Satoshi Ōmura
#1,247
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Japanese biochemist
Satoshi Ōmura's AcademicInfluence.com Rankings
Satoshi Ōmurabiology Degrees
Biology
#110
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#201
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Biochemistry
#188
World Rank
#238
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Biology
Satoshi Ōmura's Degrees
- PhD Pharmaceutical Sciences University of Tokyo
- Bachelors Pharmaceutical Sciences University of Yamanashi
Why Is Satoshi Ōmura Influential?
(Suggest an Edit or Addition)According to Wikipedia, is a Japanese biochemist. He is known for the discovery and development of hundreds of pharmaceuticals originally occurring in microorganisms. In 2015, he was awarded the Nobel Prize in Physiology or Medicine jointly with William C. Campbell for their role in the discovery of avermectins and ivermectin, the world's first endectocide and a safe and highly effective microfilaricide. It is believed that the large molecular size of ivermectin prevents it from crossing the blood/aqueous humour barrier, and renders the drug an important treatment of helminthically-derived blindness.
Satoshi Ōmura's Published Works
Number of citations in a given year to any of this author's works
Total number of citations to an author for the works they published in a given year. This highlights publication of the most important work(s) by the author
Published Works
- Degradation of CFTR by the ubiquitin-proteasome pathway (1995) (1301)
- Complete genome sequence and comparative analysis of the industrial microorganism Streptomyces avermitilis (2003) (1167)
- Avermectins, New Family of Potent Anthelmintic Agents: Producing Organism and Fermentation (1979) (818)
- Genome sequence of an industrial microorganism Streptomyces avermitilis: Deducing the ability of producing secondary metabolites (2001) (785)
- A new alkaloid AM-2282 OF Streptomyces origin. Taxonomy, fermentation, isolation and preliminary characterization. (1977) (611)
- Lactacystin, a novel microbial metabolite, induces neuritogenesis of neuroblastoma cells. (1991) (457)
- Genome-minimized Streptomyces host for the heterologous expression of secondary metabolism (2010) (433)
- The antibiotic cerulenin, a novel tool for biochemistry as an inhibitor of fatty acid synthesis. (1976) (360)
- Terpene synthases are widely distributed in bacteria (2014) (352)
- Degradation of a Mutant Secretory Protein, α1-Antitrypsin Z, in the Endoplasmic Reticulum Requires Proteasome Activity* (1996) (348)
- Production of ‘hybrid’ antibiotics by genetic engineering (1985) (315)
- The Degradation of Apolipoprotein B100 Is Mediated by the Ubiquitin-proteasome Pathway and Involves Heat Shock Protein 70* (1997) (304)
- Organization of the biosynthetic gene cluster for the polyketide anthelmintic macrolide avermectin in Streptomyces avermitilis. (1999) (289)
- Ivermectin: 25 years and still going strong. (2008) (267)
- Ivermectin, ‘Wonder drug’ from Japan: the human use perspective (2011) (253)
- Proteasome-dependent regulation of p21WAF1/CIP1 expression. (1996) (238)
- Accelerated degradation of PML-retinoic acid receptor alpha (PML-RARA) oncoprotein by all-trans-retinoic acid in acute promyelocytic leukemia: possible role of the proteasome pathway. (1996) (238)
- Novel Aspects of Degradation of T Cell Receptor Subunits from the Endoplasmic Reticulum (ER) in T Cells: Importance of Oligosaccharide Processing, Ubiquitination, and Proteasome-dependent Removal from ER Membranes (1998) (232)
- Degradation of the Met tyrosine kinase receptor by the ubiquitin-proteasome pathway (1997) (232)
- Structure of lactacystin, a new microbial metabolite which induces differentiation of neuroblastoma cells. (1991) (229)
- Agroactive compounds of microbial origin. (1993) (227)
- Lactacystin, a specific inhibitor of the proteasome, induces apoptosis in human monoblast U937 cells. (1995) (223)
- The life and times of ivermectin — a success story (2004) (217)
- Inhibition of fatty acid synthesis by the antibiotic cerulenin. Specific inactivation of beta-ketoacyl-acyl carrier protein synthetase. (1973) (215)
- Structural and Computational Analysis of the Quinone-binding Site of Complex II (Succinate-Ubiquinone Oxidoreductase) (2006) (214)
- The proteasome inhibitor lactacystin induces apoptosis and sensitizes chemo- and radioresistant human chronic lymphocytic leukaemia lymphocytes to TNF-alpha-initiated apoptosis. (1998) (210)
- Atpenins, potent and specific inhibitors of mitochondrial complex II (succinate-ubiquinone oxidoreductase) (2003) (204)
- ACAT2 Is Localized to Hepatocytes and Is the Major Cholesterol-Esterifying Enzyme in Human Liver (2004) (199)
- Staurosporine, a potentially important gift from a microorganism. (1995) (191)
- Engineered Streptomyces avermitilis host for heterologous expression of biosynthetic gene cluster for secondary metabolites. (2013) (184)
- Identification and functional analysis of genes controlling biosynthesis of 2-methylisoborneol (2008) (183)
- Inhibition of acyl-CoA: cholesterol acyltransferase activity by cyclodepsipeptide antibiotics. (1992) (174)
- mdm2 and bax, downstream mediators of the p53 response, are degraded by the ubiquitin-proteasome pathway. (1998) (171)
- Erythromycin suppresses nuclear factor-kappaB and activator protein-1 activation in human bronchial epithelial cells. (2000) (162)
- Proteasome Inhibitors Block Development ofPlasmodium spp (1998) (160)
- Chemical biology of natural indolocarbazole products: 30 years since the discovery of staurosporine (2009) (159)
- Herbimycin, a new antibiotic produced by a strain of Streptomyces. (1979) (157)
- Erythromycin and its derivatives with motilin-like biological activities inhibit the specific binding of 125I-motilin to duodenal muscle. (1988) (157)
- Binding site of cerulenin in fatty acid synthetase. (1989) (155)
- Macrolides with gastrointestinal motor stimulating activity. (1987) (155)
- Isolation of new actinomycete strains for the screening of new bioactive compounds. (2003) (154)
- Increased sensitivity of CLL‐derived lymphocytes to apoptotic death activation by the proteasome‐specific inhibitor lactacystin (1999) (150)
