Philip Kocienski
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Organic chemist and Emeritus Professor at the University of Leeds
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Why Is Philip Kocienski Influential?
(Suggest an Edit or Addition)According to Wikipedia, Philip Joseph Kocienski is a British organic chemist. He is an Emeritus Professor at the University of Leeds. Research Kocienski has made contributions to the design and development of new organometallic reagents in synthesis, and the applications of synthetic methods to complex natural products. Early work with Basil Lythgoe on the scope and stereochemistry of the Julia olefination with alpha-metallated sulphone reagents emphasised the value of this method in organic chemistry. His major contribution has been to research the synthesis and chemistry of novel metallated enol ethers, and to develop the uses of these intermediates in the synthesis of oxacyclic and geometrically defined alkene units in natural products of biological significance. Kocienski has synthesised the insecticide milbemycin beta 3, the potassium channel blocker talaromycin B, the hypotensive agent lacrimin, and the antihypertensive agent zoapatanol. His total synthesis of the insect toxin pederin, and his synthetic work toward the immunosuppressant FK 506, have made him regarded as one of the leading organic chemists in the field.
Philip Kocienski's Published Works
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Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- A Stereoselective Synthesis of trans-1,2-Disubstituted Alkenes Based on the Condensation of Aldehydes with Metallated 1-Phenyl-1H-tetrazol-5-yl Sulfones (1998) (506)
- Protecting groups (1999) (233)
- Scope and stereochemistry of an olefin synthesis from β-hydroxysulphones (1978) (101)
- Pheromone synthesis. 4. A synthesis of (.+-.)-methyl n-tetradeca-trans-2,4,5-trienoate, an allenic ester produced by the male dried bean beetle Acanthoscelides obtectus (Say) (1977) (84)
- Synthetic applications of metallate rearrangements (1990) (80)
- A stereoselective synthesis of functionalized alkenyllithiums and alkenyl cyanocuprates by the copper(I)-catalyzed coupling of organolithium reagents with .alpha.-lithiated cyclic enol ethers (1989) (76)
- A synthesis of herboxidiene (1996) (75)
- Synthesis of salinomycin (1998) (68)
- Synthesis of (S)-(-)-N-acetylcolchinol using intramolecular biaryl oxidative coupling. (2006) (66)
- The influence of chain-branching on the steric outcome of some olefin-forming reactions (1980) (64)
- A total synthesis of (±)-zoapatanol and demethyl-ORF13811 (1989) (50)
- Synthesis of (+)-manoalide via a copper(I)-mediated 1,2-metalate rearrangement. (2003) (47)
- Recent Sulphone-Based Olefination Reactions (1985) (47)
- A New approach to 1,7-dioxaspiro[5.5]undec-4-enes via metallated allenol ethers. Synthesis of Lacrimin A (1990) (47)
- Enantiospecific syntheses of pseudopterosin aglycones. Part 2. Synthesis of pseudopterosin K–L aglycone and pseudopterosin A–F aglycone via a B→BA→BAC annulation strategy (2001) (45)
- Peptide synthesis and self-assembly. (2012) (45)
- Synthetic Approaches to Rapamycin: Synthesis of a C10-C26 Fragment via a One-Pot Julia Olefination Reaction (1996) (43)
- Synthesis of (–)-Tetrahydrolipstatin (1989) (41)
- A synthesis of the C(1)-C(15) segment of tsukubaenolide (FK 506). (1988) (41)
- The First Total Synthesis of (-)-Lipstatin (1995) (41)
- Studies related to the synthesis of pederin. Part 2. Synthesis of pederol dibenzoate and benzoylpedamide. (1990) (39)
- Phenylthiomethyltrimethylsilane : a new formyl anion synthon (1980) (39)
- A practical method for N-acylation of bornane-2,10-sultam and 2-oxazolidinones (1992) (38)
- The Modified Julia Olefination in Vitamin D2 Synthesis (1999) (37)
- Vapor-phase thermolyses of 3-hydroxy-1,5-hexadienes. II. Effects of methyl substitution (1967) (37)
- Pheromone synthesis. 6. A synthesis of (-)-.alpha.-multistriatin (1977) (37)
- Solid-phase synthesis of c(RGDfK) derivatives: on-resin cyclisation and lysine functionalisation. (2002) (36)
- The in vitro biological activities of synthetic 18-O-methyl mycalamide B, 10-epi-18-O-methyl mycalamide B and pederin. (1997) (35)
- The pederin family of antitumor agents: structures, synthesis and biological activity. (2000) (34)
- A highly stereoselective and iterative approach to isoprenoid chains: synthesis of homogeraniol, homofarnesol, and homogeranylgeraniol (1989) (34)
- A Synthesis of Jaspamide Based on 1,2-Metallate Rearrangements of α-Heteroalkenylmetal Derivatives (1995) (33)
- Studies related to the synthesis of (±)-pederin. part 1. Synthesis of ethyl pederate and benzoylselenopederic acid (1990) (33)
- A convenient preparation of some 2,3,4,6-tetra-O-acetyl-1,5-anhydro-d-hexitols (1982) (32)
- A synthetic approach to the pseudopterosins (1996) (31)
- A synthesis of (aR,7S)-(−)-N-acetylcolchinol and its conjugate with a cyclic RGD peptide (2008) (30)
- A synthesis of an ionomycin calcium complex. (2009) (30)
- Terminal olefins from the fluoride-induced elimination of β-silylsulfones (1979) (30)
- Synthetic studies on the pederin family of antitumour agents. Syntheses of mycalamide B, theopederin D and pederin (2000) (28)
- Silylketenes. A bird’s eye view (1998) (28)
- Peptide-Based Materials (2012) (28)
- The Preparation and Pd(0)-Catalysed Cross Coupling Reactions of α-(Phenylthio)alkenylzinc Reagents (1992) (28)
- A new synthesis of 1,7-dioxaspiro[5.5]undecanes. Application to a rectal gland secretion of the olive fruit fly (dacus oleae). (1983) (28)
- Palladium(0)-catalysed cross-coupling reactions of α-alkoxyalkenylstannanes and α-alkoxyalkenylzincs (1994) (27)
- A synthesis of (+)-pederin. The metallated dihydropyran approach. (1990) (27)
- A directed aldol approach to (+)-milbemycin β3 (1987) (26)
- Enantiospecific syntheses of pseudopterosin aglycones. Part 1. Synthesis of the putative aglycone of pseudopterosin G–J via an A→AB→ABC annulation strategy (2001) (26)
- The 3,4-dihydro-2H-pyran approach to (+)-milbemycin β3. Part 1. An alternative synthesis of (2S,4S,6R,8R,9S)-2-formylmethyl-4-(dimethyl-t-butylsilyloxy)-8,9-dimethyl-1,7-dioxaspiro[5.5]undecane (1987) (25)
- 3-(Trimethylsilyl)oxetan-2-ones via enantioselective [2 + 2] cycloaddition of (trimethylsilyl)ketene to aldehydes catalysed by methylaluminiomidazolines (1996) (25)
- A synthesis of zoapatanol (1988) (25)
- Two syntheses of manoalide via heteroatom-assisted alkyne carbometallation (1994) (25)
- A stereoselective synthesis of trisubstituted alkenes. Part 1. Nickel-catalysed coupling of Grignard reagents with 5-alkyl-2,3-dihydrofurans (1992) (24)
- Calciferol and its relatives. Part 24. A synthesis of vitamin D4 (1979) (24)
- A new synthesis of spiroacetals via alkylidenation of ester carbonyls with metal carbene complexes (1988) (23)
- A stereoselective synthesis of tri-substituted alkenes. The nickel-catalysed coupling of Grignard reagents with 6-alkyl-3,4-dihydro-2H-pyrans (1988) (23)
- A Synthesis of the Hypocholesterolemic Agent 1233A Via Asymmetric [2 + 2] Cycloaddition (1998) (23)
- Pheromone synthesis. 5. A synthesis of 3,7-dimethylpentadec-2-yl acetate. The sex pheromone of the pine sawfly Neodiprion lecontei (1977) (23)
- An efficient and stereoselective synthesisi of homoallylic alcohols via nickel-catalysed coupling of 5-alkyl-2,3-dihydrofurans with Grignard reagents (1987) (22)
- Peracid oxidation of cyclopropenes. Evidence for 2-oxabicyclo[1.1.0]butane intermediates (1969) (22)
- Pederin: The Metallated Dihydropyran Approach. Stereoselective Reduction ofN-AcylimidatesviaRhodium-Catalysed Hydroboration (1991) (22)
- A Synthesis of Oxolenes and Furans via Oxacyclopentylidene Chromium and Molybdenum Complexes (1996) (21)
- A synthesis of pseudo-gloeosporone (1987) (21)
- The β-lactone route to α, β-unsaturated δ-lactones. Total syntheses of (′)-goniothalamin and (-)-massoialactone (2004) (21)
- Calciferol and its relatives. Part 23. An alternative synthesis of Windaus and Grundmann's C19 ketone (1978) (19)
- A synthesis of 18-O-methyl mycalamide B (1996) (19)
- An Asymmetric Synthesis of (-)-Tetrahydrolipstatin (1994) (19)
- A stereoselective total synthesis of exo- and endo-brevicomin. (1976) (19)
- 1-tert-Butyl-1H-tetrazol-5-yl Sulfones in the Modified Julia Olefination (2000) (18)
- Facile synthesis of tert-butylacetylene (1974) (18)
- Synthetic approaches to pseudopterosin G aglycone dimethyl ether (1998) (18)
- A synthesis of (Z)-6-heneicosen-11-one. The sex pheromone of the Douglas fir tussock moth. (2002) (17)
- Synthesis of D-erythro-sphingosine and D-erythro-ceramide. (2002) (17)
- Silicon-mediated annulation. Part 1. A synthesis of tetrahydropyran-4-ones, oxepan-4-ones, and oxocan-4-ones via intramolecular directed aldol reactions (1985) (17)
- Asymmetric syntheses of panclicins A–E via [2+2] cycloaddition of alkyl(trimethylsilyl)ketenes to a β-silyloxyaldehyde (1998) (16)
- Unusual stereochemistry in the copper-catalysed ring opening of a carbohydrate oxirane with vinylmagnesium bromide (1984) (16)
- PHEROMONE SYNTHESIS. 3. A SYNTHESIS OF (E)-4,6-DIMETHYL-4-OCTEN-3-ONE (MANICONE) (1976) (16)
- A Synthesis of the C24-C34 Segment of FK 506 (1990) (16)
- Synthesis of manoalide using a 1,2-metallate rearrangement (1997) (16)
- Boron-Catalyzed N-Alkylation of Amines Using Carboxylic Acids (2015) (16)
- A Practical Synthesis of (R)-(+)-Cyclohex-3-enecarboxylic Acid via an Asymmetric Diels-Alder Reaction (1993) (15)
- A Synthesis of Mycalamide B (1998) (15)
- Stereoselective Synthesis of Homoallylic Alcohols by Migratory Insertion Reactions of Higher-Order Cyanocuprates and Nickel-Catalysed Coupling Reactions Involving Enol Carbamates (1989) (15)
- A Synthesis of Theopederin D and a Formal Synthesis of Pederin (1998) (14)
- The total synthesis of (±)-pederin (1987) (14)
- Palladium(0)-Catalysed Hydrostannylation of 1-Alkoxy-1-alkynes: A Synthesis of α-Alkoxyalkenylstannanes and Their Transmetallation to α-Alkoxyalkenyllithiums (1993) (14)
- A synthesis of moenocinol (1980) (14)
