Margaret Brimble
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New Zealand chemist
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Chemistry
Why Is Margaret Brimble Influential?
(Suggest an Edit or Addition)According to Wikipedia, Dame Margaret Anne Brimble is a New Zealand chemist. Her research has included investigations of shellfish toxins and means to treat brain injuries. Early life, family, and education Brimble was born in Auckland on 20 August 1961, the daughter of Mary Anne MacMillan and Herbert MacMillan, and was encouraged by her grandmother to value education. She attended Diocesan School for Girls, Auckland from 1972 to 1978, and was dux in her final year.
Margaret Brimble's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- C-H functionalization in the synthesis of amino acids and peptides. (2014) (367)
- Molecules derived from the extremes of life. (2009) (138)
- Pyranonaphthoquinone antibiotics--isolation, structure and biological activity. (1999) (134)
- Isolation, biological activity and synthesis of benzannulated spiroketal natural products. (2010) (118)
- Natural product derived privileged scaffolds in drug discovery. (2019) (104)
- Structural Basis for Receptor Activity-Modifying Protein-Dependent Selective Peptide Recognition by a G Protein-Coupled Receptor (2015) (100)
- Effect of fungal metabolite peramine and analogs on feeding and development of argentine stem weevil (Listronotus bonariensis) (1990) (89)
- Structure-mechanical property correlations of hydrogel forming β-sheet peptides. (2016) (84)
- Synthesis of bis-spiroacetal ring systems (1999) (80)
- An Insight into FDA Approved Antibody-Drug Conjugates for Cancer Therapy (2021) (75)
- Synthesis of fish antifreeze neoglycopeptides using microwave-assisted "click chemistry". (2009) (71)
- C–H activation (2021) (71)
- Synthetic Strategies Towards Pyranonaphthoquinone Antibiotics (2000) (68)
- Structure, Function, Pharmacology, and Therapeutic Potential of the G Protein, Gα/q,11 (2015) (63)
- A one-pot approach to neoglycopeptides using orthogonal native chemical ligation and click chemistry. (2009) (63)
- Pyranonaphthoquinones--isolation, biological activity and synthesis. (2008) (63)
- Identification of Conjugated Triene Oxidation Products of .alpha.-Farnesene in Apple Skin (1995) (61)
- Methyllycaconitine analogues have mixed antagonist effects at nicotinic acetylcholine receptors. (2005) (60)
- An efficient formal synthesis of the human telomerase inhibitor (+/-)-gamma-rubromycin. (2009) (60)
- Synthesis and antifreeze activity of fish antifreeze glycoproteins and their analogues (2010) (57)
- Spiroimine shellfish poisoning (SSP) and the spirolide family of shellfish toxins: isolation, structure, biological activity and synthesis. (2010) (54)
- The Kulinkovich hydroxycyclopropanation reaction in natural product synthesis. (2012) (54)
- Allylic amination by the Lewis acid-mediated ene reactions of diethyl azodicarboxylate with alkenes (1993) (54)
- Protecting-group-free one-pot synthesis of glycoconjugates directly from reducing sugars. (2014) (54)
- Direct peptide lipidation through thiol-ene coupling enables rapid synthesis and evaluation of self-adjuvanting vaccine candidates. (2013) (52)
- Synthesis of isotopically labelled thiol volatiles and cysteine conjugates for quantification of Sauvignon Blanc wine (2007) (48)
- Grafting from Poly(3,4-ethylenedioxythiophene): A Simple Route to Versatile Electrically Addressable Surfaces (2013) (47)
- A review of neuroprotective agents. (2004) (47)
- Synthesis of the bis-spiroacetal moiety of spirolides B and D. (2005) (46)
- Supplementation of Blackcurrant Anthocyanins Increased Cyclic Glycine-Proline in the Cerebrospinal Fluid of Parkinson Patients: Potential Treatment to Improve Insulin-Like Growth Factor-1 Function (2018) (44)
- Synthesis of natural products containing spiroketals via intramolecular hydrogen abstraction. (2010) (44)
- Chemistry of Bis-spiroacetal SystemsNatural Products: Synthesis and Stereochemistry (2003) (44)
- A review of the synthesis of α-carbolines. (2015) (43)
- An improved procedure for the preparation of aminomethyl polystyrene resin and its use in solid phase (peptide) synthesis (2011) (43)
- Characterizing the mode of action of extracellular Connexin43 channel blocking mimetic peptides in an in vitro ischemia injury model. (2017) (42)
- Enhancing the Oral Bioavailability of Peptide Drugs by using ChemicalModification and Other Approaches (2014) (41)
- A phase I vaccination study with dendritic cells loaded with NY-ESO-1 and α-galactosylceramide: induction of polyfunctional T cells in high-risk melanoma patients (2018) (41)
- Synthesis of cyclic proline-containing peptides via ring-closing metathesis. (2003) (40)
- Plant antimicrobial peptides snakin-1 and snakin-2: chemical synthesis and insights into the disulfide connectivity. (2014) (40)
- Molecular Signature for Receptor Engagement in the Metabolic Peptide Hormone Amylin. (2018) (40)
- Natural products targeting telomere maintenance (2011) (40)
- Synthesis of the bis-spiroacetal moiety of the shellfish toxins spirolides B and D using an iterative oxidative radical cyclization strategy. (2006) (39)
- Gold catalysis: synthesis of spiro, bridged, and fused ketal natural products. (2017) (39)
- NKT cell-dependent glycolipid–peptide vaccines with potent anti-tumour activity† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c4sc03599b Click here for additional data file. Click here for additional data file. (2015) (39)
- Receptor Activity-modifying Proteins 2 and 3 Generate Adrenomedullin Receptor Subtypes with Distinct Molecular Properties* (2016) (38)
- Very Short and Stable Lactoferricin-Derived Antimicrobial Peptides: Design Principles and Potential Uses. (2019) (38)
- Isolation, biological activity, biosynthesis and synthetic studies towards the rubromycin family of natural products. (2015) (38)
- A convergent synthesis of the (4.4]-spiroacetal-γ-lactones cephalosporolides E and F (2011) (37)
- Addition of Silyloxydienes to 2-Substituted 1,4-Benzoquinones and 1,4-Naphthoquinones (1997) (37)
- Heteroatom-directed reverse Wacker oxidations. Synthesis of the reported structure of (-)-herbaric acid. (2010) (36)
- Gaq proteins: molecular pharmacology and therapeutic potential (2017) (36)
- Radiation Damage and Racemic Protein Crystallography Reveal the Unique Structure of the GASA/Snakin Protein Superfamily. (2016) (36)
- Identification of key residues involved in adrenomedullin binding to the AM1 receptor (2013) (35)
- Molecular Weight and Charge Density Effects of Guanidinylated Biodegradable Polycarbonates on Antimicrobial Activity and Selectivity. (2017) (35)
- The influence of microwave irradiation on lipase-catalyzed kinetic resolution of racemic secondary alcohols (2007) (35)
- Investigations into the cellular actions of the shellfish toxin gymnodimine and analogues. (2005) (35)
- The role for IGF-1-derived small neuropeptides as a therapeutic target for neurological disorders (2015) (34)
- Electrochemically-controlled grafting of hydrophilic brushes from conducting polymer substrates (2016) (34)
- Total synthesis of the cyclic depsipeptide YM-280193, a platelet aggregation inhibitor. (2015) (33)
- Use of (S)‐5‐(2‐Methylpyrrolidin‐2‐yl)‐1H‐tetrazole as a Novel and Enantioselective Organocatalyst for the Aldol Reaction (2008) (33)
- Use of a sonogashira-acetylide coupling strategy for the synthesis of the aromatic spiroketal skeleton of gamma-rubromycin. (2003) (33)
- Convergent chemoenzymatic synthesis of a library of glycosylated analogues of pramlintide: structure-activity relationships for amylin receptor agonism. (2014) (32)
- Structure–activity relationships of the N-terminus of calcitonin gene-related peptide: key roles of alanine-5 and threonine-6 in receptor activation (2013) (32)
- Peptide Lipidation – A Synthetic Strategy to Afford Peptide Based Therapeutics (2017) (32)
- Synthesis of the griseusin B framework via a one-pot annulation-methylation-double deprotection-spirocyclization sequence. (2013) (32)
- Regulation and Quality Control of Adiponectin Assembly by Endoplasmic Reticulum Chaperone ERp44* (2015) (32)
- Enduracididine, a rare amino acid component of peptide antibiotics: Natural products and synthesis (2016) (32)
- Pyranonaphthoquinone derivatives of eleutherin, ventiloquinone L, thysanone and nanaomycin A possessing a diverse topoisomerase II inhibition and cytotoxicity spectrum. (2009) (31)
- Synthesis of the insect feeding deterrent peramine via Michael addition of a pyrrole anion to a nitroalkene (1990) (31)
- Distinct Patterns of Internalization of Different Calcitonin Gene-Related Peptide Receptors. (2020) (30)
- The first enantioselective total synthesis of the anti-Helicobacter pylori agent (+)-spirolaxine methyl ether. (2005) (30)
- Fluorescent probes for bioimaging of potential biomarkers in Parkinson's disease. (2020) (30)
- Pyranonaphthoquinones - isolation, biology and synthesis: an update. (2017) (30)
- Synthesis of benzannulated spiroacetals using chiral gold–phosphine complexes and chiral anions (2013) (30)
- Access to 2-alkyl chromanones via a conjugate addition approach (2012) (30)
- The Synthesis of Phosphopeptides Using Microwave-assisted Solid Phase Peptide Synthesis (2008) (30)
- Solid-Phase Thiol-Ene Lipidation of Peptides for the Synthesis of a Potent CGRP Receptor Antagonist. (2018) (29)
- Synthesis of the cis-3a,8b-dihydrofuro[3,2-b]benzofuran-2(3H)-one ring system via a furofuran annulation to activated benzoquinones (1989) (29)
- NNZ-2566: A Gly–Pro–Glu analogue with neuroprotective efficacy in a rat model of acute focal stroke (2009) (29)
- Synthesis and activity studies of analogues of the rat selective toxicant norbormide. (2007) (29)
- Synthesis of aromatic spiroacetals related to γ-rubromycin based on a 3H-spiro[1-benzofuran-2,2′-chromane] skeleton (2007) (29)
- Toward an asymmetric synthesis of the dimeric pyranonaphthoquinone antibiotic crisamicin A. (2014) (28)
- Synthesis of macrocyclic shellfish toxins containing spiroimine moieties. (2007) (28)
- Synthesis of tricyclic analogues of methyllycaconitine using ring closing metathesis to append a B ring to an AE azabicyclic fragment. (2004) (28)
- Replacement of the CysA7-CysB7 disulfide bond with a 1,2,3-triazole linker causes unfolding in insulin glargine. (2015) (28)
- Synthesis and neuroprotective activity of analogues of glycyl-L-prolyl-L-glutamic acid (GPE) modified at the alpha-carboxylic acid. (2005) (28)
- Amylin Analog Pramlintide Induces Migraine‐like Attacks in Patients (2021) (28)
- Recent developments in transition metal-catalysed spiroketalisation. (2014) (28)
- Synthesis of the peptaibol framework of the anticancer agent culicinin D: stereochemical assignment of the AHMOD moiety. (2012) (27)
- A double alkylation - ring closing metathesis approach to spiroimines (2004) (27)
- Synthesis of multivalent neoglyconjugates of MUC1 by the conjugation of carbohydrate-centered, triazole-linked glycoclusters to MUC1 peptides using click chemistry. (2012) (27)
- Synthetic studies towards the pectenotoxins: a review. (2006) (27)
- Norborn-2-en-7-ones as physiologically-triggered carbon monoxide-releasing prodrugs† †Electronic supplementary information (ESI) available: Experimental details for the synthesis of compounds, supporting figures and schemes, and NMR spectra. See DOI: 10.1039/c7sc01647f Click here for additional data (2017) (27)
- Synthesis of proline-modified analogues of the neuroprotective agent glycyl-l-prolyl-glutamic acid (GPE) (2005) (27)
- A novel approach to the CDE ring system of pectenotoxin-4 triggered by VO(acac)(2)-induced epoxy-acetalization. (2009) (27)
- A facile synthesis of fused aromatic spiroacetals based on the 3,4,3′,4′-tetrahydro-2,2′-spirobis(2H-1-benzopyran) skeleton (2006) (27)
- Lipidation of Cysteine or Cysteine-Containing Peptides Using the Thiol-Ene Reaction (CLipPA) (2016) (27)
- Synthesis of MUC1 Neoglycopeptides using efficient microwave-enhanced chaotrope-assisted click chemistry. (2011) (27)
- Toward the total chemical synthesis of the cancer protein NY-ESO-1. (2010) (27)
- Synthesis of the C10-C22 bis-spiroacetal domain of spirolides B and D via iterative oxidative radical cyclization. (2002) (27)
- Synthesis of the ABC fragment of the pectenotoxins. (2005) (26)
- Synthesis of fluorescein-labelled O-mannosylated peptides as components for synthetic vaccines: comparison of two synthetic strategies. (2008) (26)
- Enzymatic and non-enzymatic crosslinks found in collagen and elastin and their chemical synthesis (2020) (26)
- Synthesis of pyrrolo[3,2-b]benzofurans and pyrrolo[3,2-b]naphthofurans via addition of a silyloxypyrrole to activated quinones (2004) (26)