- Avenolide, a Streptomyces hormone controlling antibiotic production in Streptomyces avermitilis (2011) (144)
- Degradation Process of Ligand-stimulated Platelet-derived Growth Factor β -Receptor Involves Ubiquitin-Proteasome Proteolytic Pathway * (1995) (138)
- The proteasome is involved in angiogenesis. (1998) (136)
- Pyripyropenes, highly potent inhibitors of acyl-CoA:cholesterol acyltransferase produced by Aspergillus fumigatus. (1993) (133)
- Defects in the Ubiquitin Pathway Induce Caspase-independent Apoptosis Blocked by Bcl-2* (1998) (130)
- Genome mining of the Streptomycesavermitilis genome and development of genome-minimized hosts for heterologous expression of biosynthetic gene clusters (2014) (129)
- Lariatins, antimycobacterial peptides produced by Rhodococcus sp. K01-B0171, have a lasso structure. (2006) (126)
- Ivermectin: panacea for resource-poor communities? (2014) (124)
- An anthelmintic compound, nafuredin, shows selective inhibition of complex I in helminth mitochondria. (2001) (121)
- Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A(H1N1)pdm09 virus infection by interfering with virus internalization process (2019) (119)
- Lactacystin, a specific inhibitor of the proteasome, inhibits human platelet lysosomal cathepsin A-like enzyme. (1997) (119)
- Identification of ACAT1- and ACAT2-specific inhibitors using a novel, cell-based fluorescence assay: individual ACAT uniqueness. (2004) (118)
- Geosmin Biosynthesis in Streptomyces avermitilis. Molecular Cloning, Expression, and Mechanistic Study of the Germacradienol/Geosmin Synthase (2006) (118)
- Xanthohumols, diacylglycerol acyltransferase inhibitors, from Humulus lupulus. (1997) (113)
- Structures and biological properties of Kinamycin A, B, C, and D. (1973) (112)
- Cloning, sequencing and deduced functions of a cluster of Streptomyces genes probably encoding biosynthesis of the polyketide antibiotic frenolicin. (1994) (112)
- Total Synthesis of (+)-Lactacystin (1996) (111)
- Specificity and affinity of natural product cyclopentapeptide inhibitors against A. fumigatus, human, and bacterial chitinases. (2004) (108)
- Deregulation of the ubiquitin system and p53 proteolysis modify the apoptotic response in B-CLL lymphocytes. (2000) (108)
- Hyper-inducible expression system for streptomycetes. (2004) (108)
- Pyripyropenes, novel inhibitors of acyl-CoA:cholesterol acyltransferase produced by Aspergillus fumigatus. I. Production, isolation, and biological properties. (1994) (108)
- Total Synthesis of (+)-Madindoline A and (−)-Madindoline B, Potent, Selective Inhibitors of Interleukin 6. Determination of the Relative and Absolute Configurations (2000) (107)
- Evidence for an essential role of long chain acyl-CoA synthetase in animal cell proliferation. Inhibition of long chain acyl-CoA synthetase by triacsins caused inhibition of Raji cell proliferation. (1991) (106)
- Degradation of 3-Hydroxy-3-methylglutaryl-CoA Reductase in Endoplasmic Reticulum Membranes Is Accelerated as a Result of Increased Susceptibility to Proteolysis* (1996) (104)
- Molecular Mechanisms of Anti-Inflammatory Action of Erythromycin in Human Bronchial Epithelial Cells: Possible Role in the Signaling Pathway That Regulates Nuclear Factor-κB Activation (2004) (104)
- Culture conditions for screening of new antibiotics. (1982) (102)
- The Search for Bioactive Compounds from Microorganisms (1992) (101)
- Argadin, a new chitinase inhibitor, produced by Clonostachys sp. FO-7314. (2000) (99)
- A new antibiotic, kinamycin. (1970) (98)
- Kitasatosporia, a new genus of the order Actinomycetales. (1982) (97)
- Potential Immunocompetence of Proteolytic Fragments Produced by Proteasomes before Evolution of the Vertebrate Immune System (1997) (97)
- A gene cluster for biosynthesis of the sesquiterpenoid antibiotic pentalenolactone in Streptomyces avermitilis. (2006) (96)
- Philosophy of new drug discovery. (1986) (95)
- In vivo treatment of mutant FLT3-transformed murine leukemia with a tyrosine kinase inhibitor (2000) (94)
- Cytochrome p450 complement (CYPome) of the avermectin-producer Streptomyces avermitilis and comparison to that of Streptomyces coelicolor A3(2). (2003) (91)
- Andrastins A-C, new protein farnesyltransferase inhibitors produced by Penicillium sp. FO-3929. II. Structure elucidation and biosynthesis. (1996) (88)
- Potent antimalarial activities of polyether antibiotic, X-206. (2001) (88)
- Letter: Nanaomycins A and B, new antibiotics produced by a strain of Streptomyces. (1974) (88)
- Proteasome regulation of activation-induced T cell death. (1997) (87)
- New lycorine-type alkaloid from Lycoris traubii and evaluation of antitrypanosomal and antimalarial activities of lycorine derivatives. (2008) (87)
- Activation of Atypical Protein Kinase C ζ by Caspase Processing and Degradation by the Ubiquitin-Proteasome System* (2000) (86)
- High-resolution structures of a chitinase complexed with natural product cyclopentapeptide inhibitors: Mimicry of carbohydrate substrate (2002) (85)
- Inhibition of farnesyl-protein transferase by gliotoxin and acetylgliotoxin. (1992) (85)
- A small-molecule inhibitor of the bacterial type III secretion system protects against in vivo infection with Citrobacter rodentium (2011) (83)
- Absolute Configuration of Staurosporine By X-Ray Analysis (1994) (83)
- The onchocerciasis chronicle: from the beginning to the end? (2012) (82)
- Lyn and Fgr Protein-tyrosine Kinases Prevent Apoptosis during Retinoic Acid-induced Granulocytic Differentiation of HL-60 Cells (*) (1996) (81)
- Pyripyropenes, novel inhibitors of acyl-CoA:cholesterol acyltransferase produced by Aspergillus fumigatus. II. Structure elucidation of pyripyropenes A, B, C and D. (1994) (81)
- Chloropeptins I and II, novel inhibitors against gp120-CD4 binding from Streptomyces sp. (1994) (81)
- Genetic studies of avermectin biosynthesis in Streptomyces avermitilis (1987) (80)
- X-Ray crystal structure of staurosporine: a new alkaloid from a Streptomyces strain (1978) (80)
- Phosalacine, a new herbicidal antibiotic containing phosphinothricin. Fermentation, isolation, biological activity and mechanism of action. (1984) (80)
- Production of new hybrid antibiotics, mederrhodins A and B, by a genetically engineered strain (1986) (79)