- An Economical Large Scale Preparation of (2S,3S)-4,5-Dimethyl-2-Phenyl-L,3-Dioxolan (1984) (14)
- The 3,4-dihydro-2H-pyran approach to (+)-milbemycin β3. Part 2. An improved synthesis of (2R,4S,6S,8R,9S)-2-[(5R)-(2E)-3-methyl-5-formyl-hex-2-en-1-yl]-8,9-dimethyl-4-(dimethyl-t-butylsilyloxy)-1,7-dioxaspiro[5.5]undecane (1987) (14)
- Isomerization of tri-tert-butylcyclopropenyl azide (1973) (14)
- Palladium(0)-Catalysed Stannylstannylation and Silylstannylation of 1-Alkoxy-1-alkynes and 1-Phenylthio-1-alkynes (1994) (13)
- Calciferol and its relatives. Part 27. A synthesis of 1 α-hydroxyvitamin D3 by way of 1 α-hydroxytachysterol3 (1980) (13)
- A synthesis of (+)-milbemycin β3. The directed aldol approach (1985) (13)
- Synthesis of the C1-C16 fragment of ionomycin using a neutral (eta3-allyl)iron complex. (2006) (13)
- A Method for the Synthesis of 6-(Trimethylstannyl)-3,4-dihydro-2H-pyrans from δ-Valerolactones (1991) (13)
- A synthetic approach to the C26-C32 fragment of rapamycin. A synthesis of allylic alcohols from allylic furylsilanes (1994) (13)
- Synthesis of phalluside-1 and Sch II using 1,2-metallate rearrangements. (2010) (13)
- A Synthesis of the Pseudopterosin A–F Aglycone (2012) (12)
- Observations on the scope of an intramolecular directed aldol condensation. A new synthesis of eight-membered rings (1983) (12)
- A stereoselective synthesis of the C(8)-C(20) fragment of premonensin B (1988) (12)
- A synthesis of 1,6-dioxaspiro[4.5]dec-3-enes. (1987) (12)
- Synthesis of 2,4,5-Trisubstituted Imidazoles (2017) (12)
- A synthetic approach to zoapatanol and related bicyclic analogues (1987) (12)
- Peroxy acid oxidation of cyclopropenes. Evidence for a dual pathway (1974) (12)
- Approaches to the 1,6,8-trioxadispiro[4.1.5.3]pentadec-13-en-15-ol ring system of salinomycin and related polyether antibiotics (1989) (12)
- Nucleophilic addition of α-metallated carbamates to planar chiral cationic η3-allylmolybdenum complexes: A stereochemical study (2004) (12)
- The hydrometallation, carbometallation, and metallometallation of heteroalkynes (1995) (12)
- Reaction of nitrimines with cyanide ions (1975) (12)
- A Synthesis of Salinomycin. Part 2. Synthesis of the Dispiroacetal Core Unit via Oxidative Rearrangement of an Acyl Furan (1994) (12)
- A Stereoselective Synthesis of trans‐1,2‐Disubstituted Alkenes Based on the Condensation of Aldehydes with Metallated 1‐Phenyl‐1H‐tetrazol‐5‐yl Sulfones. (1998) (11)
- A synthesis of (+)-milbemycin β3. The 3,4-dihydro-2H-pyran approach (1985) (11)
- A Synthesis of Salinomycin. Part 1. Synthesis of Key Fragments (1994) (11)
- The Preparation of 6-Bromo-3,4-dihydro-2H-pyrans from Tetrahydropyran-2-ones via a Ni(0)-catalysed Coupling Reaction and their Halogen-metal Exchange to 6-Lithio-3,4-dihydro-2H-pyrans. (2002) (10)
- A SYNTHESIS OF (3S*,4R*)-LUFFARIOLIDE (1995) (10)
- The Preparation of 1-Tributylstannyl Glycals from 1-Phenylsulfonyl Glycals via Ni(0)-Catalysed Coupling with Tributylstannylmagnesium Bromide (2001) (10)
- Synthetic approaches to pederin. A synthesis of pederol dibenzoate (1982) (10)
- A method for the chromatographic resolution of tetrahydropyran-2-ones (1991) (10)
- A stereoselective synthesis of trisubstituted alkenes. Part 2. The nickel-catalysed coupling of Grignard reagents with 6-alkyl-3,4-dihydro-2H-pyrans and acyclic enol ethers (1992) (10)
- A Highly Efficient Method of N-Methylation for the Amino Acid Derivatives (2010) (10)
- The nucleophilic addition of alpha-metallated 1,3-dioxanes to planar chiral cationic eta3-allylmolybdenum complexes. Synthesis of (2E,5S,6R,7E)-6-methyl-8-phenylocta-2,7-dienoic acid methyl ester, a key component of the Cryptophycins. (2004) (10)
- A new synthesis of 1,7-dioxaspiro[5.5]undec-4-enes via metallated allenol ethers. A formal synthesis of talaromycins A and B (1987) (10)
- Sulphone-based elimination reactions in synthesis. Part 1. Moenocinol (1983) (10)
- A new acetylene synthesis. Junipal (1976) (9)
- On the Julia Alkenylation Reaction in Vitamin D Synthesis. Isolation of Four Geometrical Isomers of Vitamin D4. (1999) (9)
- 1.1 Death, Taxes, and Protecting Groups (2005) (9)
- An approach to the synthesis of (–)-lipstatin by Wittig reaction and Lewis acid-promoted [2 + 2] cycloaddition (1993) (9)
- A synthesis of talaromycin B (1984) (9)
- 1,2-metallate rearrangements of α-alkoxyvinyl borates (1991) (9)
- The copper(I)-catalysed coupling of Grignard reagents with 5-lithio-2,3-dihydrofuran and 6-lithio-3,4-dihydro-2H-pyran (1991) (9)
- Rearrangement of allylic silylsulphonium ylides. A synthesis of βγ-unsaturated aldehydes (1980) (8)
- A Synthesis of Norbisabolide (1977) (8)
- Synthetic Approaches to Rapamycin. 3. Synthesis of a C1-C21 Fragment (1996) (8)
- A Synthesis of (3R*,4R*)-Luffariolide E via 1,2-Metallate Rearrangement (1995) (8)
- α-Heteroalkenyl Metallate Rearrangements in Organic Synthesis (1993) (8)
- New synthetic routes to spiroacetals. The 3,4-dihydro-2H-pyran approach to (±)-talaromycin B (1985) (7)
- A Formal Synthesis of 18-O-Methyl Mycalamide B (1999) (7)
- A 1,3-rearrangement of allylic sulphones caused by m-chloroperbenzoic acid and sodium hydrogen carbonate (1983) (7)
- Synthetic approaches to pederin. A synthesis of (±)-benzoylpedamide (1984) (7)
- The First Total Synthesis of (‐)‐Lipstatin. (1996) (7)
- New routes to 1α-hydroxyvitamin D3 (1980) (7)
- Allenol Ether Intermediates in the Synthesis of 1,7-Dioxaspiro[5.5]undec-4-enes and 1,6-Dioxaspiro[4.5]dec-3-enes (1991) (7)
- A synthesis of (-)-ebelactones A and B (2010) (6)
- Silicon-mediated annulation. Part 2. A synthesis of β-alkoxy cyclo-octanones via intramolecular directed aldol reactions (1985) (6)
- Copper(I)-Mediated 1,2-MetallateRearrangements of 1-Metallated Glycals (2012) (6)
- A synthesis of allylic alcohols from β-γ-epoxysulfones (1979) (6)
- Tri--butylcyclopropenyl azide. Degenerate isomerization (1972) (6)
- 1,2‐Metallate Rearrangement: (Z)‐4‐(2‐Propenyl)‐3‐Octen‐1‐ol (2003) (6)
- Synthesis and functionalisation of intermediates derived from allylmagnesiation of (E)-1-(trimethylsilyl)-but-1-en-3-ol (1989) (6)
- The Synthesis of Salinomycin (1997) (6)
- Synthetic approaches to pederin. A synthesis of ethyl pederate (1983) (6)
- Reductive Elimination, Vicinal Deoxygenation and Vicinal Desilylation (1991) (5)
- A Synthesis of α-Lithiated Enol Ethers from α-Arenesulfinyl Enol Ethers: Ni(0)- and Pd(0)-Catalysed Coupling of Enol Triflates and Phosphates Derived from Lactones with Sodium Arenethiolates Gives α-Arenesulfanyl Enol Ethers (2003) (5)
- A Synthesis of 1-Lithiated Glycalsand 1-Tributylstannyl Glycals from 1-Phenylsulfinyl Glycalsvia Sulfoxide-Lithium Ligand Exchange (2008) (5)
- Synthesis and Characterisation of a Doxorubicin-CNGRC Peptide Conjugate that Targets Tumour Vasculature (2002) (5)
- A Synthesis of (aR,7S)-(-)-N-Acetylcolchinol and Its Conjugate with a Cyclic RGD Peptide. (2008) (5)
- Synthesis of the C16-C23 Effector Domain of FK-506 via Copper-Catalysed Metallate Rearrangement of an α-Alkoxyalkenylcuprate (1995) (5)
- A synthesis of the C1-C9 fragment of ionomycin using cationic η3-allylicmolybdenum and -iron complexes (2005) (5)
- Conjugate addition of organolithium reagents to diphenylcyclopropenone (1969) (5)
- SYNTHETIC APPROACHES TO RAPAMYCIN. 2. A SYNTHESIS OF A C21-C42 FRAGMENT (1996) (5)
- Addition of Tri-O-benzyl-2-deoxy-d-glucosylcopper(I) to Cationic CpMo(NO)(CO)(5-methyl-2,3,4-η-hex-3-en-2-yl) Complexes. A New Approach to C-Glycosides (1998) (5)
- Synthetic applications of planar chiral cationic η3-allylmolybdenum complexes (2004) (4)
- 1-tert-Butyl-1H-tetrazol-5-yl Sulfones in the Modified Julia Olefination. (2000) (4)
- A synthesis of diumycinol (1983) (4)
- Three and one-half approaches to the synthesis of pederin (1991) (4)
- A synthesis of the spiroacetal moiety of milbemycin β3 (1984) (3)
- A Practical Method for N-Acylation of Bornane-2,10-sultam and 2- Oxazolidinones. (1992) (3)
- Synthesis Alerts 5/04 (2004) (3)
- A Synthesis of Mycalamide B. (1998) (3)
- 2-Benzothiazolyl Propargyl Sulfides:Versatile Precursors for Enantiopure Allenes, E-α,β-Unsaturated Ketonesand Z-Sulfonylalkenes (2010) (2)
- Preparation of a 1‐Alkoxy‐1‐Alkyne from Reaction of a 2,2,2‐Trifluoromethyl Ether with an Alkyllithium Reagent: 1‐Benzyloxymethoxy‐1‐Hexyne (2008) (2)
- An Approach to the Synthesis of Mycalamide B. Construction of the 2,4, 7-Trioxabicyclo(4.4.0)decane Ring System (XV). (1995) (2)
- Synthetic Approaches to Rapamycin: Synthesis of a C10‐C26 Fragment via a One‐Pot Julia Olefination Reaction. (1996) (2)
- Esterification. Methods, Reactions and Applications. By Junzo Otera. (2004) (2)
- Three and One‐Half Approaches to the Synthesis of Pederin (1992) (2)
- Synthesis Alerts 01/03 (2003) (2)
- Calciferol and its relatives. Part 26. A conversion of cholesterol into 8-hydroxymethyl-des-AB-cholest-8-ene. (1980) (2)
- A Synthesis of 6-Tributylstannyl-3,4-dihydro-2H-pyrans via Coupling of Enol Triflates with (Bu3Sn)(Bu)CuLi·LiCN (2002) (2)
- Synthesis Alerts 13/2001 (2001) (2)
- Synthesis of Raltegravir (2017) (2)
- Synthesis of PDE IVb Inhibitors (2012) (2)
- A Scalable Process for the Synthesis of 1,2-Dialkyldiselanes and 1-Alkaneselenols (2019) (2)
- Formal Synthesis of (–)-Huperzine A (2012) (2)
- Synthesis of Tafluprost (2020) (2)
- A SYNTHESIS OF (+)-HERBOXIDIENE A (1996) (2)
- Tri-tert-Butylcyclopropenyl Tetrafluoroborate (2003) (2)
- A Synthesis of Cryptophycin 4 Using a Planar Chiral Molybdenum Cationic Complex (2000) (2)
- Enantiospecific Syntheses of Pseudopterosin Aglycones. Part 1. Synthesis of the Putative Aglycone of Pseudopterosin G—J via an A→AB→ABC Annulation Strategy. (2002) (2)
- A Synthesis of Jaspamide Based on 1,2-Metallate Rearrangements of . alpha.-Heteroalkenylmetal Derivatives. (1995) (2)
- Synthesis of Efavirenz via Asymmetric Alkynylation (2018) (1)
- Synthesis Alerts 06/02 (2002) (1)
- A Stereoselective Synthesis of Trisubstituted Alkenes. The Nickel‐Catalyzed Coupling of Grignard Reagents with 6‐Alkyl‐3,4‐dihydro‐2H‐pyrans. (1988) (1)
- A Synthesis of Theopederin D and a Formal Synthesis of Pederin. (1999) (1)
- Synthesis of Dexamethasone (2020) (1)
