K. C. Nicolaou
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Cypriot-American chemist
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(Suggest an Edit or Addition)According to Wikipedia, Kyriacos Costa Nicolaou is a Cypriot-American chemist known for his research in the area of natural products total synthesis. He is currently Harry C. and Olga K. Wiess Professor of Chemistry at Rice University, having previously held academic positions at The Scripps Research Institute/UC San Diego and the University of Pennsylvania.
K. C. Nicolaou's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Palladium-catalyzed cross-coupling reactions in total synthesis. (2005) (2016)
- Cascade reactions in total synthesis. (2006) (1587)
- The Diels--Alder reaction in total synthesis. (2002) (1142)
- Metathesis reactions in total synthesis. (2005) (883)
- Total synthesis of taxol (1994) (864)
- Chemistry and Biology of the Enediyne Anticancer Antibiotics (1991) (719)
- Natural Product-like Combinatorial Libraries Based on Privileged Structures. 1. General Principles and Solid-Phase Synthesis of Benzopyrans (2000) (553)
- Palladiumkatalysierte Kreuzkupplungen in der Totalsynthese (2005) (542)
- The art of total synthesis through cascade reactions. (2009) (540)
- The Chemistry and Biology of Alkannin, Shikonin, and Related Naphthazarin Natural Products. (1999) (521)
- Chemistry and Biology of Taxol (1994) (500)
- Kaskadenreaktionen in der Totalsynthese (2006) (494)
- Chasing molecules that were never there: misassigned natural products and the role of chemical synthesis in modern structure elucidation. (2005) (451)
- Tandem reactions, cascade sequences, and biomimetic strategies in total synthesis. (2003) (443)
- Aldehyde Dehydrogenase Inhibitors: a Comprehensive Review of the Pharmacology, Mechanism of Action, Substrate Specificity, and Clinical Application (2012) (442)
- A common pharmacophore for epothilone and taxanes: molecular basis for drug resistance conferred by tubulin mutations in human cancer cells. (2000) (436)
- Efficient and mild lactonization method for the synthesis of macrolides (1974) (384)
- A chemical, genetic, and structural analysis of the nuclear bile acid receptor FXR. (2003) (351)
- Samarium diiodide mediated reactions in total synthesis. (2009) (343)
- Iodine(V) reagents in organic synthesis. Part 4. o-Iodoxybenzoic acid as a chemospecific tool for single electron transfer-based oxidation processes. (2002) (339)
- Strategic applications of named reactions in organic synthesis: background and detailed mechanisms (2005) (331)
- The enediyne antibiotics. (1996) (278)
- Chemical Biology of Epothilones. (1998) (278)
- Synthesis of epothilones A and B in solid and solution phase (1997) (271)
- Adventures in Carbohydrate Chemistry: New Synthetic Technologies, Chemical Synthesis, Molecular Design, and Chemical Biology A list of abbreviations can be found at the end of this article. Telemachos Charalambous was an inspiring teacher at the Pancyprian Gymnasium, Nicosia, Cyprus. (2001) (269)
- Metathesereaktionen in der Totalsynthese (2005) (263)
- A New Method for the One-Step Synthesis of α,β-Unsaturated Carbonyl Systems from Saturated Alcohols and Carbonyl Compounds (2000) (259)
- A mild and selective method for the hydrolysis of esters with trimethyltin hydroxide. (2005) (248)
- Activation of 6-endo over 5-exo hydroxy epoxide openings. Stereoselective and ring selective synthesis of tetrahydrofuran and tetrahydropyran systems (1989) (238)
- Die Diels‐Alder‐Reaktion in der Totalsynthese (2002) (236)
- Natural Product-like Combinatorial Libraries Based on Privileged Structures. 2. Construction of a 10 000-Membered Benzopyran Library by Directed Split-and-Pool Chemistry Using NanoKans and Optical Encoding (2000) (235)
- Practical synthesis of oligosaccharides. Partial synthesis of avermectin B1a (1984) (235)
- o-Iodoxybenzoic acid (IBX) as a viable reagent in the manipulation of nitrogen- and sulfur-containing substrates: scope, generality, and mechanism of IBX-mediated amine oxidations and dithiane deprotections. (2004) (232)
- Designed Enediynes: A New Class of DNA-Cleaving Molecules with Potent and Selective Anticancer Activity (1992) (232)
- Synthesis of macrolides (1977) (221)
- Radiofrequency Encoded Combinatorial Chemistry (1995) (217)
- Cyclic conjugated enediynes related to calicheamicins and esperamicins: calculations, synthesis, and properties (1988) (215)
- Enhanced microtubule-dependent trafficking and p53 nuclear accumulation by suppression of microtubule dynamics (2002) (210)
- Stimulation of Renin Release from Rabbit Renal Cortex by Arachidonic Acid and Prostaglandin Endoperoxides (1976) (203)
- New reactions of IBX: oxidation of nitrogen- and sulfur-containing substrates to afford useful synthetic intermediates. (2003) (202)
- A mild and general method for the synthesis of 0-glycosides (1983) (201)
- Total synthesis of rapamycin (1993) (199)
- De novo design and synthesis of somatostatin non-peptide peptidomimetics utilizing beta-D-glucose as a novel scaffolding (1993) (198)
- Iodine(V) reagents in organic synthesis. Part 3. New routes to heterocyclic compounds via o-iodoxybenzoic acid-mediated cyclizations: generality, scope, and mechanism. (2002) (198)
- Modulation of the Reactivity Profile of IBX by Ligand Complexation: Ambient Temperature Dehydrogenation of Aldehydes and Ketones to α,β‐Unsaturated Carbonyl Compounds (2002) (197)
- Chemistry and biology of natural and designed enediynes. (1993) (194)
- Chemie und Biologie von Endiin‐Cytostatica/Antibiotica (1991) (193)
- Chemie und Biologie von Endiin‐Cytostatica/Antibiotica (1991) (193)
- Nonpeptidal peptidomimetics with a β-D-glucose scaffolding. A partial somatostatin agonist bearing a close structural relationship to a potent, selective substance P antagonist (1992) (192)
- N-Phenylselenophthalimide (N-PSP) and N-phenylselenosuccinimide (N-PSS). Two versatile carriers of the phenylseleno group. Oxyselenation of olefins and a selenium-based macrolide synthesis (1979) (182)
- The Wittig and Related Reactions in Natural Product Synthesis (1997) (181)
- Enantioselective dichlorination of allylic alcohols. (2011) (179)
- A General and Highly Efficient Solid Phase Synthesis of Oligosaccharides. Total Synthesis of a Heptasaccharide Phytoalexin Elicitor (HPE) (1997) (179)
- Stereospecific 1,2-migrations in carbohydrates. Stereocontrolled synthesis of .alpha.- and .beta.-2-deoxyglycosides. (1986) (171)
- Recent advances in the chemistry and biology of naturally occurring antibiotics. (2009) (169)
- Chemical self-replication of palindromic duplex DNA (1994) (168)
- Natural Product-like Combinatorial Libraries Based on Privileged Structures. 3. The “Libraries from Libraries” Principle for Diversity Enhancement of Benzopyran Libraries (2000) (162)
- Total Synthesis of Taxol. 2. Construction of A and C Ring Intermediates and Initial Attempts To Construct the ABC Ring System (1995) (162)
- Molecular Design, Chemical Synthesis, and Biological Action of Enediynes (1992) (161)
- Constructing molecular complexity and diversity: total synthesis of natural products of biological and medicinal importance. (2012) (158)
- Identification of a novel small-molecule inhibitor of the hypoxia-inducible factor 1 pathway. (2005) (157)
- Oxidation of silyl enol ethers by using IBX and IBX.N-oxide complexes: a mild and selective reaction for the synthesis of enones. (2002) (153)
- The endiandric acid cascade. Electrocyclizations in organic synthesis. I. Stepwise, stereocontrolled total synthesis of endiandric acids A and B (1982) (150)
- Chemical synthesis and biological evaluation of cis- and trans-12,13-cyclopropyl and 12,13-cyclobutyl epothilones and related pyridine side chain analogues. (2001) (149)
- Lipoxin A. Stereochemistry and biosynthesis. (1986) (149)
- Total Syntheses of Epothilones A and B via a Macrolactonization-Based Strategy (1997) (148)
- Asymmetric total syntheses of platensimycin. (2007) (148)
- Total Synthesis of Epothilone A: The Olefin Metathesis Approach (1997) (145)
- The continuing saga of the marine polyether biotoxins. (2008) (142)
- Phenylseleno- and phenylsulfenolactonizations. Two highly efficient and synthetically useful cyclization procedures (1979) (141)
- Enantioselective intramolecular Friedel-Crafts-type alpha-arylation of aldehydes. (2009) (140)
- Chemistry and biology of diazonamide A: first total synthesis and confirmation of the true structure. (2004) (139)
- The coral-derived natural products eleutherobin and sarcodictyins A and B: effects on the assembly of purified tubulin with and without microtubule-associated proteins and binding at the polymer taxoid site. (1999) (138)
- Total synthesis of platensimycin. (2006) (136)
- Olefin Metathesis in Cyclic Ether Formation. Direct Conversion of Olefinic Esters to Cyclic Enol Ethers with Tebbe-Type Reagents (1996) (135)
- Total Synthesis of Taxol. 4. The Final Stages and Completion of the Synthesis (1995) (134)
- Total Synthesis of Taxol. 1. Retrosynthesis, Degradation, and Reconstitution (1995) (132)
- Total synthesis of brevetoxin A (1998) (131)
- The second total synthesis of diazonamide A. (2003) (129)
- Total synthesis of hamigerans and analogues thereof. Photochemical generation and Diels-Alder trapping of hydroxy-o-quinodimethanes. (2004) (127)
- Stereocontrolled total synthesis of lipoxins A (1985) (126)
- Total Synthesis of Erythromycins. 4. Total Synthesis of Erythronolide B1 (1978) (125)
- Total Synthesis of Vancomycin (1999) (123)
- Sulfated blood group Lewis(a). A superior oligosaccharide ligand for human E-selectin. (1994) (123)
- Chemie, Biologie und medizinische Anwendungen der Glycopeptid-Antibiotika (1999) (122)
- Total Synthesis of Vancomycin—Part 1: Design and Development of Methodology (1999) (122)
- Designed Epothilones: Combinatorial Synthesis, Tubulin Assembly Properties, abd Cytotoxic Action against Taxol-Resistant Tumor Cells† (1997) (121)
- Designed Epothilones: Combinatorial Synthesis, Tubulin Assembly Properties, abd Cytotoxic Action against Taxol-Resistant Tumor Cells† (1997) (121)
- Total Synthesis of Taxol. 3. Formation of Taxol's ABC Ring Skeleton (1995) (120)
- Chemistry and biology of diazonamide A: second total synthesis and biological investigations. (2004) (119)
- An expedient procedure for the oxidative cleavage of olefinic bonds with PhI(OAc)2, NMO, and catalytic OsO4. (2010) (119)
- Activation of 7-endo over 6-exo epoxide openings. Synthesis of oxepane and tetrahydropyran systems (1989) (118)
- Selective oxidation at carbon adjacent to aromatic systems with IBX. (2001) (117)
- Total synthesis of diazonamide A. (2002) (117)
- Interaction of epothilone analogs with the paclitaxel binding site: relationship between binding affinity, microtubule stabilization, and cytotoxicity. (2004) (116)
- The Olefin Metathesis Approach to Epothilone A and Its Analogues (1997) (116)
- Target-Accelerated Combinatorial Synthesis and Discovery of Highly Potent Antibiotics Effective Against Vancomycin-Resistant Bacteria. (2000) (115)
- Total synthesis of the tumor-associated Lex family of glycosphingolipids (1990) (115)
- Total synthesis of amphotericin B. 3. The final stages (1988) (114)
- Total synthesis and biological evaluation of the resveratrol-derived polyphenol natural products hopeanol and hopeahainol A. (2010) (113)
- Total synthesis of thiostrepton. Retrosynthetic analysis and construction of key building blocks. (2005) (111)
- Chemie und Biologie von Taxol (1994) (110)
- Total synthesis of platensimycin and related natural products. (2009) (110)
- Synthesis of imides, N-acyl vinylogous carbamates and ureas, and nitriles by oxidation of amides and amines with Dess-Martin periodinane. (2005) (109)
- The endiandric acid cascade. Electrocyclizations in organic synthesis. 4. Biomimetic approach to endiandric acids A-G. Total synthesis and thermal studies (1982) (109)
- Chemical synthesis and biological properties of pyridine epothilones. (2000) (109)
- Structural revision and total synthesis of azaspiracid-1, part 2: definition of the ABCD domain and total synthesis. (2004) (109)
- Additions and Corrections - Total Synthesis of Elfamycins: Aurodox and Efrotomycin. 1. Strategy and Construction of Key Intermediates (1985) (108)
- Total synthesis of englerin A. (2010) (108)
- Cyclizations of hydroxy dithioketals. New synthetic technology for the construction of oxocenes and related medium-ring systems (1989) (108)
- Total synthesis of amphoteronolide B and amphotericin B. 1. Strategy and stereocontrolled construction of key building blocks (1988) (108)
- Organoselenium-induced cyclizations in organic synthesis (1981) (107)
- Design, synthesis and biological activity of protaxols (1993) (106)
- Synergistic Effects of Peloruside A and Laulimalide with Taxoid Site Drugs, but Not with Each Other, on Tubulin Assembly (2006) (106)
- Characterization of a binding site for chemically synthesized lipo-oligosaccharidic NodRm factors in particulate fractions prepared from roots. (1995) (105)
- Total synthesis of the originally proposed and revised structures of palmerolide A and isomers thereof. (2008) (105)
- Polymer-supported selenium reagents for organic synthesis (1998) (105)
- Design, synthesis, and study of simple monocyclic conjugated enediynes. The 10-membered ring enediyne moiety of the enediyne anticancer antibiotics (1992) (104)
- The endiandric acid cascade. Electrocyclizations in organic synthesis. 3. "Biomimetic" approach to endiandric acids A-G. Synthesis of precursors (1982) (104)
- Total synthesis of calicheamicin .gamma.1I. 1. Synthesis of the oligosaccharide fragment (1993) (103)
- Palladium-Catalyzed Functionalization of Lactones via Their Cyclic Ketene Acetal Phosphates. Efficient New Synthetic Technology for the Construction of Medium and Large Cyclic Ethers (1997) (103)
- SOLID AND SOLUTION PHASE SYNTHESIS AND BIOLOGICAL EVALUATION OF COMBINATORIAL SARCODICTYIN LIBRARIES (1998) (102)
- Biomimetic Total Synthesis of Bisorbicillinol, Bisorbibutenolide, Trichodimerol, and Designed Analogues of the Bisorbicillinoids (2000) (102)
- The relationship of brevetoxin 'length' and A-ring functionality to binding and activity in neuronal sodium channels. (1995) (102)
- Total synthesis of calicheamicin .gamma.1I (1992) (101)
- Der Stand der Totalsynthese zu Beginn des 21. Jahrhunderts (2000) (100)
- Samariumdiiodid-vermittelte Reaktionen in der Totalsynthese (2009) (99)
- A practical and enantioselective synthesis of glycosphingolipids and related compounds. Total synthesis of globotriaosylceramide (Gb3) (1988) (98)
- DNA-cleavage and antitumor activity of designed molecules with conjugated phosphine oxide-allene-ene-yne functionalities (1990) (97)
- Synthesis and biological properties of a 9,11-azo-prostanoid: highly active biochemical mimic of prostaglandin endoperoxides. (1975) (96)
- Iodine(V) reagents in organic synthesis. Part 1. Synthesis of polycyclic heterocycles via Dess-Martin periodinane-mediated cascade cyclization: generality, scope, and mechanism of the reaction. (2002) (96)
- Total syntheses of anominine and tubingensin A. (2012) (96)
- Stereocontrolled Total Synthesis of Apicularen A and Its Δ17,18 Z Isomer (2002) (95)
- Synthesis and biological evaluation of vancomycin dimers with potent activity against vancomycin-resistant bacteria: target-accelerated combinatorial synthesis. (2001) (95)
- Total Synthesis of Vancomycin—Part 2: Retrosynthetic Analysis, Synthesis of Amino Acid Building Blocks and Strategy Evaluations (1999) (95)
- New Synthetic Technology for the Synthesis of Aryl Ethers: Construction of C-O-D and D-O-E Ring Model Systems of Vancomycin (1997) (95)
- Lipoxins and Related Eicosanoids: Biosynthesis, Biological Properties, and Chemical Synthesis (1991) (94)
- Total Synthesis of Vancomycin Aglycon-Part 3: Final Stages. (1998) (94)
- The Chemistry and Biology of Epothilones—The Wheel Keeps Turning (2007) (94)
- Molecules That Changed the World (2008) (93)
- Design, synthesis, and biological evaluation of platensimycin analogues with varying degrees of molecular complexity. (2008) (93)
- Synthesis and biological evaluation of epidithio-, epitetrathio-, and bis-(methylthio)diketopiperazines: synthetic methodology, enantioselective total synthesis of epicoccin G, 8,8'-epi-ent-rostratin B, gliotoxin, gliotoxin G, emethallicin E, and haematocin and discovery of new antiviral and antimal (2012) (92)