- Motilides, macrolides with gastrointestinal motor stimulating activity. I. O-substituted and tertiary N-substituted derivatives of 8,9-anhydroerythromycin A 6,9-hemiacetal. (1989) (79)
- Macrosphelide, a novel inhibitor of cell-cell adhesion molecule. I. Taxonomy, fermentation, isolation and biological activities. (1995) (78)
- Purpactins, new inhibitors of acyl-CoA:cholesterol acyltransferase produced by Penicillium purpurogenum. I. Production, isolation and physico-chemical and biological properties. (1991) (78)
- Carbon-13 nuclear magnetic resonance spectral analysis of 16-membered macrolide antibiotics. (1975) (77)
- Pyripyropene A, an Acyl–Coenzyme A: Cholesterol Acyltransferase 2–Selective Inhibitor, Attenuates Hypercholesterolemia and Atherosclerosis in Murine Models of Hyperlipidemia (2011) (76)
- Chemical and biological studies on 16-membered macrolide antibiotics. (1975) (76)
- Avermectin Biosynthesis. (1997) (76)
- EM703 improves bleomycin-induced pulmonary fibrosis in mice by the inhibition of TGF-β signaling in lung fibroblasts (2006) (75)
- Metabolism and Products of Actinomycetes - An Introduction (1990) (75)
- Triacsins, new inhibitors of acyl-CoA synthetase produced by Streptomyces sp. (1986) (75)
- Antiatherogenic activity of fungal beauveriolides, inhibitors of lipid droplet accumulation in macrophages. (2004) (75)
- Structure of virantmycin, a novel antiviral antibiotic (1981) (75)
- Selectivity of Microbial Acyl-CoA : cholesterol Acyltransferase Inhibitors toward Isozymes (2007) (75)
- A new antibiotic, kinamycin: fermentation, isolation, purification and properties. (1971) (74)
- Suppression of bone resorption by madindoline A, a novel nonpeptide antagonist to gp130 (2002) (74)
- Arisugacin, a novel and selective inhibitor of acetylcholinesterase from Penicillium sp. FO-4259. (1995) (74)
- Spoxazomicins A–C, novel antitrypanosomal alkaloids produced by an endophytic actinomycete, Streptosporangium oxazolinicum K07-0460T (2011) (74)
- Materials for the fungus flora of Japan (47) (1994) (74)
- Lariatins, Novel Anti-mycobacterial Peptides with a Lasso Structure, Produced by Rhodococcus jostii K01-B0171 (2007) (73)
- Isolation and structure of nanaomycin D, an enantiomer of the antibiotic kalafungin (1976) (73)
- Nanomycins, new antibiotics produced by a strain of Streptomyces. II. Structure and biosynthesis. (1975) (72)
- In vitro and in vivo antimalarial activities of a non-glycosidic 18-membered macrolide antibiotic, borrelidin, against drug-resistant strains of Plasmodia. (2003) (71)
- New cyclodepsipeptides, enniatins D, E and F produced by Fusarium sp. FO-1305. (1992) (70)
- Streptomyces avermectinius sp. nov., an avermectin-producing strain. (2002) (70)
- Mechanism by which the lectin actinohivin blocks HIV infection of target cells (2009) (70)
- Production of deoxyfrenolicin and a new antibiotic, frenolicin B by Streptomyces roseofulvus strain AM-3867. (1978) (69)
- Involvement of glucose catabolism in avermectin production by Streptomyces avermitilis (1988) (69)
- New beauvericins, potentiators of antifungal miconazole activity, Produced by Beauveria sp. FKI-1366. I. Taxonomy, fermentation, isolation and biological properties. (2004) (69)
- Relative and Absolute Stereochemistry of Pyripyropene A, A Potent, Bioavailable Inhibitor of Acyl-CoA:Cholesterol Acyltransferase (ACAT) (1994) (68)
- Complete inhibition of mouse macrophage-derived foam cell formation by triacsin C. (1999) (68)
- Argifin, a new chitinase inhibitor, produced by Gliocladium sp. FTD-0668. I. Taxonomy, fermentation, and biological activities. (2000) (68)
- Oxetin, a new antimetabolite from an actinomycete. Fermentation, isolation, structure and biological activity. (1984) (67)
- The structure of asukamycin, a possible shunt metabolite from 3-dehydroquinic acid in the shikimate pathway (1979) (66)
- In vitro antimalarial activity of prenylated flavonoids from Erythrina fusca (2008) (66)
- An erythromycin derivative, EM-523, induces motilin-like gastrointestinal motility in dogs. (1989) (65)
- Antiplasmodial and antitrypanosomal activity of plants from the Kingdom of Saudi Arabia (2009) (65)
- Total synthesis of (+)-lactacystin, the first non-protein neurotrophic factor (1993) (65)
- New antitumor antibiotics, OS-4742 A1, A2, B1 and B2 produced by a strain of Streptomyces. (1977) (65)
- New brominated and halogen-less derivatives and structure-activity relationship of azaphilones inhibiting gp120-CD4 binding. (1998) (65)
- Yaequinolones J1 and J2, novel insecticidal antibiotics from Penicillium sp. FKI-2140. (2005) (64)
- A combinatorial synthesis of a macrosphelide library utilizing a palladium-catalyzed carbonylation on a polymer support. (2003) (64)
- Acylated pregnane glycosides from Caralluma tuberculata and their antiparasitic activity. (2008) (63)
- Enhancement of CPP32-like activity in the TNF-treated U937 cells by the proteasome inhibitors. (1996) (63)
- Total synthesis of (-)-borrelidin. (2004) (62)
- Phthoxazolin, a specific inhibitor of cellulose biosynthesis, produced by a strain of Streptomyces sp. (1990) (62)
- Isolation and Identification of Three New 5-Alkenyl-3,3(2H)-furanones from Two Streptomyces species using a Genomic Screening Approach (2006) (62)
- Transposon mutagenesis by Tn4560 and applications with avermectin-producing Streptomyces avermitilis (1993) (61)
- Clostomicins, new antibiotics produced by Micromonospora echinospora subsp. armeniaca subsp. nov. I. Production, isolation, and physico-chemical and biological properties. (1986) (61)
- Valine as a precursor of n-butyrate unit in the biosynthesis of macrolide aglycone. (1983) (61)
- Mechanism of action of cerulenin on fatty acid synthetase. Effect of cerulenin on iodoacetamide-induced malonyl-CoA decarboxylase activity. (1982) (60)
- Oxaline, a fungal alkaloid, arrests the cell cycle in M phase by inhibition of tubulin polymerization. (2004) (60)
- Effect of ammonium ion, inorganic phosphate and amino acids on the biosynthesis of protylonolide, a precursor of tylosin aglycone. (1984) (59)
- Andrastins A-C, new protein farnesyltransferase inhibitors produced by Penicillium sp. FO-3929. I. Producing strain, fermentation, isolation, and biological activities. (1996) (59)
