Sally-Ann Poulsen
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Australian chemical biologist
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Sally-Ann Poulsenchemistry Degrees
Chemistry
#5525
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#6720
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Organic Chemistry
#1039
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#1172
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Sally-Ann Poulsenbiology Degrees
Biology
#15336
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#19292
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Biochemistry
#2748
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#2936
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Chemistry Biology
Sally-Ann Poulsen's Degrees
- PhD Chemical Biology University of Melbourne
Why Is Sally-Ann Poulsen Influential?
(Suggest an Edit or Addition)According to Wikipedia, Sally-Ann Poulsen is an Australian chemical biologist who is a Professor and Director at Griffith University. Her research considers medicinal chemistry and drug discovery. She is Chair of the Royal Australian Chemical Institute Medicinal Chemistry and Chemical Biology Division.
Sally-Ann Poulsen's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Non-zinc mediated inhibition of carbonic anhydrases: coumarins are a new class of suicide inhibitors. (2009) (421)
- Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond (2016) (324)
- Discovery of a new family of carbonic anhydrases in the malaria pathogen Plasmodium falciparum--the η-carbonic anhydrases. (2014) (279)
- Adenosine receptors: new opportunities for future drugs. (1998) (269)
- Carbonic anhydrase inhibitors: inhibition of isozymes I, II, and IX with triazole-linked O-glycosides of benzene sulfonamides. (2007) (166)
- A novel class of carbonic anhydrase inhibitors: glycoconjugate benzene sulfonamides prepared by "click-tailing". (2006) (156)
- Synthetic utility of glycosyl triazoles in carbohydrate chemistry (2006) (110)
- Targeting hypoxic tumor cell viability with carbohydrate-based carbonic anhydrase IX and XII inhibitors. (2011) (110)
- Molecular evolution: dynamic combinatorial libraries, autocatalytic networks and the quest for molecular function. (2000) (105)
- Therapeutic applications of glycosidic carbonic anhydrase inhibitors (2009) (103)
- Natural product-based phenols as novel probes for mycobacterial and fungal carbonic anhydrases. (2011) (90)
- Screening the Medicines for Malaria Venture Pathogen Box across Multiple Pathogens Reclassifies Starting Points for Open-Source Drug Discovery (2017) (89)
- Natural product coumarins that inhibit human carbonic anhydrases. (2013) (87)
- Dynamic combinatorial libraries of pseudo-peptide hydrazone macrocycles (1999) (85)
- Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes. (2014) (83)
- Metallocene-based inhibitors of cancer-associated carbonic anhydrase enzymes IX and XII. (2012) (79)
- Carbonic anhydrase inhibitors with dual-tail moieties to match the hydrophobic and hydrophilic halves of the carbonic anhydrase active site. (2015) (72)
- Microwave-accelerated Fischer glycosylation (2005) (72)
- Carbonic anhydrase inhibitors. Identification of selective inhibitors of the human mitochondrial isozymes VA and VB over the cytosolic isozymes I and II from a natural product-based phenolic library. (2010) (66)
- Inhibition of carbonic anhydrases with glycosyltriazole benzene sulfonamides. (2008) (66)
- Direct screening of a dynamic combinatorial library using mass spectrometry (2006) (65)
- Saccharin: a lead compound for structure-based drug design of carbonic anhydrase IX inhibitors. (2015) (62)
- Sulfonamide inhibition studies of the η-class carbonic anhydrase from the malaria pathogen Plasmodium falciparum. (2015) (57)
- Sulfonamide linked neoglycoconjugates--a new class of inhibitors for cancer-associated carbonic anhydrases. (2010) (57)
- Inhibition of membrane-associated carbonic anhydrase isozymes IX, XII and XIV with a library of glycoconjugate benzenesulfonamides. (2007) (54)