- Total synthesis and revised structure of biyouyanagin A. (2007) (92)
- Total Synthesis of Brevetoxin B. 2. Completion (1995) (91)
- N-phenylselenophthalimide (NPSP) : A valuable selenenylating agent (1985) (91)
- Identification of a Novel Small Molecule HIF-1α Translation Inhibitor (2009) (91)
- Phenylselenoetherification. A highly efficient cyclization process for the synthesis of oxygen- and sulfur-heterocycles (1980) (90)
- The total synthesis of coleophomones B, C, and D. (2005) (90)
- Recent developments in the chemistry, biology and medicine of the epothilones. (2001) (90)
- Synthesis of medium-sized ring ethers from thionolactones. Applications to polyether synthesis (1990) (90)
- Total synthesis of (+)-cortistatin A. (2008) (89)
- Lipoxin A-induced inhibition of human natural killer cell cytotoxicity: studies on stereospecificity of inhibition and mode of action. (1987) (88)
- Selenium in natural products synthesis (1984) (88)
- Solid-Phase Synthesis of Oligosaccharides: Construction of a Dodecasaccharide. (1998) (88)
- Total synthesis of erythromycins. 3. Stereoselective routes to intermediates corresponding to C(1) to C(9) and C(10) to C(13) fragments of erythronolide B (1978) (88)
- Total synthesis of amphoteronolide B and amphotericin B. 2. Total synthesis of amphoteronolide B (1988) (88)
- A brief history of antibiotics and select advances in their synthesis (2017) (87)
- Total Synthesis of Colombiasin A. (2001) (87)
- Reactions of glycosyl fluorides. Synthesis of O-, S-, and N-glycosides (1984) (87)
- Iodine(V) reagents in organic synthesis. Part 2. Access to complex molecular architectures via Dess-Martin periodinane-generated o-imidoquinones. (2002) (87)
- Total synthesis of ionophore antibiotic X-14547A (1985) (87)
- Superoxide ion as a synthetically useful oxygen nucleophile (1975) (87)
- Cortistatin A is a high-affinity ligand of protein kinases ROCK, CDK8, and CDK11. (2009) (87)
- Synthesis of macrocycles by intramolecular ketophosphonate reactions. Stereoselective construction of the "left-wing" of carbomycin B and a synthesis of dl-muscone from oleic acid (1979) (86)
- Total synthesis of hirsutellone B. (2009) (85)
- Total synthesis of abyssomicin C and atrop-abyssomicin C. (2006) (85)
- Bridging of macrodithionolactones to bicyclic systems. Synthesis and modeling of oxapolycyclic frameworks (1990) (85)
- Stereocontrolled total synthesis of lipoxins B (1986) (84)
- Total synthesis of the originally proposed and revised structures of palmerolide A. (2007) (84)
- A remarkably simple, highly efficient, and stereoselective synthesis of steroids and other polycyclic systems. Total synthesis of estra-1,3,5(10)-trien-17-one via intramolecular capture of o-quinodimethanes generated by cheletropic elimination of sulfur dioxide (1980) (84)
- Solid-Phase Synthesis of Macrocyclic Systems by a Cyclorelease Strategy: Application of the Stille Coupling to a Synthesis of (S)-Zearalenone. (1998) (84)
- Total synthesis of abyssomicin C, atrop-abyssomicin C, and abyssomicin D: implications for natural origins of atrop-abyssomicin C. (2007) (84)
- Total synthesis of hemibrevetoxin B and (7a.alpha.)-epi-hemibrevetoxin B (1993) (84)
- Total synthesis of calicheamicin .gamma.1I. 3. The final stages (1993) (84)
- Total synthesis of thiostrepton. Assembly of key building blocks and completion of the synthesis. (2005) (84)
- Total Synthesis of Vancomycin Aglycon-Part 2: Synthesis of Amino Acids 1-3 and Construction of the AB-COD-DOE Ring Skeleton. (1998) (83)
- Synthetic studies on the dioxepane region of brevetoxin B. New synthetic technology for the construction of oxepanes and synthesis of a model for the CDEF ring skeleton of brevetoxin B (1989) (83)
- A Novel Strategy for the Solid-Phase Synthesis of Substituted Indolines (2000) (83)
- A catalytic asymmetric three-component 1,4-addition/aldol reaction: enantioselective synthesis of the spirocyclic system of vannusal A. (2005) (83)
- Adamantaplatensimycin: a bioactive analogue of platensimycin. (2007) (83)
- Total synthesis of sialyl dimeric Lex (1992) (83)
- Total synthesis of apoptolidin: construction of enantiomerically pure fragments. (2003) (82)
- Total Synthesis of Brevetoxin B. 1. First Generation Strategies and New Approaches to Oxepane Systems (1996) (82)
- Total Synthesis of Brevetoxin B. 3. Final Strategy and Completion (1995) (82)
- Total synthesis of hybocarpone and analogues thereof. A facile dimerization of naphthazarins to pentacyclic systems. (2004) (82)
- Total Synthesis of Balanol (1994) (82)
- A Useful Method for the Conversion of Azides to Amines (1975) (81)
- DNA cleavage by a synthetic mimic of the calicheamicin-esperamicin class of antibiotics (1988) (80)
- Synthesis of the brevetoxin B IJK ring system (1989) (80)
- SYNTHESIS OF THE TRICYCLIC CORE OF ELEUTHEROBIN AND SARCODICTYINS AND TOTAL SYNTHESIS OF SARCODICTYIN A (1997) (80)
- Lipoxin A4 inhibits leukotriene B4-induced inflammation in the hamster cheek pouch. (1989) (79)
- Molecular basis for the inhibition of human alpha-thrombin by the macrocyclic peptide cyclotheonamide A. (1993) (79)
- Crystal structure of the potent natural product inhibitor balanol in complex with the catalytic subunit of cAMP-dependent protein kinase. (1999) (79)
- Formal synthesis of (+/-)-platensimycin. (2007) (79)
- Structural revision and total synthesis of azaspiracid-1, part 1: intelligence gathering and tentative proposal. (2004) (78)
- Total synthesis of thiostrepton, part 1: construction of the dehydropiperidine/thiazoline-containing macrocycle. (2004) (78)
- The essence of total synthesis. (2004) (78)
- Advancing the drug discovery and development process. (2014) (78)
- Chemistry and Biology of the Zaragozic Acids (Squalestatins) (1996) (78)
- Total synthesis of calicheamicin .gamma.1I. 2. Development of an enantioselective route to (-)-calicheamicinone (1993) (76)
- New uses for the Burgess reagent in chemical synthesis: methods for the facile and stereoselective formation of sulfamidates, glycosylamines, and sulfamides. (2004) (76)
- Total syntheses of (+/-)-platencin and (-)-platencin. (2009) (75)
- Studies toward diazonamide A: initial synthetic forays directed toward the originally proposed structure. (2004) (75)
- Letter: Synthesis of novel macrocyclic lactones in the prostaglandin and polyether antibiotic series. (1975) (75)
- Total Synthesis of the CP Molecules CP-263,114 and CP-225,917- Part 1: Synthesis of Key Intermediates and Intelligence Gathering. (1999) (74)
- Novel Reactions Initiated by Titanocene Methylidenes: Deoxygenation of Sulfoxides, N‐Oxides, and Selenoxides (2000) (74)
- Total synthesis of thiostrepton, part 2: construction of the quinaldic acid macrocycle and final stages of the synthesis. (2004) (74)
- Total synthesis of hopeahainol A and hopeanol. (2009) (74)
- Total Synthesis of Brevetoxin-B .1. Cdefg Framework (1995) (74)
- Total synthesis, revised structure, and biological evaluation of biyouyanagin A and analogues thereof. (2008) (73)
- Chemie und Biologie der Epothilone (1998) (73)
- Total synthesis and biological evaluation of cortistatins A and J and analogues thereof. (2009) (73)
- Total synthesis of kinamycins C, F, and J. (2007) (73)
- Total Synthesis of Epothilone E and Analogues with Modified Side Chains through the Stille Coupling Reaction (1998) (73)
- Total Synthesis of Hamigerans: Part 1. Development of Synthetic Technology for the Construction of Benzannulated Polycyclic Systems by the Intramolecular Trapping of Photogenerated Hydroxy-o-quinodimethanes and Synthesis of Key Building Blocks This work was financially supported by the National Inst (2001) (73)
- Total Synthesis of Sarcodictyins A and B (1998) (73)
- Biomimetic total synthesis of gambogin and rate acceleration of pericyclic reactions in aqueous media. (2005) (73)
- HIO3 and I2O5: mild and selective alternative reagents to IBX for the dehydrogenation of aldehydes and ketones. (2002) (73)
- Macrocyclic Peptide Inhibitors of Serine Proteases. Convergent Total Synthesis of Cyclotheonamides A and B via a Late-Stage Primary Amine Intermediate. Study of Thrombin Inhibition under Diverse Conditions (1995) (73)
- Total Synthesis of Swinholide A, Preswinholide A, and Hemiswinholide A (1996) (72)
- Evidence of calcium(2+)-dependent carbohydrate association through ion spray mass spectrometry (1993) (72)
- Discovery and optimization of non-steroidal FXR agonists from natural product-like libraries. (2003) (72)
- Total synthesis and structural elucidation of azaspiracid-1. Final assignment and total synthesis of the correct structure of azaspiracid-1. (2006) (72)
- Further studies of the binding specificity of the leukocyte adhesion molecule, L-selectin, towards sulphated oligosaccharides--suggestion of a link between the selectin- and the integrin-mediated lymphocyte adhesion systems. (1995) (71)
- Atropselective macrocyclization of diaryl ether ring systems: application to the synthesis of vancomycin model systems. (2002) (71)
- The Battle of Calicheamicin γ (1993) (71)
- Total synthesis of the proposed azaspiracid-1 structure, part 1: construction of the enantiomerically pure C1-C20, C21-C27, and C28-C40 fragments. (2003) (71)
- Stereocontrolled Second Generation Syntheses of the ABC and FG Ring Systems of Brevetoxin B (1990) (70)
- The Conquest of Taxol (1995) (70)
- Synthesis and biological properties of prostaglandin endoperoxides, thromboxanes and prostacyclins. (1978) (70)
- Total synthesis and antibacterial properties of carbaplatensimycin. (2007) (70)
- Total syntheses and structural revision of alpha- and beta-diversonolic esters and total syntheses of diversonol and blennolide C. (2008) (70)
- Synthesis of Zaragozic Acid A/Squalestatin S1 (1995) (70)
- Total Synthesis of Eleutherobin and Eleuthosides A and B (1998) (70)
- A GENERAL AND STEREOCONTROLLED TOTAL SYNTHESIS OF LEUKOTRIENE B4 AND ANALOGS (1984) (70)
- Total Synthesis of Eleutherobin (1997) (70)
- Total Synthesis of Vancomycin—Part 4: Attachment of the Sugar Moieties and Completion of the Synthesis (1999) (70)
- Synthesis of dynemicin A models (1990) (70)
- Total synthesis of sulfated Lex and Lea-type oligosaccharide selectin ligands (1993) (69)
- Combinatorial synthesis through disulfide exchange: discovery of potent psammaplin A type antibacterial agents active against methicillin-resistant Staphylococcus aureus (MRSA). (2001) (69)
- DNA-carbohydrate interactions. Specific binding of the calicheamicin .gamma.1I oligosaccharide with duplex DNA (1992) (69)
- A chiral pool based synthesis of platensimycin. (2008) (69)
- Synthesis of brefeldin A, carpaine, vertaline, and erythronolide B from nonmacrocyclic precursors (1975) (68)
- Synthesis of N-heterocycles via lactam-derived ketene aminal phosphates. Asymmetric synthesis of cyclic amino acids. (1998) (68)
- Synthesis of 16-membered-ring macrolide antibiotics. 4. Carbomycin B and leucomycin A3: total synthesis of cyclic key intermediate (1981) (68)
- Rhodium-catalyzed asymmetric enyne cycloisomerization of terminal alkynes and formal total synthesis of (-)-platensimycin. (2009) (68)
- Total Synthesis of Brevetoxin A: Part 4: Final Stages and Completion (1999) (67)
- An Olefin Metathesis Based Strategy for the Construction of the JKL, OPQ, and UVW Ring Systems of Maitotoxin (1996) (67)
- Total synthesis of sporolide B. (2009) (67)
- Mechanistic Studies of Periodinane-Mediated Reactions of Anilides and Related Systems. (2001) (67)
- Total synthesis of apoptolidin: completion of the synthesis and analogue synthesis and evaluation. (2003) (66)
- Synthesis and chemistry of dynemicin A models (1991) (66)
- An Approach to Epothilones Based on Olefin Metathesis (1996) (66)
- Interaction of Calicheamicin with Duplex DNA: Role of the Oligosaccharide Domain and Identification of Multiple Binding Modes (1994) (66)
- Carbohydrates in organic synthesis. Synthesis of 16-membered-ring macrolide antibiotics. 5. Total synthesis of O-mycinosyltylonolide: synthesis of key intermediates (1982) (66)
- Letter: Total synthesis of (plus or minus)-vermiculine. (1975) (66)
- A novel regio- and stereoselective synthesis of sulfamidates from 1,2-diols using Burgess and related reagents: a facile entry into beta-amino alcohols. (2002) (65)
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- Chemistry of amphotericin B: degradation studies and preparation of amphoteronolide B (1988) (65)
- Molecular design, chemical synthesis, kinetic studies, calculations, and biological studies of novel enediynes equipped with triggering, detection, and deactivating devices. Model dynemicin A epoxide and cis-diol systems (1993) (65)
- Total Synthesis of Brevetoxin A: Part 1: First Generation Strategy and Construction of BCD Ring System (1999) (65)
- A concise asymmetric total synthesis of aspidophytine. (2008) (64)
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- Total synthesis of epicoccin G. (2011) (64)
- Discovery of a biologically active thiostrepton fragment. (2005) (64)
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- Organic synthesis: the art and science of replicating the molecules of living nature and creating others like them in the laboratory (2014) (64)
- Total Synthesis of Hamigerans: Part 2. Implementation of the Intramolecular Diels-Alder Trapping of Photochemically Generated Hydroxy-o-quinodimethanes; Strategy and Completion of the Synthesis This work was financially supported by the National Institutes of Health (USA) and The Skaggs Institute fo (2001) (63)
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- Molecular design and chemical synthesis of potent enediynes. 2: Dynemicin model systems equipped with C-3 triggering devices and evidence for quinone methide formation in the mechanism of action of dynemicin A (1992) (63)
- Carbonucleotoids and carbopeptoids: New carbohydrate oligomers (1995) (63)
- Solid Phase Synthesis of Macrocycles by an Intramolecular Ketophosphonate Reaction. Synthesis of a (dl)-Muscone Library (1998) (63)
- Total Synthesis of the Novel Immunosuppressant Sanglifehrin A (2000) (63)
- Total synthesis of the NodRm-IV factors, the rhizobium nodulation signals (1992) (63)
- From nature to the laboratory and into the clinic. (2009) (63)
- Bromotyrosine-derived natural and synthetic products as inhibitors of mycothiol-S-conjugate amidase. (2002) (62)
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- Total Synthesis of Epothilone A: The Macrolactonization Approach (1997) (62)
- Total Synthesis and Biological Evaluation of Natural and Designed Tubulysins. (2016) (62)
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- Synthesis and Biopharmaceutical Evaluation of Imatinib Analogues Featuring Unusual Structural Motifs (2016) (61)
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- Palladium-Catalyzed Cross-Coupling Reactions in Total Synthesis (2005) (61)
- Total syntheses of 2,2'-epi-cytoskyrin A, rugulosin, and the alleged structure of rugulin. (2007) (61)
- Redox-controlled Bergman cycloaromatizations. Designed enediynes with DNA-cleaving properties and antitumor activity (1992) (61)
- Total synthesis and stereochemistry of uncialamycin. (2007) (61)
- Novel IBX‐Mediated Processes for the Synthesis of Amino Sugars and Libraries Thereof (2000) (61)
- Combinatorial synthesis of novel and potent inhibitors of NADH:ubiquinone oxidoreductase. (2000) (61)
- Arylsulfonamide KCN1 Inhibits In Vivo Glioma Growth and Interferes with HIF Signaling by Disrupting HIF-1α Interaction with Cofactors p300/CBP (2012) (61)
- A facile method for the solution and solid-phase synthesis of substituted [3.3.1] bicycles. (1999) (60)
- The Diels—Alder Reaction in Total Synthesis (2002) (60)
- Total synthesis of the oligosaccharide fragment of calicheamicin .gamma.1I (1990) (60)
- Stereocontrolled synthesis of sialyl Lex, the oligosaccharide binding ligand to ELAM-1 (sialyl =N-acetylneuramin) (1991) (59)
- Proteomic Signature of Fatty Acid Biosynthesis Inhibition Available for In Vivo Mechanism-of-Action Studies (2011) (59)
- Total Synthesis of the CP Molecules CP-225,917 and CP-263,114- Part 2: Evolution of the Final Strategy. (1999) (59)
- DIE TOTALSYNTHESE VON EPOTHILON A : DER ZUGANG DURCH OLEFINMETATHESE (1997) (59)