- Madindoline, a novel inhibitor of IL-6 activity from Streptomyces sp. K93-0711. I. Taxonomy, fermentation, isolation and biological activities. (1996) (59)
- Novel Mitochondrial Complex II Isolated from Trypanosoma cruzi Is Composed of 12 Peptides Including a Heterodimeric Ip Subunit* (2009) (59)
- Arisugacins A and B, novel and selective acetylcholinesterase inhibitors from Penicillium sp. FO-4259. I. Screening, taxonomy, fermentation, isolation and biological activity. (1996) (59)
- Proteasome inhibitors induce mitochondria‐independent apoptosis in human glioma cells (1999) (58)
- Relative and Absolute Stereochemistries and Total Synthesis of (+)-Macrosphelides A and B, Potent, Orally Bioavailable Inhibitors of Cell−Cell Adhesion (1997) (58)
- Isochromophilones III-VI, inhibitors of acyl-CoA:cholesterol acyltransferase produced by Penicillium multicolor FO-3216. (1995) (58)
- In vitro antimalarial activity of biflavonoids from Wikstroemia indica. (2004) (58)
- Polymyxin B identified as an inhibitor of alternative NADH dehydrogenase and malate: quinone oxidoreductase from the Gram-positive bacterium Mycobacterium smegmatis. (2009) (58)
- Actinohivin, a novel anti-HIV protein from an actinomycete that inhibits syncytium formation: isolation, characterization, and biological activities. (2001) (58)
- Guadinomines, Type III Secretion System Inhibitors, Produced by Streptomyces sp. K01-0509 (2008) (57)
- Biosynthesis of vineomycins A1 and B2. (1982) (57)
- Selective and Potent in Vitro Antitrypanosomal Activities of Ten Microbial Metabolites (2008) (57)
- Structure of herbimycin A new ansamycin antibiotic (1979) (56)
- Inhibition of acyl-CoA synthetase by triacsins. (1987) (56)
- Structure of argifin, a new chitinase inhibitor produced by Gliocladium sp. (2000) (55)
- Pentalenolactone biosynthesis. Molecular cloning and assignment of biochemical function to PtlI, a cytochrome P450 of Streptomyces avermitilis. (2006) (55)
- Effect of sea water concentration on hyphal growth and antimicrobial metabolite production in marine fungi (2001) (55)
- Virantmycin, a new antiviral antibiotic produced by a strain of Streptomyces. (1980) (55)
- Phenatic Acids A and B, New Potentiators of Antifungal Miconazole Activity Produced by Streptomyces sp. K03-0132 (2005) (55)
- Studies on the biosynthesis of 16-membered macrolide antibiotics using carbon-13 nuclear magnetic resonance spectroscopy. (1977) (55)
- The structure of phosalacine, a new herbicidal antibiotic containing phosphinothricin. (1984) (55)
- Terpendoles, novel ACAT inhibitors produced by Albophoma yamanashiensis. III. Production, isolation and structure elucidation of new components. (1995) (55)
- The structure of vineomycin B2. (1981) (55)
- Trehangelins A, B and C, novel photo-oxidative hemolysis inhibitors produced by an endophytic actinomycete, Polymorphospora rubra K07-0510 (2013) (54)
- Macrosphelide, a novel inhibitor of cell-cell adhesion molecule. II. Physiochemical properties and structural elucidation. (1996) (54)
- In vitro antitrypanosomal activity of plant terpenes against Trypanosoma brucei. (2011) (54)
- Total Synthesis of (+)-Pyripyropene A. A Potent, Orally Bioavailable Inhibitor of Acyl-CoA:Cholesterol Acyltransferase (1995) (53)
- Triacsin C: a differential inhibitor of arachidonoyl-CoA synthetase and nonspecific long chain acyl-CoA synthetase. (1989) (53)
- Antimalarial activity of radicicol, heptelidic acid and other fungal metabolites. (1998) (52)
- Total synthesis of salinosporamide A. (2008) (52)
- The expanded horizon for microbial metabolites--a review. (1992) (52)
- Terpendoles, novel ACAT inhibitors produced by Albophoma yamanashiensis. II. Structure elucidation of terpendoles A, B, C and D. (1995) (51)
- Structure elucidation of fungal beauveriolide III, a novel inhibitor of lipid droplet formation in mouse macrophages. (1999) (51)
- Cerulenin-resistant mutants of Saccharomyces cerevisiae with an altered fatty acid synthase gene (1994) (51)
- Total Synthesis of α-Pyrone Meroterpenoids, Novel Bioactive Microbial Metabolites (2005) (51)
- Potent inhibitory effect of antibiotic 1233A on cholesterol biosynthesis which specifically blocks 3-hydroxy-3-methylglutaryl coenzyme A synthase. (1987) (51)
- Novel antibiotics, furaquinocins A and B. Taxonomy, fermentation, isolation and physico-chemical and biological characteristics. (1990) (51)
- Advances in drug discovery and biochemical studies. (2007) (51)
- Cyslabdan, a New Potentiator of Imipenem Activity against Methicillin-resistant Staphylococcus aureus, Produced by Streptomyces sp. K04-0144 (2008) (50)
- Biosynthesis of furaquinocins A and B (1990) (50)
- Beauveriolides, specific inhibitors of lipid droplet formation in mouse macrophages, produced by Beauveria sp. FO-6979. (1999) (50)
- Potential therapeutics for obesity and atherosclerosis: inhibitors of neutral lipid metabolism from microorganisms. (2007) (50)
- Isolation and Structure Elucidation of Lolilline, a Possible Biosynthetic Precursor of the Lolitrem Family of Tremorgenic Mycotoxins (1997) (50)
- Neuronal differentiation of neuro 2a cells by inhibitors of cell cycle progression, trichostatin A and butyrolactone I. (1999) (49)
- Amphomycin inhibits phospho-N-acetylmuramyl-pentapeptide translocase in peptidoglycan synthesis of Bacillus. (1979) (49)
- New beauvericins, potentiators of antifungal miconazole activity, Produced by Beauveria sp. FKI-1366. II. Structure elucidation. (2004) (49)
- A new antibiotic, antimycin Ag, produced by Streptomyces sp. K01-0031. (2005) (49)
- Genome mining reveals a minimum gene set for the biosynthesis of 32-membered macrocyclic thiopeptides lactazoles. (2014) (49)
- Inhibition of sterol and fatty acid biosyntheses by cerulenin in cell-free systems of yeast. (1972) (49)
- Five new Simplicillium species (Cordycipitaceae) from soils in Tokyo, Japan (2013) (49)
- Thiotetromycin, a new antibiotic. Taxonomy, production, isolation, and physicochemical and biological properties. (1983) (49)
- Pyripyropenes, novel ACAT inhibitors produced by Aspergillus fumigatus. IV. Structure elucidation of pyripyropenes M to R. (1996) (48)
- In vitro and in vivo antimalarial activity of puberulic acid and its new analogs, viticolins A–C, produced by Penicillium sp. FKI-4410 (2011) (48)