- The Total Synthesis of (.+-.)-Pederin. (1987) (1)
- Aldolisation and Carboxylation Reactions from a-Silyl-b-lactams. A Combined Theoretical and Experimental Study (2008) (1)
- Synthesis of c-Met/ALK Inhibitor HS-10168 (2017) (1)
- cis-Mo(CO)4(Py)2: A Superior Reagent for the Preparation of η3-Allyl Molybdenum Complexes (2000) (1)
- Synthesis Alerts 02/98 (1998) (1)
- PIM Kinase Inhibitor (2021) (1)
- Synthesis of DPC 083 (2012) (1)
- Synthesis of Candesartan Cilexetil (2013) (1)
- Synthesis Alerts 09/01 (2001) (1)
- A synthesis of salinomycin. I: Synthesis of key fragments (1994) (1)
- Allenol Ether Intermediates in the Synthesis of 1,7‐Dioxaspiro(5.5) undec‐4‐enes and 1,6‐Dioxaspiro(4.5)dec‐3‐enes. (1992) (1)
- A Synthesis of 18‐O‐Methyl Mycalamide B. (1997) (1)
- A Synthesis of 1-Lithiated Glycals and 1-Tributylstannyl Glycals from 1-Phenylsulfinyl Glycals via Sulfoxide–Lithium Ligand Exchange 1-Tributylstannyl Glycals from 1-Phenylsulfinyl Glycals (2008) (1)
- Synthesis of PLK4 Inhibitor CFI-400945 (2015) (1)
- Synthesis Alerts 08/02 (2002) (1)
- Synthesis Alerts 07/02 (2002) (1)
- The Preparation of 1‐Tributylstannyl Glycals from 1‐Phenylsulfonyl Glycals via Ni(0)‐Catalyzed Coupling with Tributylstannylmagnesium Bromide. (2001) (1)
- Synthesis of Abamines (2012) (1)
- Mechanism of the oxidation of tropan-3.alpha.-ol with benzoyl chloride (1975) (1)
- Synthesis of Erlotinib (2015) (1)
- A Practical Synthesis of (R)-(+)-Cyclohex-3-enecarboxylic Acid via an Asymmetric Diels-Alder Reaction. (1993) (1)
- A Synthesis of (+)‐Milbemycin β3. The Directed Aldol Approach. (1986) (1)
- Synthesis of Bixafen (2012) (1)
- Synthesis of the C14-C28 Fragment of Tetronasin (2005) (1)
- Synthesis of an Aliskiren Intermediate (2012) (1)
- The β-Lactone Route to α,β-Unsaturated δ-Lactones. Total Syntheses of (.+-.)-Goniothalamin and (-)-Massoialactone. (2004) (1)
- Synthesis Alerts 01/98 (1998) (1)
- CALCIFEROL AND ITS RELATIVES. PART 26. A CONVERSION OF CHOLESTEROL INTO 8‐HYDROXYMETHYL‐DES‐AB‐CHOLEST‐8‐ENE (1980) (1)
- Asymmetric Synthesis of Efinaconazole and Albaconazole (2018) (1)
- Synthesis Alerts 03/97 (1997) (1)
- Synthesis Alerts 01/97 (1997) (1)
- Synthesis alerts 05/99 (1999) (1)
- Addition of Tri‐O‐benzyl‐2‐deoxy‐D‐glucosylcopper(I) to Cationic CpMo(NO)(CO)(5‐methyl‐2,3,4‐η‐hex‐3‐en‐2‐yl) Complexes. A New Approach to C‐Glycosides. (1998) (1)
- Palladium(0)-Catalyzed Cross-Coupling Reactions of α- Alkoxyalkenylstannanes and α-Alkoxyalkenylzincs. (1994) (1)
- Synthesis of AZD1656 (2018) (1)
- Approaches to the 1,6,8-Trioxadispiro(4.1.5.3)pentadec-13-en-15-ol Ring System of Salinomycin and Related Polyether Antibiotics. (1989) (1)
- Synthesis of Ziresovir (2019) (1)
- Synthesis of Filibuvir (2014) (1)
- Synthesis of Safingol (2014) (1)
- Synthesis of a DPP-4 Inhibitor (2020) (1)
- A Total Synthesis of (.+-.)-Zoapatanol and Demethyl-ORF13811. (1989) (1)
- Synthesis Alerts 04/03 (2003) (1)
- The 3,4-Dihydro-2H-pyran Approach to (+)-Milbemycin β3. Part 1. An Alternative Synthesis of (2S,4S,6R,8R,9S)-2-Formylmethyl-4-(dimethyl-t-butylsilyloxy)-8,9-dimethyl-1,7-dioxaspiro(5.5)undecane. (1988) (1)
- Synthesis of Daridorexant (2021) (1)
- A Synthesis of α‐Lithiated Enol Ethers from α‐Arenesulfinyl Enol Ethers: Ni(0)‐ and Pd(0)‐Catalyzed Coupling of Enol Triflates and Phosphates Derived from Lactones with Sodium Arenethiolates Gives α‐Arenesulfanyl Enol Ethers. (2003) (1)
- Synthesis of the Four Stereoisomers of Mefloquine (2014) (1)
- Propargyl-Linked Antifolates Overcome Resistance in S. aureus (2015) (1)
- Synthesis of Methopholine (2012) (1)
- Synthesis of a Dipeptidyl Peptidase-4 Inhibitor (2014) (1)
- Synthesis Alerts 05/98 (1998) (1)
- The Copper(I)‐Catalyzed Coupling of Grignard Reagents with 5‐Lithio‐2, 3‐dihydrofuran and 6‐Lithio‐3,4‐dihydro‐2H‐pyran. (1992) (1)
- Synthesis alerts 02/99 (1999) (1)
- Studies Related to the Synthesis of (.+-.)-Pederin. Part 1. Synthesis of Ethyl Pederate and Benzoylselenopederic Acid. (1990) (1)
- A NEW SYNTHESIS OF 1,7-DIOXASPIRO(5.5)UNDECANES. APPLICATION TO A RECTAL GLAND SECRETION OF THE OLIVE FRUIT FLY (DACUS OLEAE) (1984) (1)
- Pederin: The Metalated Dihydropyran Approach. Stereoselective Reduction of N‐Acylimidates via Rhodium‐Catalyzed Hydroboration. (2010) (1)
- Nanomolar Inhibitor of Trypanosoma brucei Trypanothione Reductase (2019) (1)
- A Formal Synthesis of IonomycinFeaturing a Permanganate-Mediated Oxidative Cyclisation (2011) (1)
- Synthesis of (+)-erythro-Mefloquine Hydrochloride (2012) (1)
- A Synthesis of Salinomycin. Part 1. Synthesis of Key Fragments. (1995) (1)
- Synthesis of Letermovir by an Asymmetric Aza-Michael Reaction (2016) (1)
- Synthesis of Cefiderocol (2018) (1)
- Absolute configuration of exo‐syn‐syn‐dicarbonyl(η5‐cyclopentadienyl)[(1,2,3‐η)‐(1R,2S,3S)‐1‐phenylbut‐2‐en‐1‐yl]molybdenum(II). Erratum (2000) (1)
- Synthesis of Epigenetic Regulator I-BET762 (GSK525762) (2014) (1)
- Synthesis Alerts 15/01 (2001) (1)
- 1,2-Metallate Rearrangements of α-Alkoxyalkyl Cuprates (2004) (1)
- Synthesis of BMS-191011 (2015) (0)
- Synthesis of (R)-(–)-Nifenalol (2012) (0)
- 4.7 Esters (2005) (0)
- Synthesis of Sergliflozin Analogues (2013) (0)
- Synthesis of (S)-(+)-Ibuprofen via Enantioselective Hydrocyanation (2013) (0)
- Synthesis of a Histone Deacetylase Inhibitor (2012) (0)
- Synthesis of MK-8150 (2019) (0)
- Syntheis of Entecavir (2012) (0)
- Synthesis of MK-6186 (2012) (0)
- Synthesis of a 5-Lipoxygenase Activating Protein (FLAP) Inhibitor (2017) (0)
- Synthesis of GSK1265744 (2015) (0)
- Synthesis of a Renin Inhibitor (2019) (0)
- Synthesis of AZD7594 (2019) (0)
- Conductively Heated Sealed-Vessel Reactor: Synthesis of Olanzapine (2017) (0)
- 8.9 Special Cases (2005) (0)
- A Short Synthesis of Molnupiravir (2020) (0)
- Synthesis of AG-270 (2021) (0)
- Synthesis of an IGF-1R Modulator (2012) (0)
- Synthesis of Thrombin Inhibitor AZD8165 (2014) (0)
- Synthesis of Parsaclisib (2020) (0)
- Synthesis of OV329 (2018) (0)
- Synthesis of Amino-Carbasugars (2017) (0)
- A Synthesis of (3R*,4R*)‐Luffariolide E via 1,2‐Metallate Rearrangement. (1995) (0)
- Asymmetric Synthesis of an AZD7594 Intermediate Using Flow Catalysis (2017) (0)
- Synthesis of SNX-5422 (2013) (0)
- Flow Synthesis of Lomustine (2019) (0)
- Synthesis of GDC-0022 (2020) (0)
- Synthesis of an Inhibitor of Histone Lysine Demethylases KDM2/7 (2018) (0)
- From 2-Phenyl-2,3-dihydrofuran or 3-Phenylisoxazole (2002) (0)
- Synthesis of the CGRP Receptor Antagonist BMS-846372 (2012) (0)
- Synthesis of GDC-0310 (2020) (0)
- Synthesis of Lanraplenib (2020) (0)
- Continuous Cryogenic Lithium–Halogen Exchange (2020) (0)
- Synthesis of a Glucosylceramide Synthase Inhibitor (2012) (0)
- Synthesis of TP-2758 (2016) (0)
- Continuous Process for the Preparation of Thiazoles (2018) (0)
- Synthesis of Vortioxetine via Catalyst-Free N-Arylation (2017) (0)
- Synthesis of PF-06873600 (2021) (0)
- Synthesis of a MAP Kinase Inhibitor (2013) (0)
- Synthesis of Mevidalen (2020) (0)
- α-Arylation of Malonate Derivatives via Oxidative Catalysis (2017) (0)
- A Method for the Synthesis of 6‐(Trimethylstannyl)‐3,4‐dihydro‐2H‐ pyrans from δ‐Valerolactones. (1991) (0)
- Synthesis of PPARα Agonist GW641597X (2020) (0)
- Synthesis of Piragliatin (2012) (0)
- Synthesis Alerts 12/97 (1997) (0)
- Asymmetric Synthesis of an 11β-HSD-1 Inhibitor (2017) (0)
- Synthesis of Gefapixant (2021) (0)
- Synthesis of a Mineralocorticoid Antagonist (2013) (0)
- Synthesis Alerts 12/99 (1999) (0)
- A Synthetic Route to the Tripeptide Unit of Geodiamolide-B. (1998) (0)
- Synthesis of Zanamivir (2012) (0)
- Synthesis of Pevonedistat (2015) (0)
- Synthesis Alerts 03/98 (1998) (0)
- Synthesis of a Dual Leucine Zipper Kinase Inhibitor (2018) (0)
- Synthesis of Gefitinib (2019) (0)
- Synthesis Alerts 1/02 (2004) (0)
- Synthesis of PF-06835919 (2021) (0)
- Synthesis of CC-90011 (2021) (0)
- Synthesis of SIPI 6398 (2019) (0)
- Synthesis of Renin Inhibitor DS-8108b (2014) (0)
- Enantioselective Synthesis of Efavirenz (2017) (0)
- Synthesis of the Indoleamine 2,3-Dioxygenase Inhibitor Linrodostat (2020) (0)
- Synthesis of (1R,3S)-HPA-12 (2013) (0)
- Synthesis of Remdesivir (2020) (0)
- Synthesis of 1′,2′-Methano-2′,3′-dideoxynucleosides (2019) (0)
- Synthesis of the Tricyclic Core of BMS-986251 (2021) (0)
- Synthesis of Giredestrant (2021) (0)
- Synthesis Alerts 06/98 (1998) (0)
- Synthesis of Brensocatib (AZD7986) (2021) (0)
- Synthesis of Solabegron (2015) (0)
- Synthesis Alerts 05/00 (2000) (0)
- Synthesis of Axelopran (2020) (0)
- Synthesis of a Non-Nucleoside Reverse Transcriptase Inhibitor (2012) (0)
- Synthesis of BAY1217224 (2021) (0)
- 6.7 Reviews (2005) (0)
- Synthesis of SN-38 (2012) (0)
- Synthesis of β-Lactamase Inhibitor Relebactam (2020) (0)
- Stereoselective Synthesis of Trisubstituted Alkenes. Part 2. Nickel- Catalyzed Coupling of Grignard Reagents with 6-Alkyl-3,4-dihydro-2H- pyrans and Acyclic Enol Ethers. (1993) (0)
- Synthesis (S)-RO4999200 (2015) (0)
- Synthesis of a Moxifloxacin Fragment (2019) (0)
- Synthesis of KAE609 via an Asymmetric aza-Diels–Alder Reaction (2015) (0)
- Development of a Commercial Synthesis of BMS-663068 (2017) (0)
- Synthesis of AZD8931 (Sapatinib) (2017) (0)
- Phase Separation Macrocyclization in the Synthesis of Vaniprevir (2017) (0)
- 8.2 Imides and Amides (2005) (0)
- Synthesis of a trans-Cyclopropoxy Building Block for Grazoprevir (2018) (0)
- Synthesis of the CHK1 Inhibitor MK-8776 (2016) (0)
- Synthesis of Tulrampator (2019) (0)
- Synthesis of Esketamine (2019) (0)
- Synthesis of AZD6738 (2019) (0)
- Synthesis of Efinaconazole (2014) (0)
- Absolute configuration of exo-syn-syn-dicarbonyl(eta(5)-cyclopentadienyl)[(1,2,3-eta)-(1R,2S,3S)-1-phenylbut-2-en-1-yl]molybdenum(II). Erratum. (2000) (0)
- Synthesis of (S)-Duloxetine (2012) (0)
- Aldolization and Carboxylation Reactions from α‐Silyl‐β‐lactams. A Combined Theoretical and Experimental Study. (2009) (0)
- A vinylic α-carbamoyloxy boran with a carbenoid-type bonding situation (2002) (0)
- Synthesis of Telmisartan (2015) (0)
- Synthesis Alerts 10/99 (1999) (0)
- Synthesis of HIV Integrase Inhibitor MK-1376 (2020) (0)