- Phenylselenolactonization. An extremely mild and synthetically useful cyclization process (1977) (59)
- A biomimetically inspired synthesis of the dehydropiperidine domain of thiostrepton. (2002) (58)
- Total synthesis of the proposed azaspiracid-1 structure, part 2: coupling of the C1-C20, C21-C27, and C28-C40 fragments and completion of the synthesis. (2003) (58)
- On the structure of maitotoxin. (2007) (58)
- Carbocyclic thromboxane A2 (1980) (58)
- Total synthesis and structural elucidation of azaspiracid-1. Construction of key building blocks for originally proposed structure. (2006) (57)
- Molecular design and chemical synthesis of potent enediynes. 1: Dynemicin model systems equipped with N-tethered triggering devices (1992) (57)
- Design, synthesis, and biological properties of highly potent epothilone B analogues. (2003) (57)
- Total synthesis of colombiasin A and determination of its absolute configuration. (2001) (57)
- A New Class of DNA‐Cleaving Molecules: pH‐Dependent DNA Cleavage by Propargylic and Allenic Sulfones (1989) (57)
- Total synthesis of hemibrevetoxin B (1992) (57)
- Total synthesis of thiopeptide antibiotics GE2270A, GE2270T, and GE2270C1. (2008) (56)
- Construction of highly functionalized medium-sized rings: synthesis of hyperforin and perforatumone model systems. (2005) (56)
- Solution and Solid‐Phase Synthesis of Functionalized 3‐Arylbenzofurans by a Novel Cyclofragmentation – Release Pathway (2000) (56)
- Total synthesis and confirmation of the revised structures of azaspiracid-2 and azaspiracid-3. (2006) (56)
- New Selenium-Based Safety-Catch Linkers: Solid-Phase Semisynthesis of Vancomycin (2000) (55)
- Total synthesis of globotriaosylceramide (Gb3) and lysoglobotriaosylceramide (lysoGb3). (1990) (55)
- Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological Investigations. (2016) (55)
- Synthesis of the ABCD Ring System of Azaspiracid. (2001) (55)
- Nucleophilic additions to thionolactones. New synthetic technology for the construction of medium and large ring ethers (1987) (55)
- Total synthesis of the CP-molecules (CP-263,114 and CP-225,917, phomoidrides B and A). 2. Model studies for the construction of key structural elements and first-generation strategy. (2002) (55)
- Carbohydrates in organic synthesis. Synthesis of 16-membered-ring macrolide antibiotics. 6. Total synthesis of O-mycinosyltylonolide: coupling of key intermediates and macrocyclization (1982) (54)
- Design, synthesis and biological evaluation of carbohydrate-based mimetics of cRGDFV (1997) (54)
- Design, synthesis and biological evaluation of nonpeptide integrin antagonists. (1998) (54)
- Synthesis of the ABC ring system of brevetoxin B (1989) (54)
- Abenteuer in der Kohlenhydratchemie: Synthesestrategien, Synthesemethoden, Moleküldesign und biologische Chemie (2001) (53)
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- Cell growth inhibition and actin cytoskeleton disorganization induced by azaspiracid-1 structure-activity studies. (2006) (53)
- Carbohydrate-Minor Groove Interactions in the Binding of Calicheamicin .gamma.1I to Duplex DNA (1994) (53)
- Synthesis of iso-epoxy-amphidinolide N and des-epoxy-caribenolide I structures. Revised strategy and final stages. (2006) (53)
- Total Synthesis of Swinholide A (1996) (53)
- Synthesis of the Fully Functionalized Bicyclic Core of Garsubellin A (1999) (53)
- TOTAL SYNTHESIS OF BREVETOXIN A : PART 2 : SECOND GENERATION STRATEGY AND CONSTRUCTION OF EFGH MODEL SYSTEM (1999) (53)
- The Role of Organic Synthesis in the Emergence and Development of Antibody-Drug Conjugates as Targeted Cancer Therapies. (2019) (52)
- Total synthesis of antibiotics GE2270A and GE2270T. (2006) (52)
- Effects of azaspiracid-1, a potent cytotoxic agent, on primary neuronal cultures. A structure-activity relationship study. (2007) (52)
- N-Phenylselenophthalimide. A useful reagent for the facile transformation of (1) carboxylic acids into either selenol esters or amides and (2) alcohols into alkyl phenyl selenides (1981) (52)
- 1,2‐Seleno Migrations in Carbohydrate Chemistry: Solution and Solid‐Phase Synthesis of 2‐Deoxy Glycosides, Orthoesters, and Allyl Orthoesters (2000) (52)
- Total synthesis and biological evaluation of halipeptins A and D and analogues. (2006) (52)
- The beta-D-glucose scaffold as a beta-turn mimetic. (2009) (51)
- Chemical synthesis and biological evaluation of palmerolide A analogues. (2008) (51)
- Inhibition of protein kinases by balanol: specificity within the serine/threonine protein kinase subfamily. (1999) (51)
- Total synthesis of 5(S),15(S)-dihydroxy-6,13-trans-8,15-cis-eicosatetraenoic acid (5,15-diHETE) and 8(S),15(S)-dihydroxy-5,11-cis-9,13-trans-eicosatetraenoic acid (8,15-DiHETE), two novel metabolites of arachidonic acid (1984) (51)
- Asymmetric synthesis and biological properties of uncialamycin and 26-epi-uncialamycin. (2008) (51)
- Classics in Total Synthesis II: More Targets, Strategies, Methods (2003) (51)
- Synthesis and Biological Activity of Sarcodictyins. (1998) (51)
- Total Synthesis of Apoptolidin: Part 1. Retrosynthetic Analysis and Construction of Building Blocks. (2001) (51)
- The action of lipoxin-A on glomerular microcirculatory dynamics in the rat. (1987) (50)
- Construction of the complete aromatic core of diazonamide A by a novel hetero pinacol macrocyclization cascade reaction (2001) (50)
- Total synthesis of marinomycins A-C and of their monomeric counterparts monomarinomycin A and iso-monomarinomycin A. (2007) (50)
- The Total Synthesis of Brevetoxin B: A Twelve‐Year Odyssey in Organic Synthesis (1996) (50)
- Chemical synthesis of the GHIJK ring system and further experimental support for the originally assigned structure of maitotoxin. (2007) (50)
- New Synthetic Technology for the Construction of N-Containing Quinones and Derivatives Thereof: Total Synthesis of Epoxyquinomycin B. (2001) (50)
- Total Synthesis of Hybocarpone (2001) (50)
- Studies toward diazonamide A: development of a hetero-pinacol macrocyclization cascade for the construction of the bis-macrocyclic framework of the originally proposed structure. (2004) (50)
- Construction of the "left domain" of haplophytine. (2007) (49)
- Total synthesis of echinopines A and B. (2010) (49)
- Biomimetically inspired total synthesis and structure activity relationships of 1-O-methyllateriflorone. 6 pi electrocyclizations in organic synthesis. (2004) (49)
- Total synthesis of (.+-.)-zoapatanol (1980) (49)
- Golfomycin A, a Novel Designed Molecule with DNA‐Cleaving Properties and Antitumor Activity (1990) (49)
- Reactions of 2,3-epoxyhalides. Synthesis of optically active allylic alcohols and homoallylic epoxides (1984) (49)
- Chemical Synthesis of the GHIJKLMNO Ring System of Maitotoxin. (2008) (48)
- A Water‐Soluble Prodrug of Taxol with Self‐Assembling Properties (1994) (48)
- TOTAL SYNTHESIS OF ZARAGOZIC ACID A/SQUALESTATIN S1 (1994) (48)
- Novel strategy for the construction of the oligosaccharide fragment of calichemicin .gamma.1.alpha.I. Synthesis of the ABC skeleton (1990) (48)
- Prostaglandin I2 as a potentiator of acute inflammation in rats. (1978) (48)
- Synthesis of the ABCDEFG ring system of maitotoxin. (2010) (47)
- New synthetic technology for the construction of oxocenes. (1986) (47)
- Molecular design and biological activity of potent and selective protein kinase inhibitors related to balanol. (1995) (47)
- Synthesis of iso-epoxy-amphidinolide N and des-epoxy-caribenolide I structures. Initial forays. (2006) (47)
- Dithiatopazine and related systems. Synthesis, chemistry, x-ray crystallographic analysis, and calculations (1990) (47)
- Total synthesis of ionophore antibiotic X-14547A. 1. Enantioselective synthesis of the tetrahydropyran and tetrahydroindan building blocks (1981) (47)
- Classics in total synthesis : targets, strategies, methods (1996) (47)
- The effects of lipoxin A and lipoxin B on functional responses of human granulocytes. (1987) (47)
- Handbook of Combinatorial Chemistry: Drugs, Catalysts, Materials (2002) (47)
- Dithiatopazine: the first stable 1,2-dithietane (1987) (46)
- Selectivity and Mechanism of Action of Novel DNA‐Cleaving Sulfones (1991) (46)
- Total synthesis of everninomicin 13,384-1--Part 1: retrosynthetic analysis and synthesis of the A1B(A)C fragment. (2000) (46)
- Total synthesis of (+)-rugulosin and (+)-2,2'-epi-cytoskyrin A through cascade reactions. (2005) (46)
- Total synthesis and structural revision of vannusals A and B: synthesis of the originally assigned structure of vannusal B. (2010) (46)
- Susceptibilities of enterovirus D68, enterovirus 71, and rhinovirus 87 strains to various antiviral compounds. (2016) (45)
- Photochemical analogue of the bergman cycloaromatization reaction (1994) (45)
- Chemical synthesis and biological evaluation of novel epothilone B and trans-12,13-cyclopropyl epothilone B analogues (2002) (45)
- A mild method for the synthesis of 2-ketopyrroles from carboxylic acids (1982) (45)
- Total Synthesis of Brevetoxin A: Part 3: Construction of GHIJ and BCDE Ring Systems (1999) (45)
- Involvement of caspase activation in azaspiracid-induced neurotoxicity in neocortical neurons. (2010) (45)
- Total synthesis and absolute configuration of the bisanthraquinone antibiotic BE-43472B. (2009) (45)
- A translactonization route to macrocyclic lactones (1977) (44)
- Total Synthesis of Tovophyllin B. (2009) (44)
- Nodule-inducing activity of synthetic Sinorhizobium meliloti nodulation factors and related lipo-chitooligosaccharides on alfalfa. Importance of the acyl chain structure. (1999) (43)
- Fortschritte in der Chemie und Biologie natürlicher Antibiotika (2009) (43)
- Total synthesis and biological evaluation of monorhizopodin and 16-epi-monorhizopodin. (2011) (43)
- The Absolute Configuration and Asymmetric Total Synthesis of the CP Molecules (CP-263,114 and CP-225,917, Phomoidrides B and A) (2000) (43)
- Total Synthesis of Balanol and Designed Analogues (1995) (43)
- Diversity-oriented organic synthesis and proteomics. New frontiers for chemistry & biology. (2002) (43)
- Antitumor efficacy of 26-fluoroepothilone B against human prostate cancer xenografts (2001) (43)
- Synthetic studies on thiostrepton: construction of thiostrepton analogues with the thiazoline-containing macrocycle. (2003) (43)
- Novel Strategies for the Construction of Complex Polycyclic Ether Frameworks. Stereocontrolled Synthesis of the FGHIJ Ring System of Brevetoxin A (1991) (43)
- Chemical Synthesis and Biological Evaluation of C-2 Taxoids (1995) (43)
- A New Method for the Stereoselective Synthesis of α- and β-Glycosylamines Using the Burgess Reagent (2004) (43)
- Probing the Ring Size of Epothilones: Total Synthesis of [14]-, [15]-, [17]-, and [18]Epothilones A (1998) (43)
- Synthesis of Novel Taxoids (1994) (42)
- New synthetic technologies for the construction of heterocycles and tryptamines. (2009) (42)
- Construction of substituted N-hydroxyindoles: synthesis of a nocathiacin I model system. (2005) (42)
- TOTAL SYNTHESIS OF (+-)-VERMICULINE (1975) (42)
- Enediyne compounds equipped with acid-, base- and photo-sensitive triggering devices. Chemical simulation of the dynemicin A reaction cascade (1991) (42)
- Total synthesis of 16-desmethylepothilone B, epothilone B10, epothilone F, and related side chain modified epothilone B analogues. (2000) (42)
- Total synthesis of the CP-molecules (CP-263,114 and CP-225,917, phomoidrides B and A). 3. Completion and synthesis of advanced analogues. (2002) (42)
- Total Synthesis of Apoptolidin: Part 2. Coupling of Key Building Blocks and Completion of the Synthesis. (2001) (42)
- Radiofrequenz‐verschlüsselte kombinatorische Chemie (1995) (42)
- Zaragozic Acid A/Squalestatin S1: Synthetic and Retrosynthetic Studies (1994) (42)
- Total synthesis and biological evaluation of (-)apicularen A and analogues thereof. (2003) (42)
- Conformational Studies of Sialyl Lewis-X in Aqueous-Solution (1992) (42)
- Reactions of hydroxyl groups with tosylchloride-dimethylaminopyridine system. Direct synthesis of chlorides from hydroxycompounds (1984) (42)
- A practical sulfenylation of 2,5-diketopiperazines. (2012) (41)
- Taxoids: new weapons against cancer. (1996) (41)
- Synthesis of the monomeric unit of the lomaiviticin aglycon. (2009) (41)
- Solid-phase combinatorial synthesis using MicroKan reactors, Rf tagging, and directed sorting. (2000) (41)
- New synthetic technology for the construction of N-hydroxyindoles and synthesis of nocathiacin I model systems. (2007) (41)
- Cell-specific regulation of apoptosis by designed enediynes. (1993) (41)
- Novel chemistry of alpha-tosyloxy ketones: applications to the solution- and solid-phase synthesis of privileged heterocycle and enediyne libraries. (2002) (41)
- Total Synthesis of Viridicatumtoxin B and Analogues Thereof: Strategy Evolution, Structural Revision, and Biological Evaluation (2014) (41)
- An expedient synthesis of a functionalized core structure of bielschowskysin. (2011) (41)
- Gezielt entworfene Epothilone: kombinatorische Synthese, Induktion der Tubulin‐Polymerisation und cytotoxische Wirkung gegen taxolresistente Tumorzellen (1997) (41)
- Total synthesis and biological evaluation of (+)- and (-)-bisanthraquinone antibiotic BE-43472B and related compounds. (2009) (41)
- The total synthesis of coleophomones B and C. (2002) (41)
- Calicheamicin θ 1I: A Rationally Designed Molecule with Extremely Potent and Selective DNA Cleaving Properties and Apoptosis Inducing Activity (1994) (40)
- Adventures in Carbohydrate Chemistry: New Synthetic Technologies, Chemical Synthesis, Molecular Design, and Chemical Biology (2001) (40)
- Total synthesis of sporolide B and 9-epi-sporolide B. (2010) (40)
- Stereospecific synthesis of 1,1-dialkylglycosides (1986) (40)
- Total synthesis and structural elucidation of azaspiracid-1. Synthesis-based analysis of originally proposed structures and indication of their non-identity to the natural product. (2006) (40)
- Irreversible cytoskeletal disarrangement is independent of caspase activation during in vitro azaspiracid toxicity in human neuroblastoma cells. (2007) (40)
- Novel strategies for the solid phase synthesis of substituted indolines and indoles. (2003) (40)
- Total synthesis and chemical biology of the sarcodictyins. (1999) (39)
- Total synthesis of the originally assigned structure of vannusal B. (2008) (39)
- Synthesis of functionalized maoecrystal V core structures. (2010) (39)
- New synthetic technology for the stereocontrolled construction of 1,1'-disaccharides and 1,1':1'',2-trisaccharides. Synthesis of the FG ring system of everninomicin 13,384-1 (1997) (39)
- Reactions of glycosyl fluorides. Synthesis of C-glycosides (1984) (39)
- Total synthesis and structural revision of vannusals A and B: synthesis of the true structures of vannusals A and B. (2010) (39)
- Total synthesis of marinomycins A-C. (2006) (38)
- Total synthesis of floresolide B and Δ6,7-Z-floresolide B (2006) (38)
- Total Synthesis and Biological Evaluation of Glycolipids Plakosides A, B and Their Analogs (2000) (38)
- 6,9-thiaprostacyclin. A stable and biologically potent analogue of prostacyclin (PGI2) (1977) (38)
- STEREOCONTROLLED SYNTHESIS OF THE EVERNINOMICIN A1B(A)C RING FRAMEWORK (1998) (37)
- Expeditious Routes to Evernitrose and Vancosamine Derivatives and Synthesis of a Model Vancomycin Aryl Glycoside (1998) (37)
- Synthesis of 16-membered-ring macrolide antibiotics. 3. Carbomycin B and leucomycin A3: retrosynthetic studies (1981) (37)
- A General Strategy for the Synthesis of Monohydroxy-eicosatetraenoic Acids: Total Synthesis of 5(S)-Hydroxy-6(E),8,11,14(Z)-eicosatetraenoic Acid (5-HETE) and 12(S)-Hydroxy-5,8,14(Z), 10(E)-eicosatetraenoic Acid (12-HETE) (1986) (37)
- Asymmetric total synthesis of cylindrocyclophanes A and F through cyclodimerization and a Ramberg-Bäcklund reaction. (2010) (37)
- Studies toward the synthesis of azadirachtin, part 1: total synthesis of a fully functionalized ABC ring framework and coupling with a norbornene domain. (2005) (37)
- Total synthesis of 26-hydroxy-epothilone B and related analogs via a macrolactonization based strategy (1998) (37)
- Totalsynthese des Vancomycin‐Aglycons – Teil 3: letzte Schritte (1998) (37)
- Sulfonamides as a new scaffold for hypoxia inducible factor pathway inhibitors. (2011) (37)
- Simple efficient synthesis of prostacyclin (PGI2)1 (1977) (37)