- Growth Habit Modification of Ice Crystals Using Antifreeze Glycoprotein (AFGP) Analogues (2010) (26)
- Total chemical synthesis of glycocin F and analogues: S-glycosylation confers improved antimicrobial activity† †Electronic supplementary information (ESI) available: Experimental details for the synthesis of all peptides, analytical LC and HR-MS, and circular dichroism data. See DOI: 10.1039/c7sc043 (2018) (26)
- Synthesis and evaluation of disulfide bond mimetics of amylin-(1-8) as agents to treat osteoporosis. (2012) (26)
- Glucose as an agent of post-translational modification in diabetes--New cardiac epigenetic insights. (2015) (26)
- Synthesis of 5-epi-7-deoxykalafungin and 5-epi-7-O-methylkalafungin (1990) (25)
- Synthesis of the monomeric unit of γ-actinorhodin (1997) (25)
- A short synthesis of deoxyfrenolicin (1994) (25)
- Total synthesis of the initially reported and revised structures of the neuroprotective agent palmyrolide A. (2012) (25)
- Synthesis of 6,6-bisbenzannulated spiroketals related to the rubromycins using a double intramolecular hetero-Michael addition (DIHMA) (2009) (25)
- A flexible asymmetric synthesis of the tetracyclic core of berkelic acid using a Horner-Wadsworth-Emmons/oxa-Michael cascade. (2010) (25)
- An approach to an enantioselective synthesis of crisamicin A via a novel double Hauser–Kraus annulation strategy (2008) (24)
- Synthesis of the antimicrobial S-linked glycopeptide, glycocin F. (2015) (24)
- A Convergent Synthesis of the 2-Formylpyrrole Spiroketal Natural Product Acortatarin A (2012) (24)
- Total synthesis of the macrocyclic N-Methyl enamides palmyrolide A and 2S-sanctolide A. (2014) (24)
- Novel preparation of chiral α-amino acids using the Mitsunobu-Tsunoda reaction. (2013) (24)
- Structure and dynamics of human Nedd4-1 WW3 in complex with the αENaC PY motif. (2013) (24)
- How do Antarctic notothenioid fishes cope with internal ice? A novel function for antifreeze glycoproteins (2010) (24)
- Synthesis of a 2-deoxyglucosyl analogue of medermycin (2001) (23)
- A new precursor for conducting polymer-based brush interfaces with electroactivity in aqueous solution (2013) (23)
- 2-Formylpyrrole natural products: origin, structural diversity, bioactivity and synthesis. (2019) (23)
- Formal synthesis of nanaomycin D via a Hauser–Kraus annulation using a chiral enone-lactone (2015) (23)
- Pyrans and their Benzo Derivatives: Synthesis (2008) (23)
- A Single Pseudoproline and Microwave Solid Phase Peptide Synthesis Facilitates an Efficient Synthesis of Human Amylin 1–37 (2013) (23)
- Unexpected Direct Synthesis of N-Vinyl Amides through Vinyl Azide-Enolate [3+2] Cycloaddition. (2017) (23)
- Total Synthesis and Stereochemical Revision of the Anti-Tuberculosis Peptaibol Trichoderin A. (2016) (23)
- Metabolic and behavioural adaptations during early development of the Antarctic silverfish, Pleuragramma antarcticum (2012) (23)
- Synthesis of the bis-spiroacetal C25-C40 moiety of the antimitotic agent spirastrellolide B using a bis-dithiane deprotection/spiroacetalisation sequence. (2010) (23)
- The enantioselective synthesis of tetracyclic methyllycaconitine analogues (2011) (23)
- Total synthesis of paecilospirone. (2011) (23)
- Synthesis of the anti-Helicobacter pylori agent (+)-spirolaxine methyl ether and the unnatural (2"S)-diastereomer. (2007) (23)
- Synthesis of the bis-spiroacetal core of the antimitotic agent spirastrellolide B. (2011) (23)
- Isolation, Structural Elucidation, and Synthesis of Lepteridine From Ma̅nuka (Leptospermum scoparium) Honey. (2016) (22)
- Synthesis and biological evaluation of novel teixobactin analogues. (2017) (22)
- Enantioselective synthesis of pyranonaphthoquinone antibiotics using a CBS reduction/cross-metathesis/oxa-Michael strategy. (2011) (22)
- Synthesis and methemoglobinemia-inducing properties of benzocaine isosteres designed as humane rodenticides. (2014) (22)
- Biomimetic studies towards the cardinalins: synthesis of (+)-ventiloquinone L and an unusual dimerisation. (2009) (22)
- Molecular Mechanisms of Class B GPCR Activation: Insights from Adrenomedullin Receptors. (2020) (22)
- Addition of silyloxydienes to 2,6-dibromo-1,4-benzoquinone: an approach to highly oxygenated bromonaphthoquinones for the synthesis of thysanone (2003) (22)
- Total synthesis of heronapyrrole C. (2014) (21)
- An enantioselective formal synthesis of berkelic acid. (2011) (21)
- Chemoenzymatic synthesis of deoxy analogues of the DNA topoisomerase II inhibitor eleutherin and the 3C-protease inhibitor thysanone (2008) (21)
- Synthesis of the FG ring fragment of pectenotoxins 1–9 (2010) (21)
- Stereoselective synthesis of deoxy analogues of the 3C-protease inhibitor thysanone (2002) (21)
- Synthesis of an Arginine Tagged [Cys155-Arg180] Fragment of NY-ESO-1: Elimination of an Undesired By-product Using ‘In House’ Resins (2009) (21)
- Synthesis of glycosylated 5-hydroxylysine, an important amino acid present in collagen-like proteins such as adiponectin. (2012) (21)
- Synthesis of two key intermediates required for the construction of the bis-spiroacetal moiety of epi-17-deoxy-(0–8)-salinomycin (1986) (21)
- Synthesis of simple analogues of methyllycaconitine - an efficient method for the preparation of the N -substituted anthranilate pharmacophore (2004) (21)
- Synthesis of triazole analogues of the nanaomycin antibiotics using ‘click chemistry’ (2010) (21)
- Maternally Administered Cyclic Glycine-Proline Increases Insulin-Like Growth Factor-1 Bioavailability and Novelty Recognition in Developing Offspring. (2016) (21)
- A Maillard Approach to 2‐Formylpyrroles: Synthesis of Magnolamide, Lobechine and Funebral (2014) (21)
- A titanium naphtholate approach for the synthesis of analogues of griseusin A (2000) (21)
- Protecting group free synthesis of glycosyl thiols from reducing sugars in water; application to the production of N-glycan glycoconjugates. (2017) (20)
- C-Glycosylation of tri-O-benzyl-2-deoxy-D-glucose: synthesis of naphthyl-substituted 3,6-dioxabicyclo[3.2.2]nonanes (2001) (20)
- A facile synthesis of aryldihydropyrans using a Sonogashira–selenoetherification strategy (2002) (20)
- Total synthesis of virgatolide B. (2013) (20)
- Synthesis of a regioisomeric analogue of the 3C-protease inhibitor thysanone via a Hauser annulation strategy (2007) (20)
- Natural Product-Inspired Pyranonaphthoquinone Inhibitors of Indoleamine 2,3-Dioxygenase-1 (IDO-1) (2013) (20)
- Anti-Helicobacter pylori activity of derivatives of the phthalide-containing antibacterial agents spirolaxine methyl ether, CJ-12,954, CJ-13,013, CJ-13,102, CJ-13,104, CJ-13,108 and CJ-13,015. (2008) (20)
- Formal synthesis of berkelic acid: a lesson in α-alkylation chemistry. (2012) (20)
- Synthesis of monolysyl advanced glycation endproducts and their incorporation into collagen model peptides. (2012) (20)
- A Convenient Method for the Asymmetric Synthesis of Fluorinated α‐Amino Acids from Alcohols (2014) (20)
- Enantioselective synthesis of the dimeric pyranonaphthoquinone core of the cardinalins using a late-stage homocoupling strategy. (2008) (20)
- Synthesis of macrocyclic analogues of the neuroprotective agent glycyl-L-prolyl-L-glutamic acid (GPE). (2006) (20)
- Synthesis of a dicarba analogue of human β-defensin-1 using a combined ring closing metathesis--native chemical ligation strategy. (2012) (20)
- Synthesis and evaluation of novel TLR2 agonists as potential adjuvants for cancer vaccines. (2020) (19)
- Cardiac troponins may be irreversibly modified by glycation: novel potential mechanisms of cardiac performance modulation (2018) (19)
- Synthesis of arizonin C1 (1995) (19)
- Synthesis of ABE tricyclic analogues of methyllycaconitine using a Wacker oxidation-aldol strategy to append the B ring to the AE fragment. (2002) (19)
- Synthesis of the ABC tricyclic fragment of the pectenotoxins via stereocontrolled cyclization of a gamma-hydroxyepoxide appended to the AB spiroacetal unit. (2006) (19)
- Synthesis and pharmacological evaluation of side chain modified glutamic acid analogues of the neuroprotective agent glycyl-L-prolyl-L-glutamic acid (GPE). (2005) (19)
- Use of bis(oxazoline)-metal complexes as chiral catalysts for asymmetric Diels-Alder reactions using 2-acetyl-1,4-naphthoquinone as a dienophile (1997) (19)
- Synthetic studies toward pyranonaphthoquinone antibiotics (2000) (19)
- Synthesis and bioactivity of antitubercular peptides and peptidomimetics: an update. (2016) (19)
- Synthesis of Analogues of Griseusin A (1999) (19)
- An efficient synthesis of 3-alkyl-1,5,3-dioxazepanes and their use as electrophiles in double-Mannich reactions (2012) (19)
- The Nedd4-1 WW Domain Recognizes the PY Motif Peptide through Coupled Folding and Binding Equilibria. (2016) (19)
- Enantioselective synthesis of an analogue of nanaomycin A (2007) (18)
- Application of olefin metathesis to the synthesis of ABE ring analogues of methyllycaconitine (2002) (18)
- Suzuki-Miyaura homocoupling of naphthyl triflates using bis(pinacolato)diboron: approaches to the biaryl skeleton of crisamicin A. (2003) (18)
- Synthesis and ene reactions of di-(−)-menthyl diazenedicarboxylate (1996) (18)
- Augmenting Influenza-Specific T Cell Memory Generation with a Natural Killer T Cell-Dependent Glycolipid-Peptide Vaccine. (2017) (18)
- Diabetes-induced alterations in tissue collagen and carboxymethyllysine in rat kidneys: Association with increased collagen-degrading proteinases and amelioration by Cu(II)-selective chelation. (2015) (18)
- Synthesis and pharmacological evaluation of glycine-modified analogues of the neuroprotective agent glycyl-L-prolyl-L-glutamic acid (GPE). (2005) (18)
- Synthesis of the spiroacetal-containing anti-Helicobacter pylori agents CJ-12,954 and CJ-13,014. (2006) (18)
- A slow gradient approach for the purification of synthetic polypeptides by reversed phase high performance liquid chromatography (2012) (18)
- Synthesis of the Bis-Spiroacetal Moiety of 17-epi-20-Deoxysalinomycin (1992) (18)
- Total Synthesis and Conformational Study of Callyaerin A: Anti-Tubercular Cyclic Peptide Bearing a Rare Rigidifying (Z)-2,3- Diaminoacrylamide Moiety. (2018) (18)
- The synthesis of dehydrotryptophan and dehydrotryptophan-containing peptides. (2011) (18)
- Synthesis of the spirocyclic framework of sesterterpenoid natural products. (2015) (18)
- Synthesis of Neoglycopeptides via Click Chemistry (2010) (18)
- SYNTHESIS OF A DIMERIC PYRANONAPHTHOQUINONE VIA A NOVEL DOUBLE FUROFURAN ANNULATION STRATEGY (1998) (17)
- Diastereoselective addition of 2-trimethylsilyloxyfuran to (S)-(+)-2-(p-tolylsulfinyl)-1,4-benzoquinone (1995) (17)
- Results of a randomized, double-blind phase II clinical trial of NY-ESO-1 vaccine with ISCOMATRIX adjuvant versus ISCOMATRIX alone in participants with high-risk resected melanoma (2020) (17)
- Double furofuran annulation to a bis-naphthoquinone: an approach to dimeric pyranonaphthoquinones (1998) (17)
- Synthetic approaches to [5,6]-benzannulated spiroketal natural products (2011) (17)
- Structure activity relationship study on the peptide hormone preptin, a novel bone-anabolic agent for the treatment of osteoporosis. (2016) (17)
- Photoaffinity Cross-Linking and Unnatural Amino Acid Mutagenesis Reveal Insights into Calcitonin Gene-Related Peptide Binding to the Calcitonin Receptor-like Receptor/Receptor Activity-Modifying Protein 1 (CLR/RAMP1) Complex. (2018) (17)
- A tandem Diels–Alder/Mannich approach to the synthesis of AE and ABE ring analogues of Delphinium alkaloids (2012) (17)
- A Facile Enantioselective Synthesis of the Dimeric Pyranonaphthoquinone Core of the Cardinalins (2008) (17)
- Synthesis of the 2-formylpyrrole spiroketal pollenopyrroside A and structural elucidation of xylapyrroside A, shensongine A and capparisine B. (2016) (17)
- Synthe1sis of 5-epi-arizonin B1 and 5-epi-arizonin C1 (1993) (17)
- Use of bis-(aminol) ethers derived from N-(S)-(−)-α-methylbenzylamine in reactions with resorcinarenes and double Mannich reactions (2005) (17)
- A facile synthesis of spiroketals (1988) (17)
- General Synthesis of the Nitropyrrolin Family of Natural Products via Regioselective CO2-Mediated Alkyne Hydration. (2017) (17)
- Using Chemical Synthesis to Probe Structure-Activity Relationships of the Glycoactive Bacteriocin Glycocin F. (2018) (17)
- Synthesis of the tetracyclic core of berkelic acid using gold(I)-catalyzed hydroarylation and oxidative radical cyclizations. (2012) (17)
- Efficient Synthesis of the Azabicyclo[3.3.1]nonane Ring System in the Alkaloid Methyllycaconitine Using Bis(alkoxymethyl)alkylamines as Aminoalkylating Agents in a Double Mannich Reaction (2005) (17)