- 7.1 Introduction (2005) (0)
- Synthesis of PSI-6130, the Nucleoside Core of Sofosbuvir (2014) (0)
- Synthesis of pan-JAK Inhibitor PF-06263276 (2019) (0)
- Rovafovir Etalafenamide (Part III): Synthesis of the Phosphonamidate Fragment (2021) (0)
- Synthesis of Rucaparib (2020) (0)
- Synthesis of Axitinib (2014) (0)
- Synthesis of Rivaroxaban (2016) (0)
- Synthesis of 5-Fluoro-1,3-oxazine β-Secretase Inhibitors (2018) (0)
- CALCIFEROL AND ITS RELATIVES. PART 27. A SYNTHESIS OF 1α-HYDROXYVITAMIN N D3 BY WAY OF 1α-HYDROXYTACHYSTEROL3 (1980) (0)
- Asymmetric Synthesis of an Imidazoline Proteasome Modulator (2020) (0)
- Synthesis of an MDM2 Antagonist (2013) (0)
- Silylketenes. A Bird′s Eye View (1998) (0)
- Synthesis of KAE609 by Catalytic Asymmetric Alkynylation (2016) (0)
- Synthesis of Entecavir (2018) (0)
- Synthesis of a CXCR7 Modulator (2018) (0)
- Synthesis of ATX Inhibitor Ziritaxestat (2020) (0)
- Synthesis of BMS-986251 (2020) (0)
- Synthesis of IPI-926 (2016) (0)
- Synthesis of Atorvastatin via NHC-Catalyzed Three-Component Coupling (2017) (0)
- Synthesis of MIDD0301 (2020) (0)
- Formal Synthesis of Clopidogrel (Plavix®) (2013) (0)
- A Synthesis of Herboxidiene. (2010) (0)
- Synthesis Alerts 07/98 (1998) (0)
- Synthesis of MK-5172 (2013) (0)
- Synthesis of BMS-986097 (2017) (0)
- Synthesis of PF-04191834 (2016) (0)
- Synthesis of Histone Acetyltransferase Inhibitor A-485 (2018) (0)
- Synthesis of Silodosin (2015) (0)
- Flow Synthesis of 3-(Mesitylthio)-1H-1,2,4-triazole (2019) (0)
- Chemoenzymatic Synthesis of a Rosuvastatin Building Block (2015) (0)
- Synthesis of an Arginase Inhibitor (2020) (0)
- Synthesis of BRD3914 via Directed C(sp3)–H Arylation (2017) (0)
- Synthesis of an Akt Kinase Inhibitor (2012) (0)
- Synthesis of an HIV-1 Integrase Allosteric Site Inhibitor (2019) (0)
- Synthesis alerts 06/99 (1999) (0)
- Synthesis of Fosdevirine (2018) (0)
- 4.8 Carbonates (2005) (0)
- Commercial Manufacture of Halaven® (2013) (0)
- Synthesis of Indolactam V (2016) (0)
- Synthesis of Flecainide (2017) (0)
- Synthesis of XL228 (2013) (0)
- Formal Synthesis of (R)-Flurbiprofen (2013) (0)
- Metal (Copper or Rhodium) Catalysis (2002) (0)
- Formal Synthesis of Atorvastatin (2015) (0)
- 4.6 Methylthiomethyl (MTM) Ethers (2005) (0)
- Synthesis of (3R,3aS,6aR)-Hexahydrofuro-[2,3-b]furan-3-ol (2017) (0)
- Formal Synthesis of Telmisartan (2021) (0)
- Synthesis of Benzo[g]indazole CK2 Inhibitors (2012) (0)
- 2.1 Introduction (2005) (0)
- Synthesis of Abrocitinib (2021) (0)
- Synthesis of a c-Kit Kinase Inhibitor Using Organocatalysis (2014) (0)
- Synthesis of MK-8742 (2014) (0)
- Synthesis of ELND007 (2013) (0)
- Synthesis Alerts 04/99 (1999) (0)
- Synthesis of JAK3 Covalent Inhibitor PF-06651600 (2019) (0)
- Synthesis of Lorlatinib (2018) (0)
- (2‐Phenylsulfonylethyl)trimethylsilane (2001) (0)
- Synthesis of Dolutegravir (2019) (0)
- Synthesis of a Fungicidal Pyrimidine Derivative (2019) (0)
- Synthesis of Remdesivir (GS-5734) — A Candidate for the Treatment of Ebola and COVID-19 Infections (2020) (0)
- Synthesis of Tofogliflozin (2016) (0)
- Synthesis Alerts 11/03 (2003) (0)
- Synthesis of BPR1K871 (2021) (0)
- Synthesis Alerts 07/97 (1997) (0)
- Synthesis of a Remdesivir Intermediate (2020) (0)
- Synthesis of a GDC-0994 Intermediate by Kumada–Corriu Cross-Coupling (2017) (0)
- Synthesis of Lonafarnib (2012) (0)
- Synthesis of Emitasvir (2021) (0)
- Synthesis Alerts 04/97 (1997) (0)
- Synthesis of SMO Inhibitor PF-04449913 (2014) (0)
- Synthesis of Glecaprevir. Part 1 (2020) (0)
- Synthesis of Islatravir (2020) (0)
- Synthesis of BACE1 Inhibitor LY3202626 (2020) (0)
- 6.6 Silyl Esters (2005) (0)
- Synthesis Alerts 13/04 (2004) (0)
- Synthesis of (S)-Naproxen (2012) (0)
- A 1,3-REARRANGEMENT OF ALLYLIC SULFONES CAUSED BY M-CHLOROPERBENZOIC ACID AND SODIUM HYDROGEN CARBONATE (1983) (0)
- Synthesis of BMS-986260 (2020) (0)
- 4.3 Alkyl Ethers (II) (2005) (0)
- Synthesis of MET Kinase Inhibitor LY2801653 (2014) (0)
- Gram-Scale Synthesis of Dolutegravir Sodium (2021) (0)
- Synthesis of a Glucokinase Activator (2019) (0)
- Route to Remdesivir’s Nucleobase via N-Amination of 2-Cyanopyrrole (2020) (0)
- Rovafovir Etalafenamide (Part IV): Synthesis of the Fluorinated Nucleoside Fragment (2021) (0)
- Asymmetric Synthesis of Chloramphenicol and Related Amphenicol Antibiotics (2021) (0)
- Continuous Flow Synthesis of Eflornithine (2018) (0)
- Synthesis Alerts 18/04 (2004) (0)
- Synthesis of an Isocitrate Dehydrogenase 1 Inhibitor (2018) (0)
- Synthesis of an αVβ6 Antagonist (2016) (0)
- Synthesis of MK-2947 (2020) (0)
- Synthesis of Doxercalciferol (2012) (0)
- Synthesis of a Bruton’s Tyrosine Kinase Inhibitor (2021) (0)
- Synthesis of an HIV-1 Protease Inhibitor (2017) (0)
- Synthesis of AZD7624 (2021) (0)
- Synthesis of HCV Protease Inhibitor MK-6325 (2015) (0)
- Synthesis of MK-7622 (2018) (0)
- Synthesis of (+)-VNI (2013) (0)
- 5.1 Introduction (2005) (0)
- Synthesis of a CCR4 Antagonist (2019) (0)
- Synthesis of AZD9742 (2020) (0)
- Synthesis of BMS-986094 (2019) (0)
- Synthesis of AMG 510 (2020) (0)
- Synthesis of EFdA via Enzymatic Desymmetrization (2017) (0)
- Synthesis of DPC 083 (2013) (0)
- PHENYLTHIOMETHYLTRIMETHYLSILANE: A NEW FORMYL ANION SYNTHON (1980) (0)
- Flow Synthesis of Ciprofloxacin (2019) (0)
- Synthesis of GK–GKRP Disruptor AMG-3969 (2014) (0)
- Synthesis of Ulimorelin (2012) (0)
- Synthesis of a TAK-480 Fragment (2019) (0)
- Synthesis of AMG 925 (2015) (0)
- CALCIFEROL AND ITS RELATIVES. PART 23. AN ALTERNATIVE SYNTHESIS OF WINDAUS AND GRUNDMANN′S C19 KETONE (1978) (0)
- Synthesis of HIV-1 Entry Inhibitor BNM-III-170 (2020) (0)
- Asymmetric Synthesis of AZD8186 (2021) (0)
- Synthesis of a Retinoic Acid Receptor Agonist (2013) (0)
- Synthesis of BMS-986104 (2017) (0)
- Synthesis of GSK3036656 (2018) (0)
- Automated Titration of Organometallic Reagents in Continuous Flow (2019) (0)
- Synthesis of BAY 1161116 (2021) (0)
- Synthesis of Dual Orexin Receptor Antagonist MK-6096 (2015) (0)
- Synthesis of LpxC Inhibitor LP-058 (2016) (0)
- Synthesis of Vismodegib through meta-Selective Nitration of Arenes (2016) (0)
- Synthesis of Olodanrigan (2020) (0)
- Oxidation of Csp3–H Bonds in Flow Using Methyl(trifluoromethyl)dioxirane (2019) (0)
- 5.5 Reviews (2005) (0)
- Synthesis of Doravirine (2015) (0)
- Synthesis of AMG 232 (2019) (0)
- Synthesis Alerts 07/99 (1999) (0)
- Synthesis of BACE1 Inhibitor PF-06751979 (2021) (0)
- Synthesis of JNJ-67569762 (2021) (0)
- Synthesis of (–)-Huperzine A (2012) (0)
- Synthesis Alerts 05/97 (1997) (0)
- Synthesis of a Glucosylceramide Inhibitor (2015) (0)
- Synthesis of the Hydroxyquinolinone Core of β2-Receptor Agonists (2015) (0)
- Synthesis of Pyrido[2,3-b]indoles Targeting DNA Gyrase and Topisomerase IV (2021) (0)
- Synthesis of a BACE1 Inhibitor (2013) (0)
- Synthesis of PF-06372865 (2019) (0)
- Synthesis of ABBV-168 (2019) (0)
- Thermolysis of (Alkoxyethynyl)silanes (1,5-Hydrogen Transfer) (2002) (0)
- Synthesis of Tofogliflozin (2019) (0)
- Synthesis of a TRPV3 Antagonist (2017) (0)
- Synthesis of a Bcl-2 Antagonist (2020) (0)
- Formal Synthesis of (R)-Silodosin (2021) (0)
- Synthesis of a HCV NS5B Nucleoside Polymerase Inhibitor (2019) (0)
- Synthesis of Darunavir (2016) (0)
- Synthesis of GDC-0810 (2018) (0)
- Synthesis of rac-Efavirenz (2015) (0)
- Synthesis of Zanamivir Phosphonate Congeners (2012) (0)
- Synthesis of NVP-HSP990 (2015) (0)
- Synthesis of an Allosteric HIV-1 Integrase Inhibitor (2020) (0)
- Synthesis of a MCH1 Receptor Antagonist (2016) (0)
- Synthesis of Tenofovir (2020) (0)
- Formal Synthesis of Rosuvastatin and Pitavastatin (2014) (0)
- Synthesis of BMS-986158 (2021) (0)
- Two Syntheses of Manoalide via Heteroatom-Assisted Alkyne Carbometalation. (1994) (0)
- Diastereoselective Synthesis of TAK-828F (2021) (0)
- Enantiospecific Syntheses of Pseudopterosin Aglycones. Part 2. Synthesis of Pseudopterosin K—L Aglycone and Pseudopterosin A—F Aglycone via a B→BA→BAC Annulation Strategy. (2002) (0)
- Synthesis of the C16-C23 Effector Domain of FK-506 via Copper- Catalyzed Metallate Rearrangement of an α-Alkoxyalkenylcuprate. (1995) (0)
- Synthesis of MK-8831 (2016) (0)
- Synthesis of Simurosertib (TAK-931) (2020) (0)
- Synthesis of GLPG2938 (2021) (0)
- Synthesis of (+)-Sertraline (2012) (0)
- Copper(I)‐Mediated 1,2‐Metallate Rearrangements of 1‐Metallated Glycals. (2012) (0)
- Synthesis of Belvarafenib (2021) (0)
- 8.6 N-Alkyl Derivatives (2005) (0)
- Synthesis of a Noradrenaline Reuptake Inhibitor (2018) (0)
- 8.3 Carbamates (II) (2005) (0)
- Synthesis of a CETP Inhibitor (2014) (0)
- The Pederin Family of Antitumor Agents: Structures, Synthesis and Biological Activity (2001) (0)
- Synthesis of a Precursor to LY2140023 (2012) (0)
- Synthesis of BI 201302 (2013) (0)
- Synthesis of (Z)-Tamoxifen (2012) (0)
- A Synthesis of (+)-Milbemycin B3. The 3,4-Dihydro-2H-pyran Approach. (1986) (0)
- Synthesis of Sisunatovir (2021) (0)
- Synthesis of a BACE1 Inhibitor (2013) (0)
- Synthesis of CD73 Inhibitor AB680 (2020) (0)
- Synthesis of Aliskiren (2016) (0)
- Synthesis of Codeine (2016) (0)
- Synthesis of Phalluside-1 and Sch II (2010) (0)
- Synthesis of Antibacterial LpxC Inhibitors (2019) (0)
- Synthesis of GDC-5338 (2020) (0)
- Synthesis of Entecavir (BMS-200475) (2012) (0)
- Synthesis of Crizotinib and Etoricoxib (2019) (0)
- Synthesis of PF-00951966 (2012) (0)
- Formal Synthesis of Beraprost (2012) (0)
- Synthesis of an Androgen Receptor Antagonist (2017) (0)
- Flow Synthesis of Vaborbactam (2019) (0)
- Synthesis of Chemokine Receptor Antagonist NIBR-1282 (2014) (0)
- Synthesis of Olopatidine Hydrochloride (2012) (0)
- Synthesis of BMS-986144 (2021) (0)
- Synthesis of an Indoleamine-2,3-dioxygenase-1 Inhibitor (2019) (0)
- Synthesis of (+)-Sertraline (2012) (0)
- Synthesis of Atorvastatin Calcium (2014) (0)
- Synthesis of DPP-4 Inhibitor Omarigliptin (2014) (0)
- Synthesis Alerts 04/98 (1998) (0)
- Synthesis of a PCSK9 Inhibitor (2018) (0)
- Synthesis of Evacetrapib (2014) (0)
- Synthesis of an Atropisomeric HIV Integrase Inhibitor (2017) (0)
- Synthesis of a SYK Inhibitor (2015) (0)