- Structure determination and total synthesis of bottromycin A2: a potent antibiotic against MRSA and VRE. (2009) (48)
- Merobatzelladines A and B, anti-infective tricyclic guanidines from a marine sponge Monanchora sp. (2009) (48)
- Microbial Metabolites: 45 Years of Wandering, Wondering and Discovering (2011) (48)
- Trends in the search for bioactive microbial metabolites (1992) (48)
- Intracellular retention and degradation of tissue-nonspecific alkaline phosphatase with a Gly317-->Asp substitution associated with lethal hypophosphatasia. (1998) (48)
- Alutenusin, a specific neutral sphingomyelinase inhibitor, produced by Penicillium sp. FO-7436. (1999) (48)
- Actinoallolides A-E, new anti-trypanosomal macrolides, produced by an endophytic actinomycete, Actinoallomurus fulvus MK10-036. (2015) (47)
- Roselipins, inhibitors of diacylglycerol acyltransferase, produced by Gliocladium roseum KF-1040. (1999) (47)
- Separation of cathepsin A-like enzyme and the proteasome: evidence that lactacystin/beta-lactone is not a specific inhibitor of the proteasome. (2000) (47)
- Biosynthesis of the manumycin group antibiotics (1990) (47)
- Control of avermectin biosynthesis in Streptomyces avermitilis for the selective production of a useful component. (1995) (47)
- Studies on bacterial cell wall inhibitors. II. Inhibition of peptidoglycan synthesis in vivo and in vitro by amphomycin. (1977) (47)
- Substitution of cellular fatty acids in yeast cells by the antibiotic cerulenin and exogenous fatty acids. (1975) (47)
- Chitinase inhibitors: extraction of the active framework from natural argifin and use of in situ click chemistry (2009) (47)
- Structure of Kinamycin C, and the Structural Relationship among Kinamycin A, B, C, and D (1971) (47)
- Atpenins, new antifungal antibiotics produced by Penicillium sp. Production, isolation, physico-chemical and biological properties. (1988) (47)
- Arthrobacter oryzae sp. nov. and Arthrobacter humicola sp. nov. (2008) (47)
- Neoxaline, a new alkaloid produced by Aspergillus japonicus. Production, isolation and properties. (1979) (47)
- Herbimycin B, a new benzoquinonoid ansamycin with anti-TMV and herbicidal activities. (1980) (47)
- Molecular insights into the biosynthesis of guadinomine: a type III secretion system inhibitor. (2012) (47)
- Terpendoles, novel ACAT inhibitors produced by Albophoma yamanashiensis. I. Production, isolation and biological properties. (1995) (47)
- Novel antibiotics, furaquinocins C, D, E, F, G and H. (1991) (47)
- ACYL DERIVATIVES OF 16-MEMBERED MACROLIDES (1981) (47)
- Ilumatobacter fluminis gen. nov., sp. nov., a novel actinobacterium isolated from the sediment of an estuary. (2009) (46)
- Structure of cypemycin, a new peptide antibiotic (1994) (46)
- Guadinomines, Type III Secretion System Inhibitors, Produced by Streptomyces sp. K01-0509 (2008) (46)
- Pyripyropenes, Novel ACAT inhibitors produced by Aspergillus fumigatus. III. Structure elucidation of pyripyropenes E to L. (1995) (46)
- Herquline, a new alkaloid produced by Penicillium herquei. Fermentation, isolation and properties. (1979) (45)
- Structure of cervinomycin, a novel xantone antibiotic active against anaerobe and mycoplasma. (1987) (45)
- Revised structure of cerulenin. (1974) (45)
- Bottromycin derivatives: efficient chemical modifications of the ester moiety and evaluation of anti-MRSA and anti-VRE activities. (2010) (45)
- Proteasome regulation of Fas ligand cytotoxicity (1997) (45)
- Inhibition of Sporulation by Cerulenin and Its Reversion by Exogenous Fatty Acids in Saccharomyces cerevisiae (1976) (45)
- Letter: Biosynthetic studies using 13C enriched precursors on the 16-membered macrolide antibiotic leucomycin A3. (1975) (44)
- Yaequinolones, New Insecticidal Antibiotics Produced by Penicillium sp. FKI-2140 (2006) (44)
- Total synthesis of (−)-physovenine from (−)-3a-hydroxyfuroindoline (2005) (44)
- Effects of herbimycin derivatives on src oncogene function in relation to antitumor activity. (1988) (43)
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- New tetrahydroquinoline and indoline compounds containing a hydroxy cyclopentenone, virantmycin B and C, produced by Streptomyces sp. AM-2504 (2018) (0)
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- Revised Structures of Epohelmins A and B Isolated as Lanosterol Synthase Inhibitors from a Fungal Strain FKI‐0929. (2006) (0)
- BIOSYNTHESIS OF VINEOMYCINS Al AND B2 (2006) (0)
- Drug Discovery as a Public Health Intervention: The Ivermectin Story (2008) (0)
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- Reaching for new heights: The Journal of Antibiotics and NPG (2009) (0)
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- Total Synthesis of Amidepsine B (I) and Revision of Its Absolute Configuration. (2009) (0)
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- P-540 SECONDARY METABOLITE PRODUCED BY A RARE FUNGUS, CALDARIOMYCES SP. FKA-35, ISOLATED FROM SUBTROPICAL SOIL (2006) (0)
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- Identification of a novel proton sensing G protein-coupled receptor and its antagonists (2017) (0)
- Activation B κ That Regulates Nuclear Factor-Possible Role in the Signaling Pathway in Human Bronchial Epithelial Cells : Anti-Inflammatory Action of Erythromycin Molecular Mechanisms of (2004) (0)
- Merobatzelladines A (I) and B (II), Antiinfective Tricyclic Guanidines from a Marine Sponge Monanchora sp. (2009) (0)
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- Megalomicins. Part 7. A Structural Revision by Carbon-l3 Nuclear Magnetic Resonance and X-Ray Crystallography. Synthesis and Conformational Analysis of 3-Dimethylamino- and 3-Azido-D- and -L-hexopyranosides, and the Crystal Structure (1979) (0)
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- Simple analytic method of diaminopimelate epimerase activity. (2013) (0)
- Foreword Celebrating the career of Professor Kuniaki Tatsuta (2013) (0)
- SYNTHESIS OF ANOMERIC METHYL 6-O-(L-MYCAROSYL)-BETA-D-GLUCOSAMINIDES AND 4-O-(L-MYCAROSYL)-BETA-D-MYCAMINOSIDES (1974) (0)
- Pentacecilides, new inhibitors of lipid droplet formation in mouse macrophages, produced by Penicillium cecidicola FKI-3765-1: II. Structure elucidation (2009) (0)