- Fragment-based drug discovery of carbonic anhydrase II inhibitors by dynamic combinatorial chemistry utilizing alkene cross metathesis. (2006) (53)
- S-glycosyl primary sulfonamides--a new structural class for selective inhibition of cancer-associated carbonic anhydrases. (2009) (50)
- A prodrug approach toward cancer-related carbonic anhydrase inhibition. (2013) (48)
- Structural Insights into Carbonic Anhydrase IX Isoform Specificity of Carbohydrate-Based Sulfamates (2014) (47)
- Pharmacological inhibition of carbonic anhydrase XII interferes with cell proliferation and induces cell apoptosis in T-cell lymphomas. (2013) (45)
- Carbonic anhydrase inhibition as a cancer therapy: a review of patent literature, 2007 – 2009 (2010) (45)
- Inhibition of carbonic anhydrase isozymes with benzene sulfonamides incorporating thio, sulfinyl and sulfonyl glycoside moieties. (2009) (42)
- Natural Product Primary Sulfonamides and Primary Sulfamates. (2015) (41)
- Promiscuity of carbonic anhydrase II. Unexpected ester hydrolysis of carbohydrate-based sulfamate inhibitors. (2011) (40)
- Protein crystal structures with ferrocene and ruthenocene-based enzyme inhibitors. (2012) (40)
- Carbonic anhydrase inhibitors developed through 'click tailing'. (2010) (40)
- Native State Mass Spectrometry, Surface Plasmon Resonance, and X-ray Crystallography Correlate Strongly as a Fragment Screening Combination. (2016) (40)
- Anti-mycobacterial activity of a bis-sulfonamide. (2007) (39)
- Inhibition of carbonic anhydrase isozymes I, II and IX with benzenesulfonamides containing an organometallic moiety. (2007) (39)
- Synthesis of S-glycosyl primary sulfonamides. (2009) (38)
- Electrospray ionisation Fourier-transform ion cyclotron resonance mass spectrometry of dynamic combinatorial libraries. (2000) (38)
- Inhibition of human mitochondrial carbonic anhydrases VA and VB with para-(4-phenyltriazole-1-yl)-benzenesulfonamide derivatives. (2008) (36)
- Fragment-based screening by X-ray crystallography, MS and isothermal titration calorimetry to identify PNMT (phenylethanolamine N-methyltransferase) inhibitors. (2010) (35)
- An Unusual Natural Product Primary Sulfonamide: Synthesis, Carbonic Anhydrase Inhibition, and Protein X-ray Structures of Psammaplin C. (2016) (34)
- P-glycoprotein-mediated chemoresistance is reversed by carbonic anhydrase XII inhibitors (2016) (32)
- Antimalarial activity of compounds comprising a primary benzene sulfonamide fragment. (2013) (32)
- Design, synthesis, and biological evaluation of novel carbohydrate-based sulfamates as carbonic anhydrase inhibitors. (2011) (31)
- Synthesis and in Vivo Biological Evaluation of (68)Ga-Labeled Carbonic Anhydrase IX Targeting Small Molecules for Positron Emission Tomography. (2016) (30)
- Solution structures in aqueous SDS micelles of two amyloid beta peptides of A beta(1-28) mutated at the alpha-secretase cleavage site (K16E, K16F). (2000) (30)
- Carbonic Anhydrase XII Inhibitors Overcome P-Glycoprotein–Mediated Resistance to Temozolomide in Glioblastoma (2018) (30)
- Synthesis and structure-activity relationship of pyrazolo[3,4-d]pyrimidines: potent and selective adenosine A1 receptor antagonists. (1996) (29)
- Screening a natural product-based combinatorial library using FTICR mass spectrometry. (2006) (27)
- Novel organometallic cationic ruthenium(II) pentamethylcyclopentadienyl benzenesulfonamide complexes targeted to inhibit carbonic anhydrase (2009) (27)
- Carbonic Anhydrase XII Inhibitors Overcome Temozolomide Resistance in Glioblastoma. (2019) (26)
- Mapping Selective Inhibition of the Cancer-Related Carbonic Anhydrase IX Using Structure-Activity Relationships of Glucosyl-Based Sulfamates. (2015) (25)
- Design and synthesis of thiourea compounds that inhibit transmembrane anchored carbonic anhydrases. (2012) (24)
- Synthesis of glycoconjugate carbonic anhydrase inhibitors by ruthenium-catalysed azide-alkyne 1,3-dipolar cycloaddition. (2011) (23)
- Synthesis and Evaluation of Antimalarial Properties of Novel 4‐Aminoquinoline Hybrid Compounds (2014) (23)
- Synthesis of acylated glycoconjugates as templates to investigate in vitro biopharmaceutical properties. (2013) (23)