- Optimization and mechanistic studies of psammaplin A type antibacterial agents active against methicillin-resistant Staphylococcus aureus (MRSA). (2001) (36)
- Total synthesis of platencin. (2008) (36)
- New synthetic strategies for the construction of medium size cyclic ethers. Stereocontrolled synthesis of the BCD ring framework of brevetoxin A (1990) (36)
- Discovery of Novel Antibacterial Agents Active Against Methicillin‐Resistant Staphylococcus aureus from Combinatorial Benzopyran Libraries (2001) (36)
- Total synthesis of everninomicin 13,384-1--Part 4: explorations of methodology; stereocontrolled synthesis of 1,1'-disaccharides, 1,2-seleno migrations in carbohydrates, and solution- and solid-phase synthesis of 2-deoxy glycosides and orthoesters. (2000) (36)
- Sequence-selective carbohydrate-DNA interaction: dimeric and monomeric forms of the calicheamicin oligosaccharide interfere with transcription factor function. (1996) (36)
- Totalsynthese von Colombiasin A (2001) (36)
- Behind enemy lines. (2001) (36)
- A Suzuki coupling–macrolactamization approach to the AB-COD bicyclic system of vancomycin (1997) (35)
- Molecular Design and Chemical Synthesis of a Highly Potent Epothilone (2006) (35)
- A novel stereocontrolled synthesis of the nonacene ring system of brevetoxin A. Conformational-reactivity effects in 9-membered rings (1990) (35)
- Synthesis and biological properties of C12,13-cyclopropyl-epothilone A and related epothilones. (1998) (35)
- Total synthesis of amphoteronolide B (1987) (35)
- The cytoskyrin cascade: a facile entry into cytoskyrin A, deoxyrubroskyrin, rugulin, skyrin, and flavoskyrin model systems. (2005) (35)
- Total synthesis of elfamycins: aurodox and efrotomycin. 2. Coupling of key intermediates and completion of the synthesis (1985) (34)
- Crossing the boundaries (1994) (34)
- Studies toward the synthesis of azadirachtin, part 2: construction of fully functionalized ABCD ring frameworks and unusual intramolecular reactions induced by close-proximity effects. (2005) (34)
- Stereocontrolled synthesis of model core systems of lomaiviticins A and B. (2006) (34)
- A new method for the synthesis of nonsymmetrical sulfamides using burgess-type reagents. (2002) (34)
- Total Syntheses of Thailanstatins A-C, Spliceostatin D, and Analogues Thereof. Stereodivergent Synthesis of Tetrasubstituted Dihydro- and Tetrahydropyrans and Design, Synthesis, Biological Evaluation, and Discovery of Potent Antitumor Agents. (2018) (34)
- Simple, stereocontrolled total synthesis fof a biologically active analog of the prostaglandin endoperoxides (PGH2, PGG2) (1976) (34)
- Ten‐Membered Ring Enediynes with Remarkable Chemical and Biological Profiles (1992) (34)
- Total synthesis of the CP-molecules (CP-263,114 and CP-225,917, phomoidrides B and A). 1. Racemic and asymmetric synthesis of bicyclo[4.3.1] key building blocks. (2002) (34)
- Totalsynthese des Vancomycin‐Aglycons – Teil 1: Synthese der Aminosäuren 4–7 und Aufbau des AB‐COD‐Ringgerüsts (1998) (34)
- An expedient entry into the fused polycyclic skeleton of vannusal AElectronic supplementary information (ESI) available: selected physical data for compounds 11 and 2. See http://www.rsc.org/suppdata/cc/b2/b208234a/Dedicated to Professor Herbert C. Brown on the occasion of his 90th birthday. (2002) (34)
- Synthesis of the First Fully Functionalized Core of the Zaragozic Acids/Squalestatins (1994) (34)
- Synthesis of C-2 taxol analogues (1994) (33)
- A novel 2'-(N-methylpyridinium acetate) prodrug of paclitaxel induces superior antitumor responses in preclinical cancer models. (2002) (33)
- Studies towards Trichodimerol: Novel Cascade Reactions and Polycyclic Frameworks (1999) (33)
- Design, synthesis, and biological evaluation of a biyouyanagin compound library (2011) (33)
- Total Synthesis of Trioxacarcins DC-45-A1, A, D, C, and C7″-epi-C and Full Structural Assignment of Trioxacarcin C. (2016) (33)
- Synthesis of C-2 taxol analogues (1994) (33)
- New synthetic technology for the synthesis of hindered alpha-diazoketones via acyl mesylates. (1999) (33)
- Thermal cycloadditions of dimethyl acetylenedicarboxylate with cyclic enolethers. An entry into medium size oxocyclic systems (1987) (33)
- Solid phase synthesis of complex natural products and libraries thereof. (2001) (33)
- Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody-Drug Conjugates. (2018) (33)
- Inspirations, discoveries, and future perspectives in total synthesis. (2009) (33)
- Total synthesis of 1-O-methyllateriflorone. (2003) (33)
- Synthesis of the WXYZA' domain of maitotoxin. (2011) (32)
- Total Synthesis of Oxazole‐ and Cyclopropane‐Containing Epothilone B Analogues by the Macrolactonization Approach (1997) (32)
- Synthesis of the Bicyclic Core of CP‐225,917 and CP‐263,114 by an Intramolecular Diels–Alder Reaction (1997) (32)
- NEW TECHNOLOGY FOR THE SYNTHESIS OF VANCOMYCIN-TYPE BIARYL RING SYSTEMS (1997) (32)
- Synthesis and antioxidant evaluation of (S,S)- and (R,R)-secoisolariciresinol diglucosides (SDGs). (2013) (32)
- Studies towards the synthesis of azadirachtin: enantioselective entry into the azadirachtin framework through cascade reactions. (2003) (32)
- The CP molecule labyrinth: a paradigm of how endeavors in total synthesis lead to discoveries and inventions in organic synthesis. (2002) (32)
- Total synthesis of myceliothermophins C, D, and E. (2014) (32)
- Total synthesis of everninomicin 13,384-1--Part 2: synthesis of the FGHA2 fragment. (2000) (32)
- Total synthesis and biological evaluation of marinopyrrole A and analogs (2011) (31)
- Bioinspired synthesis of hirsutellones A, B, and C. (2011) (31)
- Synthesis of highly substituted N-hydroxyindoles through 1,5-addition of carbon nucleophiles to in situ generated unsaturated nitrones. (2006) (31)
- Azaspiracids modulate intracellular pH levels in human lymphocytes. (2006) (31)
- Die Entdeckung und Synthese von marinen Polyethern (2008) (31)
- Total synthesis of ionophore antibiotic X-14547A. 2. Coupling of the tetrahydropyran and tetrahydroindan systems and construction of the butadienyl and ketopyrrole moieties (1981) (31)
- Total Synthesis of Shishijimicin A. (2015) (31)
- Total synthesis of Δ¹²-prostaglandin J₃, a highly potent and selective antileukemic agent. (2014) (31)
- Model studies towards azadirachtin: part 2. Construction of the crowded C8-C14 bond by transition metal chemistry. (2002) (31)
- Synthesis of a fully functionalized CD ring system of taxol (1992) (31)
- The emergence of the structure of the molecule and the art of its synthesis. (2013) (30)
- Novel chemistry of dithiatopazine (1988) (30)
- Total synthesis of novel geometric isomers of lipoxin A4 and lipoxin B4 (1989) (30)
- Die Jagd auf Moleküle, die nie existiert haben: Falsch zugeordnete Naturstoffstrukturen und die Rolle der chemischen Synthese in der modernen Strukturaufklärung (2005) (30)
- Total Synthesis of Thailanstatin A. (2016) (30)
- Cascade reactions involving formal [2+2] thermal cycloadditions: total synthesis of artochamins F, H, I, and J. (2007) (30)
- Stereoselective construction of the C18–C32 fragment of swinholide A (1994) (30)
- A Novel Approach to the CP‐225,917 and CP‐263,114 Core (1997) (30)
- Cell volume decrease as a link between azaspiracid-induced cytotoxicity and c-Jun-N-terminal kinase activation in cultured neurons. (2010) (30)
- Novel enediynes equipped with triggering and detection devices. Isolation of cis-diol models of the dynemicin a cascade (1991) (30)
- Total Synthesis and Structural Revision of Antibiotic CJ-16,264. (2015) (30)
- Selective inhibition of 5‐lipoxygenase by 5,6‐methanoleukotriene A4, a stable analogue of leukotriene A4 (1982) (30)
- Synthesis of the macrocyclic core of apoptolidin (2000) (30)
- Synthesis of macroheterocycles through intramolecular oxidative coupling of furanoid β-ketoesters. (2012) (29)
- NEW SYNTHETIC TECHNOLOGY FOR THE CONSTRUCTION OF 9-MEMBERED RING CYCLIC ETHERS. CONSTRUCTION OF THE EFGH RING SKELETON OF BREVETOXIN A (1997) (29)
- Model studies towards azadirachtin: part 1. Construction of the crowded C8-C14 bond by radical chemistry. (2002) (29)
- A New Photolabile Linker for the Photoactivation of Carboxyl Groups (2001) (29)
- Maitotoxin: An Inspiration for Synthesis. (2011) (29)
- Totalsynthese von Vancomycin (1999) (29)
- Concise and Efficient Total Syntheses of Alkannin and Shikonin. (1998) (28)
- Synthesis of (5Z)- and (5E)-6,9-thiaprostacyclins (1981) (28)
- Second-generation total synthesis of azaspiracids-1, -2, and -3. (2006) (28)
- The true structures of the vannusals, part 2: Total synthesis and revised structure of vannusal B. (2009) (28)
- Durch Olefinmetathese zum Epothilongerüst (1996) (28)
- Totalsynthese von Epothilon A durch Makrolactonisierung (1997) (28)
- An expedient synthesis of D-callipeltose (2001) (28)
- Structure toxicity relationships of synthetic azaspiracid-1 and analogs in mice (2006) (28)
- Identification of distinct thiopeptide-antibiotic precursor lead compounds using translation machinery assays. (2009) (28)
- Bridging of macrocycles to bicycles. New synthetic technology for the construction of cis- and trans-fused oxopolycyclic systems (1986) (28)
- Total synthesis of halipeptins A and D and analogues. (2005) (27)
- Total Synthesis of Oxazole‐ and Cyclopropane‐Containing Epothilone A Analogues by the Olefin Metathesis Approach (1997) (27)
- Studies towards the synthesis of esperamicinone (1994) (27)
- Total syntheses of amythiamicins A, B and C. (2008) (27)
- Bio-inspired synthesis and biological evaluation of a colchicine-related compound library. (2012) (27)
- Stereocontrolled construction of key building blocks for the total synthesis of amphoteronolide B and amphotericin B (1987) (27)
- DIE TOTALSYNTHESE VON BREVETOXIN B : EINE ZWOLF JAHRE WAHRENDE ODYSSEE IN DER ORGANISCHEN SYNTHESE (1996) (27)
- Retrosynthetic and synthetic chemistry on amphotericin B. Synthesis of C(1)–C(20) and C(21)–C(38) fragments and construction of the 38-membered macrocycle (1986) (27)
- Chemistry, biology and medicine of selected tubulin polymerizing agents (1999) (27)
- 12,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological Evaluation of Potent Antitumor Agents. (2017) (27)
- Synthesis of novel disaccharides based on glycosyltransferases: β1,4galactosyltransferase (1991) (27)
- Synthetic calicheamicin mimics with novel initiation mechanisms: DNA cleavage, cytotoxicity, and apoptosis. (1994) (26)
- Total synthesis of carboprostacyclin, a stable and biologically active analogue of prostacyclin (PGI2) (1978) (26)
- Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics. (2020) (26)
- Ionophore antibiotic X-14547A. Degradation studies and stereoselective construction of the "right wing" (C11-C25 fragment) by an intramolecular Diels-Alder reaction (1981) (26)
- Identification of a novel 7-cis-11-trans-lipoxin A4 generated by human neutrophils: total synthesis, spasmogenic activities and comparison with other geometric isomers of lipoxins A4 and B4. (1989) (26)
- The true structures of the vannusals, part 1: Initial forays into suspected structures and intelligence gathering. (2009) (26)
- Diastereomeric monocyclic diallenes. Synthesis and properties of the diastereomeric 3,4,9,10-cyclododecatetraene-1,7-diones and 3,4,10,11-cyclotetradecatetraene-1,8-diones (1973) (26)
- Synthesis and stereochemical assignment of the C1–C10 fragment of nystatin A1 (1989) (26)
- The Art and Science of Organic and Natural Products Synthesis (1998) (26)
- Synthetic Strategy for the Coupling of the Calicheamicin Oligosaccharide with Aglycons: Synthesis of Dynemicin A‐Calicheamicin Hybrid Structures (1991) (26)
- An expedient strategy for the synthesis of tryptamines and other heterocycles. (2008) (26)
- The c-Jun-N-Terminal Kinase is Involved in the Neurotoxic Effect of Azaspiracid-1 (2007) (26)
- The Emergence and Evolution of Organic Synthesis and Why It is Important to Sustain It as an Advancing Art and Science for Its Own Sake (2018) (25)
- Organoselenium-induced ring closures. Stereoselective synthesis of cyclic .alpha.,.beta.-unsaturated sulfoxides, sulfones, and sulfides and synthesis of 6,9-sulfoxa-5(E)- and -5(Z)-prostacyclin, 6,9-sulfo-5(E)- and -5(Z)-prostacyclin, 6,9-sulfo-6.alpha.- and -6.beta.-4(E)-isoprostacyclin, and 6,9-th (1978) (25)
- General synthetic approach to functionalized dihydrooxepines. (2013) (25)
- Synthesis and Biological Investigation of Δ(12)-Prostaglandin J3 (Δ(12)-PGJ3) Analogues and Related Compounds. (2016) (25)
- Asymmetric Alkylation of Anthrones, Enantioselective Total Synthesis of (-)- and (+)-Viridicatumtoxins B and Analogues Thereof: Absolute Configuration and Potent Antibacterial Agents. (2017) (25)
- Stereocontrolled Total Synthesis of (5S,6R)‐, (5S,6S)‐, (5R,6R)‐, and (5R,6S)(7E,9E,11Z,14Z)‐5,6‐Dihydroxy‐7,9,11,14‐icosatetraenoic Acid (5,6‐DiHETE) Methyl Esters (1989) (25)
- The use of PhSeCl in the synthesis of cyclic ethers (1977) (25)
- Ethanoarachidonic acids. A new class of arachidonic acid cascade modulators. 1. Monoethano compounds (1983) (24)
- Rapid Access to Complex Molecular Architectures via o-Azaquinones. (2001) (24)
- An intramolecular Diels–Alder strategy to forskolin (1985) (24)
- Total Synthesis in Search of Potent Antibody-Drug Conjugate Payloads. From the Fundamentals to the Translational. (2019) (24)
- Total Synthesis Endeavors and Their Contributions to Science and Society:A Personal Account (2019) (24)
- Der Kampf um Calicheamicin γ 1I (1993) (24)
- The Art of Total Synthesis Through Cascade Reactions (2010) (24)
- Total Synthesis of Calicheamicin–Dynemicin Hybrid Molecules (1992) (24)
- Synthesis and Biological Evaluation of 12,13‐Cyclopropyl and 12,13‐Cyclobutyl Epothilones (2001) (24)
- Stereoselective construction of the C21–C42 fragment of rapamycin (1993) (23)
- Molecules that changed the world : a brief history of the art and science of synthesis and its impact on society (2008) (23)
- Synthesis of novel heterocycles related to the dynemicin a ring skeleton (1996) (23)
- 6,9-Pyridazaprostacyclin and derivatives: the first "aromatic" prostacyclins (1979) (23)
- Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating Reagents. (2018) (23)
- DNA–Carbohydrate Recognition: Design and Synthesis of an Eight‐Base Sequence‐Selective DNA‐Binding Oligosaccharide (1995) (23)
- Synthesen und biologische Eigenschaften von Prostaglandinendoperoxiden, Thromboxanen und Prostacyclinen (1978) (23)
- Total synthesis of 26-hydroxyepothilone B and related analogues (1997) (23)
- Total Syntheses of Disorazoles A₁ and B₁ and Full Structural Elucidation of Disorazole B₁. (2017) (23)
- Total synthesis and structural revision of viridicatumtoxin B. (2013) (23)
- A total synthesis trilogy: calicheamicin γ1(I), Taxol®, and brevetoxin A. (2012) (23)
- The oxide anion accelerated retro-diels-alder reaction. (1997) (23)
- How thiostrepton was made in the laboratory. (2012) (23)
- Total Synthesis of Vancomycin Aglycon-Part 1: Synthesis of Amino Acids 4-7 and Construction of the AB-COD Ring Skeleton. (1998) (23)
- Joys of molecules. 1. Campaigns in total synthesis. (2005) (22)
- Totalsynthese der Hamigerane – Teil 2: Anwendung der intramolekularen Diels‐Alder‐Reaktion zum Abfangen photochemisch erzeugter Hydroxy‐o‐chinodimethane sowie Strategie und Abschluss der Synthese (2001) (22)
- Discoveries from the Abyss: The Abyssomicins and Their Total Synthesis. (2009) (22)
- Synthesis of ABCtaxoid ring systems via a convergent strategy (1993) (22)
- Simple stereospecific routes to 9-epi-prostaglandin F2α(PGF2β) and 11-epi-prostaglandin F2α (1975) (22)
- Synthesis and Biological Evaluation of QRSTUVWXYZA′ Domains of Maitotoxin (2014) (22)
- Synthesis of the QRSTU domain of maitotoxin and its 85-epi- and 86-epi-diastereoisomers. (2010) (22)
- Ca2+ mobilization with leukotriene A4 and epoxytetraenes in human neutrophils. (1990) (22)
- Total synthesis of halipeptins: isolation of halipeptin D and synthesis of oxazoline halipeptin analogues. (2005) (22)
- Total Synthesis of Truncated Brevetoxin B [AFGHIJK] (1994) (22)
- A convergent strategy towards taxol. A facile enantioselective entry into a fully functionalized ring A system (1992) (22)
- Stereocontrolled synthesis of the quinaldic acid macrocyclic system of thiostrepton. (2002) (22)