- Synthesis of (R)-Lisophylline (2015) (0)
- Synthesis of GDC-0339 (2019) (0)
- UNUSUAL STEREOCHEMISTRY IN THE COPPER-CATALYZED RING OPENING OF A CARBOHYDRATE OXIRANE WITH VINYLMAGNESIUM BROMIDE (1984) (0)
- Synthesis of an HCV Protease Inhibitor (2015) (0)
- Synthesis of Quetiapine via Cobalt-Catalyzed C–H Thiolation (2018) (0)
- Synthesis of Oseltamivir Phosphate (2018) (0)
- Synthesis of an HCV Replicase Inhibitor (2014) (0)
- Synthesis of AZD6906 (2012) (0)
- Synthesis Alerts 12/00 (2000) (0)
- Synthesis of Pibrentasvir (2018) (0)
- Synthesis Alerts 08/00 (2000) (0)
- Synthesis of a Tyrosinase Inhibitor (2017) (0)
- 3.6 N,O-Acetals for the Protection of 1,2- and 1,3-Amino Alcohols (2005) (0)
- Synthesis of Esketamine (2019) (0)
- Synthesis of a VLA-4 Antagonist via Electrochemical C–H Amination (2013) (0)
- Synthesis of an EGFR T790M Inhibitor (2019) (0)
- Synthesis Alerts 10/97 (1997) (0)
- Synthesis of Doravirine (2016) (0)
- Synthesis Alerts 5/05 (2005) (0)
- Synthesis of ABT-341 (2017) (0)
- Synthesis of GSK2981278A (2019) (0)
- Synthesis of BAY 1214784 (2020) (0)
- Synthesis of Ipatasertib (2015) (0)
- Manufacturing Route to Avibactam (2017) (0)
- Asymmetric Transfer Hydrogenation in the Synthesis of Lorlatinib (2017) (0)
- Synthesis of the β-Lactamase Inhibitor MK-7655 (2014) (0)
- Synthesis of Brensocatib (2020) (0)
- Synthesis of AZD1981 (2013) (0)
- Synthesis of an Estrogen Receptor Beta Agonist (2014) (0)
- A Formal Synthesis of Atorvastatin (2014) (0)
- Synthesis of (+)-BMS-820836 (2016) (0)
- Synthesis of Verubecestat (2018) (0)
- Synthesis of Taniborbactam (2020) (0)
- Synthesis of the Pyrrolidine Core of ABBV-3221 (2020) (0)
- Synthesis of Remdesivir via Diastereoselective Organocatalyzed Phosphoramidation (2021) (0)
- Stereoselective Synthesis of Homoallylic Alcohols by Migratory Insertion Reactions of Higher-Order Cyanocuprates and Nickel-Catalyzed Coupling Reactions Involving Enol Carbamates. (1990) (0)
- Synthesis of Eliglustat (2019) (0)
- 4.4 Alkoxymethyl Ethers (II) (2005) (0)
- Synthesis Alerts 06/00 (2000) (0)
- Asymmetric Synthesis of a DPP-4 Inhibitor (2015) (0)
- Synthesis of Pitavastatin (2018) (0)
- Stille Cross-Coupling Route to HIV NNRTI Doravirine Analogues (2017) (0)
- Synthesis of a Histamine-3 Receptor Antagonist (2014) (0)
- Synthesis of Manoalide Using a 1,2‐Metallate Rearrangement. (1997) (0)
- Synthesis of A-1331852 (2020) (0)
- Synthesis of BMS-919373 (2019) (0)
- Synthesis of PF-06826647 (2021) (0)
- 7.2 The Reaction of Phosphate Esters with Nucleophiles (2005) (0)
- Synthesis of AM-8553 (2012) (0)
- Synthesis of a Hepatitis C Replication Inhibitor (2014) (0)
- Synthesis of Cinacalcet by Asymmetric Hydroamination (2015) (0)
- Synthesis of a TORC 1/2 Inhibitor (2013) (0)
- Silicon-mediated Annulation. Part 2. A Synthesis of β-Alkoxy Cyclo-octanones via Intramolecular Directed Aldol Reactions. (1986) (0)
- Synthesis of Icenticaftor (2021) (0)
- Synthesis of Florfenicol (2012) (0)
- Synthesis of K777 (2016) (0)
- Synthesis of Lamivudine (2020) (0)
- Synthesis of Lamivudine (2021) (0)
- Synthesis of a Dual NK-1/Serotonin Receptor Antagonist (2013) (0)
- 8.4 Sulfonyl Derivatives (2005) (0)
- Synthesis of TAK-828F (2020) (0)
- Synthesis of a BACE1 Inhibitor (2021) (0)
- Synthesis of AM-1638 (2012) (0)
- Synthesis of MK-8718 (2016) (0)
- Synthesis of MK-7246 (2012) (0)
- Synthesis of Dasabuvir (2019) (0)
- Improved Process for 5′-O-(4,4′-Dimethoxytrityl)-N 2-isobutyryl-2′-O-(2-methoxyethyl)guanosine (2021) (0)
- Synthesis of HIV-1 Protease Inhibitors (2018) (0)
- Synthesis of (+)-Oxo-tomaymycin (2020) (0)
- Synthesis of an Inhibitor of Influenza Virus Replication (2016) (0)
- A Synthesis of Cryptophycin 4 Using a Planar Chiral Molybdenum Cationic Complex. (2000) (0)
- Synthesis of Nelfinavir (2018) (0)
- Synthesis of a Dipeptidyl Peptidase-4 Inhibitor (2019) (0)
- Synthesis Alerts 4/02 (2002) (0)
- 1,2‐Metallate Rearrangements of α‐Alkoxyvinyl Borates. (1992) (0)
- Synthesis of a PDE4 Inhibitor by C–H Activation (2016) (0)
- Synthesis of Halauxifen Methyl (2019) (0)
- Synthesis of Taselisib (2019) (0)
- Synthesis of LY426965 (2018) (0)
- Synthesis Alerts 04/01 (2001) (0)
- 8.5 N-Sulfenyl Derivatives (2005) (0)
- Synthesis of M-525 (2018) (0)
- Synthesis of a TRPV1 Antagonist (2014) (0)
- 1.5 Mutual Protection (2005) (0)
- Synthesis of PF-06409577 (2018) (0)
- Synthesis of BMS-911543 (2019) (0)
- Synthesis of a Janus Kinase Inhibitor (2020) (0)
- Synthesis of Aliskiren (2015) (0)
- Synthesis of a PDE IVb Inhibitor (2012) (0)
- Synthesis of Atorvastatin (2015) (0)
- Synthesis Alerts 18/02 (2002) (0)
- Synthesis of a TRPV1 Antagonist (2014) (0)
- Synthesis of a Bruton’s Tyrosine Kinase Inhibitor (2018) (0)
- Stereoselective Synthesis of Trisubstituted Alkenes. Part 1. Nickel- Catalyzed Coupling of Grignard Reagents with 5-Alkyl-2,3-dihydrofurans. (1993) (0)
- REARRANGEMENT OF ALLYLIC SILYLSULFONIUM YLIDES (1981) (0)
- Synthesis of Roblitinib (2021) (0)
- Synthesis of PF-04995274 (2016) (0)
- Synthesis of Palbociclib (2016) (0)
- Synthesis of Runcaciguat (2021) (0)
- 1.9 Reviews (2005) (0)
- Synthesis of Imagabalin Hydrochloride (2012) (0)
- Synthesis of Vismodegib (2016) (0)
- Synthesis of Reldesemtiv (2021) (0)
- Second-Generation Synthesis of Sulopenem (2012) (0)
- Synthesis Alerts 2/02 (2004) (0)
- Synthesis of (R)-JM 1232 by Asymmetric Alkynylation (2016) (0)
- Synthesis of E2508 (2012) (0)
- Synthesis of (+)-Asenapine (2016) (0)
- 3.2 O,O-Acetals (II) (2005) (0)
- Synthesis Alerts 11/00 (2000) (0)
- Synthesis of Heterobiaryls by Contractive C–C Coupling (2019) (0)
- Synthesis of Ceralasertib (2021) (0)
- Synthesis of Vericiguat (2017) (0)
- Synthesis of GDC-0077 (2019) (0)
- Synthesis of (R)-Rasagiline via Dynamic Kinetic Resolution (2015) (0)
- Synthesis of GNE-293 (2013) (0)
- Synthesis of MK-8876 (2016) (0)
- Synthesis of a Glycine Transporter 1 Inhibitor (2012) (0)
- 5.2 Thioether Derivatives (2005) (0)
- Synthesis Alerts 10/98 (1998) (0)
- Synthesis of Epacadostat (2017) (0)
- Synthesis of Ecopipam (2012) (0)
- 8.7 N-Silyl Derivatives (2005) (0)
- Synthesis of All Four Reboxetine Stereoisomers (2013) (0)
- NEW SYNTHETIC ROUTES TO SPIROACETALS. THE 3,4-DIHYDRO-2H-PYRAN APPROACH TO (.+-.)-TALAROMYCIN B (1985) (0)
- Synthesis of Combretastatin A-4 (2013) (0)
- Synthesis alerts 01/99 (1999) (0)
- Synthesis of Sotorasib (2021) (0)
- Synthesis of Mevidalen (2021) (0)
- Synthesis Alerts 10/01 (2004) (0)
- Synthesis of Tesirine (2018) (0)
- 2-Benzothiazolyl Propargyl Sulfides: Versatile Precursors for Enantiopure Allenes, E-α,β-Unsaturated Ketones and Z-Sulfonylalkenes. (2011) (0)
- Synthesis of (+)- and (–)-Perhexiline (2016) (0)
- Synthesis of Fosdevirine (2018) (0)
- A Synthesis of 6-Tributylstannyl-3,4-dihydro-2H-pyrans via Coupling of Enol Triflates with (Bu3Sn)(Bu)CuLi×LiCN. (2002) (0)
- 3‐(Trimethylsilyl)oxetan‐2‐ones via Enantioselective (2 + 2) Cycloaddition of (Trimethylsilyl)ketene to Aldehydes Catalyzed by Methylaluminoimidazolines. (1996) (0)
- Synthesis Alerts 02/01 (2001) (0)
- Synthesis of Thiazesim (2012) (0)
- Synthesis of (R)-Lacosamide (2016) (0)
- Synthesis of a Matrix Metalloproteinase Inhibitor (2015) (0)
- Organocatalytic Synthesis of Enantiopure 2H- and 3H-Pyrroles (2016) (0)
- Synthesis Alerts 16/01 (2004) (0)
- Synthesis of GDC-0326 (2021) (0)
- Synthesis of Acrivastine (2012) (0)
- Synthesis of a Glucokinase Activator (2013) (0)
- Synthesis of VPC01091 (2017) (0)
- Synthesis of BMS-986236 (2019) (0)
- Synthesis of TNO155 (2021) (0)
- Synthesis of Bruton’s Tyrosine Kinase Inhibitor GDC-0852 (2020) (0)
- Synthesis of Methyl- and Dimethyl-3,5-dinitropyridines via Dephosphonylation of Diethyl Pyridinephosphonates (1975) (0)
- Synthesis of Rovafovir Etalafenamide (2021) (0)
- Continuous Process for Manufacturing 5-Bromo-N-(tert-butyl)pyridine-3-sulfonamide (2019) (0)
- Synthesis of (S)-Sitagliptin (2014) (0)
- Synthesis of E2212 (2019) (0)
- Synthesis of Omarigliptin (2016) (0)
- 2.6 Cyanohydrins (2005) (0)
- Synthesis of a Tetracyclic Indolenine that Represses β-Lactam Resistance (2015) (0)
- Synthesis of BMS-932481 (2018) (0)
- Synthesis of Dihydroorotate Dehydrogenase Inhibitor BRD9185 (2017) (0)
- Synthesis Alerts 6/01 (2001) (0)
- Synthesis of LSZ102 (2020) (0)
- One-Step Synthesis of 2-Fluoroadenine in a Continuous Flow Operation (2019) (0)
- Synthesis Alerts 08/97 (1997) (0)
- Synthesis of Shld (2018) (0)
- Scalable Stereoselective Synthesis of BMT-297376 (2021) (0)
- 4.9 Reviews (2005) (0)
- An Approach to the Synthesis of (-)-Lipstatin by Wittig Reaction and Lewis Acid Promoted (2 + 2) Cycloaddition. (1993) (0)
- Synthesis of Acetyl-CoA Carboxylase Inhibitors (2013) (0)
- Synthesis of Paroxetine (2014) (0)
- STEREOSELECTIVE TOTAL SYNTHESIS OF EXO- AND ENDO-BREVICOMIN (1976) (0)
- Synthesis of BMS-741672 (2017) (0)
- Synthesis of (R)-Ruxolitinib (2015) (0)
- Synthesis of an Inhibitor of Human Arginases I and II (2013) (0)
- Asymmetric Cyclopropanation Using Engineered Myoglobin Catalysts (2017) (0)
- Synthesis of Citalopram (2016) (0)
- Synthesis of Grazoprevir (2019) (0)
- Synthesis Alerts 17/04 (2004) (0)
- Synthesis of MK-7655 (2012) (0)
- Synthesis of Sonidegib Using Palladium Catalysis in Water (2020) (0)
- Synthesis of a TRPV1 Antagonist (2014) (0)
- Synthesis of Pemigatinib (2021) (0)
- Synthesis of PF-06751979 (2018) (0)
- Pyrazolocarboxamide Inhibitors of Receptor Interacting Protein 2 Kinase (2020) (0)
- 6.2 General Comments on the Esterification of Carboxylic Acids (2005) (0)
- Synthesis of Ezetimibe (2013) (0)
- Synthesis of a BACE1 Inhibitor (2016) (0)
- A Synthesis of 1,6-Dioxaspiro(4.5)dec-3-enes. (1988) (0)
- Synthesis of Zoliflodacin (2020) (0)
- Synthesis Alerts 08/99 (1999) (0)
- Synthesis of (R)-Ramatroban (2012) (0)
- Synthesis of Molnupiravir from Uridine (2021) (0)
- Synthesis of Ubrogepant (2018) (0)
- Synthesis of Dapagliflozin (2019) (0)
- Synthesis of Birinapant (2016) (0)
- Synthesis of an Allosteric Inhibitor of the Mutant GTPase KRASG12C (2020) (0)
- SULFONE-BASED ELIMINATION REACTIONS IN SYNTHESIS. PART 1. MOENOCINOL (1983) (0)