- Chemistry and Synthetic Study of Lactacystin, the First Non‐Protein Neurotrophic Factor (1997) (0)
- Synthesis and Activity of Staurosporine Analogues with a Lactone Functionality. (1996) (0)
- Lactacystin: first-in-class proteasome inhibitor still excelling and an exemplar for future antibiotic research (2019) (0)
- Neue substanz fki-1033 und verfahren zur herstellung davon (2002) (0)
- Chemical Constituents of Erythrina suberosa (2004) (0)
- New Members of the Macrosphelides from Microsphaeropsis sp. FO-5050. Part 4. (1999) (0)
- 2S1-PM3 Discovery of microbial products with specific biological targets (2005) (0)
- Letter: A new bicyclo lactone from leukomycin-A3 by alkali treatment. (1974) (0)
- SYNTH. VON PURIN-NUCLEOSIDEN VON L-MYCAROSE UND L-CLADINOSE (1972) (0)
- A New Method for Efficient Coupling of Indole and Epoxide Catalyzed with Yb(O-Tf)3, and Application to the Total Synthesis of Kurasoin B. (2007) (0)
- Intratypic heterogeneity in adenovirus type 3. (1966) (0)
- A compound of the FO-1289 Preparation of (1994) (0)
- STRUCTURE OF PRUMYCIN (1974) (0)
- (13)C-NMR VON NATUERLICHEN UND VERWANDTEN PRODUKTEN 20. MITT. CARBON-13 NUCLEAR MAGNETIC RESONANCE SPECTRAL ANALYSIS OF 16-MEMBERED MACROLIDE ANTIBIOTICS (1975) (0)
- 717 Noninvasive Estimate Method for Intervertebral Disk Load (2013) (0)
- Nosokomycins, New Antibiotics Discovered in an in vivo-Mimic Infection Model Using Silkworm Larvae. Part 1. Fermentation, Isolation and Biological Properties. (2010) (0)
- Pharmacological characteristics of motilin agonist em 523 in gi tract in vivo and in vitro (1991) (0)
- Substances wk-5344a et wk-5344b et leur procede de production (1999) (0)
- New ft-0554A compounds and methods for their preparation (2000) (0)
- Hamuramicins A and B, 22-membered macrolides, produced by an endophytic actinomycete Allostreptomyces sp. K12-0794 (2018) (0)
- Structure Determination of Lustromycin, an Antibiotic Against Anaerobic Bacteria. (2003) (0)
- Madindoline, a Novel Inhibitor of IL-6 Activity from Streptomyces sp. K93-0711 and (0)
- A New Proteolytic Enzyme Having Milk Clotting Activity from Streptomyces sp. No. OS-1000 (1973) (0)
- Purification and Chemical Properties of Anti-complementary Polysaccharide from the Leaves of Artemisia princeps (2007) (0)
- INTRANASALLY AND ORALLY EFFECTIVE ADJUVANTS FROM CHINESE AND JAPANESE MEDICINAL HERBS FOR NASAL INFLUENZA VACCINE (2005) (0)
- A Novel Testosterone 5α-Reductase Inhibitor, 8′,9′- Dehydroascochlorin Produced by Verticillium sp. FO-2787. (1994) (0)
- DER EINFLUSS VON SCHILDDR^|^Uuml;SE UND CORPUS LUTEUM AUF DEN FETTSTOFFWECHSEL. (0)
- Absolute Configuration of Leucomycin, Spiramycin and Cerulenin. (2017) (0)
- Discovery and development of motilin agonist in nonpeptide substance (1992) (0)
- In vitro antitrypanosomal activity of bis(bibenzyls)s and bibenzyls from liverworts against Trypanosoma brucei (2011) (0)
- Chemical Modification and Structure‐Activity Relationships of Pyripyropenes. Part 1. Modification at the Four Hydroxyl Groups. (1997) (0)
- CHEMICAL AND BIOLOGICAL STUDIES ON 16-MEMBERED MACROLIDE ANTIBIOTICS 1. Isolation and Structure of 16-Membered Macrolides Following structural determination of old 16-membered macrolides such as carbomycin, (2006) (0)
- New nitrogen-compounds, penicidones E and F, produced by the fungal strain Oidiodendron sp. FKI-7498. (2022) (0)
- Serratia marcescens Chitinase B complexed with syn-triazole inhibitor (2013) (0)
- Synthetic Applications of a Three‐Component Mannich Reaction. Total Synthesis of IL‐6 Inhibitor (+)‐Madindoline A and B. (2007) (0)
- Contents Vol 88, 2011 (2011) (0)
- Staurosporine, a Potentially Important Gift from a Microorganism (1995) (0)
- [Triacsins, inhibitors of fatty acid activating enzyme]. (1993) (0)
- STRUKTUR VON PRUMYCIN, EINEM ANTIBIOTICUM MIT 2,5-DIAMINO-2,5-DIDESOXYPENTOSE (1972) (0)
- Mycophenolic Acid Inhibits Syncytium Formation Accompanied by Reduction of gp120 Expression. (2006) (0)
- Xanthoradones, New Potentiators of Imipenem Activity Against Methicillin‐Resistant Staphylococcus aureus, Produced by Penicillium Radicum FKI‐3765‐2. Part 1. Taxonomy, Fermentation, Isolation and Biological Properties. (2009) (0)
- Neuronal differentiation of neuro 2A cells by the cell cycle inhibitors lactacystin (proteasome inhibitor) and trichostatin a (histone deacetylase inhibitor) (1996) (0)
- Studies on Macrolides and New Antibiotics (1987) (0)
- KRISTALL- UND MOLEKULARSTRUKTUR DES HYDROBROMIDS VON DESMYCAROSYL-LEUCOMYCIN-A3 (1970) (0)
- Structural insightsinto potent, specific anti-HIV property of actinohivin; Crystal structure of actinohivin in complex with alpha(1-2) mannobiose moiety of high-mannose type glycan of gp120 (2012) (0)
- New Insecticidal Antibiotics, Hydroxyfungerins A and B, Produced by Metarhizium sp. FKI-1079. (2006) (0)
- Discovery of 3-Cinnamamido-N-Substituted Benzamides as Potential Antimalarial Agents. (2020) (0)
- Crystal structure of anti-HIV actinohivin in complex with alphs-1,2-mannobiose (Form II) (2013) (0)
- Total Syntheses of the AChE Inhibitors (.+-.)-Arisugacins F and G. (2004) (0)
- Corrigendum to “Microbial metabolites: 45 years of wandering, wondering and discovering” [Tetrahedron 67 (2011) 6420–6459] (2016) (0)
- DIE STRUKTUR VON CARZINOPHILIN 2. MITT. EINE NEUE AMINOSAEURE UND DEREN DERIVAT AUS CARZINOPHILIN (1972) (0)
- Quellenin, a new anti-Saprolegnia compound isolated from the deep-sea fungus, Aspergillus sp. YK-76 (2018) (0)
- Prophylactic administration of ivermectin attenuates SARS-CoV-2 induced disease in a Syrian Hamster Model (2023) (0)
- Fungal Isobisvertinol (I), a New Inhibitor of Lipid Droplet Accumulation in Mouse Macrophages. (2007) (0)
- Structure Elucidation of Fungal Sespendole (I), an Inhibitor of Lipid Droplet Synthesis in Macrophages. (2006) (0)
- New Rugulosins, anti‐MRSA Antibiotics, Produced by Penicillium radicum FKI‐3765‐2. (2010) (0)
- Chemotherapeutic efficacies of a clofazimine and diminazene aceturate combination against piroplasm parasites and their AT-rich DNA-binding activity on Babesia bovis (2017) (0)
- A NEW ADENOSINE DEAMINASE INHIBITOR CONTAINING CHLORINE PRODUCTION , ISOLATION AND PROPERTIES (2006) (0)
- Microbial Metabolites Affecting Lipid Biosynthesis. (1995) (0)