- Synthesis of 16-desmethylepothilone B: improved methodology for the rapid, highly selective and convergent construction of epothilone B and analogues (1999) (21)
- Copper(I)‐Promoted Stille Cross‐Coupling of Stannyl Enol Ethers with Enol Triflates: Construction of Complex Polyether Frameworks (1996) (21)
- A Novel Route to the Fused Maleic Anhydride Moiety of CP Molecules. (1999) (21)
- Novel Solution- and Solid-Phase Chemistry of α-Sulfonated Ketones Applicable to Combinatorial Chemistry (2000) (21)
- Phenylsulphenyl-lactonization: an easy and synthetically useful lactonization procedure (1977) (21)
- Total synthesis of (+)-haplophytine. (2009) (20)
- A convergent approach to swinholide A. Stereoselective construction of the C3–C17 fragment of swinholide A (1994) (20)
- Chemie und Biologie der Saragossasuren/Squalestatine (1996) (20)
- Totalsynthese von Eleutherobin (1997) (20)
- Enediyne Generation by a Retro‐Diels–Alder Reaction (1996) (20)
- A SHORT SYNTHETIC ROUTE TO PROSTAGLANDINS UTILIZING POSITION-SELECTIVE EPOXIDE OPENING BY THE VINYL GILMAN REAGENT (1974) (20)
- Total synthesis of coleophomone DElectronic supplementary information (ESI) available: selected physical data for compound 18. See http://www.rsc.org/suppdata/cc/b2/b208236p/ (2002) (20)
- Totalsynthese der CP-Verbindungen CP-263,114 und CP 225,917 – Teil 1: Synthese von Schlüsselintermediaten und neue präparative Erkenntnisse (1999) (20)
- Additions of chlorosulfonyl isocyanate and sulfenyl halides to benzvalene (1974) (20)
- Total synthesis and structural revision of biyouyanagin B. (2010) (20)
- Total synthesis of complex heterocyclic natural products (2008) (20)
- DNA-CARBOHYDRATE INTERACTIONS. SPECIFIC BINDING OF HEAD-TO-HEAD AND HEAD-TO-TAIL DIMERS OF THE CALICHEAMICIN OLIGOSACCHARIDE TO DUPLEX DNA (1996) (20)
- Total synthesis of trioxacarcin DC-45-A2. (2015) (19)
- Azaspiracid substituent at C1 is relevant to in vitro toxicity. (2008) (19)
- Total Synthesis of Δ(12) -Prostaglandin J3 : Evolution of Synthetic Strategies to a Streamlined Process. (2016) (19)
- In vivo arrhythmogenicity of the marine biotoxin azaspiracid-2 in rats (2014) (19)
- Organoselenium-based synthesis of oxygen-containing prostacyclins (1981) (19)
- Stereocontrolled Total Synthesis of Lipoxins As and B5 (1987) (19)
- BIOMIMETISCHE STUDIEN ZU DEN BISORBICILLINOIDEN: TOTALSYNTHESE VON BISORBICILLINOL, BISORBIBUTENOLID UND TRICHODIMEROL (1999) (19)
- Synthesis and biological evaluation of 2',4'- and 3',4'-bridged nucleoside analogues. (2011) (19)
- Perspectives from nearly five decades of total synthesis of natural products and their analogues for biology and medicine. (2020) (19)
- Total synthesis of everninomicin 13,384-1--Part 3: synthesis of the DE fragment and completion of the total synthesis. (1999) (19)
- Synthesis and biological evaluation of new paclitaxel analogs and discovery of potent antitumor agents. (2013) (19)
- Festphasensynthese von Makrocyclen mit der Strategie der Abspaltung unter Cyclisierung: Anwendung der Stille-Kupplung bei der Synthese von (S)-Zearalenon (1998) (19)
- Supercoiling affects the accessibility of glutathione to DNA-bound molecules: positive supercoiling inhibits calicheamicin-induced DNA damage. (1998) (19)
- Chemie und Biologie von Alkannin, Shikonin und verwandten Naphthazarin-Naturstoffen (1999) (18)
- Synthesis of the C'D'E'F' domain of maitotoxin. (2011) (18)
- Lipoxine und verwandte Eicosanoide: Biosynthese, biologische Eigenschaften und chemische Synthese (1991) (18)
- Synthesis of (4E)-9-deoxy-6,9α-epoxy-Δ4-PGF1α, a prostacyclin (PGX) isomer (1977) (18)
- Synthesis of the namenamicin A–C disaccharide: towards the total synthesis of namenamicin (1999) (18)
- Einfache Festphasensynthese von Oligosacchariden – Herstellung eines Dodecasaccharids (1998) (18)
- Catalyst: Synthetic Organic Chemistry as a Force for Good (2016) (18)
- Synthesis of the carboline disaccharide domain of shishijimicin A. (2011) (18)
- Synthesis of Epothilones A and B in Solid and Solution Phase. (1997) (17)
- Stereocontrolled Synthesis of the Sex Pheromones of the Green Stink Bug (1989) (17)
- Design and synthesis of a rapamycin-based high affinity binding FKBP12 ligand. (1995) (17)
- The chemistry-biology-medicine continuum and the drug discovery and development process in academia. (2014) (17)
- Conversion of thionoesters and thionolactones to ethers; a general and efficient radical desulfurisation (1995) (17)
- Carbohydrate-based syntheses of the goldinonolactone and the tetrahydrofuran fragments of aurodox and efrotomycin (1985) (17)
- Totalsynthese der CP‐Verbindungen CP‐263,114 und CP 225,917 – Teil 2: Entwicklung der Schlußstrategie (1999) (17)
- Fluorescent taxoids. (1996) (17)
- Methyl 4‐Hydroxy‐5‐iodo‐2,3‐dimethoxy‐6‐methylbenzoate: The Aromatic Fragment of Calichemicin γ 1αI. Synthesis, X‐Ray Crystallographic Analysis, and Properties (1988) (17)
- The chemical end-ligation of homopyrimidine oligodeoxyribonucleotides within a DNA triple helix. (1997) (17)
- Total Synthesis of the Carbohydrate Fragments of Esperamicin A1 (1992) (17)
- Microsphere-based immunoassay for the detection of azaspiracids. (2014) (17)
- Eine neue Klasse DNA‐spaltender Verbindungen: pH‐abhängige DNA‐Spaltung durch Propargyl‐ und Allenylsulfone (1989) (16)
- Synthesis of the sporolide ring framework through a cascade sequence involving an intramolecular [4+2] cycloaddition reaction of an o-quinone. (2008) (16)
- Perspectives in total synthesis: a personal account (2003) (16)
- RAPID AND EASY PREPARATION OF PROSTACYCLIN (1977) (16)
- Synthesis of novel oligosaccharides (1991) (16)
- Metathesis Reactions in Total Synthesis (2005) (16)
- Saragossasäure A/Squalestatin S1: synthetische und retrosynthetische Untersuchungen (1994) (16)
- Joys of molecules. 2. Endeavors in chemical biology and medicinal chemistry. (2005) (16)
- Synthesis of the CD and E ring systems of the calicheamicin γ1I oligosaccharide (1990) (16)
- Die Eroberung von Taxol (1995) (16)
- Totalsynthese der Hamigerane – Teil 1: Entwicklung einer Synthesemethode für den Aufbau benzanellierter polycyclischer Systeme durch intramolekulares Abfangen von photochemisch erzeugten Hydroxy‐o‐chinodimethanen und Synthese von Schlüsselintermediaten (2001) (16)
- Total synthesis of the potent mutagen S-3-(dodeca-1,3,5,7,9-pentaenyloxy)propane-1,2-diol (1984) (16)
- Totalsynthese von Saragossasäure A/Squalestatin S1 (1994) (16)
- Stereocontrolled Total Synthesis of (5Z,8Z,10E,12R,14Z)-12-Hydroxy-5,8,10,14-icosatetraenoic Acid [(12R)-HETE] (1989) (16)
- Novel strategies to construct the gamma-hydroxy lactone moiety of the CP molecules. Synthesis of the CP-225,917 core skeleton. (1999) (16)
- Total synthesis of atrochamins F, H, I, and J through cascade reactions. (2008) (16)
- Stereocontrolled synthesis of 1,3,5…(2n+ 1) polyols (1982) (15)
- The Enediyne Antibiotics (2010) (15)
- Ring-Closing Metathesis in the Synthesis of Epothilones and Polyether Natural Products (1998) (15)
- Differential effects of 20-trifluoromethyl leukotriene B4 on human neutrophil functions. (1989) (15)
- 5,6-Methanoleukotriene A4. A stable and biologically active analogue of leukotriene A4 (1981) (15)
- Synthetic studies on maduropeptin chromophore 2. Synthesis of the madurosamine aryl amide and the C1′C9′ fragments (1997) (15)
- In vitro chronic effects on hERG channel caused by the marine biotoxin azaspiracid-2. (2014) (15)
- De Novo Design and Synthesis of Somatostatin Non‐Peptide Peptidomimetics Utilizing β‐D‐Glucose as a Novel Scaffolding. (1994) (15)
- Stereoselektive Synthese des Everninomicin‐A1B(A)C‐Gerüsts (1998) (15)
- Origins of selectivity in pericyclic reaction cascades for the synthesis of gambogin and lateriflorone. (2006) (15)
- Synthese des ersten vollstndig funktionalisierten Gerstes der Saragossasuren/Squalestatine (1994) (15)
- Totalsynthese von Epothilon E und seitenkettenmodifizierten Epothilon‐Analoga durch Stille‐Kupplung (1998) (15)
- Synthese des bicyclischen Gerüstes von CP-225,917 und CP-263,114 durch intramolekulare Diels-Alder-Reaktion† (1997) (14)
- A highly convergent strategy towards rapamycin. Stereoselective construction of the C8–C18 fragment (1993) (14)
- Practical Synthesis of p- and o-Amino- and Methoxyphenolic Anthraquinones. (2015) (14)
- Synthesis of the Anthraquinone Framework of Dynemicin A (1994) (14)
- Cyclic Marinopyrrole Derivatives as Disruptors of Mcl-1 and Bcl-xL Binding to Bim (2014) (14)
- Origins of regioselectivity of Diels-Alder reactions for the synthesis of bisanthraquinone antibiotic BE-43472B. (2010) (14)
- Evaluation of synthetic sphingosine, lysosphingolipids and glycosphingolipids as inhibitors of functional responses of human neutrophils. (1990) (14)
- Solution Structure of the Complex between the Head-to-Tail Dimer of Calicheamicin Gamma-1-I Oligosaccharide and a DNA Duplex Containing D(Acct) and D(Tcct) High-Affinity Binding Sites (1998) (14)
- Variation der Ringgröße von Epothilonen – Totalsynthese von [14]‐, [15]‐, [17]‐ und [18]Epothilon A (1998) (14)
- Model Studies towards Diazonamide A: Synthesis of the Heterocyclic Core (2000) (14)
- Total Synthesis and Full Structural Assignment of Namenamicin. (2018) (14)
- A Photolytic Entry into Oxepane Systems (1988) (14)
- TOTALSYNTHESE VON SANGLIFEHRIN A (1999) (13)
- Constructing Molecular Complexity and Diversity: Total Synthesis of Natural Products of Biological and Medicinal Importance (2012) (13)
- Synthesis of 16-membered ring macrolide antibiotics I. Stereoselective construction of the ‘right wing” of the carbomycins and leucomycins from D-glucose (1979) (13)
- Synthetic studies on maduropeptin chromophore 1. Construction of the aryl ether and attempted synthesis of the [7.3.0] bicyclic system (1997) (13)
- Examination of the sialyl lewis X - calcium complex by electrospray mass spectrometry (1994) (13)
- SIMPLE EFFICIENT SYNTHESIS OF PROSTACYCLIN (PGI2) (1978) (13)
- Eine neuartige Strategie zum Aufbau des Vancomycin‐Biarylringsystems (1997) (13)
- Endiin‐Verbindungen mit säure‐, base‐ und lichtempfindlichen Triggergruppen; chemische Simulierung der Dynemicin‐A‐Reaktionskaskade (1991) (13)
- DNA Binding and Cleavage Modes of Shishijimicin A. (2019) (13)
- A general strategy for the total synthesis of the presumed lipoxin structures (1985) (13)
- Totalsynthese von Everninomicin 13,384‐1 – Teil 2: Synthese des FGHA2‐Fragments (1999) (13)
- A Reverse Approach to the Total Synthesis of Halichondrin B. (2021) (12)
- The Chemistry and Biology of Epothilones — The Wheel Keeps Turning (2007) (12)
- Stereokontrollierte Totalsynthesen der Lipoxine A5 und B5 (1987) (12)
- Neue Strategien zur Konstruktion komplexer polycyclischer Ethergerüste; stereokontrollierte Synthese des FGHIJ‐Ringsystems von Brevetoxin A (1991) (12)
- Novel chemistry of taxol. Retrosynthetic and synthetic studies (1994) (12)
- Enantioselective Total Synthesis of Antibiotic CJ-16,264, Synthesis and Biological Evaluation of Designed Analogues, and Discovery of Highly Potent and Simpler Antibacterial Agents. (2017) (12)
- Amphoteronolide B methyl ester. Novel oxidative deglycosidation of amphotericin B (1987) (12)
- Golfomycin A, eine neukonzipierte Verbindung mit DNA‐Spaltungs‐ und Antitumor‐Aktivität (1990) (12)
- Synthesis and biological actions of optically active enediynes related to dynemicin A (1992) (12)
- Streamlined Total Synthesis of Trioxacarcins and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues Thereof. Discovery of Simpler Designed and Potent Trioxacarcin Analogues. (2017) (12)
- Academic-industrial partnerships in drug discovery and development. (2014) (12)
- Preparation and Reactions of Glycosyl Fluorides (1988) (12)
- Solution Structure of the Head-to-Head Dimer of Calicheamicin Oligosaccharide Domain and d(CGTAGGATATCCTACG) 2 (1996) (12)
- CARDIOVASCULAR ACTIONS OF TWO THROMBOXANE A2 ANALOGS (1981) (12)
- Nonpeptidal Peptidomimetics with a β‐D‐Glucose Scaffolding. A Partial Somatostatin Agonist Bearing a Close Structural Relationship to a Potent, Selective Substance P Antagonist. (1993) (12)
- Short Total Synthesis of Δ12-Prostaglandin J2 and Related Prostaglandins. Design, Synthesis, and Biological Evaluation of Macrocyclic Δ12-Prostaglandin J2 Analogues. (2019) (12)
- Total synthesis of oestra-1,3,5(10)-trien-17-one (1979) (11)
- Total Synthesis of Δ12-Prostaglandin J3, a Highly Potent and Selective Antileukemic Agent. (2015) (11)
- Oligosaccharide Synthesis from Glycosyl Fluorides and Sulfides (1997) (11)
- Synthesis of DNA-Binding Oligosaccharides (1997) (11)
- Synthesestrategien zur Kupplung des Calicheamicin‐Oligosaccharids mit Aglyconen; die Synthese von Dynemicin‐A‐Calicheamicin‐Hybridverbindungen (1991) (10)
- Zehngliedrige cyclische Endiine mit bemerkenswerten chemischen und biologischen Eigenschaften (1992) (10)
- Stereochemistry and biosynthesis of lipoxins. (1987) (10)
- Iodine(V) Reagents in Organic Synthesis. Part 4. o‐Iodoxybenzoic Acid as a Chemospecific Tool for Single Electron Transfer‐Based Oxidation Processes. (2002) (10)
- Stereocontrolled total synthesis of (5Z,8Z11Z,13E)(15S)-15-hydroxyeicosa-5,8,11,13-tetraenoic acid (15S-HETE) and analogues (1985) (10)
- DNA–carbohydrate interactions. Design and synthesis of a head-to-tail dimer of the calicheamicin oligosaccharide (1996) (10)
- Recent Advances in the Chemistry and Biology of Naturally Occurring Antibiotics (2009) (10)
- Totalsynthese von Everninomicin 13,384‐1 – Teil 3: Synthese des DE‐Fragments und Abschluß der Totalsynthese (1999) (10)
- Totalsynthese von Apoptolidin – Teil 1: Retrosynthese und Aufbau von Schlüsselintermediaten (2001) (10)
- Synthesis and Biological Evaluation of Novel Epothilone B Side Chain Analogues (2015) (10)
- The Essence of Total Synthesis (2005) (10)
- Enantioselective Intramolecular Friedel—Crafts-Type α-Arylation of Aldehydes. (2009) (10)
- Efficient Synthesis of Dimeric Oxazoles, Piperidines and Tetrahydroisoquinolines from N-Substituted 2-Oxazolones. (2016) (10)
- 6,9-THIAPROSTACYCLIN. A STABLE AND BIOLOGICALLY POTENT ANALOG OF PROSTACYCLIN (PGI2) (1978) (10)
- Totalsynthese von Apoptolidin – Teil 2: Verknüpfung der Schlüsselintermediate und Abschluss der Synthese (2001) (9)
- EIN WASSERLOSLICHES PRODRUG VON TAXOL MIT DER FAHIGKEIT ZUR SELBSTORGANISATION (1994) (9)
- The Olefin Metathesis Approach to Epothilone A and Its Analogues. (1997) (9)
- Stereocontrolled total synthesis of methyl 12(S)-hydroxy-5Z,8E,10E-heptadecatrienoate (1989) (9)
- Design, Synthesis, and Biological Investigation of Epothilone B Analogues Featuring Lactone, Lactam, and Carbocyclic Macrocycles, Epoxide, Aziridine, and 1,1-Difluorocyclopropane and Other Fluorine Residues. (2020) (9)
- cis-3,4-Dichlorocyclobutene as a Versatile Synthon in Organic Synthesis. Rapid Entry into Complex Polycyclic Systems with Remarkably Stereospecific Reactions. (2002) (9)
- Calicheamicin θ 1I: Durch Moleküldesign zu einer Verbindung, die DNA selektiv und effizient spaltet und Zelltod auslöst (1994) (9)
- 4‐Hydroxy‐5‐iod‐2,3‐dimethoxy‐6‐methylbenzoesäuremethylester: Der aromatische Teil von Calichemicin γ 1αI; Synthese, Röntgenstrukturanalyse und Eigenschaften (1988) (9)
- The Chemical Synthesis of C‐Ring Aryl Taxoids (2006) (9)
- The endeavor of total synthesis and its impact on chemistry, biology and medicine (2014) (9)
- Designed Enediynes: A New Class of DNA‐Cleaving Molecules with Potent and Selective Anticancer Activity. (1993) (9)
- TOTALSYNTHESE VON CALICHEAMICIN-DYNEMICIN-HYBRIDMOLEKULEN (1992) (9)
- A synthetic route to forskolin (1989) (9)
- Einfache Zugänge zu Evernitrose und Vancosaminderivaten sowie Synthese eines Vancomycin-Modellglycosids (1998) (9)
- Reversal of the phenylseleno- and phenylsulpheno-cyclizations. Synthesis of olefins from phenylseleno- and phenylsulpheno-lactones, phenylselenoethers, and α-hydroxyselenides (1979) (9)
- Discovery and Optimization of Non‐steroidal FXR Agonists from Natural Product‐Like Libraries. (2003) (9)
- An Expeditious and Efficient Entry into the Aphidicolin and Related Natural Products Ring Skeleton (1981) (9)
- Synthesis of 7,13-bridged arachidonic acid analogues (1984) (8)
- Synthetic and Semisynthetic Analogs of Epothilones: Chemistry and Biological Activity (2001) (8)
- Pericyclic Reactions in Organic Synthesis and Biosynthesis: Synthetic Adventures with Endiandric Acids A–G (1984) (8)