- Synthesis of Glecaprevir. Part 2 (2020) (0)
- Synthesis of Latanoprost (2018) (0)
- Synthesis of DS79932728 (2021) (0)
- Synthesis of a Bile Acid Transporter Inhibitor (2014) (0)
- Synthesis of Olopatadine (2012) (0)
- Synthesis of Akt Inhibitor GDC-0068 (2013) (0)
- Synthesis of Ertugliflozin (2014) (0)
- The β-Lactone Route to β-Hydroxy or α,β-Unsaturated γ- and δ-Lactones. Syntheses of ()-Massoialactone and ()-Prelactone B (2002) (0)
- Synthesis Alerts 11/02 (2002) (0)
- Synthesis of M-89 (2019) (0)
- Synthesis of A-315675 (2012) (0)
- Synthesis of MK-6096 (2013) (0)
- PEROXY ACID OXIDATION OF CYCLOPROPENES, EVIDENCE FOR A DUAL PATHWAY (1974) (0)
- Synthesis of GDC-0908 (2019) (0)
- Synthesis of GPR40 Agonist AM-4668 (2014) (0)
- Synthesis of AZD9833 (2021) (0)
- Synthesis of a Phosphodiesterase 1 Inhibitor (2020) (0)
- Synthesis of Alogliptin (2021) (0)
- Synthesis of AMG 337 (2016) (0)
- Synthesis of a RORγt Inverse Agonist (2020) (0)
- Synthesis of JAK2 Inhibitor BMS-911543 (2015) (0)
- Synthesis of β-Lactamase Inhibitor ETX0282 (2021) (0)
- Synthesis of HCV Protease Inhibitor MK-1220 (2014) (0)
- Preface to the New Edition (2018) (0)
- 1.8 Protecting Groups and Solid-Phase Synthesis (2005) (0)
- Synthesis of the Bicyclic Darunavir Side Chain (2017) (0)
- Synthesis of a Bruton’s Tyrosine Kinase Inhibitor (2014) (0)
- Synthesis of Alisertib (2015) (0)
- Synthesis of a JAK1 Inhibitor (2012) (0)
- Synthesis of Anti-Malarial MMV390048 (2021) (0)
- 3.7 Reviews (2005) (0)
- Synthesis of Dactolisib (2019) (0)
- Synthesis of Verubecestat (2018) (0)
- Synthesis of the Glucocorticoid Agonist BI 653048 BS H3PO4 (2013) (0)
- A Claisen Approach to 4′-Ed4T (2015) (0)
- Synthesis of a Key Intermediate in the Manufacture of Tetracyclines (2016) (0)
- Synthesis of AMG 837 (2013) (0)
- Synthesis of Bosutinib (2016) (0)
- Synthesis of a Phosphoinositide 3-Kinase (PI3K) β Inhibitor (2018) (0)
- Formal Synthesis of Entecavir (2019) (0)
- Synthesis Alerts 03/00 (2000) (0)
- Synthesis of BMS-960 (2017) (0)
- Synthesis of CY6463 (2021) (0)
- Synthesis of Δ12-Prostaglandin J3 (2018) (0)
- Synthesis of PF-3635659 (2012) (0)
- Synthesis of MK-8282 (2018) (0)
- Synthesis Alerts 08/98 (1998) (0)
- Synthesis of Vernakalant (2014) (0)
- Synthesis of NS5B Polymerase Inhibitor GSK852A (2016) (0)
- Synthesis of LY411575 (2012) (0)
- Synthesis of a Key Subunit of HIV-1 Protease Inhibitor Darunavir (2021) (0)
- Synthesis of (–)-Oseltamivir (2014) (0)
- 6.4 Alkoxyalkyl Esters (2005) (0)
- 5.4 Disulfides as Protecting Groups and Targets (2005) (0)
- Synthesis of NVP-CGM097 (2015) (0)
- Synthesis of Marbostat-100 (2018) (0)
- C–H Arylation of Heterocyclic N-Oxides: Application to SB222200 (2016) (0)
- Synthesis of Omecamtiv Mecarbil (2012) (0)
- Synthesis of Eldecalcitol (2021) (0)
- 6.5 Esters Cleaved by β-Elimination Reactions (2005) (0)
- Synthesis of an MK2 Inhibitor (2018) (0)
- Synthesis of an HCV NS5B RNA Polymerase Inhibitor (2019) (0)
- Synthesis of Clinprost (2013) (0)
- Synthesis of an Indoleamine-2,3-Dioxygenase-1 Inhibitor (2019) (0)
- Synthesis Alerts 16/02 (2002) (0)
- Synthesis of Macrocyclic Protease Inhibitors (2014) (0)
- Synthesis of ERK1/2 Inhibitor AZD0364 (2020) (0)
- Synthesis of BMS-986143 (2021) (0)
- Synthesis of a BACE 1 Inhibitor (2019) (0)
- Synthesis of Oxadiazole-Based S1P1 Receptor Agonists (2013) (0)
- PHEROMONE SYNTHESIS. 6. A SYNTHESIS OF (-)-α-MULTISTRIATIN (1978) (0)
- Synthesis of Sofosbuvir (2018) (0)
- Synthesis of Nisoxetine (2017) (0)
- Synthesis of MRTX849 (2020) (0)
- Synthesis of YLF466D (2021) (0)
- Asymmetric Synthsis of (S)-Verapamil (2020) (0)
- Synthesis of an FXI (Factor XI) Inhibitor (2021) (0)
- 3.4 Silylene Derivatives (2005) (0)
- Synthesis of Tryptophan Hydroxylase Inhibitor LX1031 (2020) (0)
- Synthesis Alerts 02/00 (2000) (0)
- Synthesis of Verubecestat (2017) (0)
- Synthesis of Imatinib (2019) (0)
- 2.9 Reviews (2005) (0)
- Synthesis of GDC-0575 (2018) (0)
- Asymmetric Synthesis of Beraprost (2017) (0)
- Synthesis of URB597 (2013) (0)
- Synthesis of ABBC-2222 (2019) (0)
- Synthesis of a CGRP Receptor Antagonist (2016) (0)
- Synthesis of a Chemokine Receptor Antagonist (2015) (0)
- Synthesis of (S)-Baclofen (2016) (0)
- A Synthetic Approach to the Pseudopterosins. (1996) (0)
- Synthesis of P2X7 Receptor Antagonist Lu AF27139 (2021) (0)
- Synthesis of Allosteric Inhibitor BMS-986165 (2019) (0)
- Synthesis of UK-432,097 (2012) (0)
- Synthesis Alerts 12/98 (1998) (0)
- Enantioselective Sulfa-Michael Reactions (2017) (0)
- Synthesis of BRD7/9 Bromodomain Inhibitor LP99 (2015) (0)
- Synthesis of BI 201420 (2020) (0)
- Synthesis of BMS-741672 (2017) (0)
- A Directed Aldol Approach to (+)-Milbemycin β3. (1988) (0)
- Synthesis and Functionalization of Intermediates Derived from Allylmagnesiation of E-1-(Trimethylsilyl)but-3-en-1-ol. (1990) (0)
- Synthesis of MK-5204 (2020) (0)
- Synthesis of GS-9669 (2014) (0)
- Synthesis of β-Lactamase Inhibitor QPX7728 (2020) (0)
- Synthesis of LY2784544 (2012) (0)
- Thermolysis or Photolysis of Cyclobutenediones or Cyclobutenones (2002) (0)
- Industrial Production of Artemisinin (2014) (0)
- Scalable Synthesis of ELQ-300 (2021) (0)
- Synthesis of Delgocitinib (2020) (0)
- Synthesis of an HIV-1 Protease Inhibitor (2017) (0)
- Synthesis of Esomeprazole (2018) (0)
- Synthesis of Delgocitinib (2020) (0)
- Synthesis of Axitinib (2015) (0)
- Synthesis of Indolo-Phakellins (2015) (0)
- Synthesis of Silanediol FXIa Inhibitors (2018) (0)
- Synthesis of Zotatifin (2020) (0)
- Synthesis of γ-Secretase Modulator SPI-1865 (2014) (0)
- 1.7 Protecting Groups As Not-So-Innocent Bystanders (2005) (0)
- 1.4 Transprotection (2005) (0)
- Synthesis of PF-06650833 (2019) (0)
- Synthesis of GSK8175 (2019) (0)
- Synthesis of Taniborbactam (VNRX-5133) (2020) (0)
- Palladium(0)-Catalyzed Hydrostannylation of 1-Alkoxy-1-alkynes: A Synthesis of α-Alkoxyalkenylstannanes and Their Transmetalation to α-Alkoxyalkenyllithiums. (1994) (0)
- Synthesis Alerts 02/97 (1997) (0)
- Synthesis of Pictilisib (2013) (0)
- Stereospecific Amination Using Sodium Azide in Continuous Flow (2020) (0)
- Synthesis of an MDM2 Inhibitor (2013) (0)
- Synthesis of a Diacylglycerol Acyltransferase-1 (DGAT-1) Inhibitor (2015) (0)
- Synthesis of an Indoleamine-2,3-dioxygenase-1 (IDO1) Inhibitor (2020) (0)
- Synthesis of Triple Reuptake Inhibitor (1R,2S)-SIPI 5357 (2013) (0)
- Synthesis of (R)-Rolipram (2013) (0)
- Wolff–Kishner Reductions Using a Silicon Carbide Flow Reactor (2020) (0)
- Synthesis of TAK-733 (2013) (0)
- An Efficient and Stereoselective Synthesis of Homoallylic Alcohols via Nickel-Catalyzed Coupling of 5-Alkyl-2,3-dihydrofurans with Grignard Reagents. (1987) (0)
- Synthesis of (R)-(–)-Thiazesim (2016) (0)
- Synthesis of (–)-Oseltamivir (2014) (0)
- Synthesis of PARP1–DNA Trapper AZD5305 (2021) (0)
- A Method for the Chromatographic Resolution of Tetrahydropyran‐2‐ones. (1992) (0)
- Synthesis of ACT-280778 (2015) (0)
- Synthesis of IDX320 (2013) (0)
- Synthesis Alerts 06/97 (1997) (0)
- A Synthesis of Salinomycin. Part 2. Synthesis of the Dispiroacetal Core Unit via Oxidative Rearrangement of an Acyl Furan. (1995) (0)
- Synthesis of DNA Gyrase Inhibitor (2015) (0)
- Synthesis Alerts 17/03 (2003) (0)
- 5.3 Thiocarbonate Derivatives (2005) (0)
- Synthesis of Balovaptan (2020) (0)
- Synthesis of AS-3201 (Ranirestat) (2016) (0)
- Synthesis of Sonepiprazole by an Asymmetric Oxa-Michael Reaction (2015) (0)
- Synthesis of Cebranopadol (2020) (0)
- Synthesis of TEV-37440 (2017) (0)
- Synthesis of the GSK3β Inhibitor AZD8926 (2013) (0)
- Synthesis of Reverse Transcriptase Inhibitor Tenofovir (2015) (0)
- Streamlined Synthesis of Fevipiprant (2021) (0)
- Synthesis of Talazoparib (2016) (0)
- Synthesis of a Baloxavir Marboxil Fragment (2020) (0)
- Synthesis of an Inhibitor of Blood Coagulation Factor VIIa–Tissue Factor Complex (2016) (0)
- Synthesis Alerts 12/04 (2004) (0)
- Synthesis of a Glucocorticoid Receptor Modulator (2016) (0)
- A Refined ProTide Route to Uprifosbuvir (2021) (0)
- Synthesis of (–)-Cannabidiol (2020) (0)
- Synthesis Alerts 02/03 (2003) (0)
- Synthesis of MK-4256 (2012) (0)
- Synthesis of an Edoxaban Fragment (2019) (0)
- Synthesis of UCB-108770 via a Povarov Cycloaddition (2020) (0)
- Synthesis of Both Enantiomers of Mequitazine (2014) (0)
- Flow Production of Anhydrous tert-Butyl Hydroperoxide (2019) (0)
- Synthesis of Nemiralisib (2021) (0)
- Synthesis of Largazole (2018) (0)
- Synthesis Alerts 05/03 (2003) (0)
- Synthesis of a BACE1 Inhibitor (2012) (0)
- Synthesis of (S)-Duloxetine (2017) (0)
- Synthesis of Ciprofloxacin Hydrochloride in Continuous Flow (2017) (0)
- Synthesis of Abacavir by Enantioselective Hydroamination (2017) (0)
- Synthesis of a BACE1 Inhibitor (2015) (0)
- Synthesis of SGLT2 Inhibitor Canagliflozin (2015) (0)
- Synthesis of a Renin Inhibitor (2015) (0)
- 6.3 Methyl Esters and Derivatives (II) (2005) (0)
- Synthesis of Nafoxidine via Copper-Catalyzed Carboarylation (2013) (0)
- Synthesis of a Serotonin Norepinephrine Reuptake Inhibitor (2013) (0)
- Synthesis of BMS-906024 via Oxidative Enolate Coupling (2016) (0)
- Synthesis of Perampanel (2013) (0)
- Synthesis of OZ439 (2015) (0)
- Synthesis of an ORL-1 Antagonist (2016) (0)
- Synthesis of MK-0893 (2012) (0)
- Synthesis Alerts 12/96 (1996) (0)
- Synthesis of Oxolenes and Furans via Oxacyclopentylidene Chromium and Molybdenum Complexes. (1996) (0)
- Synthesis of Dengue Virus Inhibitor JNJ-A07 (2021) (0)
- Synthesis of a Dual BACE1/CYP3A4 Inhibitor (2013) (0)
- Synthesis of BAY 1895344 (2020) (0)
- Formal Synthesis of BMT-362265 (2021) (0)
- Synthesis of APD371 (2018) (0)
- Synthesis of BMS-986260 (2020) (0)
- Synthesis of Lamivudine (2020) (0)
- Flow Synthesis of a Doravirine Fragment (2018) (0)
- Formal Synthesis of Telaprevir (2015) (0)
- Synthesis of Almorexant (2013) (0)
- Regioselective Cyanomethylation of Imidazopyridines (2017) (0)
- Synthesis of a Key Intermediate of Omarigliptin (2017) (0)
- Synthesis of EEDi-5273 (2021) (0)
- Synthesis of Sitagliptin (2014) (0)
- Synthesis of PARP Inhibitor PF-01367338 (2013) (0)