- Synthesis of methyl N-Boc-(2S,4R)-4-methylpipecolate. (2010) (17)
- Synthesis and assignment of stereochemistry of the antibacterial cyclic peptide xenematide. (2011) (17)
- Nitropyrrole natural products: isolation, biosynthesis and total synthesis. (2016) (17)
- Synthesis of the spiroacetal core of the cephalosporolide family of natural products (2014) (17)
- Diastereoselective Diels-Alder reactions of optically-active vinyl sulphoxides (1985) (17)
- Synthesis of regioisomeric analogues of crisamicin A. (2003) (17)
- Synthesis and cytotoxicity of pyranonaphthoquinone natural product analogues under bioreductive conditions. (2013) (16)
- AGE-albumin enhances ABCA1 degradation by ubiquitin-proteasome and lysosomal pathways in macrophages. (2018) (16)
- Synthesis of a functionalised bis-spiroacetal (1990) (16)
- Addition of 2-tert-butyldimethylsilyloxythiophene to activated quinones: an approach to thia analogues of kalafungin (2006) (16)
- Desacetyl-α-melanocyte stimulating hormone and α-melanocyte stimulating hormone are required to regulate energy balance (2017) (16)
- Synthesis and methemoglobinemia-inducing properties of analogues of para-aminopropiophenone designed as humane rodenticides. (2013) (16)
- A comparison of Boc and Fmoc SPPS strategies for the preparation of C-terminal peptide α-thiolesters: NY-ESO-1 ³⁹Cys-⁶⁸Ala-COSR. (2013) (16)
- Peptide binding to a bacterial signal peptidase visualized by peptide tethering and carrier-driven crystallization (2016) (16)
- Synthesis of the 2-methylene analogue of the HRV 3C protease inhibitor thysanone (2-carbathysanone). (2014) (16)
- A new family of sesterterpenoids isolated around the Pacific Rim. (2018) (16)
- Short Anabolic Peptides for Bone Growth (2016) (16)
- Synthesis of AE and BE Ring Analogues of the Alkaloid Methyllycaconitine (2009) (16)
- Use of Stabilized Phthalide Anion Annulation Reactions in Synthesis: An Update (2007) (16)
- Synthesis of the phthalide-containing anti-Helicobacter pylori agents CJ-13,015, CJ-13,102, CJ-13,103, CJ-13,104 and CJ-13,108 (2005) (16)
- Synthesis and recycling of antifreeze glycoproteins in polar fishes (2012) (16)
- An update on new methods to synthesize cyclotetrapeptides. (2015) (16)
- ASYMMETRIC MICHAEL ADDITION OF 2-TRIMETHYLSILYLOXYFURAN TO CHIRAL NAPHTHOQUINONES (1998) (16)
- C-Glycosylation of Oxygenated Naphthols with 3-Dimethylamino-2,3,6-trideoxy-L-arabino-hexopyranose and 3-Azido-2,3,6-trideoxy-D-arabino-hexopyranose (2003) (16)
- Chemical synthesis of a masked analogue of the fish antifreeze potentiating protein (AFPP). (2013) (16)
- Total synthesis of chaetoquadrins A-C. (2013) (16)
- Chemical Synthesis of Peptides Containing Site-Specific Advanced Glycation Endproducts. (2016) (16)
- Improved Synthesis of the Unnatural Amino Acids AHMOD and AMD, Components of the Anticancer Peptaibol Culicinin D. (2015) (15)
- SYNTHESIS OF AN ACTINORHODIN MONOMER (1995) (15)
- Site-specific cross-linking of collagen peptides by lysyl advanced glycation endproducts. (2014) (15)
- A high yielding synthesis of anthranilate esters from sterically hindered alcohols (2001) (15)
- Synthesis of a C8 oxygenated pyranonaphthoquinone: a useful precursor to dimeric pyranonaphthoquinones (2008) (15)
- Synthesis of the 1,6,8-trioxadispiro[4.1.5.2]tetradec-11-ene ring system present in the spirolide family of shellfish toxins and its conversion into a 1,6,8-trioxadispiro[4.1.5.2]-tetradec-9-en-12-ol via base-induced rearrangement of an epoxide. (2004) (15)
- Approaches to the D-E ring of the polyether antibiotic salinomycin using sharpless asymmetric dihydroxylation (1998) (15)
- Synthesis and activity of a diselenide bond mimetic of the antimicrobial protein caenopore-5† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c5sc04187b (2015) (15)
- Synthesis of highly substituted pyranonaphthalene spiroketals related to the griseusins using a Hauser–Kraus annulation strategy (2014) (15)
- Formal synthesis of the juglomycins (1994) (15)
- A Facile Synthesis of Aryl Spirodioxines Based on a 3H,3′H-2,2′-Spiro-bi(benzo[b][1,4]dioxine) Skeleton (2007) (15)
- Synthesis of bis-2,5-linked tetrahydrofurans via iodoetherification (1995) (15)
- Virtual screening for novel Atg5–Atg16 complex inhibitors for autophagy modulation (2015) (15)
- Synthesis of the Revised Structure of Acortatarin A (2014) (14)
- Identification of anticancer agents based on the thieno[2,3-b]pyridine and 1H-pyrazole molecular scaffolds. (2016) (14)
- Synthesis of the novel 1,7,9-trioxadispiro[4.1.5.2]-tetradecane ring system present in the spirolides (2001) (14)
- Stability of polyelectrolyte-coated iron nanoparticles for T 2 -weighted magnetic resonance imaging (2017) (14)
- A comparative study of different glycosylation methods for the synthesis of D-mannopyranosides of Nalpha-fluorenylmethoxycarbonyl-trans-4-hydroxy-L-proline allyl ester. (2007) (14)
- Structure and Activity of Streptococcus pyogenes SipA: A Signal Peptidase-Like Protein Essential for Pilus Polymerisation (2014) (14)
- Design and synthesis of prodrugs of the rat selective toxicant norbormide. (2012) (14)
- A Flexible Approach to 6,5‐Benzannulated Spiroketals (2011) (14)
- Diels-Alder Addition of Acyclic Dienes to Chiral Naphthoquinones (2000) (14)
- 1,4-Addition of 2-trimethylsilyloxyfuran to quinones: a facile route to the furo[3,2-b]benzofuran nucleus (1987) (14)
- Synthesis of Azido Analogues of Medermycin (2002) (14)
- Synthesis and biological evaluation of tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R₈ERY. (2012) (14)
- A double Mannich approach to the synthesis of substituted piperidones—application to the synthesis of substituted E-ring analogues of methyllycaconitine (2010) (14)
- Total Synthesis of the Highly N-Methylated Acetylene-Containing Anticancer Peptide Jahanyne. (2018) (14)
- Total synthesis of 7',8'-dihydroaigialospirol. (2012) (14)
- Multiple Bactericidal Mechanisms of the Zinc Ionophore PBT2 (2020) (13)
- Prodrugs of N-dicarboximide derivatives of the rat selective toxicant norbormide. (2013) (13)
- Synthesis and evaluation of vasoconstrictor and vasorelaxant activity of norbormide isomers (2004) (13)
- Asymmetric Diels–Alder addition of cyclopentadiene to chiral naphthoquinones (1998) (13)
- A highly conserved tryptophan in the N‐terminal variable domain regulates disulfide bond formation and oligomeric assembly of adiponectin (2012) (13)
- Reductive thioalkylation of a pyranonaphthoquinone (2000) (13)
- Synthesis of leptosin, a glycoside isolated from mānuka honey (2013) (13)
- Stereocontrolled Synthesis of a Key Lactone Intermediate Required for the Synthesis of Salinomycin (1990) (13)
- Synthesis of the Spiroketal Core of the Pinnatifinoside Family of Natural Products (2016) (13)
- Oxidation of α-Farnesene (1993) (13)
- A peptide hydrogel derived from a fragment of human cardiac troponin C. (2016) (13)
- Influence of α-methyl substitution of proline-based organocatalysts on the asymmetric α-oxidation of aldehydes (2009) (13)
- Physicochemical studies on the copper(II) binding by glycated collagen telopeptides. (2015) (13)
- Chemical Synthesis of A Pore‐Forming Antimicrobial Protein, Caenopore‐5, by Using Native Chemical Ligation at a Glu‐Cys Site (2015) (13)
- Preparation of cis-γ-hydroxycarvone derivatives for synthesis of sesterterpenoid natural products: total synthesis of phorbin A. (2015) (13)
- Synthesis and assignment of the absolute configuration of the anti-Helicobacter pylori agents CJ-12,954 and CJ-13,014. (2007) (13)
- SYNTHESIS OF 2-METHYLPYRROLO[1,2-A]PYRAZIN-1(2H)-ONE (1988) (13)
- Using chemical synthesis to optimise antimicrobial peptides in the fight against antimicrobial resistance (2019) (13)
- Approaches to a Key Lactone Intermediate Required for the Synthesis of Pyranonaphthoquinone Antibiotics (1991) (13)
- Enantioselective access to benzannulated spiroketals using a chiral sulfoxide auxiliary. (2013) (12)
- Total synthesis and absolute configuration of (-)-berkeleyamide A. (2010) (12)
- Improved Strategy for the Synthesis of the Anticancer Agent Culicinin D (2015) (12)
- Synthesis of bicyclic pyrazinones via addition of heterocyclic amines to a nitro-alkene (1994) (12)
- The role for cyclic Glycine-Proline, a biological regulator of insulin-like growth factor-1 in pregnancy-related obesity and weight changes. (2018) (12)
- Chemical Synthesis of Bioactive Naturally Derived Cyclic Peptides Containing Ene-Like Rigidifying Motifs. (2018) (12)
- N-acetylcysteine Counteracts Adipose Tissue Macrophage Infiltration and Insulin Resistance Elicited by Advanced Glycated Albumin in Healthy Rats (2017) (12)
- Synthesis of enantiopure bicyclic alpha,alpha-disubstituted spirolactams via asymmetric Birch reductive alkylation. (2009) (12)
- Synthesis of a functionalized 7,6-bicyclic spiroimine ring fragment of the spirolides. (2010) (12)
- Replacement of the Acrid tert -Butylthiol and an Improved Isolation Protocol for Cysteine Lipidation on a Peptide or Amino Acid (CLipPA) (2020) (12)
- Total Synthesis of the Resorcyclic Acid Lactone Spiroketal Citreoviranol. (2016) (12)
- Molecules derived from the extremes of life: a decade later. (2020) (12)
- Synthesis of 3-azido-2,3,6-trideoxy-beta-D-arabino-hexopyranosyl pyranonaphthoquinone analogues of medermycin. (2003) (12)
- Glycated albumin induces lipid infiltration in mice aorta independently of DM and RAS local modulation by inducing lipid peroxidation and inflammation. (2016) (12)
- Uncatalyzed addition of N-(tert-butoxycarbonyl)-2-tert-butyldimethylsilyloxypyrrole to activated quinones (2002) (12)
- Controlling gelation with sequence: Towards programmable peptide hydrogels. (2016) (12)
- Synthesis of peramine, an insect feeding deterrent mycotoxin from Acremonium lolii (1988) (12)
- Cyclization of Linear Tetrapeptides Containing N‐Methylated Amino Acids by using 1‐Propanephosphonic Acid Anhydride (2017) (12)
- Telomerase Inhibition Studies of Novel Spiroketal- Containing Rubromycin Derivatives (2013) (11)
- Synthesis of N-(3-phenylpropyl)-substituted tricyclic ABE ring analogues of the alkaloid methyllycaconitine (2006) (11)
- Photo-induced radical thiol-ene chemistry: a versatile toolbox for peptide-based drug design. (2021) (11)
- Identification of Key Functional Motifs of Native Amelogenin Protein for Dental Enamel Remineralisation (2020) (11)
- Multifunctional thermoresponsive designer peptide hydrogels. (2017) (11)
- Pharmacological characterisation of mouse calcitonin and calcitonin receptor‐like receptors reveals differences compared with human receptors (2021) (11)
- The translocator protein (peripheral benzodiazepine receptor) mediates rat-selective activation of the mitochondrial permeability transition by norbormide. (2011) (11)
- Gold(I)-catalysed intramolecular hydroamination of α-quaternary alkynes: synthetic studies towards spiroimine marine toxins (2011) (11)
- Synthesis of spiroacetal-triazoles as privileged natural product-like scaffolds using "click chemistry". (2008) (11)
- SYNTHESIS OF TRICYCLIC ARYL SPIROACETALS RELATED TO THE PAPULACANDINS (1996) (11)
- Three Decades of Amyloid Beta Synthesis: Challenges and Advances (2019) (11)
- The synthesis of 5′-deoxyjuglomycin A and 5′-methoxyjuglomycin A. (1991) (11)
- Structure-activity relationship study of the tumour-targeting peptide A20FMDV2 via modification of Lys16, Leu13, and N- and/or C-terminal functionality. (2017) (11)
- Woodward-Prevost Reactions of 1,7-Dioxaspiro[5.5]undec-4-enes. (1996) (11)
- Discovery, Synthesis, and Optimization of Peptide-Based Antibiotics. (2021) (11)
- Synthesis and biological evaluation of analogues of the potent ADAM8 inhibitor cyclo(RLsKDK) for the treatment of inflammatory diseases and cancer metastasis. (2016) (11)
- TLR2 agonists and their structure-activity relationships. (2020) (11)
- Synthesis of the IGF-II-like hormone vesiculin using regioselective formation of disulfide bonds. (2013) (11)
- Radical oxidative cyclization of spiroacetals to bis-spiroacetals: an overview. (2004) (11)
- A versatile Boc solid phase synthesis of daptomycin and analogues using site specific, on-resin ozonolysis to install the kynurenine residue. (2019) (11)
- Total Synthesis and Stereochemical Revision of the 2-Formylpyrrole Alkaloid Hemerocallisamine I. (2017) (10)
- Improved Synthesis of the Benzyne Precursor 2-(Trimethylsilyl)phenyl Trifluoromethanesulfonate (2010) (10)
- Site-specific glycation of Aβ1–42 affects fibril formation and is neurotoxic (2019) (10)
- Synthesis of a C-Glycosylpyranonaphthoquinone Related to Medermycin (2000) (10)
- Synthesis of an Oxaspirolactone Intermediate for the Synthesis of Spirolides (2000) (10)