- An overview of Australia's compound management facility: the Queensland Compound Library. (2014) (23)
- Synthesis of cyclic oligomers of a modified sugar amino acid utilising dynamic combinatorial chemistry (2004) (22)
- Isoform-selective inhibitory profile of 2-imidazoline-substituted benzene sulfonamides against a panel of human carbonic anhydrases (2016) (22)
- Natural Product Polyamines That Inhibit Human Carbonic Anhydrases (2014) (20)
- Synthesis and structure-activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II. (2005) (19)
- Agents described in the Molecular Imaging and Contrast Agent Database for imaging carbonic anhydrase IX expression (2014) (15)
- Identification of a New Zinc Binding Chemotype by Fragment Screening. (2017) (14)
- Investigating the antiplasmodial activity of primary sulfonamide compounds identified in open source malaria data (2017) (14)
- Fragment Screening by Native State Mass Spectrometry (2014) (14)
- Pyrazolo[3,4-d]pyrimidines: C4, C6 substitution leads to adenosine A1 receptor selectivity (1996) (13)
- Synthesis of sulfonamide-bridged glycomimetics. (2011) (13)
- Synthesis, structure and bioactivity of primary sulfamate-containing natural products. (2018) (12)
- Microwave-accelerated cross-metathesis reactions of N-allyl amino acid substrates (2005) (11)
- High-Pressure Synthesis of Enantiomerically Pure C-6 Substituted Pyrazolo[3,4-d]pyrimidines (2001) (10)
- Synthesis of N-Propargyl Iminosugar Scaffolds for Compound Library Generation using Click Chemistry (2010) (9)
- Investigation of pyrimidine nucleoside analogues as chemical probes to assess compound effects on the proliferation of Trypanosoma cruzi intracellular parasites (2020) (8)
- Inhibition of Human Mitochondrial Carbonic Anhydrases VA and VB with para‐(4‐Phenyltriazole‐1‐yl)‐benzenesulfonamide Derivatives. (2009) (8)
- Natural products that inhibit carbonic anhydrase. (2014) (8)
- Phosphate Chemical Probes Designed for Location Specific Inhibition of Intracellular Carbonic Anhydrases. (2015) (8)
- Stereoselective Synthesis of Highly Functionalized Arabinosyl Nucleosides through Application of an N-Nitro Protecting Group. (2018) (7)
- Recent developments of small molecule chemical probes for fluorescence-based detection of human carbonic anhydrase II and IX (2016) (7)
- Click Chemistry in Carbohydrate Based Drug Development and Glycobiology (2007) (6)
- Women in Medicinal Chemistry Special Issue Call for Papers. (2019) (6)
- Labeling of Cellular DNA with a Cyclosal Phosphotriester Pronucleotide Analog of 5‐ethynyl‐2′‐deoxyuridine (2015) (6)
- Development of ethynyl-2'-deoxyuridine chemical probes for cell proliferation. (2016) (5)
- Carbonic anhydrase XII inhibition overcomes P-glycoprotein-mediated drug resistance: a potential new combination therapy in cancer (2021) (5)
- Characterisation of Photoaffinity‐Based Chemical Probes by Fluorescence Imaging and Native‐State Mass Spectrometry (2017) (5)
- Oxazole-Benzenesulfonamide Derivatives Inhibit HIV-1 Reverse Transcriptase Interaction with Cellular eEF1A and Reduce Viral Replication (2019) (5)
- 4-hydroxymethyl-1-(2',3',4',6'-tetra-O-acetyl-b-D-glucopyranosyl)-1,2,3-triazole. (2006) (4)
- Synthesis and Structure-Activity Relationship of Pyrazolo(3,4-d) pyrimidines: Potent and Selective Adenosine A1 Receptor Antagonists. (1997) (4)
- Women in Medicinal Chemistry: Ad Maiora! (2020) (3)
- The Key Glycolytic Enzyme Phosphofructokinase Is Involved in Resistance to Antiplasmodial Glycosides (2020) (3)
- In Situ Fragment‐Based Medicinal Chemistry: Screening by Mass Spectrometry (2008) (3)
- The Glitazone Class of Drugs as Carbonic Anhydrase Inhibitors—A Spin-Off Discovery from Fragment Screening (2021) (3)
- Synthesis of sulfonamide-conjugated glycosyl-amino acid building blocks. (2014) (3)
- N-Allyl-N-(2-nitrobenzenesulfonyl)-L-phenylalanine methyl ester (2003) (2)
- Coumarins that inhibit carbonic anhydrase (2014) (2)
- Synthesis of Novel Saccharin Derivatives (2017) (2)
- Synthesis and Structure—Activity Relationships of Novel Benzene Sulfonamides with Potent Binding Affinity for Bovine Carbonic Anhydrase II. (2006) (2)
