, Basel 1979. XIII, 248 S., Paperback Sfr. 30,– (1979) (0)
- Cooperativity of Integrin-mediated Adhesion on Nanopatterned Substrates (2007) (0)
- Inhibitors of urokinase (1998) (0)
- ANTITERMINATION FACTOR NUSB FROM ESCHERICHIA COLI, NMR, 18 STRUCTURES (1998) (0)
- Structure-activity relationship studies optimizing the antiproliferative activity of novel cyclic somatostatin analogues containing a restrained cyclic beta-amino acid. (2005) (0)
- Preparation and Transmetallation of a Triphenylstannyl β‐D‐ Glucopyranoside: Highly Stereoselective Route to β‐D‐C‐Glycosides via Glycosyl Dianions. (1995) (0)
- MESOMERIC CATIONS, V. Π‐DONOR PROPERTIES OF OXYGEN AND SULFUR ‐ DYNAMIC NMR STUDIES OF AROMATIC URONIUM‐ AND THIOURONIUM SALTS AND THE QUESTION OF PLANA INVERSION ON OXYGEN AND SULFUR (1979) (0)
- A Stereoselective Synthesis of a C-Glycosylated Peptoid Building Block. (1998) (0)
- PEPTIDE CONFORMATIONS, 36. CONFORMATIONAL STUDIES OF FOUR CYCLIC HEPTAPEPTIDES BY NMR SPECTROSCOPY (1985) (0)
- Assessment of a pro-healing stent in an animal model of early neoatherosclerosis (2020) (0)
- Fast Heteronuclear 3D NMR Spectroscopy. (1990) (0)
- Synthesis of Axinastatins 2‐5. (1996) (0)
- KONFORMATION GESCHUETZTER AMINOSAEUREN 1. MITT. NMR-UNTERSUCHUNGEN VON T-BOC-GLYCIN (1974) (0)
- CONFORMATION OF CYCLIC PENTAPEPTIDES AND HEXAPEPTIDES DERIVED FROM THYMOPOIETIN (1986) (0)
- Cyclopeptide derivatives integrin inhibiting properties. (1998) (0)
- PEPTIDE CONFORMATIONS. 6. THE BOAT CONFORMATION OF CYCLO(L-PRO2-D-PRO) (1979) (0)
- The quest towards αvβ 3-or α 5 β 1-integrin selective peptidomimetics for surface coating-History , recent advances and future perspectives (2017) (0)
- Peptide and peptide derivatives having integrin inhibitor properties II (2000) (0)
- Backbone 1H, 13C, and 15N Chemical Shift Assignments for the yeast Hsp90 Middle Domain (2011) (0)
- Additions and Corrections - Assignments of the Carbon Resonances in tert-Butylated 2-Naphthols by the Two-Dimensional C-Relayed H,C-COSY Technique. (1986) (0)
- COMMON STRUCTURAL FEATURES FOR CYTOPROTECTION ACTIVITY OF CYCLIC RETRO ANALOGUES OF SOMATOSTATIN (1987) (0)
- Modifizierte Tripelresonanz‐NMR‐Experimente mit erhöhter Empfindlichkeit für schnell austauschende Protonen (1995) (0)
- DER KONTAKT-ANTEIL BEI DER LANTHANOIDEN-INDUZIERTEN VERSCHIEBUNF VON (13)C=O-NMR-SIGNALEN (1974) (0)
- CARBON-13 NMR SPECTROSCOPY OF NORBORNANE DERIVATIVES, I. CHEMICAL SHIFT EFFECTS AND THEIR NONADDITIVITY AS EVIDENCE OF INTRAMOLECULAR INTERACTIONS (1978) (0)
- Synthesis of the 4‐Pyridine Analog of Kostanecki′s Triketone. Determination of Constitution and Stereochemistry by 2D‐NMR Spectroscopy and X‐Ray Structural Analysis. (1992) (0)
- Conformational Analysis of Didemnins (I). A Multidisciplinary Approach by Means of X-Ray, NMR, Molecular-Dynamics, and Molecular-Mechanics Techniques. (1989) (0)
- Synthesis of a New Chiral Peptide Analogue of DNA Using Ornithine Subunits and Solid‐Phase Peptide Synthesis Methodologies. (1996) (0)
- NOESY-TOCSY, an Advantageous 2D NMR Technique for the Analysis of Peptide Sequences (1988) (0)
- Structural, Electronic and Defect Properties of Chemically Modified Silicon Nanoparticles (2004) (0)
- Alanine Containing Analogues of Cyclo(-D-Pro-Phe-Thr-Lys(Z)-Trp-Phe-). Conformationally Controlled Structure-Activity-Relationships. (1988) (0)
- A comparative study on the physical and conformational state of double-tailed lipo-gastrin and -CCK derivatives (1994) (0)
- Optische Aktivität und Inversion in der 5. Hauptgruppe des Periodensystems (2004) (0)
- Solution Structure of Phalloidin (I) Obtained by NMR Spectroscopy in ( D6)DMSO and Molecular Dynamics Calculation in Vacuo and in Water. (1991) (0)
- APPLICATION OF HIGH-RESOLUTION SOLID-STATE NMR SPECTROSCOPY TO THE DETERMINATION OF THE RING-CHAIN TAUTOMERISM (1984) (0)
- Carbon-13 Nuclear Magnetic Resonance Spectroscopy. Conformational Analysis of Methyl-Substituted Cycloheptanes,. Cycloheptanols, and Cycloheptanones (1972) (0)
- Backbone 1H, 15N and 13C resonance assignments of alpha-ADT and beta-ADT. (2004) (0)
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