- How to blast osteoblasts? Novel dicarba analogues of amylin-(1-8) to treat osteoporosis. (2012) (10)
- Synthesis of the spiroacetal fragment of broussonetine H (2003) (10)
- Synthesis of an NDPK phosphocarrier domain peptide containing a novel triazolylalanine analogue of phosphohistidine using click chemistry. (2011) (10)
- Synthesis of the bis-spiroacetal moiety of the polyether antibiotic CP44,161 (2001) (10)
- Asymmetric azo-ene reactions using the chiral azo-enophile di-(−)-(1R,2S)-2-phenyl-1-cyclohexyl diazenedicarboxylate (1998) (10)
- A Facile Synthesis of 1,1′-Spirobi(3H,3′H)isobenzofurans (2007) (10)
- Receptor Activity Modifying Proteins Have Limited Effects on the Class B G Protein-Coupled Receptor Calcitonin Receptor-Like Receptor Stalk. (2018) (10)
- Direct synthesis of cyclic lipopeptides using intramolecular native chemical ligation and thiol-ene CLipPA chemistry. (2020) (10)
- Supramolecular Threading of Peptide Hydrogel Fibrils. (2018) (10)
- Synthesis of indole analogues of the anti-Helicobacter pylori compounds CJ-13,015, CJ-13,102, CJ-13,104 and CJ-13,108 (2007) (10)
- One-pot synthesis of water soluble iron nanoparticles using rationally-designed peptides and ligand release. (2013) (10)
- A Review of Advances in the Synthesis of Analogues of the Delphinium Alkaloid Methyllycaconitine (2005) (10)
- Synthesis of spiroacetal-nucleosides as privileged natural product-like scaffolds. (2009) (10)
- Regioselective asymmetric aminohydroxylation of precursors to 2,3,6-trideoxy-3-aminohexoses (2000) (10)
- Frontiers in Medicinal Chemistry (2016) (10)
- Glicentin‐related pancreatic polypeptide inhibits glucose‐stimulated insulin secretion from the isolated pancreas of adult male rats (2015) (10)
- Total synthesis of virgatolide B via exploitation of intramolecular hydrogen bonding. (2014) (10)
- Tyrosine modified analogues of the α4β7 integrin inhibitor biotin-R₈ERY prepared via Click Chemistry: synthesis and biological evaluation. (2012) (10)
- Synthesis and evaluation of 9-deoxy analogues of (-)-thysanone, an inhibitor of HRV 3C protease. (2014) (10)
- Synthesis of the All-l Cyclopentapeptides Versicoloritides A, B, and C (2012) (10)
- Genome mining, isolation, chemical synthesis and biological evaluation of a novel lanthipeptide, tikitericin, from the extremophilic microorganism Thermogemmatispora strain T81† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8sc02170h (2018) (9)
- Divergent Reactivity via Cobalt Catalysis: An Epoxide Olefination. (2016) (9)
- Synthesis of naphthyl C-glycosides of rearranged tri-O-benzyl-2-deoxy-D-glucose (2000) (9)
- Synthesis of truncated analogues of preptin-(1–16), and investigation of their ability to stimulate osteoblast proliferation. (2014) (9)
- SYNTHETIC STUDIES TOWARDS THE B, C, D, E FRAGMENT OF ANTIBIOTIC CP44, 161 (1999) (9)
- The synthesis and lectin-binding properties of novel mannose-functionalised polymers (2013) (9)
- Synthesis and reactivity of beta-methoxymethyl enecarbamates. (2009) (9)
- 'Tethering' fragment-based drug discovery to identify inhibitors of the essential respiratory membrane protein type II NADH dehydrogenase. (2018) (9)
- Chemistry of Bis‐spiroacetal Systems—Natural Products: Synthesis and Stereochemistry (2004) (9)
- Isolation and development of a HPLC method for thedetection and quantification of cryptolepine and itsapplication in the determination of the total cryptolepinecontent in the root powder of cryptolepis sanguinolenta (2012) (9)
- Cell-targeted platinum nanoparticles and nanoparticle clusters. (2015) (9)
- An Efficient Chemical Synthesis of Lassomycin Enabled by an On-Resin Lactamisation–Off-Resin Methanolysis Strategy and Preparation of Chemical Variants (2017) (9)
- Synthetic Studies Towards the Anti-inflammatory Agent, Oleocanthal using a Johnson-Claisen (Orthoester) Rearrangement Strategy (2009) (9)
- Synthetic approaches towards bedaquiline and its derivatives. (2020) (9)
- Synthesis of C-2 functionalised 1,6,8-trioxadispiro[4.1.5.3]pentadec-13-enes (1998) (9)
- Understanding the metal mediated assembly and hydrogel formation of a β-hairpin peptide. (2017) (9)
- Stereoselective synthesis of the rat selective toxicant norbormide (2016) (9)
- Total Synthesis of (-)-Peniphenone A. (2018) (9)
- 1H and 13C NMR data for C‐6 substituted 3‐azabicyclo[3.3.1]nonane‐1‐carboxylates (2006) (9)
- N-alkylsulfonylimines as dipolarophiles in cycloaddition reactions. (2013) (9)
- Reductive thioalkylation of a kalafungin analogue (1998) (9)
- Erratum: Synthesis of fish antifreeze neoglycopeptides using microwave-assisted "Click chemistry" (Organic Letters (2009) 11 (2409-2412)) (2010) (9)
- A Method for the Generation of Pam2Cys-Based Lipopeptide Mimics via CuAAC Click Chemistry (2012) (9)
- Synthesis and Herbicidal Activity of [3R,5S,6S]-3-Benzyloxy-5- methoxy-1,7-dioxaspiro[5.5]undecane and [3R,5S,6S]-3-Methoxy-5-benzyloxy-1,7-dioxaspiro[5.5]undecane. (1998) (9)
- An important side reaction using the thiol, 3,6‐dioxa‐1,8‐octanedithiol (DODT), in 9‐fluorenylmethoxycarbonyl‐based solid phase peptide synthesis (2014) (8)
- Synthetic studies toward the spiroimine unit of the spirolides (2011) (8)
- An investigation of the role of the adiponectin variable domain on the stability of the collagen‐like domain (2014) (8)
- Synthesis of arylspiroketals related to the papulacandins via generation of phthalide oxycarbenium ions (2001) (8)
- Synthesis of thiacrown and azacrown ethers based on a spiroacetal framework (2007) (8)
- Addition of cyclopentadiene and 2-trimethylsilyloxyfuran to quinones bearing a menthyl ester chiral auxiliary (1998) (8)
- Synthesis of Conjugated Trienes and Related Oxidation Products of α-Farnesene (1994) (8)
- Determination of pKa and forced degradation of the indoloquinoline antimalarial compound cryptolepine hydrochloride (2013) (8)
- Determination of the stereochemistry of 2,2-dimethyl-1,6,8-trioxadispiro(4.1.5.3)pentadec-13-ene formed by two sequential cyclization reactions using high field 1H N.M.R. spectroscopy (1985) (8)
- Structure-Activity Relationships of Wollamide Cyclic Hexapeptides with Activity against Drug-Resistant and Intracellular Mycobacterium tuberculosis (2019) (8)
- Allylic functionalization of the 1,7-dioxaspiro[5.5]-undec-4-ene and d1,6,8-trioxadispiro[4.1.5.3]-pentadec-13-ene ring systems. (1992) (8)
- Synthesis and biological evaluation of the osteoblast proliferating cyclic peptides dianthins G and H (2014) (8)
- A synthetic approach to ‘click’ neoglycoprotein analogues of EPO employing one-pot native chemical ligation and CuAAC chemistry† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c8sc03409e (2018) (8)
- Enantioselective synthesis of BE ring analogues of methyllycaconitine (2016) (8)
- Synthesis and amylin receptor activity of glycomimetics of pramlintide using click chemistry. (2016) (8)
- Synthesis and in vitro bone cell activity of analogues of the cyclohexapeptide dianthin G. (2016) (8)
- Synthesis and anti-Helicobacter pylori activity of analogues of spirolaxine methyl ether (2012) (8)
- An NBD Derivative of the Selective Rat Toxicant Norbormide as a New Probe for Living Cell Imaging (2016) (8)
- Synthesis of a pyranonaphthoquinone-spiroacetal (1992) (8)
- Synthesis and Biological Characterization of a New Norbormide Derived Bodipy FL-Conjugated Fluorescent Probe for Cell Imaging (2018) (8)
- Synthesis of 7-Methoxy-3′,4′,5′,6′-tetrahydrospiro-[isobenzofuran-1(3H),2′-pyran]-3-one and 5,7-Dimethoxy-3′,4′,5′,6′-tetrahydrospiro[isobenzofuran-1(3H),2′-pyran]-3-one (1998) (8)
- Synthesis of Psychrophilin E. (2016) (8)
- Nonsymmetrical Azocarbonamide Carboxylates as Effective Mitsunobu Reagents (2014) (8)
- Reaction of Bromonaphthofurans with Bis(pinacolato)diboron. (1999) (8)
- Studies towards development of asymmetric double-Mannich reactions of chiral 2-oxocyclohexanecarboxylate derivatives with bis(aminol)ethers (2015) (8)
- Towards eco-friendly marine antifouling biocides - Nature inspired tetrasubstituted 2,5-diketopiperazines. (2021) (8)
- Synthesis of Antimicrobial Lipopeptides Using the "CLipPA" Thiol-Ene Reaction. (2020) (8)
- Utility of the Leptospermum scoparium Compound Lepteridine as a Chemical Marker for Manuka Honey Authenticity (2020) (8)
- Synthesis of an Isotopically-labelled Antarctic Fish Antifreeze Glycoprotein Probe (2011) (8)
- Synthesis and Biological Evaluation of 7‐Deoxy Analogues of the Human Rhinovirus 3C Protease Inhibitor Thysanone (2014) (8)
- Synthesis of Natural Cyclopentapeptides Isolated from Dianthus chinensis. (2016) (8)
- “CLipP”ing on lipids to generate antibacterial lipopeptides† (2020) (7)
- Advanced Glycated apoA-IV Loses Its Ability to Prevent the LPS-Induced Reduction in Cholesterol Efflux-Related Gene Expression in Macrophages (2020) (7)
- The Bioreductive Alkylation of DNA by Kalafungin: A Theoretical Investigation (2007) (7)
- Fatty Acid‐Derived Pro‐Toxicants of the Rat Selective Toxicant Norbormide (2016) (7)
- Substituted Carbazoles – A New Class of Anthelmintic Agent (2016) (7)
- Synthesis and antiproliferative activity of culicinin D analogues containing simplified AHMOD-based residues. (2019) (7)
- A potent fluorescent calcitonin gene‐related peptide analogue enables visualization of receptor internalization (2019) (7)
- Bioinspired Total Synthesis and Stereochemical Revision of the Fungal Metabolite Pestalospirane B. (2017) (7)
- Solid-Phase Thiol-Ene Lipidation of Peptides for the Synthesis of a Potent CGRP Receptor Antagonist (2018) (7)
- Chemistry of bis-spiroacetals. Synthesis of the 1,6,8-trioxadispiro[4.1.5.3]pentadecane ring system (1988) (7)
- Intermolecular Peptide Cross-Linking by Using Diaminodicarboxylic Acids. (2016) (7)
- Regioselective iridium(I)-catalysed remote borylation of oxygenated naphthalenes (2012) (7)
- Novel Phosphopeptides as Surface-Active Agents in Iron Nanoparticle Synthesis (2012) (7)
- The chemistry of spiroacetals. Approaches to the novel 1,6,8-trioxadispiro[4.1.5.3]pentadecane ring system (1985) (7)
- A Convergent Synthesis of Gonytolide C Using an Intramolecular Oxa‐Michael Addition (2016) (7)
- Substituted sulfonamide bioisosteres of 8-hydroxyquinoline as zinc-dependent antibacterial compounds. (2020) (7)
- Synthesis of an azido precursor to (2S,5R)-5-hydroxylysine using an asymmetric organocatalytic chlorination/reduction sequence. (2013) (7)
- Thiol-ene Enabled Chemical Synthesis of Truncated S-Lipidated Teixobactin Analogs (2020) (7)
- Stereochemical Characterization of Polyketide Stereotriads Synthesized via Hydrogen-Mediated Asymmetric syn-Crotylation. (2017) (7)
- Assessing the molecular basis for rat-selective induction of the mitochondrial permeability transition by norbormide. (2007) (7)
- Deprotonation and alkylation of 2-methyl-4,5,6,7-tetrahydro-3H-azepine (1999) (7)
- Benzannulated spiroketal natural products: isolation, biological activity, biosynthesis, and total synthesis. (2019) (7)
- Enhancing T cell responses and tumour immunity by vaccination with peptides conjugated to a weak NKT cell agonist. (2019) (7)
- Alanine scan-guided synthesis and biological evaluation of analogues of culicinin D, a potent anticancer peptaibol. (2020) (7)
- Synthesis of 5,6- and 6,6-Spirocyclic Compounds (2014) (7)
- Two stereoisomers of the rat toxicant norbormide. (2004) (7)
- Synthetic studies toward shellfish toxins containing spiroacetal units (2007) (7)
- Reactivity of 2-Nitropyrrole Systems: Development of Improved Synthetic Approaches to Nitropyrrole Natural Products. (2018) (7)
- Synthesis and biological evaluation of S-lipidated lipopeptides of a connexin 43 channel inhibitory peptide. (2020) (7)
- Synthesis of (±) Wine Lactone and Its Analogues by a Diels–Alder Approach (2009) (7)
- Oxidation of α-Farnesene. (1994) (7)
- Addition of Silyloxydienes to 2,6‐Dibromo‐1,4‐benzoquinone: An Approach to Highly Oxygenated Bromonaphthoquinones for the Synthesis of Thysanone. (2003) (6)
- DIRECTED ORTHO METALATIONS OF TERTIARY BENZAMIDES USING LACTONES AS ELECTROPHILES (1994) (6)
- Kinetic resolution in the asymmetric dihydroxylation of 1,7-dioxaspiro[5.5]under-4-enes (1997) (6)
- Synthesis of stable isotope-labelled monolysyl advanced glycation endproducts (2013) (6)
- On resin synthesis and cross-linking of collagen peptides containing the advanced glycation end-product pyrraline via Maillard condensation. (2015) (6)
- Synthesis of a novel cage compound via oxidative rearrangement of a dihydronaphthofuran (1998) (6)
- A double-click approach to the protecting group free synthesis of glycoconjugates. (2018) (6)
- A review of agents patented for their neuroprotective properties. (2006) (6)
- Total Synthesis of Danshenspiroketallactone (2012) (6)