- N‐Cinnamoyl‐l‐valine methyl ester (2007) (2)
- (η5-Pentamethylcyclopentadienyl)(η6-p-toluenesulfonamide)ruthenium(II) tetraphenylborate (2008) (1)
- Bifunctional copper(II) chelators from the coupling of the encapsulating ligand 1-methyl-8-amino-3,13,16-trithia-6,10,19-triazabicyclo[6.6.6]icosane (AMN3S3sar) with carboxylic acids; applications of the coupling agent DMT-MM (2015) (1)
- Methyl 2,3,4-tri-O-acetyl-1-azido-1-deoxy-β-d-glucopyranuronate at room temperature (2005) (1)
- N-(2-Nitrophenylsulfonyl)glycine methyl ester (2005) (1)
- Novel Organometallic Ruthenium(II)Cp* Benzenesulphonamides for the Inhibition of Carbonic Anhydrases (2008) (1)
- N-{2-(4-(Aminosulfonyl)phenyl)ethyl}-2-(4-hydroxy- phenyl)acetamide (2007) (1)
- Human Carbonic anhydrases II in complex with a acetazolamide derivative comprising one hydrophobic and one hydrophilic tail moiety (2015) (0)
- Synthesis of ferrocene and ruthenocene-based arylsulfonamides and the elucidation of their crystal structures with human carbonic anhydrase II (2009) (0)
- Attenuating the solubility of carbohydrate-based drugs for improved delivery and targeting. (2007) (0)
- In situ click synthesis of glycosyltriazole arylsulfonamides: Hydrophilic carbonic anhydrase II inhibitors. (2006) (0)
- Synthesis of 5‐Alkynyl Substituted 2ʹ‐Arabinosyl 2ʹ‐Halogenated Uridine Nucleosides (2019) (0)
- Orgamometallic-Based Inhibitors of Carbonic Anhydrases Targeting Hypoxic Tumors (2008) (0)
- Selective inhibition of carbonic anhydrase isozymes I, II and IX with novel metallocene-based triazole-linked sulfonamides (2008) (0)
- Human carbonic anhydrase II in complex with 1-S-D-Galactopyranosylsulfonamide (2009) (0)
- Pyrazolo(3,4-d)pyrimidines: Synthesis and Structure-Activity Relationships for Binding to Adenosine Receptors (1996) (0)
- Structure-based drug design of novel inhibitors of carbonic anhydrase for treatment of glaucoma (2009) (0)
- Carbonic anhydrase 2 in complex with [(2R,3S,4R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-3,4-DIHYDROXYTETRAHYDRO-2-FURANYL]METHYL SULFAMATE inhibitor (2018) (0)
- Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond Citation (2016) (0)
- Human carbonic anhydrase II in complex with (2,3,4,6-Tetra-O-acetyl-beta-D-galactopyranosyl) -(1-4)-1,2,3,6-tetra-O-acetyl-1-thio-beta-D-glucopyranosylsulfonamide (2009) (0)
- Carbonic anhydrase 2 in complex with 2-chloro-5'-O-sulfamoyladenosine (2018) (0)
- Identification of a New Zinc Binding Chemotype of by Fragment Screening on human carbonic anhydrase (2017) (0)
- Dynamic combinatorial chemistry and mass spectrometry: a combined strategy for high-performance lead discovery (2009) (0)
- Operationally Simple Regioselective 5′-Phosphorylation of Unprotected 5-Ethynyl-2′-deoxyuridine Analogues (2020) (0)
- High-pressure synthesis of enantiomerically pure C-6 substituted pyrazol. (2001) (0)
- SOLUTION NMR STRUCTURE OF AMYLOID BETA[E16], RESIDUES 1-28, 14 STRUCTURES (1998) (0)
- Synthesis, carbonic anhydrase inhibition and protein X-ray structure of the unusual natural product primary sulfonamide Psammaplin C (2016) (0)
- Human carbonic anhydrase II in complex with topiramate (2009) (0)
- N-Cinnamoyl-l-phenylalanine methyl ester (2007) (0)
- High-Pressure Synthesis of Enantiomerically Pure C-6 Substituted Pyrazolo[3,4-d]pyrimidines. (2001) (0)
- L-phenylalanine methyl ester (2003) (0)
- Editorial: Excellence in Medicinal Chemistry from Australia. (2017) (0)
- Human carbonic anhydrase II in complex with alpha-D-Glucopyranosyl-(1->4)-1-thio-beta-D-glucopyranosylsulfonamide (2009) (0)
- Microwave‐Accelerated Fischer Glycosylation. (2005) (0)
- Synthesis of Glycoconjugate Carbonic Anhydrase Inhibitors by Ruthenium-Catalyzed Azide-Alkyne 1,3-Dipolar Cycloaddition. (2012) (0)
- Thymidine kinase-independent click chemistry DNADetect™ probes for DNA proliferation assessment in malaria parasites (2023) (0)
- Microwave‐Accelerated Cross‐Metathesis Reactions of N‐Allyl Amino Acid Substrates. (2006) (0)
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