- Ein photolytischer Zugang zu Oxepansystemen (1988) (8)
- Click Triazoles (2012) (8)
- On the mechanism of activation of designed enediynes with selective cytotoxicity (1992) (8)
- Ein neuartiger Zugang zum zentralen Gerüst von CP‐225,917 und CP‐263,114 (1997) (8)
- Total synthesis and biological evaluation of marinopyrrole A and analogues. (2011) (8)
- Chemistry and Biology of Diazonamide A: First Total Synthesis and Confirmation of the True Structure [J. Am. Chem. Soc. 2004, 126, 12888−12896]. (2004) (8)
- Enantioselective Intramolecular Friedel-Crafts-Type α-Arylation of Aldehydes (Journal of the American Chemical Society (2009) 131 (2086-2087)) (2009) (8)
- Chemistry and Biology of Alkannin, Shikonin, and Related Naphthazarin Natural Products (1999) (8)
- Stereoselective total synthesis of the presumed biosynthetic precursor to lipoxins A and B: methyl (7E,9E,11Z,13E,5S,6S,15S)-5,6-epoxy-15-hydroxyicosa-7,9,11,13-tetra-enoate and its 5,6-methano analogue (1986) (8)
- Synthesis of sulphur-containing prostacyclin PGI1 analogues 6,9-epithio-PGI1, its S-oxide stereoisomers, and its SS-dioxide (1978) (8)
- A general and stereocontrolled total synthesis of leukotriene B4 and analogues (1984) (8)
- Reaction of Phenylselenenyl Chloride with Enol Ethers and 1,2-Ethanediyl Acetals. Synthesis of α-Phenylseleno-aldehydes and α-Phenylseleno-acetals (1979) (8)
- Total Synthesis of 20‐Hydroxy‐ and 20‐Carboxy‐leukotrienes B4. (1986) (8)
- Total Synthesis of Vancomycin Aglycon. Part 2. Synthesis of Amino Acids 1—3 and Construction of the AB-COD-DOE Ring Skeleton. (1999) (7)
- In vivo efficacy of novel synthetic enediynes 1. (1995) (7)
- Synthesis of stable thromboxane A2 analogs: pinane thromboxane A2 (PTA2) and carbocyclic thromboxane A2 (CTA2). (1982) (7)
- Kurze und effiziente Totalsynthesen von Alkannin und Shikonin (1998) (7)
- DNA-Kohlenhydrat-Erkennung: Design und Synthese eines an eine DNA-Sequenz aus acht Basen selektiv bindenden Oligosaccharids† (1995) (7)
- Marinopyrrole Derivatives with Sulfide Spacers as Selective Disruptors of Mcl-1 Binding to Pro-Apoptotic Protein Bim (2014) (7)
- Progress towards the total synthesis of the enediyne anticancer antibiotics (1993) (7)
- Cationization of organometallo carbonyl compounds by fast ion bombardment (1992) (7)
- Profile. K. C. Nicolaou. (2003) (7)
- Synthesis of Imides, N‐Acyl Vinylogous Carbamates and Ureas, and Nitriles by Oxidation of Amides and Amines with Dess—Martin Periodinane. (2006) (7)
- Stereospecific 1,2-Migrations in Carbohydrates. Stereocontrolled Synthesis of α- and β-2-Deoxyglycosides. (1986) (7)
- Palladium-Catalyzed Cross-Coupling Reactions in Total (2005) (7)
- Total Synthesis of Hamigerans. Part 2. Implementation of the Intramolecular Diels—Alder Trapping of Photochemically Generated Hydroxy-o-quinodimethanes; Strategy and Completion of the Synthesis. (2002) (7)
- Ein außergewöhnlicher Zugang zur anellierten Maleinsäureanhydrid‐Einheit der CP‐Moleküle (1999) (7)
- Synthese und biologische Aktivität von Sarcodictyinen (1998) (7)
- Synthese von Makroheterocyclen durch intramolekulare oxidative Kupplung von furanoiden β‐Ketoestern (2012) (7)
- Monocyclic allenes. Synthesis of 3,8,9-cycloundecatriene-1,6-dione and 12-oxabicyclo[7.2.1]dodeca-5,6,9,11-tetraen-3-one, a furanophane containing an allene group (1973) (6)
- Total Synthesis of Hamigerans. Part 1. Development of Synthetic Technology for the Construction of Benzannulated Polycyclic Systems by the Intramolecular Trapping of Photogenerated Hydroxy-o-quinodimethanes and Synthesis of Key Building Blocks. (2002) (6)
- Synthesis of thromboxane A2 analogs. (1980) (6)
- Syntheses of Cyclopropyl Analogues of Disorazoles A1 and B1 and Their Thiazole Counterparts. (2018) (6)
- Structural assignment and total synthesis of azaspiracid-1 (2007) (6)
- The art and science of constructing the molecules of nature. (2004) (6)
- Total Synthesis of the Monomeric Unit of Lomaiviticin A. (2020) (6)
- A new designed tumor selective daunomycin derivative (1993) (6)
- Asymmetric Synthesis of 3-Substituted 4-Oxoesters Using the SAMP-/RAMP-Hydrazone Method (1998) (6)
- Zur Struktur des Maitotoxins (2007) (6)
- Vom Aufkommen des Molekülkonzepts zur Kunst der Molekülsynthese (2013) (6)
- Novel IBX-Mediated Processes for the Synthesis of Amino Sugars and Libraries Thereof. (2000) (6)
- Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates. (2020) (6)
- Chapter 17 Prostacyclin, Thromboxanes and the Arachidonic Acid Cascade (1979) (6)
- SYNTHESIS OF NOVEL MACROCYCLIC LACTONES IN THE PROSTAGLANDIN AND POLYETHER ANTIBIOTIC SERIES (1975) (5)
- TOTAL SYNTHESIS OF ERYTHROMYCINS. 4. TOTAL SYNTHESIS OF ERYTHRONOLIDE B (1978) (5)
- Die Totalsynthese der Kohlenhydratbausteine von Esperamicin A1 (1992) (5)
- Synthese von C‐2‐analogen Taxolen (1994) (5)
- Experimental Evolution of Diverse Strains as a Method for the Determination of Biochemical Mechanisms of Action for Novel Pyrrolizidinone Antibiotics. (2017) (5)
- Synthesis of 3,4,5,10,11,12-cyclotetradecahexaene-1,8-dione, a monocyclic dicumulenedione (1973) (5)
- Stereokontrollierte Totalsynthese von (5S,6R)‐, (5S,6S)‐, (5R,6R)‐ und (5R,6S)‐ (7E,9E,11Z,14Z)‐5,6‐Dihydroxy‐7,9,11,14‐icosatetraensäure‐(5,6‐DiHETE)methylester (1989) (5)
- Total Synthesis of the NodRm-IV Factors, the Rhizobium Nodulation Signals. (1993) (5)
- Activation of 6-Endo Over 5-Exo Hydroxy Epoxide Openings. Stereoselective and Ring Selective Synthesis of Tetrahydrofuran and Tetrahydropyran Systems. (1989) (5)
- The total synthesis of the lipoxins and related compounds. (1988) (5)
- Sulfur and the enediyne antibiotics (1993) (5)
- The Total Synthesis of Paclitaxel by Assembly of the Ring System (1994) (5)
- Total Synthesis of Sialyl Dimeric Lex. (1992) (5)
- Diastereomeric monocyclic diallenes. The synthesis of cyclododeca-3,4,9,10-tetraene-1,7-dione (1970) (5)
- Total synthesis of selected natural products (1997) (5)
- The β‐D‐Glucose Scaffold as a β‐Turn Mimetic (2010) (5)
- The Evolution and Impact of Total Synthesis on Chemistry, Biology and Medicine (2017) (5)
- Total Synthesis of the Proposed Azaspiracid-1 Structure. Part 2. Coupling of the C1-C20, C21-C27, and C28-C40 Fragments and Completion of the Synthesis. (2003) (5)
- New Synthetic Technology for the Synthesis of Aryl Ethers: Construction of C‐O‐D and D‐O‐E Ring Model Systems of Vancomycin. (1997) (4)
- Pharmacodynamics of lipoxin A4 in airway smooth muscle (2005) (4)
- Total Synthesis of Sulfated Lex and Lea‐Type Oligosaccharide Selectin Ligands. (1994) (4)
- Enantioselective Total Synthesis of (‐)‐Calicheamicinone. (1992) (4)
- Construction of the Complete Aromatic Core of Diazonamide A by a Novel Hetero Pinacol Macrocyclization Cascade Reaction. (2002) (4)
- New Synthetic Technology for the Synthesis of Hindered α-Diazoketones via Acyl Mesylates. (1999) (4)
- Design, Synthesis, and Study of Simple Monocyclic Conjugated Enediynes. The 10-Membered Ring Enediyne Moiety of the Enediyne Anticancer Antibiotics. (1993) (4)
- ASPECTS OF EICOSANOIDS IN INFLAMMATION (1989) (4)
- New Synthetic Technology for the Construction of 9-Membered Ring Cyclic Ethers. Construction of the EFGH Ring Skeleton of Brevetoxin A. (1997) (4)
- Macrocyclic Peptide Inhibitors of Serine Proteases. Convergent Total Synthesis of Cyclotheonamides A and B via a Late-Stage Primary Amine Intermediate. Study of Thrombin Inhibition under Diverse Conditions. [Erratum to document cited in CA122:161323] (1995) (4)
- Total Synthesis of the CP Molecules CP‐225,917 and CP‐263,114. Part 2. Evolution of the Final Strategy. (1999) (4)
- Total Synthesis of Hemibrevetoxin B and (7aα)-epi-Hemibrevetoxin B (2010) (4)
- A General Strategy for the Synthesis of Monohydroxyeicosatetraenoic Acids: Total Synthesis of 5(S)-Hydroxy-6(E),8,11,14(Z)-eicosatetraenoic Acid (5-HETE) and 12(S)-Hydroxy-5,8,14(Z),10(E)-eicosatetraenoic Acid (12-HETE). (1986) (4)
- Total Synthesis of Abyssomicin C and atrop‐Abyssomicin C. (2006) (4)
- Chemistry and biology of selected natural products (1996) (4)
- Diastereomeric monocyclic diallenes. The stereochemistry of formation of racemic and meso-3,4,9,10-cyclodecatetraene-1,7-dione (1972) (4)
- Chemical Synthesis of Complex Carbohydrates (2000) (4)
- Synthesis of Novel Heterocycles Related to the Dynemicin A Ring Skeleton. (1996) (4)
- A new journal for an expanding field (1994) (4)
- A Novel Regio‐ and Stereoselective Synthesis of Sulfamidates from 1,2‐Diols Using Burgess and Related Reagents: A Facile Entry into β‐Amino Alcohols. (2002) (4)
- Totalsynthese und Revidierung der Struktur von Viridicatumtoxin B (2013) (4)
- Total Synthesis of the CP-Molecules (CP-263,114 and CP-225,917, Phomoidrides B and A). Part 3. Completion and Synthesis of Advanced Analogues. (2002) (4)
- A Highly Convergent Total Synthesis of Norhalichondrin B. (2021) (4)
- Synthesis and Structural Elucidation of Azaspiracid-1 (2006) (4)
- Synthesis of the Tricyclic Core of Eleutherobin and Sarcodictyins and Total Synthesis of Sarcodictyin A. (1998) (4)
- Solid Phase Synthesis of Complex Natural Products and Libraries Thereof (2002) (4)
- Total Synthesis of Gukulenin B via Sequential Tropolone Functionalizations. (2022) (4)
- Synthesis and biological evaluation of dimeric furanoid macroheterocycles: discovery of new anticancer agents. (2015) (4)
- Lipoxin A4-induced release of thromboxane in the guinea-pig lung: studies of its characteristics using lipoxin A4-methyl ester. (1992) (4)
- SYNTHESIS AND BIOLOGICAL PROPERTIES OF PROSTACYCLINS AND PROSTAGLANDIN ENDOPEROXIDE ANALOGS (1979) (4)
- Total Syntheses of Epothilones A and B via a Macrolactonization-Based Strategy. (1997) (3)
- Novel Reactions Initiated by Titanocene Methylidenes: Deoxygenation of Sulfoxides, N‐Oxides, and Selenoxides. (2000) (3)
- The Battle of Calicheamicin γI 1 (1994) (3)
- Total Synthesis of Calicheamicin γ1I (1993) (3)
- Redox-Controlled Bergman Cycloaromatizations. Designed Enediynes with DNA-Cleaving Properties and Antitumor Activity. (2010) (3)
- Total Synthesis of Amphoteronolide B and Amphotericin B. Part 1. Strategy and Stereocontrolled Construction of Key Building Blocks. (1988) (3)
- Wie Thiostrepton im Labor synthetisiert wurde (2012) (3)
- Solution and Solid-Phase Synthesis of Functionalized 3-Arylbenzofurans by a Novel Cyclofragmentation—Release Pathway. (2000) (3)
- Kupfer(I)‐unterstützte Stille‐Kupplung von α‐stannylsubstituierten Enolethern mit Enoltriflaten: Aufbau von komplexen Polyethergerüsten (1996) (3)
- Synthesis of Zaragozic Acid A/Squalestatin S1. (1996) (3)
- Streamlined Symmetrical Total Synthesis of Disorazole B1 and Design, Synthesis, and Biological Investigation of Disorazole Analogues. (2020) (3)
- Novel Strategy for the Construction of the Oligosaccharide Fragment of Calicheamicin γ1αI. Synthesis of the ABC Skeleton. (1990) (3)
- Combinatorial Chemistry in Perspective (2005) (3)
- Practical Synthesis ofp-ando-Amino- and Methoxyphenolic Anthraquinones (2015) (3)
- Total Synthesis of Hamigerans and Analogues Thereof. Photochemical Generation and Diels—Alder Trapping of Hydroxy-o-quinodimethanes. (2004) (3)
- Synthesis of prostaglandin H2 (PGH2) and prostacyclin (PGI2) analogs: tetrathia-PGH2 and PGI2-ketal methyl ester. (1978) (3)
- Total Synthesis of Swinholide A. (1996) (3)
- Oxidation of Silyl Enol Ethers by Using IBX and IBX×N‐Oxide Complexes: A Mild and Selective Reaction for the Synthesis of Enones. (2002) (3)
- SIMPLE, STEREOCONTROLLED TOTAL SYNTHESIS OF A BIOLOGICALLY ACTIVE ANALOG OF THE PROSTAGLANDIN ENDOPEROXIDES (PGH2, PGG2) (1976) (3)
- Cover Picture: Palladium‐Catalyzed Cross‐Coupling Reactions in Total Synthesis / Metathesis Reactions in Total Synthesis (Angew. Chem. Int. Ed. 29/2005) (2005) (3)
- Molecular basis for the inhibition of human a-thrombin by the macrocyclic peptide cyclotheonamide A ( serine protease / a-keto amide / transition-state analogue / x-ray crystallography / total synthesis ) (2005) (3)
- Lipoxin A4 causes generation of thromboxane A2 in the guinea-pig lung (2005) (3)
- Molecular Design, Chemical Synthesis, Kinetic Studies, Calculations, and Biological Studies of Novel Enediynes Equipped with Triggering, Detection, and Deactivating Devices. Model Dynemicin A Epoxide and cis‐ Diol Systems. (1993) (3)
- Bridging of Macrodithionolactones to Bicyclic Systems. Synthesis and Modeling of Oxapolycyclic Frameworks. (1990) (3)
- Synthesis of cyclotetradeca-3,4,5,10,11,12-hexaene-1,8-dione, a monocyclic dicurnulenedione (1971) (3)
- Formal Synthesis of Platencin (2009) (3)
- Das Labyrinth der CP‐Verbindungen: ein Musterbeispiel dafür, wie Bemühungen in der Totalsynthese zu Entdeckungen und Erfindungen in der Organischen Synthese führen (2002) (3)
- Lassen sich Moleküle mit mehreren stereogenen Elementen nach der CIP‐Nomenklatur angemessen beschreiben? Eine Fallstudie mit Vancomycin und verwandten Verbindungen (2001) (3)
- Stereocontrolled Synthesis of the Everninomicin A1B(A)C Ring Framework. (1998) (3)
- Total Synthesis of Vancomycin Aglycon. Part 3. Final Stages. (1999) (3)
- SYNTHETIC TECHNOLOGY AND TOTAL SYNTHESIS: THE ELFAMYCINS (1985) (3)
- 5,6-methano leukotriene A4: a potent specific inhibitor for 5-lipoxygenase. (1983) (2)
- Total Synthesis of Coleophomone D. (2003) (2)
- Total Synthesis of Viridicatumtoxin B and Analogues Thereof: Strategy Evolution, Structural Revision, and Biological Evaluation. (2015) (2)
- Chemical Synthesis of Glycosphingolipids (1991) (2)
- Total Synthesis of Amphotericin B (X). (1987) (2)
- Epothilones and Sarcodictyins: From Combinatorial Libraries to Designed Analogs (2001) (2)
- Total Synthesis of Balanol and Designed Analogues. (1996) (2)
- New Synthetic Technology for the Stereocontrolled Construction of 1,1′‐Disaccharides and 1,1′:1′′,2‐Trisaccharides. Synthesis of the FG Ring System of Everninomicin 13,384‐1. (1998) (2)
- Total Synthesis of Epothilone A: The Macrolactonization Approach. (1997) (2)
- Structural Revision and Total Synthesis of Azaspiracid‐1. Part 2. Definition of the ABCD Domain and Total Synthesis. (2004) (2)
- Endiine durch Retro-Diels-Alder-Reaktion† (1996) (2)
- Conformational Studies of Sialyl Lewis X in Aqueous Solution. (1992) (2)
- Novel Strategies to Construct the γ-Hydroxy Lactone Moiety of the CP Molecules. Synthesis of the CP-225,917 Core Skeleton. (1999) (2)
- A Novel Approach to the CP-225,917 and CP-263,114 Core. (1998) (2)
- SYNTHESIS OF BREFELDIN A, CARPAINE, VERTALINE AND ERYTHRONOLIDE B FROM NONMACROCYCLIC PRECURSORS (1975) (2)
- Total Synthesis of Taxol. Part 4. The Final Stages and Completion of the Synthesis (1995) (2)
- Molecular Design and Chemical Synthesis of a Highly Potent Epothilone. (2006) (2)
- Total Synthesis of Brevetoxin B. Part 1. CDEFG Framework. (1995) (2)
- Titelbild: Palladiumkatalysierte Kreuzkupplungen in der Totalsynthese / Metathesereaktionen in der Totalsynthese (Angew. Chem. 29/2005) (2005) (2)
- High‐Throughput Combinatorial Synthesis of Discrete Compounds in Multimilligram Quantities: Non‐Chemical Encoding and Directed Sorting (2001) (2)
- Synthesis of the Macrocyclic Core of Apoptolidin. (2000) (2)
- Solid‐Phase Synthesis of Natural Products and Natural Product‐Like Libraries (2005) (2)
- Selektivität und Wirkungsmechanismus neuer DNA‐spaltender Sulfone (1991) (2)
- A REMARKABLY SIMPLE, HIGHLY EFFICIENT, AND STEREOSELECTIVE SYNTHESIS OF STEROIDS AND OTHER POLYCYCLIC SYSTEMS. TOTAL SYNTHESIS OF ESTRA-1,3,5(10)-TRIEN-17-ONE VIA INTRAMOLECULAR CAPTURE OF O-QUINODIMETHANES GENERATED BY CHELETROPIC EL (1980) (2)
- AN EFFICIENT AND MILD LACTONIZATION METHOD FOR THE SYNTHESIS OF MACROLIDES (1974) (2)
- Discoveries from the Abyss: The Abyssomicins and Their Total Synthesis (2009) (2)
- Correction: Synthesis of epothilones A and B in solid and solution phase (1997) (2)
- Ten-Membered Ring Enediynes with Remarkable Chemical and Biological Properties. (1992) (2)
- An Expedient Entry into the Fused Polycyclic Skeleton of Vannusal A. (2003) (2)
- Total Synthesis of (+)‐Rugulosin and (+)‐2,2′‐epi‐Cytoskyrin A Through Cascade Reactions. (2006) (2)
- Stereocontrolled total synthesis of apicularen A and its delta(17,18) Z isomer. (2002) (2)
- Total Synthesis of Marinomycins A‐C and of Their Monomeric Counterparts Monomarinomycin A and iso‐Monomarinomycin A. (2007) (2)
- Effect of 6,9-thia prostaglandin I2 (a stable PGI2 analogue) on passive cutaneous anaphylaxis (PCA) in rats. (1979) (2)