- Synthesis and Self-Assembly of a Peptide)Amphiphile as a Drug Delivery Vehicle (2013) (6)
- Live applications of norbormide-based fluorescent probes in Drosophila melanogaster (2019) (6)
- Nanoribbon Self-assembly and Hydrogel Formation from an N-Octanoyl Octapeptide Derived from the Antiparallel β-Interface of a Protein Homotetramer. (2020) (6)
- Synthesis of Benzannulated SpiroketalsUsing an Oxidative Radical Cyclization (2011) (6)
- Synthesis of the Tetracyclic Cores of the Integrastatins, Epicoccolide A and Epicocconigrone A. (2019) (6)
- Solid‐Phase Synthesis of the Peptaibol Alamethicin U‐22324 by Using a Double‐Linker Strategy (2017) (6)
- Total Synthesis and Structural Confirmation of the Antimalarial Naphthopyrone Lasionectrin. (2015) (6)
- Characterisation of agonist signalling profiles and agonist‐dependent antagonism at PACAP‐responsive receptors: Implications for drug discovery (2021) (6)
- Efficient synthesis of the spiroacetal core of paecilospirone via oxidative radical cyclisation (2011) (6)
- A Facile Cross Metathesis-Radical Cyclisation Approach to Monobenzannulated Spiroketals (2009) (6)
- Variable-length Ester-based Staples for α-Helical Peptides Using A Double Thiol-ene Reaction. (2020) (6)
- The Chemical Synthesis of the Collagenous Domain of the Hormone Adiponectin (2012) (6)
- Pharmacological characterization and investigation of N-terminal loop amino acids of adrenomedullin 2 that are important for receptor activation. (2019) (6)
- Synthesis of the Griseusin A Ring System (1990) (6)
- Synthesis of crown ethers based on a spiro acetal framework (1998) (5)
- Synthetic Studies Towards Natural Products Containing Bis‐spiroacetals (1999) (5)
- ALLYLIC OXIDATION OF UNSATURATED SPIROKETALS (1990) (5)
- Spiroimine Shellfish Poisoning (SSP) and the Spirolide Family of Shellfish Toxins: Isolation, Structure, Biological Activity and Synthesis (2010) (5)
- Analysis of Advanced Glycation End products in ribose-, glucose- and lactose-crosslinked gelatin to correlate the physical changes induced by Maillard reaction in films (2021) (5)
- Naturally Occurring Lumazines. (2019) (5)
- Synthesis of a C-Terminal Thioester Derivative of the Lipopeptide Pam2CSKKKKG Using Fmoc SPPS (2007) (5)
- Intermolecular Diels-Alder Cycloaddition/Cross-Coupling Sequences of 2-Bromo-1,3-butadienes. (2020) (5)
- A simple solid phase, peptide-based fluorescent assay for the efficient and universal screening of HRV 3C protease inhibitors. (2012) (5)
- Metal binding studies using spiroacetal thiacrown ethers (2010) (5)
- Synthesis of Spiroketals Related to Griseusin A (1996) (5)
- Addition of allylstannanes to an oxy-stabilized carbenium ion on a 1,7-dioxaspiro[5.5]undecane ring system (1998) (5)
- Synthesis of endolides A and B: naturally occurring N-methylated cyclic tetrapeptides. (2019) (5)
- Synthesis of (E)-1-Bromo-3-ethyl-3-pentene (1996) (5)
- Synthesis of 8-bromokalafungin as an intermediate for the preparation of C-glycoside derivatives (1997) (5)
- Cyclic Peptide Callyaerin A Bearing a Rare Rigidifying (Z)-2,3- Diaminoacrylamide Moiety (2018) (5)
- Efficient synthesis and characterisation of the amyloid beta peptide, Aβ1-42, using a double linker system. (2018) (5)
- MALDI-imaging enables direct observation of kinetic and thermodynamic products of mixed peptide fiber assembly. (2017) (5)
- Total chemical synthesis of glycocin F and analogues: S-glycosylation confers improved antimicrobial activity (2018) (5)
- Determining the regio- and typo-selectivity of calf pregastric lipase (2001) (5)
- Neoglycoprotein Synthesis Using the Copper‐Catalyzed Azide–Alkyne Click Reaction and Native Chemical Ligation (2013) (5)
- 2-Nitropyrrole cross-coupling enables a second generation synthesis of the heronapyrrole antibiotic natural product family. (2016) (5)
- Directed self-assembly of peptide-diketopyrrolopyrrole conjugates - a platform for bio-organic thin film preparation. (2020) (5)
- Iridium-Catalysed C–H Borylation Facilitates a Total Synthesis of the HRV 3C Protease Inhibitor (±)-Thysanone (2014) (5)
- Guanidinylated Amphiphilic Polycarbonates with Enhanced Antimicrobial Activity by Extending the Length of the Spacer Arm and Micelle Self-Assembly. (2020) (5)
- Synthesis of Leptosin, a Glycoside Isolated from Manuka Honey. (2014) (5)
- C-Glycosylation of naphthols using glucosyl donors (2001) (5)
- Cyclic Enecarbamates as Precursors of α,β-Unsaturated Iminium Ions: Reactivity and Synthesis of 6,6-Spirocyclic Ring Systems. (2016) (5)
- Norborn-2-en-7-ones as physiologically-triggered carbon monoxide-releasing prodrugs † (2017) (5)
- Synthesis of the Antifungal Cyclic Peptides Tunicyclins C and D (2012) (5)
- Anthranilate phosphoribosyltransferase: Binding determinants for 5'-phospho-alpha-d-ribosyl-1'-pyrophosphate (PRPP) and the implications for inhibitor design. (2018) (5)
- Synthesis of paenipeptin C' analogues employing solution-phase CLipPA chemistry. (2020) (5)
- Synthesis of a 6,6-spiroketal amino acid and its incorporation into a peptide turn sequence using solid-phase peptide synthesis. (2013) (5)
- The post-lockdown period should be used to acquire effective therapies for future resurgence in SARS-Cov-2 infections. (2020) (5)
- Synthesis of AHMOD-containing aminolipopeptides, unique bioactive peptaibiotics. (2017) (5)
- Addition of 2-((trimethylsilyloxy))furan to 2-acetyl-1,4- benzoquinone using chiral non-racemic copper(II)-pybox catalysts (2003) (5)
- Remarkable Influence of Cobalt Catalysis on Epoxide Ring-Opening with Sulfoxonium Ylides (2017) (5)
- Synthesis of a Novel Polyaniline Glycopolymer and its Lectin Binding Studies (2014) (5)
- Synthesis of aryl spiroketals related to the papulacandins via allylation of phthalides (2000) (5)
- Synthesis of a new spiroacetal based herbicide (1997) (4)
- Asymmetric dihydroxylation of a- and -farnesene (1994) (4)
- Synthesis of aromatic spiroacetals (1996) (4)
- Divalent cannabinoid-1 receptor ligands: A linker attachment point survey of SR141716A for development of high-affinity CB1R molecular probes. (2019) (4)
- Antibody responses to Collagen Peptides and Streptococcal Collagen-like 1 Proteins in Acute Rheumatic Fever Patients. (2021) (4)
- A Novel Approach to MonobenzannulatedSpiroketals Using Styrenes in the Kulinkovich Reaction (2009) (4)
- The chemistry of bis-spiroacetals. Synthesis of the novel 1,7,9-trioxadispiro[5.1.5.3]hexadecane ring system (1990) (4)
- 6,8′-Dimethoxy-2,2′-spirobichroman (2005) (4)
- Synthesis of spirolactams via Diels-Alder addition of 1,3-butadienes to an α-methylene lactam (2004) (4)
- Synthetic Studies Towards the Pectenotoxins: A Review (2007) (4)
- Fluorescent IGF-II analogues for FRET-based investigations into the binding of IGF-II to the IGF-1R. (2016) (4)
- Lipidated Calcitonin Gene-Related Peptide (CGRP) Peptide Antagonists Retain CGRP Receptor Activity and Attenuate CGRP Action In Vivo (2022) (4)
- Synthesis of Chiral Hydroxylated Farnesene Derivatives (1996) (4)
- Chemical synthesis of a polypeptide backbone derived from the primary sequence of the cancer protein NY‐ESO‐1 enabled by kinetically controlled ligation and pseudoprolines (2015) (4)
- Glycolipid‐peptide conjugate vaccines elicit CD8 + T‐cell responses and prevent breast cancer metastasis (2022) (4)
- On-resin Preparation of Allenamidyl Peptides: a Versatile Chemoselective Conjugation and Intramolecular Cyclisation Tool. (2020) (4)
- Novel Use of N-Carboalkoxy α,β-Unsaturated Iminium Ions as Dienophiles in Diels-Alder Reactions (2008) (4)
- Synthesis and structural insight into ESX‐1 Substrate Protein C, an immunodominant Mycobacterium tuberculosis‐secreted antigen (2016) (4)
- C—H Functionalization in the Synthesis of Amino Acids and Peptides (2014) (4)
- Enantioselective Synthesis of the Apple Aroma Constituent 1,3,3-Trimethyl-2,7-dioxabicyclo[2.2.1]heptane via Asymmetric Dihydroxylation (1995) (4)
- Synthesis of the carbon skeleton of the griseorhodins (2015) (4)
- Buchwald-Hartwig Mono-N-arylation with 2,6-Dihaloisonicotinic Acid Derivatives : A Convenient Desymmetrization Method (2008) (4)
- Synthesis of Enediamino Amino Acid Analogues and Peptides (2017) (4)
- Retaining or retrieving older and trying to identify novel rodenticides (2012) (4)
- Synthesis of Spirocyclic Imines: Key Pharmacophores in the Shellfish Toxins Spirolides and Gymnodimine (2003) (4)
- Synthesis and activity of a diselenide bond mimetic of the antimicrobial protein caenopore-5 (2016) (4)
- One‐Pot Synthesis of Functionalized Noble Metal Nanoparticles Using a Rationally Designed Phosphopeptide (2014) (4)
- Design, characterization and evaluation of β-hairpin peptide hydrogels as a support for osteoblast cell growth and bovine lactoferrin delivery (2020) (4)
- Asymmetric Total Synthesis of the Naturally Occurring Antibiotic Anthracimycin. (2020) (4)
- Enantioselective Synthesis ofthe 3C-Protease Inhibitor (-)-Thysanone by a Staunton-WeinrebAnnulation Strategy (2009) (4)
- Naturally occurring antitubercular cyclic peptides (2019) (4)
- Chemical synthesis of γ‐secretase activating protein using pseudoglutamines as ligation sites (2015) (4)
- Synthesis of trans- and cis-14-phenylsulfonyl-1,7,9-trioxadispiro[5.1.5.3]hexadecane (1994) (4)
- Facile Bisarylation of Aldehydes Using Titanium Naphtholates (1997) (4)
- Use of ‘Click Chemistry’ forthe Synthesis of Tetrazole-Containing Analogues of the NeuroprotectiveAgent Glycyl-l-prolyl-l-glutamicAcid (2009) (4)
- A short enantioselective synthesis of the topoisomerase II inhibitor (+)-eleutherin (2007) (4)
- Synthetic Studies Towards Spirocyclic Imine Marine Toxins Using N-Acyl Iminium Ions as Dienophiles in Diels–Alder Reactions (2020) (4)
- Synthesis of Novel Triazole-Containing Phosphonate Polymers (2015) (4)
- Enantioselective Synthesis of the 3C-Protease Inhibitor (–)-Thysanone by a Staunton–Weinreb Annulation Strategy (2009) (3)
- Synthesis of a Novel Nucleoside Based on a Spiroacetal Framework (2004) (3)
- Reactions of semiquinones in aqueous solution. A comparison of the one electron reduction of kalafungin and analogues with other semiquinones using pulse radiolysis (1999) (3)
- Synthesis of Chiral Diazanedicarboxylates (1998) (3)
- Synthesis of the Bicyclic Lactone Core of Leonuketal, Enabled by a Telescoped Diels-Alder Reaction Sequence. (2018) (3)
- seco-Labdanes: a Study of Terpenoid Structural Diversity Resulting from Biosynthetic C-C Bond Cleavage. (2020) (3)
- Synthesis of DOHNAA, a Mycobacterium tuberculosis Cholesterol CD Ring Catabolite and FadD3 Substrate (2015) (3)
- Synthesis and Biological Evaluation of the Osteoblast Proliferating Cyclic Peptides Dianthins G and H. (2015) (3)
- Synthesis of the PyranonaphthoquinonesDehydroherbarin, (+)-Astropaquinone B and (+)-AstropaquinoneC en Route to Ascomycones A and B (2010) (3)
- DNA adduct formation of mitomycin C. A test case for DFT calculations on model systems (2013) (3)
- Synthesis and antiproliferative activity of C- and N-terminal analogues of culicinin D. (2020) (3)
- The Synthesis of Oxygenated Naphthyl Stannanes Possessing ortho-Methoxy Substituents for Use in Stille Coupling Reactions (1999) (3)
- ent-Atisane diterpenoids: isolation, structure and bioactivity. (2020) (3)
- Highly Diastereoselective Synthesis of Syn-1,3-Dihydroxyketone Motifs from Propargylic Alcohols via Unusual Spiroepoxide Intermediates. (2019) (3)
- 1H and 13C NMR spectra of methylmaleimido‐ and methylsuccinimidoanthranilate esters of 1‐hydroxymethyl‐6‐methoxy‐3‐azabicyclo[3.3.1]nonanes (2007) (3)
- Recent Progress in the Synthesis of Homogeneous Erythropoietin (EPO) Glycoforms (2020) (3)
- N-Vinyl Acrylamides: Versatile Heterobifunctional Electrophiles for Thiol-Thiol Bioconjugations. (2022) (3)
- TRENDS IN VERTEBRATE PESTICIDE USE AND NEW DEVELOPMENTS: NEW ZEALAND INITIATIVES AND INTERNATIONAL IMPLICATIONS (2010) (3)
- Enantioselective synthesis of C-linked spiroacetal-triazoles as privileged natural product-like scaffolds. (2012) (3)
- A Ring Closing Metathesis Approach to the Formal Synthesis of (+)‐Callyspongiolide (2020) (3)
- Investigations of the key macrolactamisation step in the synthesis of cyclic tetrapeptide pseudoxylallemycin A. (2019) (3)
- Dihydroxylation of 1,7-Dioxaspiro[5.5]undec-4-enes (1993) (3)
- Microwave-Assisted Synthesisof Fluorescein-Labelled GalNAcα1-O-Ser/Thr (Tn)Glycopeptides as Immunological Probes (2010) (3)
- Addition of a Grignard reagent to bis-spiroacetal aldehydes: appendage of a tetrahydrofuran ring (1999) (3)
- Novel Preparation of Chiral α‐Amino Acids Using the Mitsunobu—Tsunoda Reaction. (2013) (3)
- Stereoselective Synthesis of 4-Substituted 4-Hydroxypiperidines via Epoxidation-Ring Opening of 4-Methylenepiperidines (2010) (3)