- Synthesis of the Indole Core of MK-3281 (2013) (0)
- Synthesis of Monobactam 1 (2020) (0)
- Synthesis of a Histone Deacetylase Inhibitor (2012) (0)
- Synthesis Alerts 15/02 (2002) (0)
- Asymmetric Copper-Catalyzed Hydroamination of Aryl Alkynes (2015) (0)
- Synthesis of P4Q-391 (2017) (0)
- Synthetic Approaches to Rapamycin. Part 2. A Synthesis of a C21‐C42 Fragment. (1997) (0)
- Synthesis of (–)-Benzolactam-V8 (2012) (0)
- Formation of Aza-Allenic Derivatives and Their Further Electrocyclization (2002) (0)
- Synthesis of a CB1 Cannabinoid Receptor Antagonist (2012) (0)
- Synthesis of BMS-665053 (2012) (0)
- Synthesis of Bimatoprost (2015) (0)
- Synthesis of Taxadienone (2015) (0)
- Synthesis of QCA570 (2018) (0)
- Synthesis of Filorexant (2016) (0)
- Synthesis of Florfenicol (2012) (0)
- Synthesis of VX-787 (2014) (0)
- Synthesis of BMS-986235/LAR-1219 (2020) (0)
- Synthesis of an Aurora Kinase B Inhibitor (2015) (0)
- Reductive Amination of β-Tetralones Catalyzed by a Chiral Phosphoric Acid (2018) (0)
- Synthesis of Chitinase Inhibitor OATD-01 (2021) (0)
- 2.8 Oxazolines (2005) (0)
- Synthesis of a Glucokinase Activator (2014) (0)
- RECENT SULFONE-BASED OLEFINATION REACTIONS (1985) (0)
- Formal Synthesis of Ezetimibe (2012) (0)
- Synthesis of (–)-Oseltamivir (2012) (0)
- 8.1 Introduction (2005) (0)
- Synthesis Alerts 15/03 (2003) (0)
- Synthesis of Voriconazole (2014) (0)
- Synthesis of PDE4 Inhibitors (2016) (0)
- Synthesis of an ORL-1 Antagonist (2016) (0)
- Synthesis of AZD7545 (2012) (0)
- Generation and Cross-Coupling of Organozinc Reagents in Flow (2019) (0)
- Synthesis of a Ghrelin Receptor Agonist (2018) (0)
- Synthesis of GSK2137305 (2012) (0)
- Synthesis of Sotagliflozin (2021) (0)
- Synthesis of BMS-986278 (2021) (0)
- Synthesis of (1R,3S)-HPA-12 (2013) (0)
- Synthesis Alerts 1/04 (2003) (0)
- Synthesis of a Boceprevir Fragment (2012) (0)
- Synthesis of ACT-334441 (2016) (0)
- Synthesis of MK-7145 (2021) (0)
- Synthesis of BMS-978587 (2018) (0)
- Synthesis of AT13387 (2013) (0)
- Synthesis of Neobenodrine (2012) (0)
- 3.1 Introduction (2005) (0)
- Synthesis of GDC-4379 (2021) (0)
- Synthesis of Fluorinated BACE Inhibitors (2018) (0)
- Synthesis of PF-00610355 (2012) (0)
- The 3,4‐Dihydro‐2H‐pyran Approach to (+)‐Milbemycin β3. Part 2. An Improved Synthesis of (2R,4S,6S,8R,9S)‐2‐((5R)‐(2E)‐3‐Methyl‐5‐formylhex‐2‐en‐1‐yl)‐8,9‐dimethyl‐4‐(dimethyl‐t‐butylsilyloxy)‐1,7‐dioxaspiro(5.5)undecane. (1988) (0)
- Synthesis of (R)-(–)-Sumanirole (2012) (0)
- Synthesis of a P2X7 Inhibitor (2016) (0)
- Synthesis of Maxipost (2013) (0)
- Synthesis of a SIRT1 Inhibitor (2014) (0)
- Synthesis of TP-808 (2017) (0)
- Synthesis of GDC-0853 (2018) (0)
- Synthesis of UM171 (2017) (0)
- Synthesis of an HDM2 Inhibitor (2014) (0)
- Synthesis of Pregabalin (2013) (0)
- A Synthesis of (3S*,4R*)‐Luffariolide. (1996) (0)
- Synthesis of Tesirine (2018) (0)
- Synthesis of (S)-Pregabalin (2015) (0)
- Synthesis of a BACE1 Inhibitor (2019) (0)
- Formal Synthesis of (–)-Indatraline (2012) (0)
- 2-Sulfinyl-Diazabicyclooctane Derivatives as β-Lactamase Inhibitors (2021) (0)
- Synthesis of CEP-28122 (2012) (0)
- Photoredox Catalysis in the Synthesis of JAK2 Inhibitor LY2784544 (2015) (0)
- 4-(Difluoromethyl)pyridin-2-amine, a Key Intermediate for Lipid Kinase Inhibitors PQR620 and PQR530 (2020) (0)
- Synthesis of TAK-071 Using Flash Chemistry (2019) (0)
- Synthesis of PF-06815189 (2018) (0)
- Asymmetric Synthesis of an hNK1 Inhibitor (2020) (0)
- Synthesis of HIV-1 Protease Inhibitors (2018) (0)
- Synthesis of Flibanserin (2018) (0)
- Synthesis of a Cyclic Glutamine Analogue Used in Antiviral Agents (2021) (0)
- Synthesis of 4-(Aminomethyl)quinolin-2(1H)-ones (2020) (0)
- Flow Synthesis of Anilines through Photoredox/Ni(II)-Catalyzed C–N Cross-Coupling: Tetracaine (2020) (0)
- Synthesis of Aminocyclohexenes from 7-Azanorbornenes (2018) (0)
- A New Synthesis of a-Methylene Carbinols (1979) (0)
- Synthesis of Ivosidenib (2018) (0)
- Palladium(0)‐Catalyzed Stannylstannylation and Silylstannylation of 1‐ Alkoxy‐1‐alkynes and 1‐Phenylthio‐1‐alkynes. (1995) (0)
- Synthesis of DZ-2384 (2015) (0)
- Synthesis of Remibrutinib (2020) (0)
- Synthesis of a Key Subunit of HIV-1 Protease Inhibitor Darunavir (2021) (0)
- Silicon-mediated Annulation. Part 1. A Synthesis of Tetrahydropyran-4-ones, Oxepan-4-ones, and Oxocan-4-ones via Intramolecular Directed Aldol Reactions. (1986) (0)
- Synthesis of β-Lactamase Inhibitor IID572 (2020) (0)
- Synthesis of DS-8108b (2012) (0)
- Synthesis of a Key Building Block for Anti-AIDS Drugs (2016) (0)
- Synthesis of Letermovir via Asymmetric Hydrogen Bonding Catalysis (2017) (0)
- Asymmetric Copper-Catalyzed Hydroamination: Maraviroc (2019) (0)
- Synthesis of Ataciguat via Sulfoximine-Directed Sulfamidation (2013) (0)
- Synthesis Alerts 07/03 (2003) (0)
- Synthesis Alerts 09/97 (1997) (0)
- Synthesis of (–)-Oxycodone (2019) (0)
- Synthesis of Eravacycline (2013) (0)
- A Synthetic Approach to Zoapatanol (I) and Related Bicyclic Analogues. (1987) (0)
- Synthesis of Sacubitril (2016) (0)
- Synthesis of 2′-Fluoro-6′-methylene-carbocyclic Adenosine (FMCA) (2019) (0)
- Synthesis of a Macrocyclic Mcl-1 Inhibitor (2020) (0)
- Synthesis of Δ9-Tetrahydrocannabinol (2018) (0)
- Synthesis of LY500307 (2012) (0)
- Asymmetric Synthesis of Ipatasertib (2017) (0)
- Synthesis of GSK1324726A (2015) (0)
- Synthesis of Entecavir (2013) (0)
- Synthesis of Aztreonam (2020) (0)
- Synthesis of PF-07059013 (2021) (0)
- Synthesis of MK-8666 (2017) (0)
- Synthesis of AMG 232 (2019) (0)
- Synthesis of (–)-Oseltamivir Phosphate (2013) (0)
- Synthesis of Eravacycline (2013) (0)
- Synthesis of ent-Ketorfanol (2016) (0)
- Synthesis alerts 03/99 (1999) (0)
- Book Reviews, Comprehensive Natural Products Chemistry 08/99 (1999) (0)
- Synthesis of Diaryl Sulfones: GSK 742457 (2014) (0)
- SYNTHETIC APPROACHES TO PEDERIN. A SYNTHESIS OF (.+-.)-BENZOYLPEDAMIDE (1984) (0)
- Synthesis of (–)-Galanthamine (2012) (0)
- Synthesis of Suvorexant (2012) (0)
- Synthesis of a Topisomerase I Inhibitor (2012) (0)
- Asymmetric Synthesis of cis-2,5-Disubstituted Pyrrolidines (2013) (0)
- A New Synthesis of 1,7-Dioxaspiro(5.5)undec-4-enes via Metallated Allenol Ethers. A Formal Synthesis of Talaromycins A and B. (1988) (0)
- The Preparation of 6-Bromo-3,4-dihydro-2H-pyrans from Tetrahydropyran-2-ones via a Ni(0)-Catalyzed Coupling Reaction and Their Halogen—Metal Exchange to 6-Lithio-3,4-dihydro-2H-pyrans. (2002) (0)
- Asymmetric Synthesis of a Carbapenem Intermediate (2019) (0)
- Synthesis of Nilotinib (2012) (0)
- Synthesis of Tucatinib (2019) (0)
- Synthesis of a HIV Integrase Inhibitor (2014) (0)
- Synthesis of Chk1 Inhibitor GDC-0425 (2015) (0)
- Synthesis Alerts 7/04 (2004) (0)
- Synthesis of Tyclopyrazoflor (2019) (0)
- Continuous Palladium-Catalyzed Carbonylative Cyclization Using Iron Pentacarbonyl as a CO Source (2020) (0)
- Synthesis of Monobactam Antibiotic LYS228 (2020) (0)
- Synthesis Alerts 3/05 (2005) (0)
- 7.4 Esters Cleaved by β-Elimination Reactions (2005) (0)
- Enantioselective Synthesis of (2R,6R)-Hydroxynorketamine (2017) (0)
- Formal Synthesis of Neratinib (2013) (0)
- Synthesis of GDC-0810 (2018) (0)
- Synthesis of Trifluorinated Thiazolines That Target Prohibitins (2014) (0)
- Synthesis of LY2623091 (2017) (0)
- Synthesis of DPA-714 (2012) (0)
- Synthesis of an Adenosine A2A Receptor Antagonist (2013) (0)
- Synthesis of BMS-986118 (2018) (0)
- Synthesis of Venetoclax (2019) (0)
- Synthesis of an EGFR Inhibitor (2016) (0)
- Synthesis Alerts 10/00 (2000) (0)
- Synthesis of SGLT-2 Inhibitor Empagliflozin (2014) (0)
- Synthesis of GSK2798745 (2019) (0)
- Synthesis Alerts 01/02 (2000) (0)
- Synthesis of Beclabuvir (2018) (0)
- Synthesis of Levamisole (2014) (0)
- Synthesis of a Glucokinase Activator (2020) (0)
- The Synthesis of α-Heteroalkenylmetals via Hydrometalation and Metallometalation of Alkynes (1995) (0)
- 8.10 Reviews (2005) (0)
- Cooperative Catalysis in the Synthesis of Chroman-2-ones: NNC 45-0781 (2018) (0)
- Synthesis of PF-06815345 (2019) (0)
- Synthesis of Omecamtiv Mecarbil (2019) (0)
- Synthesis of a Glucagon Receptor Antagonist (2013) (0)
- 7.5 Reviews (2005) (0)
- Synthesis Alerts 09/99 (1999) (0)
- SCOPE AND STEREOCHEMISTRY OF AN OLEFIN SYNTHESIS FROM β-HYDROXY-SULFONES (1978) (0)
- Synthetic Studies on the Pederin Family of Antitumor Agents. Syntheses of Mycalamide B (XIII), Theopederin D (XVI) and Pederin (XVIII). (2000) (0)
- Synthesis of (–)-Huperzine A (2012) (0)
- Synthesis of BMS-929075 (2020) (0)
- Synthesis of Fibrinolysis Inhibitor AZD6564 (2014) (0)
- Synthesis of a GPR40 Modulator (2017) (0)
- A NEW SYNTHESIS OF α‐METHYLENE CARBINOLS (1979) (0)
- Synthesis Alerts 3/04 (2004) (0)
- Synthesis of a GPR40 Superagonist (2019) (0)
- Synthesis of ABBV-744 (2020) (0)
- One-Pot Synthesis of a TGFβRI Inhibitor (2020) (0)
- Synthesis of Artemisinin (2017) (0)
- Synthesis of Imatinib (2013) (0)
- Formal Synthesis of HIV Integrase Inhibitor BI 224436 (2016) (0)
- Synthesis of a Carfilzomib Fragment (2020) (0)
- Synthesis of (R)-Sitagliptin (2016) (0)
- Synthesis of Idasanutlin (RG7388) (2017) (0)
- Formation of β-Lactones via Lewis Acid Promoted [2+2]-Cycloaddition Reaction (2002) (0)
- Synthesis of a BACE1 Inhibitor (2013) (0)
- Synthesis of the JAK2 Kinase Inhibitor AZD1480 (2013) (0)
- Third-Generation Synthesis of Sulopenem (2012) (0)
- Synthesis Alerts 14/00 (2000) (0)
- Synthesis of β-Secretase Inhibitor NB-360 (2021) (0)
- Synthesis of a PDE10A Inhibitor (2019) (0)
- Synthesis of ACT-209905 (2012) (0)
- Rearrangement by 1,3-Silyl Shift (2002) (0)
- Synthesis of (–)-Galanthamine (2013) (0)
- Synthesis of an Atropisomeric HIV Integrase Inhibitor (2015) (0)
- Synthesis of Vixotrigine (2021) (0)
- Synthesis of 1,3-Oxazine Based β-Secretase Inhibitors (2018) (0)
- Synthesis of Huprine Derivatives (2016) (0)
- Synthesis of Pamiparib (2021) (0)
- Synthesis of (3S,5R)-3-Aminomethyl-5-methyloctanoic Acid (2012) (0)
- Synthesis of TAK-063 (2019) (0)
- Synthesis of BACE1 Inhibitors (2015) (0)
- Synthesis of Vabicaserin (2013) (0)
- Synthesis of Taselisib (2019) (0)