- PB115 TOTAL SYNTHESIS AND ABSOLUTE CONFIGURATION OF VIRANTMYCIN (1988) (0)
- CHEMIE DER LEUCOMYCINE 10. MITT. KONFORM. VON LEUCOMYCIN (1972) (0)
- Macrolides with Promotive Activity of Monocyte to Macrophage Differentiation. (2005) (0)
- DER EINFLUSS VON SCHILDDR^|^Uuml;SE UND NEBENNIERENRINDE ODER VON NEBENNIERENRINDE UND INSULIN AUF DEN FETTSTOFFWECHSEL (0)
- PC13 INHIBITION MECHANISM OF CERULENIN ON FATTY ACID SYNTHETASE (1988) (0)
- Geological analysis based on tunnel monitoring in Taiwan High Speed Railway Project (2003) (0)
- Crystal structure of a potent anti-HIV lectin actinohivin in complex with alpha-1,2-mannotriose (2013) (0)
- Erythromycin derivative and method for its production. (1986) (0)
- Structure—Activity Relationships Study of Pyripyropenes: Reversal of Cancer Cell Multidrug Resistance. (2000) (0)
- Complex II (Succinate Dehydrogenase) From E. Coli with carboxin inhibitor docked at the ubiquinone binding site (2006) (0)
- Mixing of pharmaceutical powders and granules. II. Mixing degree of granules and various kinds of powders. (1982) (0)
- Structure—Activity Relationships of Stemphones, Potentiators of Imipenem Activity Against Methicillin‐Resistant Staphylococcus aureus. (2009) (0)
- Xanthoradones, New Potentiators of Imipenem Activity Against Methicillin‐Resistant Staphylococcus aureus, Produced by Penicillium radicum FKI‐3765‐2. Part 2. Structure Elucidation. (2009) (0)
- Formation of Phosphinothricin from Phosalacine by Cell-free Extracts from B . subtilis and Spinach (2006) (0)
- Detection and characterization of new mangromicin analogs by tandem mass spectrometry. (2022) (0)
- CELL-FREE BIOSYNTHESIS OF MACROLIDES AND OTHER “POLYKETIDE” ANTIBIOTICS (1981) (0)
- New Analogues of the Pyripyropene Family of ACAT Inhibitors via α-Pyrone Fragmentation and γ-Acylation/Cyclization. (1998) (0)
- Corrigendum: Micromonospora pelagivivens sp. nov., a new species of the genus Micromonospora isolated from deep-sea sediment in Japan. (2020) (0)
- FO-1289 compound and their preparation. (1993) (0)
- ‘Click Chemistry’ Synthesis of Macrolide Derivatives with Anti-MRSA and Anti-VRE Activity (2008) (0)
- 53(P-21) The Production of Novel Polyketide Compounds by Engineered Biosynthesis (2003) (0)
- Relative and Absolute Stereochemistry of the Melanogenesis Inhibitors OH-3984 K1 and K2. Partial Synthesis from Albocycline. (1994) (0)
- An Effect of Novel Non-Antibiotic Macrolide EM900 in HDM-Induced Airway Inflammation Mice Model (2019) (0)
- NOVEL DIMERIC DERIVATIVES OF LEUCOMYCINS AND TYLOSIN, SIXTEEN-MEMBERED MACROLIDES (1982) (0)
- Crystal Structure of PtlH with AKG and ent-1PL bound (2007) (0)
- 4′′′-N-Demethylspiramycin Derivatives: Synthesis and Evaluation of Effectiveness Against Drug-Resistant Bacteria. (2008) (0)
- 502 Noninvasive estimation of load on the intervertebral disk to evaluate lumbago (2014) (0)
- Ammonia Trapping and Stimulation of l-Serine Production from Glycine by Magnesium Phosphate (1982) (0)
- Substance fo-1289 et sa production (1993) (0)
- Inhibitor of electron transport system complex II of (2002) (0)
- Kurasoins A and B, New Protein Farnesyltransferase Inhibitors Produced by Paecilomyces sp. FO‐3684. Part 2. Structure Elucidation and Total Synthesis. (1997) (0)
- Cipralphelin, a new anti-oxidative N-cinnamoyl tripeptide produced by the deep sea-derived fungal strain Penicillium brevicompactum FKJ-0123 (2019) (0)
- Identification of an antibiotic I-1431 isolated from a Streptomyces strain. (1965) (0)
- New substance fki-1083 and process for their preparation (2001) (0)
- Azithromycin, a 15-membered macrolide antibiotic, inhibits influenza A(H1N1)pdm09 virus infection by interfering with virus internalization process (2019) (0)
- Mixing of pharmaceutical powders and granules. I. Effect of grain size on the manufacturing process. (1982) (0)
- Specificity and affnity of natural product cyclopentapeptide inhibitor Argadin against Aspergillus fumigatus chitinase (2004) (0)
- Crystal structures of actinohivin, an anti-HIV protein from an actinomycete, and its complex with mannobiose (2009) (0)
- P-491 Total synthesis and determination of stereochemistry of Verticilide, an anthelmintic cyclodepsipeptide (2006) (0)
- Unearthing Beneficial Microbial Compounds: Discovery, Development & International Partnerships (2016) (0)
- New KF-1040 substance and process for their preparation (1998) (0)
- [Action of EM900 on mucus secretion by the respiratory epithelial cells]. (2009) (0)
- [Feature of antibiotics in the 21st century]. (1996) (0)
- To the genus Streptomyces belonging, for production of nemadictin capable originating and process for production of nemadictin using strain (2003) (0)
- Purification and Chemical Properties of Anti-complementary Polysaccharide from the Leaves of Artemisia princeps (2007) (0)
- Isochromophilones I and II, Novel Inhibitors Against gp120-CD4 Binding Produced by Penicillium multicolor FO-2338. Part 2. Structure Elucidation. (1996) (0)
- Toward the Total Synthesis of Luminamicin, a Specific Anti-Anaerobic Bacteriacide (2013) (0)
- Chemical Modification and Structure-Activity Relationships of Pyripyropenes. Part 2. 1,11-Cyclic Analogues. (1997) (0)
- Structure and Biosynthesis of Novel Antibiotics, Aurantinins A and B, Produced by Bacillus aurantinus. (1988) (0)
- Synthesis and Biological Evaluation of Novel 4′′-Alkoxy Avermectin Derivatives. (2004) (0)
- Complex of a chitinase with the natural product cyclopentapeptide argadin from Clonostachys (2002) (0)
- Contents Vol. 79, 2007 (2007) (0)
- P-525 Efficient production of the anti-HIV protein actinohivin in recombinant Streptomyces strain (2006) (0)
- Pyridindolols K1 and K2, new alkaloids from Streptomyces sp. K93-0711. (1997) (0)
- (+)-Trienomycins A (Ia), B (Ib), C (Ic), and F (Id) and (+)- Mycotrienins I (II) and II (Ie): Relative and Absolute Stereochemistry. (1997) (0)
- [Suppression of endotoxic shock by macrolide derivative, EM900, and the mechanism involved in the process]. (2009) (0)
- Selection Media for beauveriolide I or III and process for selectively preparing these substances (2001) (0)
- SYNTHESIS OF ANOMERIC METHYL-6-O-(L-MYCAROSYL)-BETA-D-GLUCOSAMINIDES (1973) (0)