- Synthesis of New Aza‐C‐disaccharides Linking 4‐Deoxy‐4‐amino‐β‐L‐erythro‐furanose to C‐2 of D‐Glucose and D‐Allose (2006) (3)
- Chemistry of bis-spiroacetals: synthesis of cis- and trans-1-(2-methyl-1,6,8-trioxadispiro[4.1.5.3]pentadec-13-en-2-yl)methanol (1991) (3)
- Pyranonaphthoquinones—Isolation, Biological Activity and Synthesis (2008) (3)
- Aminovinyl Cysteine Containing Peptides: A Unique Motif That Imparts Key Biological Activity (2021) (3)
- A Chemometric Analysis of Compounds from Native New Zealand Medicinal Flora. (2018) (3)
- A Catalytic Asymmetric Ene Reaction for Direct Preparation of α-Hydroxy 1,4-Diketones as Intermediates in Natural Product Synthesis (2020) (3)
- Recent Developments in Neoglycopeptide Synthesis (2011) (3)
- Disruption of Metallostasis in the Anaerobic Human Pathogen Fusobacterium nucleatum by the Zinc Ionophore PBT2. (2021) (3)
- A new high-capacity metal ion-complexing gel containing cyclen ligands (2016) (3)
- Total Synthesis of (±)-Leonuketal. (2020) (3)
- Stereochemical Effects on the Antimicrobial Properties of Tetrasubstituted 2,5-Diketopiperazines. (2022) (2)
- Synthesis of the Phthalide-Containing anti-Helicobacter pylori Agents CJ-13,015 (Ia), CJ-13,102 (Ib), CJ-13,103 (Ic), CJ-13,104 (Id) and CJ-13,108 (Ie). (2006) (2)
- In vitro metabolism of norbormide in rat, mouse and guinea pig liver preparations. (2009) (2)
- A High-Yielding Synthesis of Anthranilate Esters from Sterically Hindered Alcohols. (2010) (2)
- Evolution of Peptide-Based Prostate-Specific Membrane Antigen (PSMA) Inhibitors: An Approach to Novel Prostate Cancer Therapeutics. (2020) (2)
- Total synthesis of the proposed structure of talarolide A. (2018) (2)
- Polyether antibiotic CP44,161. (2001) (2)
- Building trans-bicyclo[4.4.0]decanes/decenes in complex multifunctional frameworks: the case for antibiotic development. (2020) (2)
- Application Of A Double Mannich Reaction Using Bis(Aminol) Ethers In The Synthesis Of Ae Ring Analogues Of Methyl Lycaconitine (2004) (2)
- Using mass spectrometry to detect, differentiate, and semiquantitate closely related peptide hormones in complex milieu: measurement of IGF-II and vesiculin. (2015) (2)
- The tryptophan connection: cyclic peptide natural products linked via the tryptophan side chain. (2021) (2)
- Microtiter Screening Reveals Oxygen-Dependent Antimicrobial Activity of Natural Products Against Mastitis-Causing Bacteria (2019) (2)
- Stability of 5(6)-carboxyfluorescein in microwave-assisted synthesis of fluorescein-labelled O-dimannosylated peptides (2009) (2)
- Incorporation of 'click' chemistry glycomimetics dramatically alters triple-helix stability in an adiponectin model peptide. (2017) (2)
- Expedient Synthesis of Peptides Containing N ε-Carboxymethyllysine (2014) (2)
- The Selective Rat Toxicant Norbormide Blocks KATP Channels in Smooth Muscle Cells But Not in Insulin-Secreting Cells (2019) (2)
- Synthesis of deuterium labelled hexenols (1992) (2)
- C-2 derivatized 8-sulfonamidoquinolines as antibacterial compounds. (2020) (2)
- Synthesis of Aromatic Spiroacetals. (1996) (2)
- Highly stereoselective syn-hydroxylation of spiroketals (1991) (2)
- Synthesis of isotopically labelled αCGRP8-37 and its lipidated analogue. (2020) (2)
- Synthesis of the Spiroacetal Fragment of Broussonetine H. (2003) (2)
- Total Synthesis of the Macrocyclic N‐Methyl Enamides Palmyrolide A and 2S‐Sanctolide A. (2015) (2)
- Total chemical synthesis of an Orf virus protein, ORFV002, an inhibitor of the master gene regulator NF‐κB (2014) (2)
- (1R,6R)-1-Methyl-8-azaspiro[5.6]dodecan-7-one (2008) (2)
- Screening a Natural Product-Inspired Library for Anti-Phytophthora Activities (2021) (2)
- Synthesis of Aryl Spiroketals Related to the Papulacandins via Allylation of Phthalides. (2000) (2)
- Synthesis of Bis‐Spiroacetal Ring Systems (1999) (2)
- A Concise Synthetic Strategy Towards the Novel Calcium-dependent Lipopeptide Antibiotic, Malacidin A and Analogues (2021) (2)
- Spectral Assignments and Reference Data (2008) (2)
- An Efficient Enantioselective Synthesis of the 3C Protease Inhibitor (-)-Thysanone (2008) (2)
- (1S,2S)‐1‐{2‐[(4‐Methoxybenzyl)oxy]ethyl}‐2‐methyl‐3‐butenyl (1S,4R)‐4,7,7‐trimethyl‐3‐oxo‐2‐oxabicyclo[2.2.1]heptane‐1‐carboxylate (2005) (2)
- Synthesis of mannosylated glycopeptides as components for synthetic vaccines. (2009) (2)
- Diels-Alder Cycloaddition of Cyclopentadiene to a Bis-naphthoquinone (2000) (2)
- Synthesis of Benzannulated Spiroketals Using an Oxidative Radical Cyclization. (2011) (2)
- An Improved Method for the Synthesis of Lipopeptide TLR2-Agonists Using Click Chemistry (2013) (2)
- Preparation of truncated orf virus entry fusion complex proteins by chemical synthesis (2014) (2)
- Synthesis of peptide homo‐ and heterodimers as potential mimics of platelet‐derived growth factor BB (2020) (2)
- The Total Chemical Synthesis and Biological Evaluation of the Cationic Antimicrobial Peptides, Laterocidine and Brevicidine. (2021) (2)
- Datasets, processing and refinement details for Mtb-AnPRT: inhibitor structures with various space groups (2017) (2)
- A Highly Efficient N-Mesityl Thiazolylidene for the Aliphatic Stetter Reaction: Stereoelectronic Quantification for Comparison of N‑Heterocyclic Carbene Organocatalysts (2021) (2)
- Synthesis and SAR analysis of lipovelutibols B and D and their lipid analogues. (2019) (2)
- (±)-1-{8′-(tert-Butyldiphenylsilyloxymethyl)-1′,7′-dioxaspiro[5.5]undecan-2′-yl}uridine (2008) (2)
- 1H and 13C NMR spectra of C‐6 and C‐9 substituted 3‐azabicyclco[3.3.1]nonanes (2008) (2)
- Anticholinesterase Inhibition, Drug-Likeness Assessment, and Molecular Docking Evaluation of Milk Protein-Derived Opioid Peptides for the Control of Alzheimer’s Disease (2022) (1)
- Cardiac troponins may be irreversibly modified by glycation: novel potential mechanisms of cardiac performance modulation (2018) (1)
- Book Review, Organic Synthesis Highlights II (1996) (1)
- Convenient access to 5-membered cyclic iminium ions: evidence for a stepwise [4 + 2] cycloaddition mechanism. (2019) (1)
- Crystal Structures of (3S*,4S*,5S*,6S*)-3,4-Epoxy- 1,7-dioxaspiro[5.5]undecan-5-ol, (3R*,5S*,6S*)-1,7- Dioxaspiro[5.5]undecane-3,5-diyl Diacetate and (4S*,5S*,6S*)-1,7-Dioxaspiro[5.5]undecane-4,5-diol (1997) (1)
- Back Cover: Rapid and simultaneous analysis of advanced glycation end products on silica hydride column: Comparison of ultraviolet, fluorescence, and mass spectrometry detectors (2020) (1)
- Synthesis and SAR of a Library of Cell-Permeable Biotin-R8ERY* Peptidomimetics Inhibiting α4β7 Integrin Mediated Adhesion of TK-1 Cells to MAdCAM-1-Fc (2012) (1)
- Synthesis and incorporation of an advanced lipid peroxidation end-product building block into collagen mimetic peptides. (2017) (1)
- Asymmetric Diels—Alder Addition of Cyclopentadiene to Chiral Naphthoquinones. (1998) (1)
- Synthesis of isotopically labelled glycyl‐L‐prolyl‐L‐glutamic acid (Glypromate®) and derivatives (2006) (1)
- A convenient synthesis of 2-(3-methyl-2,5-dioxopyrrolidin-1-yl)benzoic acid (2003) (1)
- Synthesis of Conjugated Trienes and Related Oxidation Products of . alpha.-Farnesene. (1995) (1)
- Diastereoselective Synthesis of Substituted 4-Piperidones and 4-Piperidols Using a Double Mannich Reaction. (2009) (1)
- (1R,1′R,3S,3′S)-5,5′,10,10′-Tetramethoxy-1,1′,3,3′-tetramethyl-3,3′,4,4′-tetrahydro-1H,1′H-8,8′-bi[benzo[g]isochromene] (2008) (1)
- Total Synthesis of Novel Antimicrobial β-Hairpin Capitellacin Via Rapid Flow-Based SPPS Assembly and Regioselective On-Resin Disulfide Cyclisation (2021) (1)
- 5,8'-Dimethoxy-3H-1-benzofuran-2-spiro-2'-chroman (2005) (1)
- Diastereoselective Synthesisof Substituted 4-Piperidones and 4-Piperidols Using a Double MannichReaction (2008) (1)
- (2′′S,5′′R,7′′S)-2-[2′-(2′′-Methyl-1′′,6′′-dioxaspiro[4.5]dec-7′′-yl)ethylsulfonyl]-1,3-benzothiazole (2006) (1)
- Towards Eco-Friendly Marine Antifouling Biocides – Nature Inspired Tetrasubstituted 2,5-Diketopiperazines (2021) (1)
- Synthesis of Pharmaceuticals Using Molecular Chess and Automated Synthesis (2005) (1)
- Instant Insight: Life at the Extremes (2008) (1)
- Rules for abbreviation of protecting groups (IUPAC Technical Report) (2012) (1)
- Glucoregulatory activity of vesiculin in insulin sensitive and resistant mice (2019) (1)
- Synthesis, Antibacterial Activity, and Nephrotoxicity of Polymyxin B Analogues Modified at Leu-7, d-Phe-6, and the N-Terminus Enabled by S-Lipidation. (2022) (1)
- A Facile Synthesis of a Spironitrone and a Study of Its Cycloaddition and Nucleophilic Addition Reactions (2008) (1)
- Organic Synthesis: Where to from Now? A Personal Perspective from Down Under. (2019) (1)
- Novel Fluorescently Labeled PACAP and VIP Highlight Differences between Peptide Internalization and Receptor Pharmacology. (2022) (1)
- C-Glycosylation of Tri-O-benzyl-2-deoxy-D-glucose: Synthesis of Naphthyl-Substituted 3,6-Dioxabicyclo[3.2.2]nonanes. (2001) (1)
- Enantioselective synthesis of a cyclopentannulated kalafungin analogue (2000) (1)
- An Update on New Methods to Synthesize Cyclotetrapeptides (2015) (1)
- Nitrobenzoxadiazole derivatives of the rat selective toxicant norbormide as fluorescent probes for live cell imaging. (2022) (1)
- An Efficient Fmoc Solid-Phase Synthesis of an Amphiphile of the Neuroprotective Agent Glycyl-prolyl-glutamic Acid (2014) (1)
- [2R*,5S*,6S*]-2-Methyl-1,7-dioxaspiro[5.5]undec-2-en-5-ol (1997) (1)
- An Efficient Synthesis of 3-Alkyl-1,5,3-dioxazepanes and Their Use as Electrophiles in Double-Mannich Reactions. (2012) (1)
- A chiral auxiliary-based synthesis of the C5–C17 trans-decalin framework of anthracimycin (2019) (1)
- Application of a Double Mannich Reaction Using Bis(aminol) Ethers in the Synthesis of AE Ring Analogues of Methyl Lycaconitine. (2005) (1)
- Highly Diastereoselective Synthesis of Syn ‐1,3‐Dihydroxyketone Motifs from Propargylic Alcohols via Spiroepoxide Intermediates (2019) (1)
- Synthesis of a 2-Deoxyglucosyl Analogue of Medermycin. (2001) (1)
- Metabolic and behavioural adaptations during early development of the Antarctic silverfish, Pleuragramma antarcticum (2011) (1)
- Allylic Amination by the Lewis-Acid-Mediated Ene Reaction of Diethyl Azodicarboxylate with Alkenes. (2010) (1)
- Addition of a chiral non-racemic silyloxypyrrole to an activated 1,4-benzoquinone (2002) (1)
- Synthesis of Lipopeptides by CLipPA Chemistry. (2021) (1)
- endo‐(1′R,2′R,5′S,7′R,9′S)‐2‐(9′‐Benzyloxy‐2′‐phenyl‐3′,6′‐dioxabicyclo[3.2.2]nonan‐7′‐yl)‐7‐bromo‐5,8‐dimethoxynaphthalen‐1‐yl acetate (2001) (1)
- Total Synthesis of Chaetoquadrins H and I (2013) (1)
- Site-specific glycations of Aβ1–42 affect fibril formation and are neurotoxic (2019) (1)
- Recent Developments in Transition Metal-Catalyzed Spiroketalisation (2014) (1)
- Fourth-Generation Analogues of the Anticancer Peptaibol Culicinin D: Probing the Effects of Hydrophobicity and Halogenation on Cytotoxicity (2021) (1)
- Frontispiece: Chemical Synthesis of Bioactive Naturally Derived Cyclic Peptides Containing Ene‐Like Rigidifying Motifs (2018) (1)
- Enantioselective Synthesis of BE Ring Analogues of Methyllycaconitine. (2016) (1)
- Use of a Sonogashira—Acetylide Coupling Strategy for the Synthesis of the Aromatic Spiroketal Skeleton of γ‐Rubromycin (VII). (2004) (1)
- Differential internalisation of the CGRP and AMY1 receptor (2020) (1)
- Synthesis of Naphthyl C-Glycosides of Rearranged Tri-O-benzyl-2-deoxy-D-glucose. (2000) (1)
- The synthesis and bioactivity of the marine macrolide callyspongiolide. (2020) (1)
- A novel bromine-induced ring expansion of the spiroimine moiety of the shellfish toxin gymnodimine (2006) (1)
- PAC1, VPAC1, and VPAC2 Receptor Expression in Rat and Human Trigeminal Ganglia: Characterization of PACAP-Responsive Receptor Antibodies (2022) (1)
- Synthesis of Benzotriazole Analogues of the Helicobactericidal Agents CJ-13,015, CJ-13,102, CJ-13,108, and CJ-13,104 Using a Regioselective 1,3-Dipolar Cycloaddition (2011) (1)
- Directed ortho‐Metalations of Tertiary Benzamides Using Lactones as Electrophiles (1994) (1)
- Radical Oxidative Cyclization of Spiroacetals to Bis-spiroacetals (2005) (1)
- A Convenient Synthesis of 2‐(3‐Methyl‐2,5‐dioxopyrrolidin‐1‐yl)benzoic Acid. (2003) (1)
- Synthesis of Triazole Analogues of the Nanaomycin Antibiotics Using “Click Chemistry”. (2010) (0)
- A Single Pseudoproline and Microwave Solid Phase Peptide Synthesis Facilitates an Efficient Synthesis of Human Amylin 1–37 (2012) (0)
- Molecules Derived from the Extremes of Life (2009) (0)
- [3R*,5S*,6S*]-1,7-Dioxaspiro[5.5]undecane-3,5-diyl Bis(3,5-dinitrobenzoate) (1997) (0)
- A solid support-based synthetic strategy for the site-selective functionalization of peptides with organometallic half-sandwich moieties. (2021) (0)