- Synthesis of the macrocyclic core of sanglifehrin A (1999) (2)
- Synthesis of the Namenamicin A—C Disaccharide: Towards the Total Synthesis of Namenamicin. (1999) (2)
- THE ENDIANDRIC ACID CASCADE. ELECTROCYCLIZATIONS IN ORGANIC SYNTHESIS. 4. BIOMIMETIC APPROACH TO ENDIANDRIC ACIDS A‐G. TOTAL SYNTHESIS AND THERMAL STUDIES (1983) (2)
- Novel Stereocontrolled Synthesis of the Nonacene Ring System of Brevetoxin A. Conformational-Reactivity Effects in Nine-Membered Rings. (1990) (2)
- The Absolute Configuration and Asymmetric Total Synthesis of the CP Molecules (CP-263,114 and CP-225,917, Phomoidrides B and A). (2010) (2)
- Total Synthesis of the CP Molecules CP-263,114 and CP-225,917. Part 1. Synthesis of Key Intermediates and Intelligence Gathering. (1999) (2)
- Model Studies Towards Azadirachtin. Part 1. Construction of the Crowded C8—C14 Bond by Radical Chemistry. (2002) (2)
- Total Synthesis of Brevetoxin A. Part 1. First Generation Strategy and Construction of BCD Ring System. (1999) (2)
- A Practical and Enantioselective Synthesis of Glycosphingolipids and Related Compounds. Total Synthesis of Globotriaosylceramide (Gb3). (1989) (2)
- Total Synthesis and Structural Elucidation of Azaspiracid‐1. Synthesis‐Based Analysis of Originally Proposed Structures and Indication of Their Non‐Identity to the Natural Product. (2006) (2)
- Total Synthesis of Swinholide A, Preswinholide A, and Hemiswinholide A. (1996) (2)
- Chemistry and biology of the calicheamicins (1994) (2)
- Synthesis of (+)-BE-43472B (2009) (2)
- Recent Advances in the Synthesis of Cyclic Polyether Marine Natural Products (2005) (2)
- Activation of 7-Endo Over 6-Exo Epoxide Openings. Synthesis of Oxepane and Tetrahydropyran Systems. (1989) (2)
- Die Bedeutung der organischen Synthese bei der Entstehung und Entwicklung von Antikörper‐Wirkstoff‐Konjugaten als gezielte Krebstherapien (2019) (2)
- The Total Synthesis of the Lipoxins and Related Compounds (1989) (1)
- Total Synthesis of Δ12-Prostaglandin J3: Evolution of Synthetic Strategies to a Streamlined Process. (2016) (1)
- Synthesis of Palmerolide A (2008) (1)
- Total Synthesis of Biyouyanagin A (2007) (1)
- Total Synthesis of the Oligosaccharide Fragment of Calicheamicin . gamma.I 1. (1991) (1)
- How Thiostrepton Was Made in the Laboratory (2013) (1)
- Synthesis of Uncialamycin (2007) (1)
- Modern Synthetic Technology and Total Synthesis of Bioactive Molecules (1986) (1)
- Vignette 1: The Olefin Metathesis Reaction in Complex Molecule Construction (2008) (1)
- Progress in the Total Synthesis of Brevetoxins (2010) (1)
- The Art and Science of Total Synthesis and the Dawn of the Twenty‐First Century (2010) (1)
- Design, Synthesis, and Biological Evaluation of Tubulysin Analogues, Linker-Drugs, and Antibody-Drug Conjugates, Insights into Structure-Activity Relationships, and Tubulysin-Tubulin Binding Derived from X-ray Crystallographic Analysis. (2021) (1)
- Structural Revision and Total Synthesis of Azaspiracid-1. Part 1. Intelligence Gathering and Tentative Proposal. (2004) (1)
- Dithiatopazine and Related Systems. Synthesis, Chemistry, X-Ray Crystallographic Analysis and Calculations. (1990) (1)
- Molecular Design and Chemical Synthesis of Potent Enediynes. Part 2. Dynemicin Model Systems Equipped with C‐3 Triggering Devices and Evidence for Quinone Methide Formation in the Mechanism of Action of Dynemicin A. (1993) (1)
- DIASTEREOMERIC MONOCYCLIC DIALLENES, SYNTHESIS AND PROPERTIES OF THE DIASTEREOMERIC 3,4,9,10-CYCLODODECATETRAENE-1,7-DIONES AND 3,4,10,11-CYCLOTETRADECATETRAENE-1,8-DIONES (1973) (1)
- Dithiatopazine: The First Stable 1,2‐Dithietane. (1987) (1)
- Invigorating education. (2011) (1)
- Model Studies Towards Azadirachtin. Part 2. Construction of the Crowded C8—C14 Bond by Transition Metal Chemistry. (2002) (1)
- DNA Cleavage by a Synthetic Mimic of the Calicheamicin-Esperamicin Class of Antibiotics. (1989) (1)
- Cascade Reactions in Total Synthesis: Recent Advances (2004) (1)
- Synthesis of the FGHI Ring System of Azaspiracid. (2010) (1)
- Rhodium-Catalyzed Asymmetric Enyne Cycloisomerization (2009) (1)
- The Structure of Maitotoxin. (2007) (1)
- Novel Chemistry of Taxol. Retrosynthetic and Synthetic Studies. (1994) (1)
- Total Synthesis of Oxazole‐ and Cyclopropane‐Containing Epothilone B Analogues by the Macrolactonization Approach. (1998) (1)
- Book Review: Total Synthesis of Natural Products: The “Chiron” Approach. By S. Hanessian (1986) (1)
- Creating complexity: the beauty and logic of synthesis (2003) (1)
- Synthesis of the WXYZA′ Domain of Maitotoxin. (2011) (1)
- Titelbild: Structural Revision and Total Synthesis of Azaspiracid‐1, Part 1: Intelligence Gathering and Tentative Proposal (Angew. Chem. 33/2004) (2004) (1)
- Total Synthesis of Epothilone A: The Olefin Metathesis Approach. (1997) (1)
- REACTIONS OF 2,3-EPOXY HALIDES. SYNTHESIS OF OPTICALLY ACTIVE ALLYLIC ALCOHOLS AND HOMOALLYLIC EPOXIDES (1984) (1)
- Total Synthesis of Everninomicin 13,384-1. Part 1. Synthesis of the A1B(A)C Fragment. (2000) (1)
- Total synthesis of Taxol. 2. construction of A and C ring intermediates and initial attempts to construct the ABC ring system. [Erratum to document cited in CA122:160984] (1995) (1)
- Cover Picture: Angew. Chem. Int. Ed. 10/2002 (2002) (1)
- Novel Enediynes Equipped with Triggering and Detection Devices. Isolation of cis‐Diol Models of the Dynemicin A Cascade. (1992) (1)
- Synthesis of (+)-Cortistatin A (2009) (1)
- HIGHLY ACTIVE PROSTACYCLIN ANALOG SYNTHESIZED (1978) (1)
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- Total Synthesis of Calicheamicin γI 1. Part 1. Synthesis of the Oligosaccharide Fragment. (1993) (1)
- Stereocontrolled Total Synthesis of Lipoxins A5 and B5. (1988) (1)
- Methyl 4‐Hydroxy‐5‐iodo‐2,3‐dimethoxy‐6‐methylbenzoate: The Aromatic Fragment of Calichemicin γI 1α. Synthesis, X‐Ray Crystallographic Analysis, and Properties. (1988) (1)
- A triple test for screening biological activity of prostacyclin analogues (1978) (1)
- Synthesis of (-)-Platensimycin (2007) (1)
- Retrosynthetic and Synthetic Chemistry on Amphotericin B. Synthesis of C(1) - C(20) and C(21)- C(38) Fragments and Construction of the 38-Membered Macrocycle (1986) (1)
- A unified strategy for the total syntheses of eribulin and a macrolactam analogue of halichondrin B (2022) (1)
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- An Olefin Metathesis Based Strategy for the Construction of the JKL, OPQ, and UVW Ring Systems of Maitotoxin. (1997) (1)
- A Facile Method for the Solution and Solid‐Phase Synthesis of Substituted [3.3.1] Bicycles. (1999) (1)
- SYNTHESIS OF 16-MEMBERED RING MACROLIDE ANTIBIOTICS. I. STEREOSELECTIVE CONSTRUCTION OF THE “RIGHT WING” OF THE CARBOMYCINS AND LEUCOMYCINS FROM D-GLUCOSE (1979) (1)
- Stereocontrolled Total Synthesis of (5S,6R)-, (5S,6S)-, (5R,6R)- and (5R,6S)-(7E,9E,11Z,14Z)-5,6-Dihydroxy-7,9,11,14-icosatetraenic Acid (5,6-DiHETE) Methyl Esters (1989) (1)
- Total Synthesis of Natural Products and Designed Molecules: Brevetoxin B (1998) (1)
- Synthesis of Kinamycin C (2007) (1)
- Cover Picture: Molecular Design and Chemical Synthesis of a Highly Potent Epothilone (ChemMedChem 1/2006) (2006) (1)
- Total Synthesis of Calicheamicin‐Dynemicin Hybrid Molecules. (1992) (1)
- Photochemical Analogue of the Bergman Cycloaromatization Reaction. (2010) (1)
- Synthesis and Chemistry of Dynemicin A Models. (1991) (1)
- Nucleophilic Additions to Thionolactones. New Synthetic Technology for the Construction of Medium- and Large-Ring Ethers. (1987) (1)
- New Synthetic Technology for the Rapid Construction of Novel Heterocycles. Part 2. The Reaction of IBX with Anilides and Related Compounds. (2000) (1)
- Synthesis of the Macrocyclic Core of Sanglifehrin A. (1999) (1)
- Total Synthesis of Brevetoxin B. Part 2. Completion. (1995) (1)
- A New Class of DNA-Cleaving Molecules: pH-Dependent DNA Cleavage by Propargylic and Allenic Sulfones. (1989) (1)
- Asymmetric Reactions in Total Synthesis (2010) (1)
- Total Synthesis of Amphotericin B. Part 3. The Final Stages. (1988) (1)
- Total Synthesis of the CP‐Molecules (CP‐263,114 and CP‐225,917, Phomoidrides B and A). Part 2. Model Studies for the Construction of Key Structural Elements and First‐Generation Strategy. (2002) (1)
- Book Review: Robert Burns Woodward Architect and Artist in the World of Molecules. Edited by Otto T. Benfey and Peter J. T Morris (2003) (1)
- Design, Synthesis, and Biological Evaluation of Carbohydrate-Based Mimetics of cRGDFV. (1997) (1)
- Stereocontrolled Construction of Key Building Blocks for the Total Synthesis of Amphoteronolide B and Amphotericin B. (1987) (1)
- Total Synthesis and Chemical Biology of the Sarcodictyins (2000) (1)
- Design, Synthesis, and Biological Investigation of Thailanstatin A and Spliceostatin D Analogues Containing Tetrahydropyran, Tetrahydrooxazine, and Fluorinated Structural Motifs. (2021) (1)
- Synthesis of Hirsutellone B (2010) (1)
- Cyclic Conjugated Enediynes (II) Related to Calicheamicins and Esperamicins: Calculations, Synthesis, and Properties. (1988) (1)
- ChemInform Abstract: Novel Chemistry of α-Tosyloxy Ketones: Applications to the Solution- and Solid-Phase Synthesis of Privileged Heterocycle and Enediyne Libraries. (2002) (1)
- Stereoselective Total Synthesis of the Presumed Biosynthetic Precursor to Lipoxins A and B: Methyl (7E,9E,11Z,13E,5S,6S,15S)-5,6-Epoxy-15-hydroxyicosa-7,9,11,13-tetraenoate (Ia) and its 5,6-Methano Analogue (Ib). (1987) (1)
- Iodine(V) Reagents in Organic Synthesis. Part 2. Access to Complex Molecular Architectures via Dess—Martin Periodinane Generated o-Imidoquinones. (2002) (1)
- Cover Picture: Maitotoxin: An Inspiration for Synthesis (Isr. J. Chem. 3‐4/2011) (2011) (1)
- Probing the Ring Size of Epothilones: Total Synthesis of [14]-, [15]-, [17]-, and [18]Epothilones A. (1998) (1)
- Total Synthesis of the Originally Proposed and Revised Structures (I) of Palmerolide A. (2007) (1)
- Total Synthesis of the Carbohydrate Fragments of Esperamicin A1. (1992) (1)
- Subject Index, Vol. 25, 1980 (1980) (1)
- Lipoxins and Related Eicosanoids: Biosynthesis, Chemical Synthesis and Biological Properties (1991) (1)
- Titelbild: Total Synthesis and Revised Structure of Biyouyanagin A (Angew. Chem. 25/2007) (2007) (1)
- Conversion of Thionoesters and Thionolactones to Ethers; a General and Efficient Radical Desulfurization. (1995) (1)
- Total Synthesis of Calicheamicin γI 1. Part 3. The Final Stages. (1993) (1)
- New Synthetic Technology for the Rapid Construction of Novel Heterocycles. Part 1. The Reaction of Dess—Martin Periodinane with Anilides and Related Compounds. (2000) (1)
- Cascade Reactions Involving Formal [2 + 2] Thermal Cycloadditions: Total Synthesis of Artochamins F, H, I, and J. (2008) (1)
- SIMPLE STEREOSPECIFIC ROUTES TO 9-EPI-PROSTAGLANDIN F(2ALPHA)(PGF(2BETA)) AND 11-EPI-PROSTAGLANDIN F(2ALPHA) (1975) (1)
- Olefin Metathesis in Cyclic Ether Formation. Direct Conversion of Olefinic Esters to Cyclic Enol Ethers with Tebbe-Type Reagents. (1996) (1)
- Eine schnelle und ergiebige Synthese des Ringgerüsts von Aphidicolin und ähnlichen Naturstoffen (1981) (1)
- Die Stärkung des Bildungswesens (2011) (1)
- ORGANOSELENIUM-INDUCED RING CLOSURES. STEREOSELECTIVE SYNT (1978) (1)
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- Stereocontrolled Total Synthesis of Methyl (12S)-Hydroxy-5Z,8E,10E-heptadecatrienoate (1990) (0)
- NEW SYNTHETIC TECHNOLOGY AND TOTAL SYNTHESIS(天然物化学のニュ-トピックス) (1988) (0)
- Self-total taxol-diterpenoid nanostructures (1995) (0)
- Novel Strategies of Construction of Complex Polycyclic Ether Frameworks. Stereo‐Controlled Synthesis of the FGHIJ Ring System of Brevetoxin A. (1991) (0)
- A Highly Convergent Strategy Towards Rapamycin. Stereoselective Construction of the C8-C18 Fragment (I). (1993) (0)
- A New Method for the Stereoselective Synthesis of α- and β-Glycosylamines Using the Burgess Reagent. (2004) (0)
- Iodine(V) Reagents in Organic Synthesis. Part 1. Synthesis of Polycyclic Heterocycles via Dess—Martin Periodinane Mediated Cascade Cyclization: Generality, Scope, and Mechanism of the Reaction. (2002) (0)
- REACTIONS OF HYDROXYL GROUPS WITH THE TOSYL CHLORIDE-DIMETHYLAMINOPYRIDINE SYSTEM. DIRECT SYNTHESIS OF CHLORIDES FROM HYDROXY COMPOUNDS (1984) (0)
- Synthetic Strategies for the Coupling of the Calicheamicine‐ Oligosaccharide with Aglycones. Synthesis of Dynemicine‐A‐ Calicheamicine Hybrid Compounds. (1991) (0)
- Synthesis of Coleophomone B (2006) (0)
- Total Synthesis of the Tumor-Associated LeX Family of Glycosphingolipids. (1990) (0)
- 1,2‐Benziodoxol‐3(1H)‐one, 1‐Hydroxy, 1‐Oxide (2012) (0)
- Biomimetic Total Synthesis of Bisorbicillinol, Bisorbibutenolide, Trichodimerol, and Designed Analogues of the Bisorbicillinoids. (2000) (0)
- Comprar Molecules That Changed the World | K. C. Nicolaou | 9783527309832 | Wiley (2007) (0)
- Synthesis of Thiostrepton (2006) (0)
- Bridging of Macrocycles to Bicycles. New Synthetic Technology for the Construction of cis- and trans-Fused Oxopolycyclic Systems. (1987) (0)
- Structure of Tubulin Tyrosine Ligase in Complex with Tb116 (2021) (0)
- Polymer-Supported Selenium Reagents for Organic Synthesis. (2010) (0)
- Synthesis and Biological Actions of Optically Active Enediynes Related to Dynemicin A. (1993) (0)
- Synthesis of the Bicyclic Core or CP-225,917 and CP-263,114 by an Intramolecular Diels-Alder Reaction. (1997) (0)
- Thermal Cycloadditions of Dimethyl Acetylenedicarboxylate with Cyclic Enol Ethers. An Entry into Medium Size Oxocyclic Systems. (1987) (0)
- Construction of the “Left Domain” of Haplophytine (I). (2007) (0)
- Total Synthesis of Colombiasin A (I) and Determination of Its Absolute Configuration. (2002) (0)
- Total Syntheses of 2,2′‐epi‐Cytoskyrin A (Ia), Rugulosin (Ib), and the Alleged Structure (II) of Rugulin. (2007) (0)
- Total Synthesis of Floresolide B and Δ6,7‐Z‐Floresolide B. (2006) (0)
- TOTAL SYNTHESIS OF ESTRA-1,3,5(10)-TRIEN-17-ONE (1980) (0)
- Dynemisiinianalogien enantiomers, their preparation and use (1994) (0)
- Total Synthesis of Thiostrepton. Part 1. Construction of the Dehydropiperidine/Thiazoline-Containing Macrocycle. (2004) (0)
- Total Synthesis of Eleutherobin (IX) and Eleuthosides A (X) and B (XI). (1999) (0)
- Synthesis of Marinomycin A (2007) (0)
- Synthesis of the ABC Ring System of Brevetoxin B. (1989) (0)
- Synthesis of a- and -Diversonolic Esters (2009) (0)
- Cascade Reactions in Total Synthesis (2007) (0)
- Total Synthesis and Biological Evaluation of (-)-Apicularen A and Analogues Thereof (2004) (0)
- 5,6-METHANOLEUKOTRIENE A4. A STABLE AND BIOLOGICALLY ACTIVE ANALOG OF LEUKOTRIENE A4 (1982) (0)
- Preparation of sarcodictyin and eleutherobin and analogs useful for stabilizing microtubules (1999) (0)
- Professor K. C. Nicolaou (2002) (0)
- Cover Picture: Total Synthesis and Revised Structure of Biyouyanagin A (Angew. Chem. Int. Ed. 25/2007) (2007) (0)
- ORGANOSELENIUM-INDUCED RING CLOSURES: CYCLIZATION OF DIENES WITH “PHSEOH” TO FORM CYCLIC ETHERS (1979) (0)
- Patent Number : 5 , 274 , 137 45 Date of Patent : 54 INTERMEDIATES FOR PREPARATION OF TAXOLS 76 Inventors : (2017) (0)
- Chemistry, Biology, and Medicine of the Glycopeptide Antibiotics (1999) (0)
- Synthesis of Highly Substituted N‐Hydroxyindoles Through 1,5‐Addition of Carbon Nucleophiles to in situ Generated Unsaturated Nitrones. (2006) (0)
- Erratum: Studies toward diazonamide A: Development of a hetero-pinacol macrocyclization cascade for the construction of the bis-macrocyclic framework of the originally proposed structure (Journal of the American Chemical Society (2004) 126 (10174-10182)) (2004) (0)
- Reactions of Glycosyl Fluorides. Synthesis of C-Glycosides. Synthesis of O-, S- and N-Glycosides. (1985) (0)
- Total Synthesis of Taxol. Part 1. Retrosynthesis, Degradation, and Reconstitution. (1995) (0)
- PERICYCLIC REACTIONS IN ORGANIC SYNTHESIS AND BIOSYNTHESIS: SYNTHETIC ADVENTURES WITH ENDIANDRIC ACIDS A-G (1985) (0)
- Total Synthesis of Brevetoxin A. Part 3. Construction of GHIJ and BCDE Ring Systems. (1999) (0)
- Cover Picture: The Continuing Saga of the Marine Polyether Biotoxins (Angew. Chem. Int. Ed. 38/2008) (2008) (0)
- Total Synthesis of Marinomycins A—C. (2007) (0)