- Corrigendum: Streptomyces lactacystinicus sp. nov. and Streptomyces cyslabdanicus sp. nov., producing lactacystin and cyslabdan, respectively (2017) (0)
- Aogacillins A (Ia) and B (Ib) Produced by Simplicillium sp. FKI‐5985: New Circumventors of Arbekacin Resistance in MRSA. (2014) (0)
- CARBOHYDRATE MIMICRY IN COMPLEXES OF CHITINASES WITH NATURAL PRODUCT CYCLOPENTAPEPTIDE INHIBITORS (2002) (0)
- Antibiotics. Structure, Elucidation, and Production of New Substances Using Biosynthetic Means (1988) (0)
- 62(P-35) Lanosterol Synthase Inhibitors from Streptomyces sp. K99-5041 (2002) (0)
- Serratia marcescens Chitinase B complexed with azide inhibitor and quinoline compound (2013) (0)
- Transcriptional analysis of genes encoding proteins significantly increased in Kitasatospora setae KM-6054(T) under submerged culture. (2014) (0)
- Welcoming the addition of the SAJ to the JA publishing enterprise (2011) (0)
- アクチノヒビン多量体を含む融合タンパク質からなる抗ＨＩＶ薬、これを構成するポリペプチド、ポリペプチドをコードする遺伝子および抗ＨＩＶ薬の製造法 (2008) (0)
- Foreword Celebrating the career of Professor Arnold Demain (2010) (0)
- An Effect of Non-Antibiotic Macrolide EM900 in Obese Asthma Model (2020) (0)
- Letter: Fast liquid chromatography of macrolide antibiotics. (1973) (0)
- PC82 ISOLATION, STRUCTURAL AND SYNTHETIC STUDIES ON JIETACINS A AND B, NEW NEMATOCIDAL ANTIBIOTICS (1988) (0)
- Synthesis and Biological Activities of Novel 4′′-Alkylidene Avermectin Derivatives. (2004) (0)
- The erythromycin derivatives and process for their preparation (1986) (0)
- Tolyprolinol, a new dipeptide from Tolypocladium sp. FKI-7981 (2018) (0)
- Afidopyropen, a novel insecticide originating from microbial secondary extracts (2022) (0)
- A New Antimicrobial Antibiotic from Actinoplanes capillaceus sp. K95‐5561T (2001) (0)
- P-490 Total synthesis of (+)-guadinomines C, potent, selective inhibitors of Type III secretion system. Determination of the absolute configurations (2006) (0)
- Antibiotics for Emerging and Re-emerging Diseases (2015) (0)
- Dinapinones, Novel Inhibitors of Triacylglycerol Synthesis in Mammalian Cells, Produced by Penicillium pinophilum FKI-3864. (2011) (0)
- P-523 SELECTIVITY OF BEAUVERIOLIDE ANALOGS, ACAT INHIBITORS, TO THE ISOZYMES (2006) (0)
- New antibiotic am-1042 (1977) (0)
- A microorganism for the selective production of a specific component of avermectin and selective production method for this. (1990) (0)
- CHEMISTRY OF LEUCOMYCINS PART 11, CHEMICAL TRANSFORMATION OF A BASIC MACROLIDE TO A NEUTRAL MACROLIDE (1974) (0)
- P9 The potency of a new erythromycin (EM) derivative, EM900, to reduce the density of the nasopharyngeal Streptococcus pneumoniae colonization (2013) (0)
- Chloropeptins, New Anti-HIV Antibiotics Inhibiting gp120-CD4 Binding from Streptomyces sp. Part 2. Structure Elucidation of Chloropeptin I. (2010) (0)
- Pyripyropenes , Novel ACATInhibitors Produced by Aspergillus fumigatus IV . Structure Elucidation of Pyripyropenes Mto (2006) (0)
- 5,9-Diacetyl (3,6)bicycloleuconolide A3 (1977) (0)
- Serratia marcescens Chitinase B, tetragonal form (2013) (0)
- Anthelmintic substance fki-1033 and methods for production thereof (2002) (0)
- Complex of a chitinase with the natural product cyclopentapeptide argifin from Gliocladium (2002) (0)
- Pyrizomicin A and B: structure and bioactivity of new thiazolyl pyridines from Lechevalieria aerocolonigenes K10-0216 (2018) (0)
- Synthesis and stereochemical determination of an antiparasitic pseudo-aminal type monoterpene indole alkaloid (2016) (0)
- Total Synthesis of Pinellic Acid, a Potent Oral Adjuvant for Nasal Influenza Vaccine. Determination of the Relative and Absolute Configuration. (2002) (0)
- Identification and heterologous expression of the actinoallolide biosynthetic gene cluster (2018) (0)
- Crystal Structure of PtlH with Fe/alpha ketoglutarate bound (2007) (0)
- Compound FO-1289 and a process for its preparation (1994) (0)
- Antimalarial troponoids, puberulic acid and viticolins; divergent synthesis and structure-activity relationship studies (2017) (0)
- Acknowledgement to Referees for Pharmacology 2011 (2011) (0)
- P-539 ISOBISVERTINOL, A NOVEL INHIBITOR OF LIPID DROPLET ACCUMULATION IN MOUSE MACROPHAGES PRODUCED BY Aspergillus sp. FKI-1746 (2006) (0)
- Synthetic Study of α‐Pyrone Meroterpenoids, Pyripyropens (1998) (0)
- THE SYNTHESIS OF ANOMERIC METHYL-4-O-L-MYCAROSYL-BETA-D-MYCAMINOSIDES (1973) (0)
- Mechanism of the motor-stimulating action of motilin and motilide (EM523) in the dog (1992) (0)
- Tensidols, New Potentiators of Antifungal Miconazole Activity, Produced by Aspergillus niger FKI-2342. (2007) (0)
- A process for preparing avermectin derivatives (2001) (0)
- Synthesis and Biological Activities of New HMG‐COA Synthase Inhibitors: 2‐Oxetanones with a Side Chain Containing Biphenyl, Terphenyl, or Phenylpyridine. (1994) (0)
- A NEW PEPTIDE ANTIBIOTIC BY STREPTOMYCES SP (2006) (0)
- P-41 Novel Anti-FLU Antibiotics, Wickerols, Produced by Trichoderma sp.(Poster Presentation) (2008) (0)
- Use of a Chiral Praseodymium Shift Reagent in Predicting the Complete Stereostructure of Glisoprenin A (2005) (0)
- Pyripyropenes, Novel Inhibitors of Acyl-CoA: Cholesterol Acyltransferase Produced by Aspergillus fumigatus. Part 1. Production, Isolation, and Biological Properties. (1994) (0)
- Isolation, Total Synthesis and Determination of the Absolute Configuration of Guadinomines; Potent Inhibitors of a Bacterial Type III Secretion System (2012) (0)
- A Concise Total Synthesis of Dehydroantofine and the Antimalarial Activity against Chloroquine-Resistant P. falciparum. (2021) (0)
- Synthesis and insecticidal efficacy of pyripyropene derivatives focusing on the C-1, C-7, and C-11 positions’ substituent groups (2018) (0)
- Takanawaenes, Novel Antifungal Antibiotics Produced by Streptomyces sp. K99-5278. Part 1. Taxonomy, Fermentation, Isolation and Biological Properties. (2003) (0)
- Crystal structure of anti-HIV actinohivin in complex with alpha-1,2-mannobiose (P 2 21 21 form) (2013) (0)
- Anthelmintic substance FKI-1033 and process for production thereof. (2002) (0)
- Metapochonia hahajimaensis (Clavicipitaceae, Hypocreales), a new species from soil in Hahajima Island, Tokyo, Japan (2020) (0)
- Enantioselective Total Synthesis of Atpenin A5. (2009) (0)
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