- The Synthesis of Potential Chemotherapeutic Agents Based on Leads from Nature (2010) (0)
- Chemistry Research: Making Molecules for Medicines (2008) (0)
- ASYMMETRIC DIHYDROXYLATION OF ALPHA - AND BETA -FARNESENE (1994) (0)
- tert-Butyl methoxy(2-propynyl)carbamate (2001) (0)
- Deprotonation and Alkylation of 2-Methyl-4,5,6,7-tetrahydro-3H-azepine. (2000) (0)
- Photoa ffi nity Cross-Linking and Unnatural Amino Acid Mutagenesis Reveal Insights into Calcitonin Gene-Related Peptide Binding to the Calcitonin Receptor-like Receptor / Receptor Activity-Modifying Protein 1 ( CLR / RAMP 1 ) Complex (2018) (0)
- Synthesis of Macrocyclic Shellfish Toxins Containing Spiroimine Moieties (2007) (0)
- C‐Glycosylation of Oxygenated Naphthols with 3‐Dimethylamino‐2,3,6‐trideoxy‐L‐arabino‐hexopyranose and 3‐Azido‐2,3,6‐trideoxy‐D‐arabino‐hexopyranose. (2003) (0)
- 196 Strategies for Inhibiting Advanced Glycation Endproduct (Age) Induced Vascular Calcification in a Smooth Muscle Cell Culture Model (2016) (0)
- Synthesis of a Novel Cage Compound via Oxidative Rearrangement of a Dihydronaphthofuran. (1999) (0)
- Asymmetric Dihydroxylation of a- and -Farnesence. (1995) (0)
- Double Furofuran Annulation to a Bis-naphthoquinone: An Approach to Dimeric Pyranonaphthoquinones. (2010) (0)
- Cover Picture: Radiation Damage and Racemic Protein Crystallography Reveal the Unique Structure of the GASA/Snakin Protein Superfamily (Angew. Chem. Int. Ed. 28/2016) (2016) (0)
- Total Synthesis of the Fungal Metabolite Virgatolide B (2015) (0)
- Synthesis of Spiroketals Related to Griseusin A. (1998) (0)
- Synthesis of 7‐Methoxy‐3′,4′,5′,6′‐tetrahydrospiro [isobenzofuran‐1(3H),2′‐pyran]‐3‐one and 5,7‐Dimethoxy‐3′,4′,5′,6′‐tetrahydrospiro [isobenzofuran‐1(3H),2′‐pyran]‐3‐one. (1998) (0)
- (6bR*,9aR*)-6-(2-benzyloxy-1-oxoethyl)-6b,9a-dihydro-5-hydroxy- 4-methoxyfuro[3,2-b]naphtho[2,1-d]furan-8(9H)-one (2000) (0)
- Equilibrated structures for the MD simulations (2017) (0)
- Norbormide-Based and Their Application for Mitochondrial Imaging in (2021) (0)
- Species specific stimulation of the mitochondrial permeability transition by norbormide and its derivatives (2006) (0)
- A Review of the Synthesis of α-Carbolines (2015) (0)
- Innenrücktitelbild: Total Synthesis and Conformational Study of Callyaerin A: Anti‐Tubercular Cyclic Peptide Bearing a Rare Rigidifying (Z)‐2,3‐ Diaminoacrylamide Moiety (Angew. Chem. 14/2018) (2018) (0)
- A novel tyrosine hyperoxidation enables selective peptide cleavage (2022) (0)
- Engineering a stable complex of ERp44 with a designed peptide ligand for analyzing the mode of interaction of ERp44 with its clients (2021) (0)
- A Facile Synthesis of Spiroacetals. (1989) (0)
- Regioselective Iridium(I)‐Catalyzed Remote Borylation of Oxygenated Naphthalenes. (2012) (0)
- (4R,2'R,3'R,5'R)-3-[3,5-Bis(tert-butyldimethylsilyloxy)-1-oxo-2-(phenylmethoxy)hexyl]-4-(phenylmethyl)-2-oxazolidinone (2000) (0)
- Approaches to a Key Lactone Intermediate Required for the Synthesis of Pyranonaphthoquinone Antibiotics. (1991) (0)
- Asymmetric Michael Addition of 2-Trimethylsilyloxyfuran to Chiral Naphthoquinones. (1998) (0)
- Redevelopment of a Rat Specific Rodenticide Norbormide (2018) (0)
- Characterising the mode of action of Connexin43 mimetic Peptide5 to target retinal ischemia-reperfusion injury (2016) (0)
- Synthesis of stable isotope-labelled monolysyl advanced glycation endproducts (2013) (0)
- Pyridine-3-carboxaldehyde O-methyloxime (2001) (0)
- Synthesis of Arizonin C1. (1996) (0)
- Natural Resources Proceedings of the Vertebrate Pest Conference Title Toxicodynamics of Methemoglobin ( MtHb ) Inducers Permalink (2011) (0)
- Synthesis of a Pyranonaphthoquinone Spiroacetal. (1992) (0)
- (±)-2′-Phenylcyclohexanespiro-4′-(azepano[1,2-b]isoxazolidine) (2008) (0)
- N‐Alkylsulfonylimines as Dipolarophiles in Cycloaddition Reactions (2013) (0)
- Nonsymmetrical Azocarbonamide Carboxylates as Effective Mitsunobu Reagents. (2015) (0)
- Synthesis of the Revised Structure of Acortatarin A. (2015) (0)
- Allylic Oxidation of Unsaturated Spiroketals. (2010) (0)
- THE CHEMISTRY OF SPIROACETALS. APPROACHES TO THE NOVEL 1,6,8-TRIOXADISPIRO(4.1.5.3)PENTADECANE RING SYSTEM (1985) (0)
- A Novel Approach to Monobenzannulated Spiroketals Using Styrenes in the Kulinkovich Reaction. (2010) (0)
- NOVEL LIPIDATED CGRP PEPTIDE ANTAGONISTS FOR THE TREATMENT OF MIGRAINE AND PAIN (2018) (0)
- Synthesis of Tricyclic Aryl Spiroacetals Related to the Papulacandins. (1996) (0)
- Synthesis of 5-epi-7-Deoxykalafungin and 5-epi-7-O-Methylkalafungin. (1990) (0)
- ’ neoglycoprotein analogues of EPO employing one-pot native chemical ligation and CuAAC chemistry † (2019) (0)
- Synthesis of Indole Analogues of the anti‐Helicobacter pylori Compounds CJ‐13,015, CJ‐13,102, CJ‐13,104 and CJ‐13,108. (2007) (0)
- Synthesis and characterization of mono S-lipidated peptide hydrogels: a platform for the preparation of reactive oxygen species responsive materials. (2021) (0)
- (1R,6R,13R,18R)-(Z,Z)-1,18-Bis[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]-3,16-dimethylene-8,20-diazadispiro[5.6.5.6]tetracosa-7,19-diene (2010) (0)
- A Double Alkylation—Ring Closing Metathesis Approach to Spiroimines. (2004) (0)
- A randomised trial of dentric cell vaccination with NY-ESO-1 and alpha- galactosylceramide in patients with metastatic melanoma (ACTRN12612001101875) (2021) (0)
- [3S*,5S*,6S*]-1,7-Dioxaspiro[5.5]undecane-3,5-diyl Diacetate (1997) (0)
- The Kulinkovich Hydroxycyclopropanation Reaction in Natural Product Synthesis (2013) (0)
- Synthesis of the Bis‐spiroacetal C25—C40 Moiety of the Antimitotic Agent Spirastrellolide B Using a Bis‐dithiane Deprotection/Spiroacetalisation Sequence. (2010) (0)
- Editorial Advisory Board Members Progress in Heterocyclic Chemistry 2008-2009 (2009) (0)
- Total Synthesis of Spiroketal Alkaloids Lycibarbarines A-C. (2023) (0)
- Reductive Thioalkylation of a Pyranonaphthoquinone. (2000) (0)
- Frontispiece: seco ‐Labdanes: A Study of Terpenoid Structural Diversity Resulting from Biosynthetic C−C Bond Cleavage (2021) (0)
- Inside Back Cover: Total Synthesis and Conformational Study of Callyaerin A: Anti‐Tubercular Cyclic Peptide Bearing a Rare Rigidifying (Z)‐2,3‐ Diaminoacrylamide Moiety (Angew. Chem. Int. Ed. 14/2018) (2018) (0)
- Addition of 2-tert-Butyldimethylsilyloxythiophene to Activated Quinones: An Approach to Thia Analogues of Kalafungin. (2006) (0)
- A Flexible Approach to 6,5-Benzannulated Spiroketals. (2011) (0)
- Microsoft Word-Manuscript.docx (2013) (0)
- Buchwald—Hartwig Mono-N-Arylation with 2,6-Dihaloisonicotinic Acid Derivatives: A Convenient Desymmetrization Method. (2009) (0)
- Synthesis of an Actinorhodin Monomer. (1996) (0)
- A Tribute to Prof. Jim Coxon (2005) (0)
- Analogues de glycyl-prolyl-glutamate (2006) (0)
- Synthesis of Spirocyclic Imines: Key Pharmacophores in the Shellfish Toxins Spirolides and Gymnodimine. (2004) (0)
- Corrigendum to ‘Electrochemically-controlled grafting of hydrophilic brushes from conducting polymer substrates’ [Electrochimica Acta 188 (2016) 57–70] (2016) (0)
- [2R*,5S*,6S*]-2-Methyl-1,7-dioxaspiro[5.5]undec-3-en-5-ol§ (1997) (0)
- (±)-Cyclohexane-1,2-diyl bis(4-nitrobenzoate) (2008) (0)
- Mle-Phe-Mle-Phe. Linear precursor of pseudoxylallemycin A. (2019) (0)
- A Novel Approach toMonobenzannulated Spiroketals Using Styrenes in the KulinkovichReaction (2009) (0)
- Novel Use of N‐Carboalkoxy α,β‐Unsaturated Iminium Ions as Dienophiles in Diels—Alder Reactions. (2008) (0)
- Synthesis of Highly Substituted Pyranonaphthalene Spiroketals Related to the Griseusins Using a Hauser—Kraus Annulation Strategy. (2014) (0)
- Targeting synthetic glycopeptides to MGL on Dermal Dendritic cells (2011) (0)
- 1-(2-Vinyl-pyridin-3-yl)propanal O-methyloxime and 1-(6-Vinyl-pyridin-3-yl)propanal O-methyloxime (2001) (0)
- Thiol-ene enabled preparation of S-lipidated anti-HBV peptides. (2020) (0)
- A randomised controlled trial of long NY-ESO-1 peptide-pulsed autologous dendritic cells with or without alpha-galactosylceramide in high-risk melanoma. (2023) (0)
- Reductive Thioalkylation of a Kalafungin Analogue. (1998) (0)
- Synthesis of the Griseusin A Ring System. (1990) (0)
- Total Synthesis of Allene-Containing Cyclic Tetrapeptide Pseudoxylallemycin C (2020) (0)
- Synthesis of C‐2 Functionalized 1,6,8‐Trioxadispiro[4.1.5.3]pentadec‐13‐enes. (1998) (0)
- A Titanium Naphtholate Approach for the Synthesis of Analogues of Griseusin A. (2000) (0)
- Facile Bisarylation of Aldehydes Using Titanium Naphtholates. (1997) (0)
- Nitropyrrole Natural Products: Isolation, Biosynthesis and Total Synthesis (2016) (0)
- Rearrangement of a Furo(3,2‐b)naphtho(2,1‐d)furan to a Pyranonaphthoquinone. (1989) (0)
- 2-Trimethylsilyloxyfuran, CAS No: 61550-02- Update (2008) (0)
- The Synthesis of 5′-Deoxyjuglomycin A (Ia) and 5′-Methoxyjuglomycin A ( Ib). (1992) (0)
- Synthesis of the cis-3a,8b-Dihydrofuro(3,2-b)benzofuran-2(3H)-one Ring System via a Furofuran Annulation to Activated Benzoquinones. (1989) (0)
- MGL as a Target for Vaccine Design (2010) (0)
- Flow-Based Fmoc-SPPS Preparation and SAR Study of Cathelicidin-PY Reveals Selective Antimicrobial Activity (2023) (0)
- Synthesis of (.+‐.) Wine Lactone and Its Analogues by a Diels—Alder Approach. (2010) (0)
- Synthesis of N-Linked Glycopeptides Using Convergent Enzymatic Glycosylation Combined with SPPS (2018) (0)
- Synthesis of Cyclic Proline‐Containing Peptides via Ring‐Closing Metathesis. (2003) (0)
- Synthesis and Development of Seven-Membered Constrained Cyclic Urea Based PSMA Inhibitors Via RCM (2022) (0)
- Effects of a self-adjuvanting Synthetic Long Peptide targeting TLR2 on human immune cells (2010) (0)
- Stereoselective synthesis of the spirocyclic core of 13-desmethyl spirolide C using an aza-Claisen rearrangement and an exo-selective Diels-Alder cycloaddition. (2023) (0)
- Structure and dynamics of the human Nedd4-1 WW3* domain (2013) (0)
- Cover Feature: A Versatile Boc Solid Phase Synthesis of Daptomycin and Analogues Using Site Specific, On‐Resin Ozonolysis to Install the Kynurenine Residue (Chem. Eur. J. 62/2019) (2019) (0)
- Synthesis of Two Key Intermediates Required for the Construction of the Bis-spiroacetal Moiety of epi-17-Deoxy-(O-8)-salinomycin. (1986) (0)
- The First Enantioselective Total Synthesis of the anti‐Helicobacter pylori Agent (+)‐Spirolaxine Methyl Ether. (2005) (0)
- Rapid and simultaneous analysis of advanced glycation end products on silica hydride column: Comparison of ultraviolet, fluorescence, and mass spectrometry detectors (2020) (0)
- Synthesis of 2-Methylpyrrolo(1,2-a)pyrazin-1(2H)-one. (1989) (0)
- trans-2-(2-Naphthyl)-3-(phenylselenyl)tetrahydropyran (2002) (0)
- Highly Stereoselective syn‐Hydroxylation of Spiroacetals. (1992) (0)
- Uncatalyzed Addition of N‐(tert‐Butoxycarbonyl)‐2‐tert‐butyldimethylsilyloxypyrrole to Activated Quinones. (2002) (0)
- A Maillard Approach to 2‐Formylpyrroles: Synthesis of Magnolamide, Lobechine and Funebral. (2014) (0)
- Technology Advances for Vertebrate Pest Eradication (2020) (0)
- A Facile Synthesis of a Spironitrone and a Study of Its Cycloaddition and Nucleophilic Addition Reactions. (2009) (0)
- Global Trends in the Development of Rodenticides and Mammalian Pest Control Technologies (2018) (0)
- Addition of Silyloxydienes to 2-Substituted 1,4-Benzoquinones and 1,4- Naphthoquinones. (1997) (0)
- A Short Synthesis of Deoxyfrenolicin. (1994) (0)
- Professor Jim Coxon. A Tribute (2006) (0)
- Toxicodynamics of Methemoglobin (MtHb) Inducers (2010) (0)
- Diastereoselective Mannich-Based Synthesis of Piperidones (2009) (0)
- Spectral Assignments and Reference Data 1 Ha nd 13 C NMR data for C-6 substituted 3-azabicyclo(3.3.1)nonane-1-carboxylates (2006) (0)
- Formal Synthesis of the Juglomycins. (1995) (0)
- The Synthesis of Dehydrotryptophan and Dehydrotryptophan‐Containing Peptides. (2012) (0)
- STRUCTURE OF A BIS-SPIROACETAL, CIS-14-PHENYLSULFONYL-1,7,9-TRIOXADISPIRO[5.1.5.3]-HEXADECANE (1993) (0)
- Investigation into the racemic X-ray structure of the antimicrobial protein snakin-1 (2015) (0)
- (±)-N-(3-Hydroxy-1,2-diphenylpropyl)-4-methylbenzenesulfonamide (2008) (0)
- Synthesis of Analogues of Griseusin A. (2000) (0)
- Back Cover: On‐Resin Preparation of Allenamidyl Peptides: A Versatile Chemoselective Conjugation and Intramolecular Cyclisation Tool (Angew. Chem. Int. Ed. 41/2020) (2020) (0)
- Norbormide-Based Probes and Their Application for Mitochondrial Imaging in Drosophila Melanogaster. (2021) (0)
- Synthesis of 6,6-Bisbenzannulated Spiroketals Related to the Rubromycins Using a Double Intramolecular Hetero-Michael Addition (DIHMA). (2009) (0)