- Synthesis of a CXCR Antagonist (2018) (0)
- Synthesis of β-Adrenergic Blockers (2012) (0)
- Crystallization-Induced Dynamic Resolution of a Dibenzoazepinone (2017) (0)
- Synthesis of a β-Secretase Inhibitor (2013) (0)
- Synthesis of Aficamten (2021) (0)
- Synthesis of a Hydroxamic Acid LpxC Inhibitor (2012) (0)
- Synthesis of 2-Amino-4H-chromene Antibacterial Agents (2012) (0)
- Synthesis of MK-4688 (2021) (0)
- AN ECONOMICAL LARGE SCALE PREPARATION OF (2S,3S)-4,5-DIMETHYL-2-PHENYL-1,3-DIOXOLAN (1985) (0)
- cis-Mo(CO)4(Py)2: A Superior Reagent for the Preparation of η3-Allyl Molybdenum Complexes. (2001) (0)
- Synthesis of a Selective Estrogen Receptor β Agonist (2013) (0)
- Synthesis of AZD7762 (2017) (0)
- Synthesis of (R)-Verapamil by Enantioselective Heck Arylation (2016) (0)
- 7.3 Alkyl Esters (2005) (0)
- Synthesis of a p38 Kinase Inhibitor (2013) (0)
- Synthesis of (Z)-Tamoxifen (2012) (0)
- 2.7 Orthoester Derivatives (2005) (0)
- Synthesis of Efavirenz (2012) (0)
- Synthesis of GPI 16539 (2013) (0)
- Flow Synthesis of Dolutegravir (2018) (0)
- Synthesis Alerts 13/02 (2002) (0)
- Synthesis of O-GlcNAcase Inhibitor MK-8719 (2020) (0)
- Synthesis of LX2761 (2019) (0)
- Synthesis of Tetrahydrolipstatin (2014) (0)
- Synthesis of a Serine Hydroxymethyltransferase Inhibitor (2017) (0)
- Synthesis of an Estrogen-Related Receptor 1 Inhibitor (2014) (0)
- Synthesis of l-Carbidopa via Enantioselective α-Amination (2013) (0)
- Synthesis of GGDC-0994 (2017) (0)
- Asymmetric Synthesis of Netarsudil (2019) (0)
- A New Approach to 1,7-Dioxaspiro(5.5)undec-4-enes via Metalated Allenol Ethers. Synthesis of Lacrimin A. (1990) (0)
- Continuous Flow Synthesis of a Lamivudine Intermediate (2020) (0)
- Synthesis Alerts 5/01 (2001) (0)
- Synthesis Alerts 11/96 (1996) (0)
- A Synthesis of the Hypocholesterolemic Agent 1233A via Asymmetric [2 + 2] Cycloaddition. (1999) (0)
- Synthesis of an HCV NS5B Polymerase Inhibitor (2012) (0)
- 1.2 Deprotection: The Concept of Orthogonal Sets (2005) (0)
- Concise Synthesis of Molnupiravir (2021) (0)
- Synthesis of a FLAP Inhibitor (2015) (0)
- Synthesis of a CGRP Receptor Inhibitor (2013) (0)
- Asymmetric Fluorination Approach to an SYK Inhibitor (2015) (0)
- Synthesis of BMS-663068 (2014) (0)
- A vinylic α‐carbamoyloxyborane with a carbenoid‐type bonding arrangement (2002) (0)
- Synthesis of GNE-834 (2020) (0)
- Synthesis of a NaV 1.7 inhibitor (2020) (0)
- Synthesis of CH4930808 (2018) (0)
- Synthesis of (S)-Omeprazole (2018) (0)
- Synthesis of Serine Hydrolase Inhibitor ABL303 (2012) (0)
- Synthesis of GSK2263167 (2014) (0)
- Synthesis of CPI-0610 (2016) (0)
- Synthesis of AB928 (2020) (0)
- Synthesis of the 2-Fluoroadenine Nucleobase of Islatravir (2021) (0)
- CCDC 762203: Experimental Crystal Structure Determination (2011) (0)
- Synthesis of Tropifexor (2018) (0)
- Synthesis of MK-8831 (2016) (0)
- 4.2 Silyl Ethers (II) (2005) (0)
- Synthesis of AZD6738 (2019) (0)
- 6.1 Introduction (2005) (0)
- Synthesis of a MK-8876 Fragment (2016) (0)
- Artificial Intelligence Guides the Synthesis of SCH 47949 (2019) (0)
- 3.5 1,1,3,3-Tetraisopropyldisiloxanylidene Derivatives (2005) (0)
- Synthesis of AZD4121 (2012) (0)
- Synthetic Approaches to Pseudopterosin G Aglycone Dimethyl Ether. (1998) (0)
- Synthesis of LY2784544 (2013) (0)
- Thermolytic Deprotection of N-Boc Groups (2019) (0)
- Synthesis Alerts 04/00 (2000) (0)
- Synthesis of an 11-β-HSD-1 Inhibitor via Asymmetric Methallylation (2016) (0)
- Synthesis of (+)-Lithospermic Acid (2013) (0)
- Synthesis of PF-06843195 (2021) (0)
- Synthesis of EPZ015666 (2018) (0)
- Synthesis of Vaniprevir (MK-7009) (2012) (0)
- Synthesis of 1,1-Diphenylpropyl-1-amines via Hydroaminomethylation (2013) (0)
- Synthesis of (–)-Chloramphenicol (2016) (0)
- Synthesis of BMS-986318 (2021) (0)
- The Preparation and Pd(0)‐Catalyzed Cross Coupling Reactions of α ‐(Phenylthio)alkenylzinc. (1993) (0)
- Synthesis of Monobactam Antibiotic LYS228 (2020) (0)
- Synthesis Alerts 11/97 (1997) (0)
- Synthesis Alerts 08/03 (2003) (0)
- Peptide Synthesis and Self‐Assembly (2013) (0)
- Synthesis of PF-00835231 (2021) (0)
- Synthesis of an H3 Antagonist (2012) (0)
- Synthesis of Sacubitril (2016) (0)
- Synthesis of the Cyclohexane Dicarboxylate Fragment of BMS-986251 (2021) (0)
- Synthesis of Dantrolene (2014) (0)
- Synthesis of Salinomycin. (1998) (0)
- Synthesis of Synosutine via Asymmetric Cyclopropanation (2014) (0)
- 1.3 Relay Deprotection (2005) (0)
- Synthesis of Olutasidenib (2020) (0)
- Synthesis of (+)-Ambrisentan (2012) (0)
- Synthesis of AMD15548 (2012) (0)
- Synthesis of Daclatasvir by C–H Activation (2016) (0)
- Synthesis Alerts 03/01 (2001) (0)
- Synthesis of (R)-Baclofen (2015) (0)
- Synthesis of ALK Inhibitor PF-06463922 (2014) (0)
- A Scalable Ring-Closing Metathesis for the Manufacture of AMG 176 (2021) (0)
- Synthesis of the Corey Lactone and Latanoprost (2020) (0)
- Continuous-Flow Diazotization (2019) (0)
- Synthesis of (+)-CP-99,994 (2018) (0)
- Synthesis of Dolutegravir (2019) (0)
- Synthesis of a Glucokinase Activator (2012) (0)
- 4.1 Introduction (2005) (0)
- 1.6 Temporary Protection (2005) (0)
- Continuous Flow Photo-oxidation of Cyclopentadiene (2020) (0)
- Synthesis of Tofogliflozin Hydrate (2017) (0)
- 8.8 Imine and Enamine Derivatives (2005) (0)
- Synthesis of Veliparib (2019) (0)
- Synthessis of Tipifarnib (2015) (0)
- Synthesis of BMS-214662 (2018) (0)
- Asymmetric Alkynylation in the Synthesis of Efavirenz Intermediates (2018) (0)
- Synthesis of LY541850 and Its C4 Epimer (2012) (0)
- Synthesis of (–)-Nutlin-3 (2014) (0)
- Synthesis Alerts 09/98 (1998) (0)
- Synthesis Alerts 09/00 (2000) (0)
- Cyanoamidine Cyclization Approach to Remdesivir’s Nucleobase (2020) (0)
- Diastereoselective Pyrrolidine Synthesis Using a Sulfinamide Annulating Agent (2020) (0)
- Synthesis Alerts 12/03 (2003) (0)
- Flow Synthesis of Ceramide d-erythro-CER[NDS] (2019) (0)
- Enantioselective Synthesis of AC-7954 (2013) (0)
- Stereoselective Synthesis of Functionalized Alkenyllithiums and Alkenyl Cyanocuprates by the Cu(I)-Catalyzed Coupling of Organolithium Reagents with α-Lithiated Cyclic Enol Ethers. (1989) (0)
- Synthesis of Escitalopram (2016) (0)
- Synthesis of d 9-Ivacaftor Using o-Quinone Methide Chemistry (2020) (0)
- Synthesis of the C14—C28 Fragment of Tetronasin. (2006) (0)
- (3R*,4S*)-4-[(S*)-2-Cyclohexyl-2-(tert-butyldimethylsiloxy)ethyl]-3-hexyl-3-(trimethylsilyl)oxetan-2-one (1996) (0)
- A Synthetic Approach to the C26-C32 Fragment of Rapamycin. A Synthesis of Allylic Alcohols from Allylic Furylsilanes. (1994) (0)
- Pilot-Scale Synthesis of TV-45070 (2018) (0)
- Synthesis Alerts 10/02 (2002) (0)
- Synthesis of rac-Naproxen (2012) (0)
- Synthesis of Vismodegib via Directed C–H Chlorination (2017) (0)
- Synthesis of PF-06424439 (2018) (0)
- Synthesis of Pexidartinib (2019) (0)
- Synthesis of (–)-Huperzine A (2013) (0)
- Synthesis of SUVN-911 (2020) (0)
- Synthesis of a Sodium–Hydrogen Exchange Type 1 Inhibitor (2013) (0)
- Synthesis of GDC-0276 by a Highly Regioselective SNAr Reaction (2019) (0)
- Synthesis of Glacaprevir by Ring-Closing Metathesis (2020) (0)
- Synthesis of a Telithromycin Analogue (2012) (0)
- Synthesis of a Squaramide-Based CXCR2 Receptor Antagonist (2015) (0)
- A New Synthesis of Spiroacetals via Alkylidenation of Ester Carbonyls with Metal Carbene Complexes. (1988) (0)
- Synthesis of a Key Building Block for HCV Protease Inhibitor Telaprevir (2015) (0)
- Synthesis of JAK Inhibitor ASP3627 (2020) (0)
- Synthesis of AZD7648 (2020) (0)
- Synthesis Alerts 11/98 (1998) (0)
- Synthesis of MK-3207 (2013) (0)
- Asymmetric Syntheses of Panclicins A-E via [2 + 2] Cycloaddition of Alkyl(trimethylsilyl)ketenes to a β-Silyloxyaldehyde. (1998) (0)
- The β-Lactone Route to β-Hydroxy of α,β-Unsaturated γ- and δ-Lactones. Syntheses of (.+-.)-Massoialactone (I) and (.+-.)-Prelactone B (II). (2003) (0)
- Commercial Synthesis of BMS-663068 (2017) (0)
- A Synthesis of the C24-C34 Segment of FK 506. (1990) (0)
- Synthesis of Niraparib (2014) (0)
- Synthesis of BMS-986020 by a Tandem Borylation–Suzuki Procedure (2018) (0)
- A SYNTHESIS OF ALLYLIC ALCOHOLS FROM β,Γ-EPOXYSULFONES (1979) (0)
- Synthesis of MK-8262 (2021) (0)
- Synthesis of an Androgen Receptor Modulator (2014) (0)
- Synthesis of LY2886721 (2015) (0)
- Synthesis of an H-PGDS Inhibitor (2013) (0)
- Synthesis of the Antifungal Agent ASP9726 (2014) (0)
- Synthesis of Encequidar (2021) (0)
- Synthesis Alerts 11/99 (1999) (0)
- 2.2 O,O- Acetals (2005) (0)
- Synthesis Alerts 12/01 (2001) (0)
- 4.5 Tetrahydropyranyl (THP) and Related Ethers (2005) (0)
- Recent Progress in Research on the Immunosuppressant FK-506 (1990) (0)
- Synthesis of All Four Mefloquine Diastereoisomers (2013) (0)
- Synthesis of Canagliflozin (2018) (0)
- Synthesis of AG-041 Analogues (2015) (0)
- Synthesis of Olmesartan Medoxomil (2015) (0)
- Synthesis of Tacalcitol (2021) (0)
- Synthesis of Lobucavir (2012) (0)
- Synthesis of Spiropiperidine BACE-1 Inhibitors (2013) (0)
- Formal Synthesis of Oseltamivir Phosphate (2013) (0)
- Synthesis of a Saxagliptin Fragment (2014) (0)
- A NEW AND USEFUL OLEFIN SYNTHESIS BASED ON SULFONES (1981) (0)
- Synthesis of MK-8248 (2017) (0)
- Synthesis of a PI3VIIδ Inhibitor via Alkyne Cyclotrimerization (2016) (0)
- The Hydrometalation, Carbometalation, and Metallometalation of Heteroalkynes (1995) (0)
- Synthesis of PF-06869206 (2018) (0)
- Synthesis of a CGRP Receptor Antagonist (2016) (0)
- Synthesis of SCH 900229 (2013) (0)
- Synthesis of Vaniprevir (2012) (0)
- Synthesis of Ritobegron Ethyl Hydrochloride (2020) (0)
- Synthesis of a tRNA–Guanine Transglycosylase Inhibitor (2016) (0)
- Formal Synthesis of Omarigliptin (2017) (0)
- Synthesis of Atabecestat (2021) (0)
- Synthetic Approaches to Rapamycin. Part 3. Synthesis of a C1-C21 Fragment. (1997) (0)
- From Diazo Compounds via Wolff Rearrangement (2002) (0)
- Synthesis of Atuveciclib (2019) (0)
- Synthesis of Atorvastatin (2013) (0)
- Synthesis Alerts 10/05 (2005) (0)
- Synthesis of Lotronex through anti-Azacarboxylation of a 2-Alkynylaniline (2016) (0)
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