- Activation of 6-endo- over S-exo Epoxide Openings. Ring-Selective Formation of Tetrahydropyran Systems and Stereocontrolled Synthesis of the ABC Ring Framework of Brevetoxin B. (1986) (0)
- Stereocontrolled Total Synthesis of (5Z,8Z,11Z,13E)(15S)-15-Hydroxyeicosa-5,8,11,13-tetraenoic Acid (15S-HETE) and Analogues. (1986) (0)
- Frontispiece: Efficient Synthesis of Dimeric Oxazoles, Piperidines and Tetrahydroisoquinolines from N -Substituted 2-Oxazolones (2016) (0)
- Cancer Therapy : Preclinical Arylsulfonamide KCN 1 Inhibits In Vivo Glioma Growth and Interfereswith HIF Signaling byDisrupting HIF-1 a Interaction with Cofactors p 300 / CBP (2012) (0)
- SYNTHESIS OF SULFUR-CONTAINING PROSTACYCLIN PGI1 ANALOGS, 6,9-EPITHIO-PGI1, ITS S-OXIDE STEREOISOMERS, AND ITS SS-DIOXIDE (1978) (0)
- Enediyne Compounds with Acid‐, Base‐ and Photo‐Sensitive Trigger Groups. Chemical Simulation of the Dynemicin A Reaction Cascade. (1991) (0)
- Masthead: ChemistryOpen 1/2015 (2015) (0)
- Copper(I)-Promoted Stille Cross-Coupling of α-Stannyl Enol Ethers with Enol Triflates: Construction of Complex Polyether Frameworks. (1996) (0)
- Total Synthesis of Natural Products: The „Chiron”︁ Approach. Von S. Hanessian. Pergamon Press, Oxford 1983. XVII, 291 S., Paperback 11.25. – ISBN 0‐08‐030715‐9 (1985) (0)
- Total Synthesis of Calicheamicin γI 1. Part 2. Development of an Enantioselective Route to (-)-Calicheamicinone. (1993) (0)
- Total Synthesis of Oxazole‐ and Cyclopropane‐Containing Epothilone A Analogues by the Olefin Metathesis Approach. (1998) (0)
- Stereospecific Synthesis of 1,1-Dialkylglycosides. (1986) (0)
- SIR DEREK BARTON'S 80TH BIRTHDAY (2000) (0)
- N-Phenylselenophthalimide (NPSP), a Valuable Selenenylating Agent. (1986) (0)
- The Continuing Saga of the Marine Polyether Biotoxins (2008) (0)
- Cover Picture: Structural Revision and Total Synthesis of Azaspiracid‐1, Part 1: Intelligence Gathering and Tentative Proposal (Angew. Chem. Int. Ed. 33/2004) (2004) (0)
- United States Patent ( 19 ) Nicolaou et al . ( 54 ) PHARMACEUTICALLY ACTIVE 6 , 9-THIAPROSTACYCLIN ANALOGS AND DERVATIVES THEREOF (2017) (0)
- Synthesis of Complex Carbohydrates: Everninomicin (2005) (0)
- Total Synthesis of 20-Hydroxy- and 20-Carboxy-leukotrienes B4. (1986) (0)
- A Photolytic Access to Oxepane Systems. (1989) (0)
- SYNTHESIS OF 7,13-BRIDGED ARACHIDONIC ACID ANALOGS (1984) (0)
- Nicolaou creating others like them in the laboratory replicating the molecules of living nature and Organic synthesis : the art and science of (2014) (0)
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- A RAPID AND PRODUCTIVE SYNTHESIS OF THE RING FRAMEWORK OF APHIDICOLIN AND SIMILAR NATURAL COMPOUNDS (1981) (0)
- 1,2‐Seleno Migrations in Carbohydrate Chemistry: Solution and Solid‐Phase Synthesis of 2‐Deoxy Glycosides, Orthoesters, and Allyl Orthoesters. (2000) (0)
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- Titelbild: Angew. Chem. 10/2002 (2002) (0)
- Synthetic Studies on Maduropeptin Chromophore. Part 1. Construction of the Aryl Ether and Attempted Synthesis of the (7.3.0) Bicyclic System. (1997) (0)
- Total Synthesis of Sarcodictyins A (Xa) and B (Xb). (1999) (0)
- Formal synthesis of (±)-platensmiycin (2007) (0)
- Synthesis of Dynemicin A Models. (1991) (0)
- The CP Molecule Labyrinth: A Paradigm of How Endeavors in Total Synthesis Lead to Discoveries and Inventions in Organic Synthesis (2002) (0)
- The Total Synthesis of Brevetoxin B: A Twelve-Year Odyssey in Organic Synthesis (1996) (0)
- Synthesis of Medium-Sized Ring Ethers from Thionolactones. Applications to Polyether Synthesis. (1990) (0)
- Synthesis of Abyssomicin C (2006) (0)
- TOTAL SYNTHESIS OF CARBOPROSTACYCLIN, A STABLE AND BIOLOGICALLY ACTIVE ANALOG OF PROSTACYCLIN (PGI2) (1979) (0)
- Buchbesprechung: Robert Burns Woodward Architect and Artist in the World of Molecules. Herausgegeben von Otto T. Benfey und Peter J. T. Morris (2003) (0)
- Cover Picture: Angew. Chem. Int. Ed. 15/2002 (2002) (0)
- Samarium Diiodide Mediated Reactions in Total Synthesis (2009) (0)
- REACTION OF PHENYLSELENENYL CHLORIDE WITH ENOL ETHERS AND 1,2-ETHANEDIYL ACETALS. SYNTHESIS OF α-PHENYLSELENO ALDEHYDES AND α-PHENYLSELENO ACETALS (1980) (0)
- Conference Report : Chemical Synthesis and Drug Discovery : ICS Symposium Honoring (2016) (0)
- Total Synthesis of Amphoteronolide B. (1987) (0)
- Modulation of the Reactivity Profile of IBX by Ligand Complexation: Ambient Temperature Dehydrogenation of Aldehydes and Ketones to α,β-Unsaturated Carbonyl Compounds. (2002) (0)
- Metathesis reactions in the synthesis of complex molecules (2007) (0)
- Total Synthesis of Taxol. Part 3. Formation of Taxol′s ABC Ring Skeleton (1995) (0)
- STEREOCONTROLLED SYNTHESIS OF 1,3,5...(2N + 1) POLYOLS (1983) (0)
- Analogs of epothilone cyclobutyl and cyclopropyl. (2002) (0)
- Stereocontrolled Total Synthesis of Apicularen A (I) and Its Δ17,18 Z Isomer. (2003) (0)
- TOTAL SYNTHESIS OF THE POTENT MUTAGEN (S)-3-(DODECA-1,3,5,7,9-PENTAENYLOXY)PROPANE-1,2-DIOL (1984) (0)
- Solid‐ and Solution‐Phase Synthesis of Vancomycin and Vancomycin Analogues with Activity Against Vancomycin‐Resistant Bacteria. (2002) (0)
- New Synthetic Technology for the Construction of N‐Containing Quinones and Derivatives Thereof: Total Synthesis of Epoxyquinomycin B. (2001) (0)
- Palladium‐Catalyzed Functionalization of Lactones via Their Cyclic Ketene Acetal Phosphates. Efficient New Synthetic Technology for the Construction of Medium and Large Cyclic Ethers. (1997) (0)
- Recent Developments in the Chemistry, Biology and Medicine of the Epothilones (2001) (0)
- Total Synthesis of the Proposed Azaspiracid‐1 Structure (I). Part 1. Construction of the Enantiomerically Pure C1—C20, C21—C27, and C28—C40 Fragments. (2003) (0)
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- Synthesis of the Brevetoxin B IJK Ring System. (1989) (0)
- DIASTEREOMERE MONOCYCLISCHE DIALLENE, SYNTH. VON CYCLODODECA-3,4,9,10-TETRAEN-1,7-DION (1970) (0)
- Synthesis of the C′D′E′F′ Domain of Maitotoxin. (2011) (0)
- Structure of Tubulin Tyrosine Ligase in Complex with Tb111 (2021) (0)
- Synthetic Studies on Maduropeptin Chromophore. Part 2. Synthesis of the Madurosamine Aryl Amide and the C1′—C9′ Fragments. (1997) (0)
- The True Structures of the Vannusals. Part 2. Total Synthesis and Revised Structure of Vannusal B. (2009) (0)
- Erratum: Chemistry and biology of diazonamide A: First total synthesis and confirmation of the true structure (Journal of the American Chemical Society (2004) 126 (12888-12896)) (2004) (0)
- Correction to The Art and Science of Organic and Natural Products Synthesis (1999) (0)
- Synthesis of Complex Carbohydrates: Everninomicin 13,384-1 (2004) (0)
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- Molecular Design and Chemical Synthesis of Potent Enediynes. Part 1. Dynemicin Model Systems Equipped with N-Tethered Triggering Devices. (1993) (0)
- Chemical Synthesis and Biological Evaluation of Novel Epothilone B and trans-12,13-Cyclopropyl Epothilone B Analogues. (2002) (0)
- The Synthesis of Bisorbicillinoids: An Amazing Self‐Assembly of Simple Compounds into Highly Complex Natural Products (2000) (0)
- Chemistry and Biology of Diazonamide A: Second Total Synthesis and Biological Investigations [J. Am. Chem. Soc. 2004, 126, 12897−12906]. (2004) (0)
- Total Synthesis of Eleutherobin (I) (2010) (0)
- Total Synthesis of Brevetoxin B. Part 3. Final Strategy and Completion. (1996) (0)
- A new method for the stereoselective synthesis of alpha- and beta-glycosylamines using the Burgess reagent. (2004) (0)
- Synthesis of Halipeptins A and D (2006) (0)
- Golfomycin A, a Novel Designed Molecule with DNA-Cleaving Properties and Antitumor Activity. (1990) (0)
- Modulation of the reactivity profile of IBX by ligand complexation: ambient temperature dehydrogenation of aldehydes and ketones to alpha,beta-unsaturated carbonyl compounds. (2002) (0)
- Chemistry of Amphotericin B. Degradation Studies and Preparation of Amphoteronolide B. (1988) (0)
- New Synthetic Strategies for the Construction of Medium-Size Cyclic Ethers. Stereocontrolled Synthesis of the BCD Ring Framework of Brevetoxin A. (1990) (0)
- Total synthesis of floresolide B and Delta(6,7)-Z-floresolide B. (2006) (0)
- Synthese des Anthrachinongerüsts von Dynemicin A (1994) (0)
- Ethanoarachidonic Acids. A New Class of Arachidonic Acid Cascade Modulators. Part 1. Monoethano Compounds. Part 2. Polyethano Compounds. (1984) (0)
- Cover Picture: Total Synthesis and Absolute Configuration of the Bisanthraquinone Antibiotic BE-43472B (Angew. Chem. Int. Ed. 19/2009) (2009) (0)
- Stereoselective Construction of the C18-C32 Fragment of Swinholide A. (1994) (0)
- Stereocontrolled Total Synthesis of (5Z,8Z,10E,12R,14Z)-12-Hydroxy-5,8,10,14-icosatetraenoic Acid ((12R)-HETE). (1990) (0)
- Synthesis of (+)-Rugulosin (2006) (0)
- Novel Chemistry of Dithiatopazine. (1988) (0)
- A New Method for the Synthesis of Nonsymmetrical Sulfamides Using Burgess‐Type Reagents. (2003) (0)
- Synthesis of the CDEFDomain of Maitotoxin (2012) (0)
- Studies Toward the Synthesis of Azadirachtin. Part 1. Total Synthesis of a Fully Functionalized ABC Ring Framework and Coupling with a Norbornene Domain (2005) (0)
- Efficient Synthesis of Dimeric Oxazoles, Piperidines and Tetrahydroisoquinolines from N‐Substituted 2‐Oxazolones. (2016) (0)
- creating others like them in the laboratory replicating the molecules of living nature and Organic synthesis: the art and science of (2014) (0)
- Total Synthesis of Brevetoxin A. Part 2. Second Generation Strategy and Construction of EFGH Model System. (1999) (0)
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- Optimization and Mechanistic Studies of Psammaplin A Type Antibacterial Agents Active Against Methicillin‐Resistant Staphylococcus aureus (MRSA). (2002) (0)
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- Total Synthesis of Amphoteronolide B and Amphotericin B. Part 2. Total Synthesis of Amphoteronolide B. (1988) (0)
- Studies Towards the Synthesis of Esperamicinone (XVI). (1995) (0)
- Expeditious Routes to Evernitrose and Vancosamine Derivatives and Synthesis of a Model Vancomycin Aryl Glycoside. (1998) (0)
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- Stereoselective Construction of the C21-C42 Fragment (I) of Rapamycin. (1993) (0)
- Synthetic Studies on the Dioxepane Region of Brevetoxin B. New Synthetic Technology for the Construction of Oxepanes and Synthesis of a Model for the CDEF Ring Skeleton of Brevetoxin B. (1989) (0)
- New Synthetic Technology for the Construction of N‐Hydroxyindoles and Synthesis of Nocathiacin I Model Systems. (2007) (0)
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- A Convergent Approach to Swinholide A. Stereoselective Construction of the C3‐C17 Fragment of Swinholide A. (1994) (0)
- Total Synthesis of the Originally Proposed (I) and Revised Structures (II) of Palmerolide A and Isomers Thereof. (2008) (0)
- Adamantaplatensimycin (II): A Bioactive Analogue of Platensimycin (I). (2007) (0)
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- Total Synthesis of 26‐Hydroxy‐epothilone B and Related Analogues via a Macrolactonization Based Strategy. (1998) (0)
- 6,9-Thiaprostacyclin. A stable and biologically potent analogue of proracyclin (PGI2) (1978) (0)
- Combinatorial Chemistry in Perspectives (2004) (0)
- Total Synthesis of Zaragozic Acid A/Squalestatin S1. (1995) (0)
- Total Synthesis of Everninomicin 13,384-1. Part 3. Synthesis of the DE Fragment and Completion of the Total Synthesis. (2000) (0)
- Total Synthesis of Halipeptins A (Ia) and D (Ib) and Analogues. (2005) (0)
- Synthesis of (-)-Platencin (2008) (0)
- Studies Toward Diazonamide A: Development of a Hetero‐Pinacol Macrocyclization Cascade for the Construction of the Bis‐Macrocyclic Framework of the Originally Proposed Structure. (2004) (0)
- Titelbild: Angew. Chem. 15/2002 (2002) (0)
- Synthesis of C‐2 Taxol Analogues. (1995) (0)
- soluble onium salt of taxo-diterpenoid. (1995) (0)
- MONOCYCLISCHE ALLENE, DIE SYNTH. VON 3,8,9-CYCLOUNDECATRIEN-1,6-DION UND 12-OXABICYCLO(7,2,1)DODECA-5,6,9,11-TETRAEN-3-ON, EINEM FURANOPHAN MIT EINER ALLENGRUPPE (1973) (0)
- DIASTEREOMERE MONOCYCLISCHE DIALLENE, DIE STEREOCHEMIE DER BLDG. VON RACEMISCHEM UND MESO-3,4,9,10-CYCLODECATETRAEN-1,7-DION (1972) (0)
- Synthesis of 16-Desmethylepothilone B: Improved Methodology for the Rapid, Highly Selective and Convergent Construction of Epothilone B and Analogues. (1999) (0)
- Total Synthesis of Hybocarpone (I). (2001) (0)
- Stereocontrolled Second Generation Syntheses of the ABC and FG Ring Systems of Brevetoxin B. (1990) (0)
- Synthesis of Biologically Active Taxoids (2008) (0)
- An Approach to Epothilones Based on Olefin Metathesis. (1997) (0)
- Synthesis of Antibiotic GE2270A (2007) (0)
- 2 . Current State of Affairs in the Drug Discovery and Development Process (2014) (0)
- Cover Picture: Total Synthesis and Structural Revision of Viridicatumtoxin B (Angew. Chem. Int. Ed. 33/2013) (2013) (0)
- Zaragozic Acid A/Squalestatin S1(I): Synthetic and Retrosynthetic Studies. (1995) (0)
- Berichtigung: Die Bedeutung der organischen Synthese bei der Entstehung und Entwicklung von Antikörper‐Wirkstoff‐Konjugaten als gezielte Krebstherapien (2021) (0)
- A Suzuki Coupling—Macrolactamization Approach to the AB‐COD Bicyclic System of Vancomycin. (1998) (0)
- Studies Toward the Synthesis of Azadirachtin. Part 2. Construction of Fully Functionalized ABCD Ring Frameworks and Unusual Intramolecular Reactions Induced by Close-Proximity Effects. (2005) (0)
- Synthesis of Novel Taxoids. (1994) (0)
- Tandem Reactions, Cascade Sequences, and Biomimetic Strategies in Total Synthesis (2003) (0)
- Total Synthesis of Natural and Designed Molecules of Biological and Medical Importance (2013) (0)
- Synthesis of Artochamins H, I, and J (2008) (0)
- Synthesis of Vannusal B (2010) (0)
- Total Synthesis of 26-Hydroxyepothilone B and Related Analogues. (1998) (0)
- Synthesis of Sporolide B (2009) (0)
- Synthesis of (+)-Haplophytine (2010) (0)
- Total Synthesis of the Novel Immunosuppressant Sanglifehrin A (I). (2000) (0)
- Total Synthesis and Biological Evaluation of Cortistatins A (I) and J (II) and Analogues Thereof. (2010) (0)
- Synthesis of DNA‐Binding Oligosaccharides (1997) (0)
- The Oxide Anion Accelerated Retro-Diels-Alder Reaction (1997) (0)
- AN INTRAMOLECULAR DIELS-ALDER STRATEGY TO FORSKOLIN (1985) (0)
- Total Synthesis of Natural Products and the Synergy with Synthetic Methodology (2012) (0)
- Amphoteronolide B Methyl Ester (I). Novel Oxidative Deglycosidation of Amphotericin B. (1987) (0)
- Inspirations, Discoveries, and Future Perspectives in Total Synthesis (2009) (0)
- Studies toward Diazonamide A: Development of a Hetero-Pinacol Macrocyclization Cascade for the Construction of the Bis-Macrocyclic Framework of the Originally Proposed Structure [J. Am. Chem. Soc. 2004, 126, 10174−10182]. (2004) (0)
- Catalytic Asymmetric Dichlorination of Allylic Alcohols (2011) (0)
- Enhancement of the sensitivity of hamster cheek pouch arterioles to beta-adrenergic stimulus during pregnancy (1982) (0)
- SYNTHESIS AND BIOLOGICAL PROPERTIES OF PROSTAGLANDIN ENDOPEROXIDES, THROMBOXANES, AND PROSTACYCLINS (1978) (0)
- United States Patent ( 19 ) Nicolaou et al . 54 PYRIDOZA PROSTACYCLIN ANALOGUES (2017) (0)
- Total Synthesis of Brevetoxin B. Part 2. Second Generation Strategies and Construction of the Dioxepane Region (DEFG). (1996) (0)
- Total Synthesis and Structural Elucidation of Azaspiracid‐1. Construction of Key Building Blocks for Originally Proposed Structure. (2006) (0)
- Synthesis of Aspidophytine (2009) (0)
- REVERSAL OF THE PHENYLSELENO- AND PHENYLSULFENO-CYCLIZATIONS. SYNTHESIS OF OLEFINS FROM PHENYLSELENO- AND PHENYLSULFENO-LACTONES, PHENYLSELENOETHERS, AND α-HYDROXYSELENIDES (1979) (0)
- Total Synthesis of Taxol. Part 2. Construction of A and C Ring Intermediates and Initial Attempts to Construct the ABC Ring System (1995) (0)
- Titelbild: Total Synthesis and Absolute Configuration of the Bisanthraquinone Antibiotic BE‐43472B (Angew. Chem. 19/2009) (2009) (0)
- Total Synthesis of the CP‐Molecules (CP‐263,114 and CP‐225,917, Phomoidrides B and A). Part 1. Racemic and Asymmetric Synthesis of Bicyclo[4.3.1] Key Building Blocks. (2002) (0)
- New Technology for the Synthesis of Vancomycin-Type Biaryl Ring Systems. (1997) (0)
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