- The Chemistry of Bis-spiroactals. Synthesis of the Novel 1,7,9-Trioxadispiro(5.1.5.3)hexadecane Ring System. (1990) (0)
- Synthesis of Bis-2,5-Linked Tetrahydrofurans via Iodoetherification. (1996) (0)
- Gpe-analogues and peptidomimetics (2002) (0)
- The Synthesis of Oxygenated Naphthyl Stannanes Possessing ortho-Methoxy Substituents for Use in Stille Coupling Reactions. (1999) (0)
- Diels—Alder Addition of Acyclic Dienes to Chiral Naphthoquinones. (2001) (0)
- 1,4‐Addition of 2‐Trimethylsilyloxyfuran to Quinones: A Facile Route to the Furo(3,2‐b)benzofuran Nucleus. (1988) (0)
- Vesiculin derived from IGF-II drives increased islet cell mass in a mouse model of pre-diabetes (2021) (0)
- DETERMINATION OF THE STEREOCHEMISTRY OF 2,2-DIMETHYL-1,6,8-TRIOXADISPIRO(4.1.5.3)PENTADEC-13-ENE FORMED BY TWO SEQUENTIAL CYCLIZATION REACTIONS USING HIGH-FIELD PROTON NMR SPECTROSCOPY (1985) (0)
- Chemistry of Bis-spiroacetals. Synthesis of the 1,6,8-Trioxadispiro(4.1.5.3)pentadecane Ring System. (1988) (0)
- [4R*,5R*,6S*]-1,7-Dioxaspiro[5.5]undecane-4,5-diol (1997) (0)
- Chemoenzymatic Synthesis of Deoxy Analogues of the DNA Topoisomerase II Inhibitor Eleutherin and the 3C‐Protease Inhibitor Thysanone. (2008) (0)
- Effect of regio- and stereoisomerism on antifouling 2,5-diketopiperazines. (2022) (0)
- Synthesis of the Insect Feeding Deterrent Peramine (VIII) via Michael Addition of a Pyrrole Anion to a Nitroalkene. (1990) (0)
- Synthesis of a Functionalized Bisspiro Acetal. (1991) (0)
- Synthesis of Pyrrolo[3,2-b]benzofurans and Pyrrolo[3,2-b]naphthofurans via Addition of a Silyloxypyrrole to Activated Quinones. (2004) (0)
- Synthesis of 8‐Bromokalafungin as an Intermediate for the Preparation of C‐Glycoside Derivatives. (1997) (0)
- Allylic Functionalization of the 1,7-Dioxaspiro(5.5)undec-4-ene and 1, 6,8-Trioxadispiro(4.1.5.3)pentadec-13-ene Ring Systems. (1992) (0)
- Di‐(−)‐(1R,2S)‐2‐phenyl‐1‐cyclohexyl Diazenedicarboxylate (2002) (0)
- A Facile Cross‐Metathesis—Radical‐Cyclization Approach to Monobenzannulated Spiroketals. (2009) (0)
- Synthesis of Arylspiroketals Related to the Papulacandins via Generation of Phthalide Oxycarbenium Ions. (2001) (0)
- Azide-Enolate Cycloaddition-Rearrangement Enables Direct α-Amination of Amides and Enelactam Synthesis from Esters. (2023) (0)
- Synthesis of a spiroacetal intermediate for the synthesis of the anti- Helicobacter pylori agent CJ-12, 954 (2001) (0)
- Live applications of norbormide-based fluorescent probes in 2 Drosophila melanogaster 3 4 (2021) (0)
- The Effect of Glycosylation on the Potency of Pramlintide, An Anti-Diabetic Drug (2013) (0)
- A Facile Synthesis of 1,1′‐Spirobi(3H,3′H)isobenzofurans (2007) (0)
- Electrical conductivity of Self-assembling Peptide-semiconducting dye Conjugate nanofibre networks (2021) (0)
- Scalable Biomimetic Syntheses of Paeciloketal B, 1-epi-Paeciloketal B, and Bysspectin A. (2021) (0)
- (4R,2'R,3'R,5'R)-3-[5-(tert-Butyldimethylsilyloxy)-1-oxo-2,3-bis(phenylmethoxy)hexyl]-4-(phenylmethyl)-2-oxazolidinone (2000) (0)
- A Facile Synthesis of Aryldihydropyrans Using a Sonogashira—Selenoetherification Strategy. (2002) (0)
- Cover Picture: Synthesis of Chiral Tertiary Alcohols by CuI-Catalyzed Enantioselective Addition of Organomagnesium Reagents to Ketones / Emergence of the First Catalytic Oligonucleotides in a Formamide-Based Origin Scenario / Intermolecular Peptide Cross- (2016) (0)
- Enantioselective Synthesis of the Apple Aroma Constituent 1,3,3‐ Trimethyl‐2,7‐dioxabicyclo(2.2.1)heptane (III) via Asymmetric Dihydroxylation. (1996) (0)
- Titelbild: Radiation Damage and Racemic Protein Crystallography Reveal the Unique Structure of the GASA/Snakin Protein Superfamily (Angew. Chem. 28/2016) (2016) (0)
- Access to 2‐Alkyl Chromanones via a Conjugate Addition Approach. (2013) (0)
- The Chemical Synthesis of the Collagenous Domain of the Hormone Adiponectin (2011) (0)
- Stereocontrolled Synthesis of a Key Lactone Intermediate Required for the Synthesis of Salinomycin. (1990) (0)
- 1-(Pyridin-3-yl)-4-(triethylsilyloxy)-2-butyn-1-ol (2001) (0)
- Synthesis of trans- and cis-14-Phenylsulfonyl-1,7,9-trioxadispiro(5.1. 5.3)hexadecane. (1994) (0)
- Science of Synthesis, Volume 28: Compounds with Two Carbon-Heteroatom Bonds: Quinones and Heteroatom Analogues (2007) (0)
- Separation, characterisation and biological evaluation of the individual isomers of the rat selective toxicant norbormide – isolated using a chemical derivatization strategy (2021) (0)
- [4R*,5R*,6S*]-1,7-Dioxaspiro[5.5]undec-4,5-diyl Diacetate (1997) (0)
- Synthesis of Bicyclic Pyrazinones via Addition of Heterocyclic Amines to a Nitroalkene. (1994) (0)
- Racemic snakin-1 in P21/c (2016) (0)
- Synthesis of Benzannulated Spiroacetals Using Chiral Gold—Phosphine Complexes and Chiral Anions. (2014) (0)
- Quasi-racemic snakin-1 in P1 before radiation damage (2016) (0)
- 水中における還元糖からのグリコシルチオール類の無保護基合成;N‐グリカン糖複合体製造への応用 (2017) (0)
- Synthesis of the Novel 1,7,9-Trioxadispiro[4.1.5.2]-tetradecane Ring System Present in the Spirolides. (2001) (0)
- Chemistry of Bis‐spiroacetals: Synthesis of cis‐ and trans‐1‐(2‐Methyl‐ 1,6,8‐trioxadispiro(4.1.5.3)pentadec‐13‐en‐2‐yl)methanol. (1991) (0)
- cyclo-Mle-Phe-Mle-Phe. Pseudoxylallemycin A. (2019) (0)
- Synthesis and Reactivity of -Methoxymethyl Enecarbamates (2010) (0)
- Rücktitelbild: On‐Resin Preparation of Allenamidyl Peptides: A Versatile Chemoselective Conjugation and Intramolecular Cyclisation Tool (Angew. Chem. 41/2020) (2020) (0)
- On‐Resin Preparation of Allenamidyl Peptides: A Versatile Chemoselective Conjugation and Intramolecular Cyclisation Tool (2020) (0)
- ( )-1-{ 8 0-( tert-Butyldiphenylsilyloxy-methyl )-1 0 , 7 0-dioxaspiro [ 5 . 5 ] undecan-2 0-yl } uridine (2008) (0)
- Guanidinylated Amphiphilic Polycarbonates with Enhanced Antimicrobial Activity by Extending the Length of the Spacer Arm and Micelle Self‐Assembly (2020) (0)
- Use of Bis(oxazoline)-Metal Complexes as Chiral Catalysts for Asymmetric Diels—Alder Reactions Using 2-Acetyl-1,4-naphthoquinone as a Dienophile. (1998) (0)
- A Convenient Method for the Asymmetric Synthesis of Fluorinated α‐Amino Acids from Alcohols. (2014) (0)
- 1-(Pyridin-3-yl)but-2-yn-1,4-diol (2001) (0)
- A Convenient Method for the Asymmetric Synthesis of Fluorinated α‐Amino Acids from Alcohols (Eur. J. Org. Chem. 6/2014) (2014) (0)
- Equipment Access for Graduate Students - The First Hurdle (2007) (0)
- Synthesis and Bioactivity of Antitubercular Peptides and Peptidomimetics: An Update (2016) (0)
- Synthesis of Novel Nucleoside Analogues based on a Spiroacetal Framework (2003) (0)
- cis-2-(2-Methoxyphenyl)-3-(phenylselenyl)tetrahydropyran (2002) (0)
- Synthesis and Systematic Study on the Effect of Different PEG Units on Stability of PEGylated, Integrin-αvβ6-Specific A20FMDV2 Analogues in Rat Serum and Human Plasma (2022) (0)
- A synthetic study towards aryl 6,6-spiroacetal analogues of rubromycin (2008) (0)
- Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents (2023) (0)
- Weight loss after pregnancy is associated with reduced IGFBP-3 and increased cGP/IGF-1 ratio (2016) (0)
- A Double Mannich Approach to the Synthesis of Substituted Piperidones—Application to the Synthesis of Substituted E-Ring Analogues of Methyllycaconitine. (2011) (0)
- Application of Olefin Metathesis to the Synthesis of ABE Ring Analogues of Methyllycaconitine. (2002) (0)
- Synthesis of Spiroacetal‐Triazoles as Privileged Natural Product‐Like Scaffolds Using “Click Chemistry”. (2009) (0)
- Neuroprotective effects of diketopiperazines, potential clinical application of small cyclic form of neuropeptide following ischemic brain injury (2005) (0)
- Addition of Allylstannanes to an Oxy-Stabilized Carbenium Ion on a 1,7-Dioxaspiro[5.5]undecane Ring System. (1998) (0)
- Synthesis of Simple Analogues of Methyllycaconitine — An Efficient Method for the Preparation of the N-Substituted Anthranilate Pharmacophore. (2004) (0)
- [3R*,5S*,6S*]-5-Hydroxy-1,7-dioxaspiro[5.5]undec-3-yl 3,5-Dinitrobenzoate (1997) (0)
- Synthesis of Glycosylated 5‐Hydroxylsine, an Important Amino Acid Present in Collagen‐Like Proteins such as Adiponectin. (2012) (0)
- Thia-Michael addition: the route to promising opportunities for fast and cysteine-specific modification. (2023) (0)
- Alkylarsenic, -antimony, and -bismuth Compounds (2005) (0)
- Total Synthesis of Virgatolide B (I). (2014) (0)
- Synthesis of the C4-C16 Polyketide Fragment of Portimines A and B. (2021) (0)
- Synthetic Studies Towards the Calcium-Dependent Lipopeptide Antibiotic Cadaside B. (2022) (0)
- Synthesis of a New Spiroacetal Based Herbicide. (1997) (0)
- A Short Enantioselective Synthesis of the Topoisomerase II Inhibitor (+)‐Eleutherin. (2008) (0)
- Use of (S)-5-(2-Methylpyrrolidin-2-yl)-1H-tetrazole as a Novel and Enantioselective Organocatalyst for the Aldol Reaction. (2008) (0)
- Synthesis and Herbicidal Activity of [3R*,5S*,6S*]‐3‐Benzyloxy‐5‐methoxy‐1,7‐dioxaspiro[5.5]undecane and [3R*,5S*,6S*]‐3‐Methoxy‐5‐benzyloxy‐1,7‐dioxaspiro[5.5]undecane. (1998) (0)
- 3-[5-(tert-Butyldimethylsilyloxy)-3-(3,5-dinitrobenzoyl)-1-oxo- 2-(phenylmethoxy)hexyl]-4-(phenylmethyl)-2-oxazolidinone (2000) (0)
- Synthetic Studies Towards The Rubromycins (2003) (0)
- Factors influencing on-resin depsipeptide bond formation: case studies on daptomycin- and brevicidine-derived sequences. (2023) (0)
- Neuroprotection with Glycine-2-Methylproline-Glutamate (G-2MePE) after hypoxic-ischemic brain injury in adult rats (2014) (0)
- Synthesis of Enantiopure Bicyclic α,α-Disubstituted Spirolactams via Asymmetric Birch Reductive Alkylation. (2009) (0)
- Structure and dynamics of a human Nedd4 WW domain-ENaC complex (2013) (0)
- cyclo-Mle-Phe-Mle-D-Phe. D-Phe analogue of pseudoxylallemycin A. (2019) (0)
- Synthesis of Aromatic Spiroacetals Related to γ‐Rubromycin Based on a 3H‐Spiro[1‐benzofuran‐2,2′‐chroman] Skeleton. (2007) (0)
- Synthesis of the Monomeric Unit of γ-Actinorhodin. (1997) (0)
- Investigating the individual importance of the Pam2Cys ester motifs on TLR2 activity (2021) (0)
- Synthesis of the Cysteine Protease Inhibitors CPI-2081a and CPI-2081b Using a Controlled SPPS Byproduct Forming Reaction (2013) (0)
- Synthesis of a C-Glycosylpyranonaphthoquinone Related to Medermycin. (2000) (0)
- Dihydroxylation of 1,7‐Dioxaspiro(5.5)undec‐4‐enes. (1993) (0)
- Intermolecular Peptide Cross‐Linking by Using Diaminodicarboxylic Acids (2016) (0)
- Synthesis of the anti‐Helicobacter pylori Agent (+)‐Spirolaxine Methyl Ether (Ia) and the Unnatural (2′′S)‐Diastereomer (Ib). (2007) (0)
- Addition of a Grignard Reagent to Bis-spiroacetal Aldehydes: Appendage of a Tetrahydrofuran Ring. (2000) (0)
- 3-Allyl-2-hydroxy-5,6,8-trimethoxynaphthalene-1,4-dione (2008) (0)
- Synthesis of (±) Wine Lactone and Its Analogues by a Diels–Alder Approach (Eur. J. Org. Chem. 26/2009) (2009) (0)
- Synthesis of the Spiroacetal Core of the Cephalosporolide Family of Natural Products. (2014) (0)
- Synthesis of ABE Tricyclic Analogues (IX) of Methyllycaconitine Using a Wacker Oxidation—Aldol Strategy to Append the B Ring to the AE Fragment. (2002) (0)
- A Tribute to Don Cameron (2005) (0)
- IGF‐IIのIGF1Rへの結合を対象としたFRETベース研究のための蛍光IGF‐IIアナログ類 (2016) (0)
- Synthesis and Biological Evaluation of Termini-Modified and Cyclic Variants of the Connexin43 Inhibitor Peptide5 (2022) (0)
- Synthesis of the Bis‐spiroacetal Moiety of the Polyether Antibiotic CP44,161. (2001) (0)
- Enantioselective Synthesis of an Analogue of Nanaomycin A. (2008) (0)
- Diastereoselective Diels-Alder Reactions of Optically Active Vinyl Sulphoxides. (1986) (0)
- Studies Towards Development of Asymmetric Double‐Mannich Reactions of Chiral 2‐Oxocyclohexanecarboxylate Derivatives with Bis(aminol)ethers. (2015) (0)
- Synthetic Studies Towards Spirolaxine (2003) (0)
- Synthesis of a pyranonaphtoquinone-spiroacetal (1992) (0)
- Synthetic peptide analogs of neuronal regeneration (2008) (0)
- Diastereoselective Addition of 2‐Trimethylsilyloxyfuran to (S)‐(+)‐2‐( p‐Tolylsulfinyl)‐1,4‐benzoquinone. (1995) (0)
- Synthesis of (E)-1-Bromo-3-ethyl-3-pentene. (1996) (0)
- The Anti-Tubercular Aminolipopeptide Trichoderin A Displays Selective Toxicity against Human Pancreatic Ductal Adenocarcinoma Cells Cultured under Glucose Starvation (2023) (0)
- Synthesis and Ene Reactions of Di-(-)-menthyl Diazenedicarboxylate. (1996) (0)
- Isolation, Biological Activity and Synthesis of Benzannulated Spiroketal Natural Products (2010) (0)
- Mle-Phe-Mle-D-Phe. Linear tetrapeptide related to pseudoxylallemycin A. (2019) (0)
- 8′-Methoxy-3H-spiro[1-naphthofuran-2,2′-chroman] (2006) (0)
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